IP Library Granted Patent US 9,441,049
Granted Patent B2
US 9,441,049 · App. 14/331,876 · Granted Sep 13, 2016

Antibodies reactive with B7-H3 and uses thereof

Inventors: Leslie S. Johnson (Darnestown, MD); Ling Huang (Bethesda, MD); Paul A. Moore (North Bethesda, MD); Deryk T. Loo (Belmont, CA); Francine Z. Chen (San Francisco, CA)
Assignee: MacroGenics, Inc.
C07K16/30A61K39/39558A61K45/06A61K47/48561A61K47/48569C07K16/2809C07K16/2827G01N33/57484A61K2039/505C07K2317/24C07K2317/31C07K2317/33C07K2317/73C07K2317/77C07K2317/94
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Quick Facts
Patent No.
US 9,441,049
App. No.
14/331,876
Granted
Sep 13, 2016
Kind
B2
Abstract

The present invention relates to antibodies that are immunoreactive to the mammalian, and more particularly, the human B7-H3 receptor and to uses thereof, particularly in the treatment of cancer and inflammation. The invention thus particularly concerns humanized B7-H3-reactive antibodies that are capable of mediating, and more preferably enhancing the activation of the immune system against cancer cells that are associated with a variety of human cancers.

Claims (11)

1. A method of treating cancer in a patient having a cancer, comprising administering to said patient a therapeutically effective amount of a polypeptide comprising the amino acid sequence of SEQ ID NO: 117 and a polypeptide comprising the amino acid sequence of SEQ ID NO: 119, and wherein said cancer is characterized by the presence of a cancer cell that expresses B7-H3.

2. The method of claim 1 , wherein said polypeptides bind to B7-H3 that is endogenously expressed on the surface of a cancer cell.

3. The method of claim 1 , wherein said polypeptides bind to B7-H3 expressed on the surface of a cancer cell and are internalized into said cell upon binding to said B7-H3.

4. The method of claim 1 , wherein said cancer cell is selected from the group consisting of a cell of a bladder cancer, a cervical cancer, a colon cancer, a colorectal cancer, a gastric cancer, a liver cancer, a lung cancer, an ovarian cancer, a pancreatic cancer, a prostate cancer, a kidney cancer, a breast cancer, a head and neck cancer, a skin cancer, a sarcoma, a brain tumor, a brain and a spinal cord cancer, an adrenal cancer, a uterine cancer, a neuroblastoma, a small round cell tumor, a peripheral nerve sheath tumor, a bone cancer, a rhabdoid tumor, a lymphoma, a multiple myeloma, a leukemia, a neuroendocrine tumor, and a melanoma.

5. The method of claim 1 , wherein said patient is human.

6. The method of claim 1 , wherein said polypeptides are an antibody.

7. The method of claim 6 , wherein said polypeptides are a humanized antibody.

8. The method of claim 6 , wherein said polypeptides are a monoclonal antibody, or a bispecific antibody.

9. The method of claim 1 , wherein said method further comprises administering to said patient one or more additional anti-cancer agents.

10. The method of claim 9 , wherein said additional anti-cancer agent is a chemotherapeutic agent, a radiation therapeutic agent, a hormonal therapeutic agent, a toxin, or an immunotherapeutic agent.

11. The method of claim 10 , wherein said additional anti-cancer agent is a toxin selected from the group consisting of: a taxane, a maytansinoid, an auristatin, a calicheamicin, an anthracycline, a CC-1065 analog, docetaxel, a cathepsin, ricin, gelonin, Pseudomonas exotoxin, diphtheria toxin, RNase, and a toxic radioisotope.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 28, 2014
From: JOHNSON, LESLIE S; HUANG, LING; MOORE, PAUL A; LOO, DERYK T; CHEN, FRANCINE Z
To: MACROGENICS, INC.
Reel/Frame 034047/0112 →
Continuity (7)
Division 13463924 · May 4, 2012
Continuation In Part PCTUS2011026689 · Mar 1, 2011
Provisional Application 61482771 · May 5, 2011
Provisional Application 61311057 · Mar 5, 2010
Provisional Application 61310695 · Mar 4, 2010
Provisional Application 61310692 · Mar 4, 2010
Related Publication 20140328750A1 · Nov 6, 2014