IP Library Granted Patent US 9,446,034
Granted Patent B2
US 9,446,034 · App. 14/887,763 · Granted Sep 20, 2016

Pyrazolylaminopyridines as inhibitors of FAK

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Quick Facts
Patent No.
US 9,446,034
App. No.
14/887,763
Granted
Sep 20, 2016
Kind
B2
Abstract

The present invention relates to a compound of formula (I): or a pharmaceutically acceptable salt thereof, wherein R 1 , R 2 , R 3 , R 11 , R 12 , R 13 , Q, Z, and p are as described herein. Compounds of the present invention are useful for the treatment of cancers.

Claims (6)

1. A method of treating or lessening the severity of mesothelioma in a human in need thereof, which comprises administering to such human a therapeutically effective amount of the compound:

2-[(5-Chloro-2-{[3-methyl-1-(1-methylethyl)-1H-pyrazol-5-yl]amino}-4-pyridinyl)amino]-N-(methyloxy)benzamide;

or a pharmaceutically acceptable salt thereof.

2. A method of treating or lessening the severity of pancreatic cancer in a human in need thereof, which comprises administering to such human a therapeutically effective amount of the compound:

2-[(5-Chloro-2-{[3-methyl-1-(1-methylethyl)-1H-pyrazol-5-yl]amino}-4-pyridinyl)amino]-N-(methyloxy)benzamide;

or a pharmaceutically acceptable salt thereof.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 4, 2016
From: ADAMS, JERRY LEROY; FAITG, THOMAS H.; JOHNSON, NEIL W.; KASPAREC, JIRI; LIN, HONG; MELLINGER, MARK; PENG, XIN; XIE, REN
To: GLAXOSMITHKLINE LLC
Reel/Frame 037666/0380 →