IP Library Granted Patent US 9,533,984
Granted Patent B2
US 9,533,984 · App. 14/256,438 · Granted Jan 3, 2017

Bicyclic heterocycles as FGFR inhibitors

Inventors: Yaping Sun (Hockessin, DE); Liang Lu (Hockessin, DE); Wenqing Yao (Chadds Ford, PA); Jincong Zhuo (Garnet Valley, PA); Liangxing Wu (Wilmington, PA); Meizhong Xu (Hockessin, DE); Ding-Quan Qian (Newark, DE); Chunhong He (Chadds Ford, PA); Fenglei Zhang (Ambler, PA)
Assignees: Incyte Holdings Corporation; Incyte Corporation
C07D471/04
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Quick Facts
Patent No.
US 9,533,984
App. No.
14/256,438
Granted
Jan 3, 2017
Kind
B2
Abstract

The present invention relates to bicyclic heterocycles, and pharmaceutical compositions of the same, that are inhibitors of one or more FGFR enzymes and are useful in the treatment of FGFR-associated diseases such as cancer.

Claims (7)

1. A compound which is:

2′-(2,6-difluoro-3,5-dimethoxyphenyl)-6′-[(2-morpholin-4-ylethyl)amino]-1′,2′-dihydro-3′H-spiro[cyclopropane-1,4′-[2,4]naphthyridin]-3′-one or a pharmaceutically acceptable salt thereof.

2. A pharmaceutical composition comprising the compound of claim 1 , or a pharmaceutically acceptable salt thereof, and at least one pharmaceutically acceptable carrier or excipient.

3. A compound which is 2′-( 2 , 6 -difluoro- 3 , 5 -dimethoxyphenyl)- 6 ′-[(2-morpholin-4-ylethyl)amino]-1′,2′-dihydro-3′H-spiro]cyclopropane-1,4′-[2,7]naphthyridin]-3′-one.

4. A pharmaceutical composition comprising the compound of claim 3 and at least one pharmaceutically acceptable carrier or excipient.

5. A pharmaceutically acceptable salt of 2′-(2,6-difluoro-3,5-dimethoxyphenyl) -6′-[(2-morpholin-4-ylethyl)amino]-1′,2′-dihydro-3′H -spiro[cyclopropane-1,4′-[2,7]naphthyridin]-3′-one.

6. A pharmaceutical composition comprising the pharmaceutically acceptable salt of claim 5 , and at least one pharmaceutically accceptable carrier or excipient.

Assignments (5)
CORRECTIVE ASSIGNMENT TO CORRECT THE RECEIVING PARTY INFORMATION PREVIOUSLY RECORDED ON REEL 035920 FRAME 0576. ASSIGNOR(S) HEREBY CONFIRMS THE RECEIVING PARTY NAME SHOULD BE RECORDED AS TWO PARTIES. Recorded Jul 2, 2015
From: INCYTE CORPORATION
To: INCYTE HOLDINGS CORPORATION; INCYTE CORPORATION
Reel/Frame 036054/0740 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jun 16, 2015
From: INCYTE CORPORATION
To: INCYTE HOLDINGS CORPORATION AND INCYTE CORPORATION
Reel/Frame 035920/0576 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded May 6, 2014
From: HE, CHUNHONG
To: INCYTE CORPORATION
Reel/Frame 032830/0181 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 18, 2014
From: SUN, YAPING; LU, LIANG; YAO, WENQING; ZHUO, JINCONG; WU, LIANGXING; XU, MEIZHONG; QIAN, DING-QUAN; ZHANG, FENGLEI
To: INCYTE CORPORATION
Reel/Frame 032710/0317 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 18, 2014
From: SUN, YAPING; LU, LIANG; YAO, WENQING; ZHUO, JINCONG; WU, LIANGXING; XU, MEIZHONG; QIAN, DING-QUAN; ZHANG, FENGLEI
To: INCYTE CORPORATION
Reel/Frame 032710/0479 →
Continuity (2)
Provisional Application 61813782 · Apr 19, 2013
Related Publication 20140315902A1 · Oct 23, 2014