IP Library Granted Patent US 9,545,426
Granted Patent B2
US 9,545,426 · App. 14/812,148 · Granted Jan 17, 2017

Use of amisulpride as an anti-emetic

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Quick Facts
Patent No.
US 9,545,426
App. No.
14/812,148
Granted
Jan 17, 2017
Kind
B2
Abstract

Amisulpride is used in the therapy of nausea, vomiting or retches. The therapy may utilize a novel injectable formulation, in unit dosage form, comprising less than 50 mg amisulpride.

Claims (25)

1. A method for the prevention and/or treatment of post-operative nausea and vomiting, wherein said method comprises administering amisulpride at a dose of 1 mg to 20 mg to a subject of a surgical procedure and in need of such prevention and/or treatment.

2. The method of claim 1 , wherein the subject is also administered an emetogenic agent.

3. The method of claim 2 , wherein the emetogenic agent is an opiate.

4. The method of claim 2 , wherein the emetogenic agent is morphine.

5. The method of claim 1 , wherein the subject is a human.

6. The method of claim 1 , wherein the amisulpride is in the form of an acceptable pharmaceutical salt.

7. The method of claim 1 , wherein the amisulpride is administered in combination with another anti-emetic drug.

8. The method of claim 7 , wherein the another anti-emetic drug is a 5HT3 antagonist.

9. The method of claim 8 , wherein the 5HT3 antagonist is ondansetron.

10. The method of claim 1 , wherein the amisulpride is administered in combination with dexamethasone.

11. The method of claim 1 , wherein the amisulpride is administered at a dose of 2.5 mg to 20 mg.

12. The method of claim 1 , wherein the amisulpride is administered at a dose of 2.5 mg.

13. The method of claim 1 , wherein the amisulpride is administered at a dose of 5 mg.

14. The method of claim 1 , wherein the amisulpride is administered at a dose of 20 mg.

15. The method of claim 1 , wherein the subject has received an anesthetic.

16. The method of claim 1 , wherein the surgical procedure is chosen from procedures of the eye or ear, laparoscopic cholecystectomy, hysterectomy, breast surgery, abdominal surgery, and gynecological surgery.

17. The method of claim 1 , wherein the amisulpride is administered by intravenous injection.

18. The method of claim 1 , wherein the amisulpride is administered by intramuscular injection.

19. The method of claim 1 , wherein the amisulpride is administered by subcutaneous injection.

20. The method of claim 1 , wherein the amisulpride is administered orally.

21. The method of claim 1 , wherein the amisulpride is administered topically.

22. The method of claim 1 , wherein the amisulpride is administered rectally.

23. The method of claim 1 , wherein the amisulpride is administered intranasally.

24. The method of claim 1 , wherein the amisulpride is administered transdermally.

25. The method of claim 1 , wherein the amisulpride is (S—)-amisulpride.

Assignments (5)
SECURITY INTEREST Recorded Apr 27, 2026
From: LXO IRELAND DESIGNATED ACTIVITY COMPANY
To: KROLL TRUSTEE SERVICES LIMITED, AS SECURITY AGENT
Reel/Frame 074483/0163 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 4, 2026
From: ACACIA PHARMA LIMITED; ACACIA PHARMA, INC.; EAGLE PHARMACEUTICALS, INC.
To: LXO IRELAND DESIGNATED ACTIVITY COMPANY; LXO US, INC.
Reel/Frame 073967/0303 →
RELEASE OF SECURITY INTEREST Recorded Apr 1, 2025
From: JPMORGAN CHASE BANK, N.A., AS ADMINISTRATIVE AGENT
To: ACACIA PHARMA LIMITED
Reel/Frame 070698/0351 →
SECURITY INTEREST Recorded Apr 28, 2023
From: ACACIA PHARMA LIMITED
To: JPMORGAN CHASE BANK, N.A., AS ADMINISTRATIVE AGENT
Reel/Frame 063476/0631 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Aug 5, 2015
From: GILBERT, JULIAN CLIVE; GRISTWOOD, ROBERT WILLIAM; COOPER, NICOLA; FOX, GABRIEL
To: ACACIA PHARMA LIMITED
Reel/Frame 036255/0411 →