IP Library Granted Patent US 9,012,479
Granted Patent B2
US 9,012,479 · App. 14/047,688 · Granted Apr 21, 2015

Pyrazolylaminopyridines as inhibitors of FAK

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Quick Facts
Patent No.
US 9,012,479
App. No.
14/047,688
Granted
Apr 21, 2015
Kind
B2
Abstract

The present invention relates to a compound of formula (I): or a pharmaceutically acceptable salt thereof, wherein R 1 , R 2 , R 3 , R 11 , R 12 , R 13 , Q, Z, and p are as described herein. Compounds of the present invention are useful for the treatment of cancers.

Claims (14)

1. A compound that is:

2-[(5-Chloro-2-{[3-methyl-1-(1-methylethyl)-1H-pyrazol-5-yl]amino}-4-pyridinyl)amino]-N-(methyloxy)benzamide;

or a pharmaceutically acceptable salt thereof.

2. The compound of claim 1 that is:

2-[(5-Chloro-2-{[3-methyl-1-(1-methylethyl)-1H-pyrazol-5-yl]amino}-4-pyridinyl)amino]-N-(methyloxy)benzamide.

3. A pharmaceutical composition comprising a compound according to claim 1 and one or more pharmaceutically acceptable carriers, diluents or excipients.

4. A pharmaceutical composition comprising the compound according to claim 2 and one or more pharmaceutically acceptable carriers, diluents or excipients.

5. A process for preparing a pharmaceutical composition containing a pharmaceutically acceptable carrier and the compound of claim 1 which process comprises bringing the compound of claim 1 into association with one or more pharmaceutically acceptable carriers, diluents or excipients.

6. A pharmaceutical composition according to claim 3 , wherein the composition is in tablet form.

7. A pharmaceutical composition according to claim 4 , wherein the composition is in tablet form.

8. A compound that is:

9. A pharmaceutical composition comprising the compound according to claim 8 and one or more pharmaceutically acceptable carriers, diluents or excipients.

10. A pharmaceutical composition according to claim 9 , wherein the composition is in tablet form.

11. A process for preparing a pharmaceutical composition containing a pharmaceutically acceptable carrier and the compound of claim 8 which process comprises bringing the compound of claim 8 into association with the pharmaceutically acceptable carrier.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 14, 2015
From: ADAMS, JERRY LEROY; FAITG, THOMAS H.; JOHNSON, NEIL W.; LIN, HONG; PENG, XIN
To: GLAXOSMITHKLINE LLC
Reel/Frame 034705/0551 →