IP Library Granted Patent US 9,598,374
Granted Patent B2
US 9,598,374 · App. 14/775,794 · Granted Mar 21, 2017

Arginine methyltransferase inhibitors and uses thereof

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Quick Facts
Patent No.
US 9,598,374
App. No.
14/775,794
Granted
Mar 21, 2017
Kind
B2
Abstract

Described herein are compounds of Formula (I), pharmaceutically acceptable salts thereof, and pharmaceutical compositions thereof. Compounds described herein are useful for inhibiting arginine methyltransferase activity. Methods of using the compounds for treating arginine methyltransferase-mediated disorders are also described.

Claims (10)

1. A compound of formula:

or a pharmaceutically acceptable salt thereof.

2. The compound of claim 1 , wherein the compound is:

3. The compound of claim 1 , wherein the compound is a pharmaceutically acceptable salt of:

4. A pharmaceutical composition comprising a compound of claim 1 , or a pharmaceutically acceptable salt thereof, and a pharmaceutically acceptable excipient.

5. A pharmaceutical composition comprising a compound of claim 2 , and a pharmaceutically acceptable excipient.

6. A pharmaceutical composition comprising a compound of claim 3 , and a pharmaceutically acceptable excipient.

7. A kit or packaged pharmaceutical comprising a compound of claim 1 , or a pharmaceutically acceptable salt thereof, and instructions for use thereof.

8. A kit or packaged pharmaceutical comprising a compound of claim 2 , and instructions for use thereof.

9. A kit or packaged pharmaceutical comprising a compound of claim 3 , and instructions for use thereof.

Assignments (3)
TERMINATION AND RELEASE OF SECURITY INTEREST IN PATENTS AT REEL/FRAME: 051057/0848 Recorded Aug 13, 2022
From: BIOPHARMA CREDIT PLC
To: EPIZYME, INC.
Reel/Frame 061165/0501 →
SECURITY INTEREST Recorded Nov 19, 2019
From: EPIZYME, INC.
To: BIOPHARMA CREDIT PLC
Reel/Frame 051057/0848 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Sep 16, 2015
From: CHESWORTH, RICHARD; MITCHELL, LORNA HELEN; SHAPIRO, GIDEON; SWINGER, KERREN K.
To: EPIZYME, INC.
Reel/Frame 036578/0568 →