IP Library Granted Patent US 10,201,585
Granted Patent B2
US 10,201,585 · App. 14/418,809 · Granted Feb 12, 2019

Methods for treatment of atherosclerosis

Inventors: D. Travis Wilson (Newton, MA); Mark Bamberger (South Glastonbury, CT); Brian Blakey (Doylestown, PA)
Assignee: Stealth Biotherapeutics Corp
A61K38/07A61K31/215A61K31/22A61K31/351A61K31/366A61K31/40A61K31/404A61K31/505A61K45/06A61P9/10
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Quick Facts
Patent No.
US 10,201,585
App. No.
14/418,809
Granted
Feb 12, 2019
Kind
B2
Abstract

Disclosed herein are methods and compositions for preventing or treating atherosclerosis in a mammalian subject. The methods comprise administering to the subject an effective amount of an aromatic-cationic peptide and, in some applications, a second active agent, to subjects in need thereof. The present technology relates to the treatment or prevention of atherosclerosis in mammals through the administration of a therapeutically effective amount of aromatic cationic peptides and, in some embodiments, a second active agent.

Claims (5)

1. A method for delaying onset, ameliorating or eliminating statin side effects in a subject in need thereof, the method comprising administering simultaneously, separately or sequentially with the statin, an effective amount of a peptide D-Arg-2′6′-Dmt-Lys-Phe-NH 2 or a pharmaceutically acceptable salt thereof, wherein the statin side effect comprises one or more of rhabdomyolysis, kidney failure, diabetes, memory loss, and decreased coenzyme Q10 levels.

2. The method of claim 1 , wherein the statin is selected from the group consisting of: atorvastatin, simvastatin, pravastatin, fluvastatin, lovastatin, pitavastatin, rosuvastatin, niacin extended-release/lovastatin, lovastatin extended-release, amlodipine, atorvastatin, rosuvastatin, sitagliptin/simvastatin, fluvastatin, fluvastatin extended-release, atorvastatin, pitavastatin, lovastatin, pravastatin, niacin extended-release/simvastatin, ezetimibe/simvastatin, and simvastatin.

3. The method of claim 1 , wherein the peptide and statin are administered sequentially in either order.

4. The method of claim 1 , wherein the pharmaceutically acceptable salt comprises acetate salt or trifluoroacetate salt.

5. The method of claim 1 , wherein the statin comprises rosuvastatin or atorvastatin.

Assignments (3)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Nov 17, 2021
From: STEALTH BIOTHERAPEUTICS CORP
To: STEALTH BIOTHERAPEUTICS INC.
Reel/Frame 058164/0305 →
CHANGE OF NAME Recorded Mar 23, 2017
From: STEALTH PEPTIDES INTERNATIONAL, INC.
To: STEALTH BIOTHERAPEUTICS CORP
Reel/Frame 042157/0448 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 20, 2017
From: WILSON, D. TRAVIS; BAMBERGER, MARK; BLAKEY, BRIAN; ANDERSEN, MARC W.
To: STEALTH PEPTIDES INTERNATIONAL, INC.
Reel/Frame 041025/0946 →
Continuity (4)
Provisional Application 61678992 · Aug 2, 2012
Provisional Application 61695807 · Aug 31, 2012
Provisional Application 61695850 · Aug 31, 2012
Related Publication 20150283200A1 · Oct 8, 2015