IP Library Granted Patent US 9,585,887
Granted Patent B2
US 9,585,887 · App. 14/723,225 · Granted Mar 7, 2017

Modulators of androgen synthesis

Inventors: Suzanne Dilly (Oxfordshire, GB); Gregory Stoloff (London, GB); Paul Taylor (London, GB)
Assignee: Tangent Reprofiling Limited
A61K31/519A61K31/201A61K31/454A61K45/06
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Quick Facts
Patent No.
US 9,585,887
App. No.
14/723,225
Granted
Mar 7, 2017
Kind
B2
Abstract

The present specification discloses compositions comprising at least one therapeutic compound capable of modulating androgen production and methods and uses for treating a disorder associated with androgen production using such compositions and/or compounds.

Claims (32)

1. A method of treating an individual with a lung cancer, the method comprising the step of administering to the individual a therapeutically effective amount of risperidone and about 0.01 mg/kg/day to about 0.5 mg/kg/day of 9Z, 11E conjugated Linoleic acid,

wherein there is a synergistic effect between risperidone and 9Z, 11E conjugated Linoleic Acid; and

wherein administration the risperidone and the 9Z, 11E conjugated Linoleic acid reduces a symptom associated with the lung cancer, thereby treating the individual.

2. The method according to claim 1 , wherein the therapeutically effective amount of risperidone is from about 0.1 mg/day to about 20 mg/day.

3. The method according to claim 1 , wherein the therapeutically effective amount of risperidone is from about 0.01 mg/kg/day to about 0.5 mg/kg/day.

4. The method according to claim 1 , wherein 9Z, 11E conjugated Linoleic acid is in an amount from about 1 mg/day to about 20 mg/day.

5. The method according to claim 1 , wherein the lung cancer is a non-small cell lung adenocarcinoma.

6. The method according to claim 1 , wherein risperidone and 9Z, 11E conjugated Linoleic Acid are sequentially or simultaneously administered to the individual as separate compositions.

7. The method according to claim 1 , wherein risperidone and 9Z, 11E conjugated Linoleic Acid are administered as a single composition to the individual.

8. A method of treating an individual with a lung cancer, the method comprising the step of administering to the individual a therapeutically effective amount of risperidone and about 1 mg/day to about 20 mg/day of 9Z, 11E conjugated Linoleic Acid, wherein there is a synergistic effect between the risperidone and 9Z, 11 E conjugated Linoleic Acid; and wherein administration of risperidone and 9Z, 11E conjugated Linoleic acid reduces a symptom associated with the lung cancer, thereby treating the individual.

9. The method according to claim 8 , wherein the therapeutically effective amount of risperidone is in an amount from about 0.1 mg/day to about 20 mg/day.

10. The method according to claim 8 , wherein the therapeutically effective amount of risperidone is in an amount from about 0.01 mg/kg/day to about 0.5 mg/kg/day.

11. The method according to claim 8 , wherein 9Z, 11E conjugated Linoleic acid is in an amount from about 0.01 mg/kg/day to about 0.5 mg/kg/day.

12. The method according to claim 8 , wherein the lung cancer is a non-small cell lung adenocarcinoma.

13. The method according to claim 8 , wherein risperidone and 9Z, 11E conjugated Linoleic Acid are sequentially or simultaneously administered to the individual as separate compositions.

14. The method according to claim 8 , wherein risperidone and 9Z, 11E conjugated Linoleic Acid are administered as a single composition to the individual.

15. A method of treating an individual with a lung cancer, the method comprising the step of administering to the individual about 1 mg/day to about 20 mg/day of risperidone and about 1 mg/day to about 20 mg/day of 9Z, 11E conjugated Linoleic acid,

wherein there is a synergistic effect between risperidone and 9Z, 11E conjugated Linoleic Acid; and

wherein administration risperidone and 9Z, 11E conjugated Linoleic acid reduces a symptom associated with the lung cancer, thereby treating the individual.

16. The method according to claim 15 , wherein the lung cancer is a non-small cell lung adenocarcinoma.

17. The method according to claim 15 , wherein risperidone and 9Z, 11E conjugated Linoleic Acid are sequentially or simultaneously administered to the individual as separate compositions.

18. The method according to claim 15 , wherein risperidone and 9Z, 11E conjugated Linoleic Acid are administered as a single composition to the individual.

19. The method according to claim 15 , wherein the therapeutically effective amount of risperidone is from about 0.01 mg/kg/day to about 0.5 mg/kg/day.

20. The method according to claim 15 , wherein 9Z, 11E conjugated Linoleic acid is in an amount from about 0.01 mg/kg/day to about 0.5 mg/kg/day.

21. A method of treating an individual with a lung cancer, the method comprising the step of administering to the individual about 0.01 mg/kg/day to about 0.5 mg/kg/day of risperidone and about 0.01 mg/kg/day to about 0.5 mg/kg/day of 9Z, 11E conjugated Linoleic acid,

wherein there is a synergistic effect between risperidone and 9Z, 11E conjugated Linoleic Acid; and

wherein administration risperidone and 9Z, 11E conjugated Linoleic acid reduces a symptom associated with the lung cancer, thereby treating the individual.

22. The method according to claim 21 , wherein risperidone is in an amount from about 0.1 mg/day to about 20 mg/day.

23. The method according to claim 21 , wherein 9Z, 11E conjugated Linoleic acid is in an amount from about 1 mg/day to about 20 mg/day.

24. The method according to claim 21 , wherein the lung cancer is a non-small cell lung adenocarcinoma.

25. The method according to claim 21 , wherein risperidone and 9Z, 11E conjugated Linoleic Acid are sequentially or simultaneously administered to the individual as separate compositions.

26. The method according to claim 21 , wherein risperidone and 9Z, 11E conjugated Linoleic Acid are administered as a single composition to the individual.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 11, 2016
From: DILLY, SUZANNE; STOLOFF, GREGORY A.; TAYLOR, PAUL
To: TANGENT REPROFILING LIMITED
Reel/Frame 038247/0501 →
Continuity (4)
Division 14037481 · Sep 26, 2013
Provisional Application 61871662 · Aug 29, 2013
Provisional Application 61705790 · Sep 26, 2012
Related Publication 20150258095A1 · Sep 17, 2015