IP Library Granted Patent US 10,392,439
Granted Patent B2
US 10,392,439 · App. 14/294,544 · Granted Aug 27, 2019

Methods for treating allergy and enhancing allergen-specific immunotherapy by administering an IL-4R inhibitor

Inventors: Neil Stahl (Carmel, NY); Jamie M Orengo (Cortlandt Manor, NY); Andrew J. Murphy (Croton-on-Hudson, NY); Namita Gandhi (New York, NY); Neil Graham (Croton-on-Hudson, NY)
Assignee: Regeneron Pharmaceuticals, Inc.
C07K16/2866A61K45/06A61K2039/505A61K2039/577
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Quick Facts
Patent No.
US 10,392,439
App. No.
14/294,544
Granted
Aug 27, 2019
Kind
B2
Abstract

The present invention provides methods for treating, preventing or reducing the severity of allergic reactions. The present invention also provides methods for enhancing the efficacy and/or safety of an allergen-specific immunotherapy (SIT) regimen. The methods of the present invention comprise administering to a subject in need thereof a therapeutic composition comprising an interleukin-4 receptor (IL-4Rα) antagonist such as an anti-IL-4Rα antibody.

Claims (11)

1. A method for treating or reducing the severity of an allergic reaction, the method comprising administering a therapeutically effective amount of a pharmaceutical composition comprising an interleukin-4 receptor (IL-4R) antagonist to a subject in need thereof, wherein the IL-4R antagonist is an antibody or antigen-binding fragment thereof, wherein the antibody or antigen-binding fragment thereof comprises three heavy chain complementarity determining regions (HCDRs) (HCDR1, HCDR2 and HCDR3) and three light chain complementarity determining regions (LCDRs) (LCDR1, LCDR2 and LCDR3), wherein the HCDR1 comprises the amino acid sequence of SEQ ID NO:3; the HCDR2 comprises the amino acid sequence of SEQ ID NO:4; the HCDR3 comprises the amino acid sequence of SEQ ID NO:5; the LCDR1 comprises the amino acid sequence of SEQ ID NO:6; the LCDR2 comprises the amino acid sequence of SEQ ID NO:7; and the LCDR3 comprises the amino acid sequence of SEQ ID NO:8, wherein the allergic reaction is triggered by a food allergen, and wherein the composition is administered to the subject less than 4 hours before allergen exposure, less than 4 hours after allergen exposure, or less than 4 hours after manifestation of one or more allergic symptoms in the subject.

2. The method of claim 1 , wherein the antibody or antigen-binding fragment thereof binds IL-4Rα and prevents the interaction of IL-4 and/or IL-13 with a type 1 or type 2 IL-4 receptor.

3. The method of claim 2 , wherein the antibody or antigen-binding fragment thereof prevents the interaction of IL-4 with both type 1 and type 2 IL-4 receptors.

4. The method of claim 3 , wherein the antibody or antigen-binding fragment thereof comprises a heavy chain variable region (HCVR) comprising the amino acid sequence of SEQ ID NO:1 and a light chain variable region (LCVR) comprising the amino acid sequence of SEQ ID NO:2.

5. The method of claim 1 , wherein the IL-4R antagonist is dupilumab or a bioequivalent thereof.

6. The method of claim 1 , wherein the allergic symptoms are selected from the group consisting of urticaria, angioedema, rhinitis, asthma, vomiting, respiratory compromise, swollen lips, swollen tongue, and reduced blood pressure.

7. The method of claim 1 , wherein the allergic reaction is anaphylaxis.

8. The method of claim 1 , wherein the food allergen is selected from the group consisting of dairy product, egg, wheat, soy, fish, shellfish, peanut and tree nut.

9. The method of claim 1 , wherein the pharmaceutical composition is administered to the subject as part of a therapeutic dosing regimen comprising once a week, once every two weeks, once every three weeks, or once a month dosing of the pharmaceutical composition.

10. The method of claim 1 , wherein the pharmaceutical composition is administered to the subject in combination with a second therapeutic agent selected from the group consisting of steroids, antihistamines, decongestants, and anti-IgE agents.

11. The method of claim 2 , wherein the antibody or antigen-binding fragment thereof prevents the interaction of IL-13 with a type 2 IL-4 receptor.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jun 3, 2014
From: STAHL, NEIL; ORENGO, JAMIE M.; MURPHY, ANDREW J.; GANDHI, NAMITA; GRAHAM, NEIL
To: REGENERON PHARMACEUTICALS, INC.
Reel/Frame 033019/0840 →
Continuity (2)
Provisional Application 61830919 · Jun 4, 2013
Related Publication 20140356372A1 · Dec 4, 2014
Cited By (7)
US 12,291,571 US 12,440,562 US 12,502,429 US 12,685,771 US 12,702,709 US 12,708,666 US 12,709,642