IP Library Granted Patent US 9,745,635
Granted Patent B2
US 9,745,635 · App. 14/864,466 · Granted Aug 29, 2017

Recurrent gene fusions in prostate cancer

Inventors: Scott Tomlins (Ann Arbor, MI); Daniel Rhodes (Ann Arbor, MI); Arul Chinnaiyan (Ann Arbor, MI); Rohit Mehra (Ann Arbor, MI); Mark A. Rubin (New York, NY); Xiao-Wei Sun (New York, NY); Sven Perner (Ellwaugen, DE); Charles Lee (Marlborough, MA); Francesca Demichelis (New York, NY)
Assignees: THE REGENTS OF THE UNIVERSITY OF MICHIGAN; THE BRIGHAM AND WOMEN'S HOSPITAL, INC.
C12Q1/6886C12N15/113G01N33/57434C12N2310/11C12N2310/14C12Q2600/112C12Q2600/156C12Q2600/158Y10S435/81
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Quick Facts
Patent No.
US 9,745,635
App. No.
14/864,466
Granted
Aug 29, 2017
Kind
B2
Abstract

Recurrent gene fusions of androgen regulated genes and ETS family member genes in prostate cancer are described. Compositions and methods having utility in prostate cancer diagnosis, research, and therapy are also provided.

Claims (20)

1. A composition comprising a hybridized oligonucleotide:target gene fusion duplex, wherein the target gene fusion comprises a chimeric nucleic acid molecule in which a 5′ portion of the chimeric nucleic acid molecule is from a TMPRSS2 gene and a 3′ portion of the chimeric nucleic acid molecule is from an ETS family member gene, wherein the ETS family member gene is selected from the group consisting of ERG, ETV1 (ER81), FLI1, ETS1, ETS2, ELK1, ETV6 (TEL1), ETV7 (TEL2), GABPα, ELF1, ETV4 (E1AF; PEA3), ETV5 (ERM), ERF, PEA3/E1AF, PU.1, ESE1/ESX, SAP1 (ELK4), ETV3 (METS), EWS/FLI1, ESE1, ESE2 (ELF5), ESE3, PDEF, NET (ELK3; SAP2), NERF (ELF2), and FEV; and wherein the oligonucleotide is covalently labeled with a detectable label.

2. The composition of claim 1 wherein the ETS family member gene is an ERG gene.

3. The composition of claim 1 wherein the ETS family member gene is an ETV1 gene.

4. The composition of claim 1 wherein the ETS family member gene is an ETV4 gene.

5. The composition of claim 1 wherein the ETS family member gene is an FLI1 gene.

6. The composition of claim 1 wherein the target gene fusion is obtained from a tissue, blood, urine, semen, prostatic secretion, plasma, serum, urine supernatant, urine cell pellet, or prostate cell sample.

7. The composition of claim 1 wherein the 5′ portion of the chimeric nucleic acid molecule is from a transcriptional regulatory region of the TMPRSS2 gene.

8. The composition of claim 1 wherein the transcriptional regulatory region comprises a promoter region of the TMPRSS2 gene.

9. The composition of claim 1 wherein the oligonucleotide is hybridized to a junction at which the 5′ portion of the chimeric nucleic acid molecule is fused to the 3′ portion of the chimeric nucleic acid molecule.

10. The composition of claim 1 wherein:

a) the oligonucleotide is hybridized to the 5′ portion of the chimeric nucleic acid molecule and the composition further comprises a second oligonucleotide hybridized to the 3′ portion of the chimeric nucleic acid molecule; or

b) the oligonucleotide is hybridized to the 3′ portion of the chimeric nucleic acid molecule and the composition further comprises a second oligonucleotide hybridized to the 5′ portion of the chimeric nucleic acid molecule, wherein the second oligonucleotide is covalently labeled with a detectable label.

11. The composition of claim 10 further comprising a polymerase.

12. The composition of claim 10 further comprising a third oligonucleotide covalently labeled with a detectable label.

13. The composition of claim 1 further comprising a detectably labeled oligonucleotide probe that hybridizes to a nucleic acid molecule selected from one or more of the group consisting of PCA3, PSA, AMACR/P504S, PCGEM1, prostein/P501S, P503S, P504S, P509S, P510S, prostase/P703P, and P710P.

14. The composition of claim 1 further comprising a detectably labeled oligonucleotide probe that hybridizes to PSA.

15. The composition of claim 1 further comprising a detectably labeled oligonucleotide probe that hybridizes to PCA3.

16. A method of producing a hybridized oligonucleotide:target gene fusion duplex, the method comprising contacting a sample comprising a target gene fusion comprising a chimeric nucleic acid molecule in which a 5′ portion of the chimeric nucleic acid molecule is from a TMPRSS2 gene and a 3′ portion of the chimeric nucleic acid molecule is from an ETS family member gene with an oligonucleotide covalently labeled with a detectable label and having a sequence that hybridizes to a junction at which the 5′ portion of the chimeric nucleic acid molecule is fused to the 3′ portion of the chimeric nucleic acid molecule.

17. The method of claim 16 wherein the 5′ portion of the chimeric nucleic acid molecule is from a TMPRSS2 gene and the 3′ portion of the chimeric nucleic acid molecule is from an ETS family member gene, wherein the ETS family member gene is selected from the group consisting of ERG, ETV1 (ER81), FLI1, ETS1, ETS2, ELK1, ETV6 (TEL1), ETV7 (TEL2), GABPα, ELF1, ETV4 (E1AF; PEA3), ETV5 (ERM), ERF, PEA3/E1AF, PU.1, ESE1/ESX, SAP1 (ELK4), ETV3 (METS), EWS/FLI1, ESE1, ESE2 (ELF5), ESE3, PDEF, NET (ELK3; SAP2), NERF (ELF2), and FEV.

18. The method of claim 16 wherein the sample comprises tissue, blood, urine, semen, prostatic secretion, plasma, serum, urine supernatant, urine cell pellet, or a prostate cell.

Assignments (2)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 9, 2015
From: DEMICHELIS, FRANCESCA; RUBIN, MARK A.; PERNER, SVEN; LEE, CHARLES; SUN, XIAO-WEI
To: THE BRIGHAM AND WOMEN'S HOSPITAL, INC.
Reel/Frame 036768/0091 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 9, 2015
From: CHINNAIYAN, ARUL; TOMLINS, SCOTT; RHODES, DANIEL; MEHRA, ROHIT
To: THE REGENTS OF THE UNIVERSITY OF MICHIGAN
Reel/Frame 036768/0099 →
Continuity (8)
Continuation 13483157 · May 30, 2012
Division 12650164 · Dec 30, 2009
Division 11519397 · Sep 12, 2006
Provisional Application 60716436 · Sep 12, 2005
Provisional Application 60779041 · Mar 3, 2006
Provisional Application 60730358 · Oct 27, 2005
Provisional Application 60795590 · Apr 28, 2006
Related Publication 20160097104A1 · Apr 7, 2016