IP Library Granted Patent US 11,554,229
Granted Patent B2
US 11,554,229 · App. 14/315,132 · Granted Jan 17, 2023

Nasal administration

Inventors: Per Gisle Djupesland (Oslo, NO); Ramy A. Mahmoud (Skillman, NJ); John Messina (Downingtown, PA)
Assignee: OptiNose Inc.
A61M15/08A61M15/0098A61M16/0057A61M16/14A61M16/20A61M11/003A61M15/009A61M15/0021A61M15/0041A61M16/0045A61M16/107A61M16/1055A61M2202/0225A61M2202/0275A61M2202/0468A61M2202/064A61M2205/3324A61M2205/3334
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Quick Facts
Patent No.
US 11,554,229
App. No.
14/315,132
Granted
Jan 17, 2023
Kind
B2
Abstract

A method of delivering a substance, such as one or more of a triptan, a nasal steroid or carbon dioxide gas, to the nasal cavity of a subject, in particular for the treatment of headaches, for example, migraine, or rhinosinusitis, for example, chronic rhinosinusitis, optionally with polyps, the method comprising the steps of fitting a nosepiece to one nostril of the subject, delivering the substance through the nosepiece to the posterior region of the nasal cavity of the subject.

Claims (32)

1. A method of treating nasal polyps in a patient comprising:

placing a nosepiece into a first nostril of the patient;

placing a mouthpiece into a mouth of the patient, the mouthpiece being fluidly connected to the nosepiece, wherein exhalation by the patient into the mouthpiece and out of the nosepiece produces a bi-directional fluid flow of exhalation air into a first nasal passageway of the patient and out of a second nasal passageway of the patient;

administering fluticasone during exhalation by the patient through the nosepiece;

delivering carbon dioxide during exhalation by the patient through the nosepiece, to a location at an upper posterior region of the first nasal passageway of the patient; and

reducing a pH at the location at the upper posterior region of the first nasal passageway of the patient by an amount ranging from about 0.1 pH units to about 0.2 pH units by controlling the fluid flow to deliver the carbon dioxide at a concentration of from about 5% vol/vol to about 6% vol/vol carbon dioxide and at a fluid flow rate of at least 20 L/min for a duration of from about 2 seconds to about 3 seconds, wherein the carbon dioxide is delivered before or at the same time as the fluticasone.

2. The method of claim 1 , wherein the fluticasone is fluticasone propionate.

3. The method of claim 1 , wherein the fluticasone is administered as a liquid aerosol.

4. The method of claim 1 , wherein the fluticasone is administered in an amount of about 400 μg b.i.d.

5. The method of claim 1 , wherein the fluticasone is administered in an amount of 100 μg to 400 μg b.i.d.

6. The method of claim 1 , wherein the fluticasone is administered in an amount of at least 200 μg daily.

7. The method of claim 1 , wherein the fluticasone is administered in an amount of at least 400 μg daily.

8. The method of claim 1 , wherein the fluticasone is administered in an amount of at least 200 μg daily delivered in two doses.

9. The method of claim 1 , wherein the fluticasone is administered in an amount of at least 400 μg daily delivered in two doses.

10. The method of claim 1 , wherein the fluticasone is fluticasone propionate administered as a liquid aerosol in an amount of 100 μg to 400 μg b.i.d.

11. The method of claim 1 , wherein the fluticasone is fluticasone propionate administered as a liquid aerosol in an amount of at least 200 μg b.i.d.

12. A method of treating chronic rhinosinusitis with or without nasal polyps in a patient comprising:

placing a nosepiece into a first nostril of the patient;

placing a mouthpiece into a mouth of the patient, the mouthpiece being fluidly connected to the nosepiece, wherein exhalation by the patient into the mouthpiece and out of the nosepiece produces a bi-directional fluid flow of exhalation air into a first nasal passageway of the patient and out of a second nasal passageway of the patient;

administering fluticasone during exhalation by the patient through the nosepiece;

delivering carbon dioxide during exhalation by the patient through the nosepiece, to a location at an upper posterior region of the first nasal passageway of the patient; and

reducing a pH at the location at the upper posterior region of the first nasal passageway of the patient by an amount ranging from about 0.1 pH units to about 0.2 pH units by controlling the fluid flow to deliver the carbon dioxide at a concentration of from about 5% vol/vol to about 6% vol/vol carbon dioxide and at a fluid flow rate of at least 20 L/min for a duration of from about 2 seconds to about 3 seconds, wherein the carbon dioxide is delivered before or at the same time as the fluticasone.

13. The method of claim 12 , wherein the fluticasone is fluticasone propionate.

14. The method of claim 12 , wherein the fluticasone propionate is administered as a liquid aerosol.

15. The method of claim 12 , wherein the fluticasone propionate is administered in an amount of about 400 μg b.i.d.

16. The method of claim 13 , wherein the fluticasone is administered in an amount of 100 μg to 400 μg b.i.d.

17. The method of claim 13 , wherein the fluticasone is administered in an amount of at least 200 μg daily.

18. The method of claim 13 , wherein the fluticasone is administered in an amount of at least 400 μg daily.

19. The method of claim 13 , wherein the fluticasone is administered in an amount of at least 200 μg daily delivered in two doses.

20. The method of claim 13 , wherein the fluticasone is administered in an amount of at least 400 μg daily delivered in two doses.

21. The method of claim 13 , wherein the fluticasone is fluticasone propionate administered as a liquid aerosol in an amount of 100 μg to 400 μg b.i.d.

22. The method of claim 13 , wherein the fluticasone is fluticasone propionate administered as a liquid aerosol in an amount of at least 200 μg b.i.d.

Assignments (10)
RELEASE OF SECURITY INTEREST IN PATENTS RECORDED AT REEL/FRAME 71337/0132 Recorded Mar 17, 2026
From: OAKTREE FUND ADMINISTRATION, LLC
To: OPTINOSE, INC.
Reel/Frame 075101/0804 →
PATENT SECURITY AGREEMENT Recorded Mar 16, 2026
From: OPTINOSE, INC.
To: WILMINGTON TRUST, NATIONAL ASSOCIATION, AS ADMINISTRATIVE AGENT
Reel/Frame 075111/0018 →
SECURITY INTEREST Recorded May 22, 2025
From: OPTINOSE, INC.
To: OAKTREE FUND ADMINISTRATION, LLC
Reel/Frame 071337/0132 →
RELEASE OF SECURITY INTEREST Recorded May 21, 2025
From: BIOPHARMA CREDIT PLC, AS COLLATERAL AGENT
To: OPTINOSE INC.
Reel/Frame 071547/0979 →
CHANGE OF ADDRESS Recorded Jan 6, 2025
From: OPTINOSE, INC.
To: OPTINOSE, INC.
Reel/Frame 069825/0322 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Sep 27, 2022
From: OPTINOSE AS
To: OPTINOSE INC
Reel/Frame 061546/0424 →
SECURITY INTEREST Recorded Sep 13, 2019
From: OPTINOSE AS
To: BIOPHARMA CREDIT PLC, AS COLLATERAL AGENT
Reel/Frame 050371/0913 →
RELEASE OF SECURITY AGREEMENT RECORDED AT REEL 044976 FRAME 0505 Recorded Sep 13, 2019
From: ATHYRIUM OPPORTUNITIES III ACQUISITION LP
To: OPTINOSE AS
Reel/Frame 050371/0894 →
SECURITY INTEREST Recorded Dec 29, 2017
From: OPTINOSE AS
To: ATHYRIUM OPPORTUNITIES III ACQUISITION LP
Reel/Frame 044976/0505 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 29, 2016
From: DJUPESLAND, PER GISLE; MAHMOUD, RAMY A.; MESSINA, JOHN
To: OPTINOSE AS
Reel/Frame 037616/0854 →
Continuity (3)
Continuation In Part 14226287 · Mar 26, 2014
Provisional Application 61805400 · Mar 26, 2013
Related Publication 20150144129A1 · May 28, 2015
Cited By (1)
US 12,616,806