IP Library Granted Patent US 10,004,745
Granted Patent B2
US 10,004,745 · App. 15/066,600 · Granted Jun 26, 2018

Use of inhibitors of Bruton'S tyrosine kinase (Btk)

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Quick Facts
Patent No.
US 10,004,745
App. No.
15/066,600
Granted
Jun 26, 2018
Kind
B2
Abstract

Disclosed herein are methods for treating a cancer comprising: a. administering a Btk inhibitor to a subject sufficient to result in an increase or appearance in the blood of a subpopulation of lymphocytes defined by immunophenotyping; b. determining the expression profile of one or more biomarkers from one or more subpopulation of lymphocytes; and c. administering a second agent based on the determined expression profile.

Claims (8)

1. A method for treating follicular lymphoma in an individual who has failed at least one prior therapy for follicular lymphoma, comprising:

administering to the individual once per day about 560 mg of an oral dose of a compound having the structure:

2. The method of claim 1 , wherein the follicular lymphoma is follicular small cleaved cell lymphoma, follicular mixed small cleaved and large cell lymphoma, or follicular large cell lymphoma.

3. The method of claim 1 , wherein, following administration of the compound, the individual achieves a stable disease, a partial response, or a complete response.

4. The method of claim 1 , wherein, following administration of the compound, the individual achieves a partial response or a complete response.

5. The method of claim 1 , wherein, following administration of the compound, the individual achieves a complete response.

6. The method of claim 1 , wherein, following administration of the compound, the individual does not experience a progressive disease.

7. The method of claim 1 , wherein the prior therapy comprised administration of rituximab.

Assignments (3)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 10, 2017
From: BUGGY, JOSEPH J.; ELIAS, LAURENCE; FYFE, GWEN; HEDRICK, ERIC; LOURY, DAVID J.; MODY, TARAK D.
To: PHARMACYCLICS, INC.
Reel/Frame 040934/0712 →
MERGER Recorded Jan 10, 2017
From: OXFORD AMHERST CORPORATION; PHARMACYCLICS, INC.
To: PHARMACYCLICS, INC.
Reel/Frame 040934/0759 →
MERGER AND CHANGE OF NAME Recorded Jan 10, 2017
From: PHARMACYCLICS, INC.; OXFORD AMHERST LLC; PHARMACYCLICS LLC
To: PHARMACYCLICS LLC
Reel/Frame 040934/0827 →