IP Library Granted Patent US 9,707,219
Granted Patent B2
US 9,707,219 · App. 14/903,694 · Granted Jul 18, 2017

Losmapimod for use in treating glomerular disease

Inventors: Dennis Sprecher (Pennsylvania, PA); Robert Nicholas Willette (Pennsylvania, PA)
Assignee: GlaxoSmithKline Intellectual Property (No.2) Limited
A61K31/455A61K45/06
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Quick Facts
Patent No.
US 9,707,219
App. No.
14/903,694
Granted
Jul 18, 2017
Kind
B2
Abstract

The present invention relates to a method of treating a glomerular disease with 6-(5-cyclopropylcarbamoyl-3-fluoro-2-methyl-phenyl)-N-(2,2-dimethylpropyl)-nicotinamide or a pharmaceutically acceptable salt thereof.

Claims (6)

1. A method for treating focal segmental glomerulosclerosis (FSGS) in a subject in need thereof comprising administering to said subject a pharmaceutical formulation comprising the compound 6-(5-cyclopropylcarbamoyl-3-fluoro-2-methyl-phenyl)-N-(2,2-dimethylpropyl)-nicotinamide or a pharmaceutically acceptable salt thereof.

2. The method of claim 1 , wherein the pharmaceutical formulation is adapted for oral administration.

3. The method of claim 1 , wherein the pharmaceutical formulation comprises one or more other therapeutic agents which are suitable for the treatment of focal segmental glomerulosclerosis (FSGS).

4. The method of claim 1 , wherein the compound 6-(5-cyclopropylcarbamoyl-3-fluoro-2-methyl-phenyl)-N-(2,2-dimethylpropyl)-nicotinamide is in the form of a free base.

5. The method of claim 4 , wherein the pharmaceutical formulation is adapted for oral administration.

6. The method of claim 4 , wherein the pharmaceutical formulation further comprises one or more other therapeutic agents which are suitable for the treatment of focal segmental glomerulosclerosis (FSGS).

Assignments (2)
CHANGE OF ADDRESS Recorded Apr 16, 2025
From: GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO.2) LIMITED
To: GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO.2) LIMITED
Reel/Frame 070854/0469 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 8, 2016
From: SPRECHER, DENNIS; WILLETTE, ROBERT NICHOLAS
To: GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO.2) LIMITED
Reel/Frame 037439/0176 →
Continuity (2)
Provisional Application 61844491 · Jul 10, 2013
Related Publication 20160220550A1 · Aug 4, 2016