IP Library Granted Patent US 10,058,522
Granted Patent B2
US 10,058,522 · App. 14/113,547 · Granted Aug 28, 2018

Oxidative retinal diseases

Inventor: Mikhail S. Shchepinov (Kingston Upon Thames, GB)
Assignee: Retrotope, Inc.
A61K31/201A61K31/12A61K31/122A61K31/202A61K31/231A61K31/355A61K31/375A61K31/66
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Quick Facts
Patent No.
US 10,058,522
App. No.
14/113,547
Granted
Aug 28, 2018
Kind
B2
Abstract

Some aspects of the invention provide for a method of treating Wet and/or Dry Age-related Macular Degeneration, Retinitis Pigmentosa, Diabetic Retinopathy, cataracts, and/or Stargardt Disease using polyunsaturated fatty acids which are modified in certain positions to attenuate oxidative damage by Reactive Oxygen Species (ROS) and/or suppress the rate of formation of reactive products and toxic compounds.

Claims (23)

1. A method of treating or inhibiting progression of an oxidative retinal disease, comprising:

treating a patient having a Wet or Dry Age-related Macular Degeneration (AMD), Retinitis Pigmentosa (RP), Diabetic Retinopathy (DR), or Stargardt Disease (SD) over a time period by repeatedly administering an effective amount of a polyunsaturated fatty acid or fatty acid ester during a treatment period, wherein the polyunsaturated fatty acid or fatty acid ester is deuterated at one or more bis-allylic positions, wherein the amount of deuterated polyunsaturated fatty acid or fatty acid ester administered to or ingested by the patient is in the range of about 5% to about 75% of the total amount of polyunsaturated fatty acid or fatty acid ester administered to or ingested by the patient, and wherein over the treatment period a significant amount of deuterated polyunsaturated fatty acid or fatty acid ester is incorporated into the patient's eye such that the amount of deuterated polyunsaturated fatty acid or fatty acid ester in the patient's eye is sufficient to reduce or prevent autoxidation and cancel toxicity of undeuterated polyunsaturated fatty acid or fatty acid ester in the patient's eye.

2. The method of claim 1 , wherein the at least one deuterium atom is present at a level greater than 0.02%.

3. The method of claim 2 , wherein over the treatment period the deuterated polyunsaturated fatty acid or fatty acid ester comprises between about 10% and 50% of the total amount of fatty acids or fatty acid esters in the patient's eye.

4. The method of claim 2 , wherein over the treatment period the deuterated polyunsaturated fatty acid or fatty acid ester comprises between about 10% and 30% of the total amount of fatty acids or fatty acid esters in the patient's eye.

5. The method of claim 2 , wherein over the treatment period the deuterated polyunsaturated fatty acid or fatty acid ester comprises about 20% to about 50% of the total amount of fatty acids or fatty acid esters in the patient's eye.

6. The method of claim 2 , wherein the deuterated polyunsaturated-fatty acid or fatty acid ester is an omega-3 fatty acid or fatty acid ester, or an omega-6 fatty acid or fatty acid ester.

7. The method of claim 6 , wherein the deuterated polyunsaturated fatty acid or fatty acid ester is selected from the group consisting of 11,11-D2-linolenic acid, 14,14-D2-linolenic acid, 11,11,14,14-D4-linolenic acid, 11,11-D2-linoleic acid, 11-D-linolenic acid, 14-D-linolenic acid, 11,14-D2-linolenic acid, and 11-D-linoleic acid.

8. The method of claim 6 , wherein the deuterated polyunsaturated fatty acid or fatty acid ester is further deuterated at at least one saturated methylene group that is adjacent to a second saturated methylene group.

9. The method of claim 1 , wherein the ester is a triglyceride, diglyceride, or monoglyceride.

10. The method of claim 1 further comprising co-administering an antioxidant.

11. The method of claim 10 , wherein the antioxidant is idebenone, mitoquinone, mitoquinol, vitamin C, or vitamin E.

12. The method of claim 1 , wherein the deuterated polyunsaturated fatty acid or fatty acid ester is administered topically to the patient's eye.

13. The method of claim 1 , wherein the deuterated polyunsaturated fatty acid or fatty acid ester is administered orally.

14. The method of claim 1 , wherein the deuterated polyunsaturated fatty acid or fatty acid ester is arachidonic acid or an ester thereof.

15. The method of claim 1 , wherein the deuterated fatty acid or fatty acid ester is eicosapentaenoic acid or an ester thereof.

16. The method of claim 1 , wherein the deuterated fatty acid or fatty acid ester is docosahexaenoic acid or an ester thereof.

17. The method of claim 1 , wherein the deuterated fatty acid or fatty acid ester is a linoleic acid or an ester thereof.

18. The method of claim 1 , wherein the deuterated fatty acid or fatty acid ester is a linolenic acid or an ester thereof.

19. The method of claim 1 , wherein the deuterated fatty acid or fatty acid ester is an ethyl ester.

20. The method of claim 1 , wherein the amount of deuterated polyunsaturated fatty acid or fatty acid ester administered to or ingested by the patient is in the range of about 0.1 mg/kg to about 100 mg/kg per day.

21. The method of claim 1 , wherein the deuterated polyunsaturated fatty acid or fatty acid ester is 11,11-D2-linoleic acid or ethyl ester thereof.

22. The method of claim 1 , wherein the deuterated polyunsaturated fatty acid or fatty acid ester is 11,11,14,14-D4-linolenic acid or ethyl ester thereof.

Assignments (5)
RELEASE OF SECURITY INTEREST Recorded Sep 9, 2022
From: RTMFP ENTERPRISES INC.
To: RETROTOPE, INC.
Reel/Frame 061403/0670 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Sep 9, 2022
From: RETROTOPE, INC.
To: RTMFP ENTERPRISES INC.
Reel/Frame 061403/0835 →
CHANGE OF NAME Recorded Sep 9, 2022
From: RTMFP ENTERPRISES INC.
To: BIOJIVA LLC
Reel/Frame 061405/0819 →
SECURITY INTEREST Recorded Mar 30, 2022
From: RETROTOPE, INC.
To: RTMFP ENTERPRISES, INC.
Reel/Frame 059442/0414 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Nov 8, 2016
From: SHCHEPINOV, MIKHAIL SERGEEVICH
To: RETROTOPE, INC.
Reel/Frame 040258/0507 →
Continuity (2)
Provisional Application 61479281 · Apr 26, 2011
Related Publication 20140044693A1 · Feb 13, 2014
Cited By (2)
US 12,673,037 US 12,697,319