IP Library Granted Patent US 10,016,437
Granted Patent B2
US 10,016,437 · App. 14/287,017 · Granted Jul 10, 2018

Drug combinations and uses in treating a coughing condition

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Quick Facts
Patent No.
US 10,016,437
App. No.
14/287,017
Granted
Jul 10, 2018
Kind
B2
Abstract

The present specification discloses compositions comprising a plurality of therapeutic compound having antitussive activity and methods and uses for treating a coughing condition with such compositions.

Claims (10)

1. An oral pharmaceutical composition comprising 0.5 mg/mL to 10 mg/mL of Theobromine, 0.25 mg/mL to 7.5 mg/mL of Diphenhydramine, and 0.1 mg/mL to 5 mg/mL of Phenylephrine, wherein the pharmaceutical composition does not include a non-opiate antitussive agent and wherein the therapeutically-effective amount of the theobromine is at least 60 mg/day and at most 150 mg/day.

2. The oral pharmaceutical composition according to claim 1 , wherein the oral pharmaceutical composition comprises 0.5 mg/mL to 6 mg/mL of Theobromine, 0.5 mg/mL to 5 mg/mL of Diphenhydramine, and 0.1 mg/mL to 2 mg/mL of Phenylephrine.

3. The oral pharmaceutical composition according to claim 2 , wherein the oral pharmaceutical composition comprises 1 mg/mL to 3 mg/mL of Theobromine, 1 mg/mL to 3 mg/mL of Diphenhydramine, and 0.1 mg/mL to 1 mg/mL of Phenylephrine.

4. The oral pharmaceutical composition according to claim 3 , wherein the oral pharmaceutical composition comprises 2 mg/mL of Theobromine, 1.25 mg/mL of Diphenhydramine, and 0.5 mg/mL of Phenylephrine.

5. A method of treating cough due to a cold, the method comprising the step of administering a therapeutically-effective amount of the oral pharmaceutical composition of claim 1 .

6. The method according to claim 5 , wherein the oral pharmaceutical composition comprises 0.5 mg/mL to 6 mg/mL of Theobromine, 0.5 mg/mL to 5 mg/mL of Diphenhydramine, and 0.1 mg/mL to 2 mg/mL of Phenylephrine.

7. The method according to claim 6 , wherein the oral pharmaceutical composition comprises 1 mg/mL to 3 mg/mL of, 1 mg/mL to 3 mg/mL of Diphenhydramine, and 0.1 mg/mL to 1 mg/mL of Phenylephrine.

8. The method according to claim 7 , wherein the oral pharmaceutical composition comprises 2 mg/mL of Theobromine, 1.25 mg/mL of Diphenhydramine, and 0.5 mg/mL of Phenylephrine.

9. The method according to claim 5 , wherein the therapeutically-effective amount of the oral pharmaceutical composition comprises between 60 mg/day and 150 mg/day of Theobromine, 20 mg/day and 100 mg/day of Diphenhydramine, and 5 mg/day and 50 mg/day of Phenylephrine.

10. The method according to claim 9 , wherein the therapeutically-effective amount of the oral pharmaceutical composition comprises between 60 mg/day and 120 mg/day of Theobromine, 37.5 mg/day and 75 mg/day of Diphenhydramine, and 15 mg/day and 30 mg/day of Phenylephrine.

Assignments (7)
SECURITY INTEREST Recorded Jun 10, 2025
From: BIOMAX HEALTH PRODUCTS, LLC; INFIRST HEALTHCARE INC.
To: AXOS BANK
Reel/Frame 071376/0454 →
CORRECTIVE ASSIGNMENT TO CORRECT THE SECOND CONVEYING PARTY NAME PREVIOUSLY RECORDED ON REEL 67526 FRAME 735. ASSIGNOR(S) HEREBY CONFIRMS THE SECURITY INTEREST. Recorded Jun 5, 2024
From: BIOMAX HEALTH PRODUCTS, LLC; INFIRST HEALTHCARE INC.
To: HAYFIN SERVICES LLP, AS THE COLLATERAL AGENT
Reel/Frame 067636/0356 →
SECURITY INTEREST Recorded Apr 23, 2024
From: BIOMAX HEALTH PRODUCTS, LLC; LNFIRST HEALTHCARE LNC.
To: HAYFIN SERVICES LLP, AS THE COLLATERAL AGENT
Reel/Frame 067526/0735 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Dec 7, 2023
From: INFIRST HEALTHCARE LIMITED
To: INFIRST HEALTHCARE INC.
Reel/Frame 065801/0688 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 13, 2016
From: BREW, JOHN; BANNISTER, ROBIN MARK
To: BIOCOPEA LIMITED
Reel/Frame 038274/0051 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Sep 15, 2014
From: BIOCOPEA LIMITED
To: RESPICOPEA LIMITED
Reel/Frame 033740/0403 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Sep 15, 2014
From: RESPICOPEA LIMITED
To: INFIRST HEALTHCARE LIMITED
Reel/Frame 033740/0512 →