IP Library Granted Patent US 9,320,732
Granted Patent B2
US 9,320,732 · App. 14/661,191 · Granted Apr 26, 2016

1,2,5-oxadiazoles as inhibitors of indoleamine 2,3-dioxygenase

Inventors: Andrew P. Combs (Kennett Square, PA); Eddy W. Yue (Landenberg, PA); Richard B. Sparks (Wilmington, DE); Wenyu Zhu (Media, PA)
Assignees: Incyte Corporation; Incyte Holdings Corporation
A61K31/4245A61K39/3955C07D271/08C07D413/04C07D413/12
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Quick Facts
Patent No.
US 9,320,732
App. No.
14/661,191
Granted
Apr 26, 2016
Kind
B2
Abstract

The present invention is directed to 1,2,5-oxadiazole derivatives, and compositions of the same, which are inhibitors of indoleamine 2,3-dioxygenase and are useful in the treatment of cancer and other disorders, and to the processes and intermediates for making such 1,2,5-oxadiazole derivatives.

Claims (10)

1. A pharmaceutical composition comprising a compound of the formula:

and at least one pharmaceutically acceptable carrier.

2. The pharmaceutical composition of claim 1 , wherein the composition is a unit dosage form.

3. The pharmaceutical composition of claim 2 , wherein the unit dosage form is a tablet.

4. The pharmaceutical composition of claim 2 , wherein the unit dosage form is a capsule.

5. A pharmaceutically acceptable salt of the compound of formula:

6. A pharmaceutical composition comprising the pharmaceutically acceptable salt of claim 5 and at least one pharmaceutically acceptable carrier.

7. The pharmaceutical composition of claim 6 , wherein the composition is a unit dosage form.

8. The pharmaceutical composition of claim 7 , wherein the unit dosage form is a tablet.

9. The pharmaceutical composition of claim 7 , wherein the unit dosage form is a capsule.

Assignments (2)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Nov 30, 2015
From: INCYTE CORPORATION
To: INCYTE HOLDINGS CORPORATION; INCYTE CORPORATION
Reel/Frame 037166/0164 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jul 1, 2015
From: COMBS, ANDREW P.; YUE, EDDY W.; SPARKS, RICHARD B.; ZHU, WENYU; ZHOU, JIACHENG; LIN, QIYAN; WENG, LINGKAI; YUE, TAI-YUEN; LIU, PINGLI
To: INCYTE CORPORATION
Reel/Frame 035999/0179 →
Continuity (6)
Continuation 14322362 · Jul 2, 2014
Continuation 13294711 · Nov 11, 2011
Division 12498782 · Jul 7, 2009
Provisional Application 61150873 · Feb 9, 2009
Provisional Application 61078876 · Jul 8, 2008
Related Publication 20150190378A1 · Jul 9, 2015