IP Library Granted Patent US 8,969,420
Granted Patent B2
US 8,969,420 · App. 14/155,288 · Granted Mar 3, 2015

Treatment of pervasive developmental disorders with redox-active therapeutics

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Quick Facts
Patent No.
US 8,969,420
App. No.
14/155,288
Granted
Mar 3, 2015
Kind
B2
Abstract

Methods of treating or suppressing pervasive developmental disorders (PDDs) including; autistic disorder, Asperger's syndrome, childhood disintegrative disorder (CDD), Rett's disorder, and PDD—not otherwise specified (PDD-NOS) or attention deficit/hyperactivity disorder (ADHD) comprising administering to a subject in need thereof a therapeutically effective amount of one or more compounds as disclosed herein.

Claims (28)

1. A method of reducing a symptom associated with, or for treating or suppressing a pervasive developmental disorder (PDD) or attention deficit/hyperactivity disorder (ADHD) in a patient in need of such treatment, comprising administering to the patient a therapeutically or physiologically effective amount of a compound of Formula III,

wherein,

the bonds indicated with a dashed line are independently single bonds or double bonds; and

R 1 , R 2 , and R 3 are independently selected from the group consisting of H, (C 1 -C 6 )alkyl, (C 1 -C 6 )haloalkyl, (C 1 -C 6 )alkoxy, halogen and CN;

or a stereoisomer, a mixture of stereoisomers, a solvate or a hydrate thereof.

2. The method according to claim 1 , wherein the compound of Formula III has the formula:

or a stereoisomer, a mixture of stereoisomers, a solvate or a hydrate thereof.

3. The method according to claim 2 , wherein the compound is:

or a stereoisomer, or a mixture of stereoisomers, a solvate or a hydrate thereof.

4. The method of claim 1 , wherein the bonds indicated with a dashed line are all single bonds.

5. The method of claim 1 , wherein the bonds indicated with a dashed line are all double bonds.

6. The method of claim 3 , wherein the bonds indicated with a dashed line are all single bonds.

7. The method of claim 3 , wherein the bonds indicated with a dashed line are all double bonds.

8. The method of claim 1 , wherein R 1 , R 2 , and R 3 are independently selected from the group consisting of H, (C 1 -C 6 )alkyl, and (C 1 -C 6 )alkoxy.

9. The method of claim 1 , wherein R 1 , R 2 , and R 3 are independently selected from (C 1 -C 4 )alkyl.

10. The method of claim 1 , wherein R 1 , R 2 , and R 3 are methyl.

11. The method of claim 1 , wherein at least one of R 1 , R 2 , and R 3 is not methyl.

12. The method of claim 1 , wherein R 1 and R 2 are methoxy, and R 3 is methyl.

13. The method of claim 4 , wherein the method is for treating the PDD, wherein the PDD is autistic spectrum disorder (ASD).

14. The method according to claim 5 , wherein the method is for treating the PDD, wherein the PDD is autistic spectrum disorder (ASD).

15. The method of claim 6 , wherein the method is for treating the PDD, wherein the PDD is autistic spectrum disorder (ASD).

16. The method according to claim 7 , wherein the method is for treating the PDD, wherein the PDD is autistic spectrum disorder (ASD).

17. The method according to claim 4 , wherein the method is for treating attention deficit/hyperactivity disorder (ADHD).

18. The method according to claim 5 , wherein the method is for treating attention deficit/hyperactivity disorder (ADHD).

19. The method according to claim 6 , wherein the method is for treating attention deficit/hyperactivity disorder (ADHD).

20. The method according to claim 7 , wherein the method is for treating attention deficit/hyperactivity disorder (ADHD).

21. The method according to claim 6 , wherein the method is for treating Rett's disorder.

22. The method according to claim 7 , wherein the method is for treating Rett's disorder.

Assignments (3)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Nov 15, 2019
From: BIOELECTRON TECHNOLOGY CORPORATION
To: PTC THERAPEUTICS, INC.
Reel/Frame 051041/0478 →
CHANGE OF NAME Recorded Feb 8, 2017
From: EDISON PHARMACEUTICALS, INC.
To: BIOELECTRON TECHNOLOGY CORPORATION
Reel/Frame 041660/0644 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 19, 2014
From: MILLER, GUY M.; KHEIFETS, VIKTORIA
To: EDISON PHARMACEUTICALS, INC.
Reel/Frame 032249/0631 →