IP Library › Granted Patent US 9,944,655
Granted Patent B2
US 9,944,655 · App. 15/067,634 · Granted Apr 17, 2018

ACC inhibitors and uses thereof

Inventors: Geraldine C. Harriman (Charlestown, RI); Craig E. Masse (Cambridge, MA); H. James Harwood (Ledyard, CT); Sathesh Bhat (West New York, NY); Jeremy Robert Greenwood (Brooklyn, NY)
Assignee: Gilead Apollo, LLC
C07D495/04A01N43/90A61K31/519
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Quick Facts
Patent No.
US 9,944,655
App. No.
15/067,634
Granted
Apr 17, 2018
Kind
B2
Abstract

The present invention provides compounds useful as inhibitors of Acetyl CoA Carboxylase (ACC), compositions thereof, and methods of using the same.

Claims (10)

1. A compound of formula:

or a pharmaceutically acceptable salt thereof.

2. The compound according to claim 1 , wherein the compound is:

3. The compound according to claim 1 , wherein the compound is:

4. The compound according to claim 1 , wherein the compound is:

5. The compound according to claim 1 , wherein the compound is:

6. The compound according to claim 1 , wherein the compound is:

7. The compound according to claim 1 , wherein the compound is:

8. The compound according to claim 1 , wherein the compound is:

9. A composition comprising a compound according to claim 1 and a pharmaceutically acceptable carrier, adjuvant, or vehicle.

Assignments (10)
CHANGE OF NAME Recorded Oct 3, 2016
From: GILEAD APOLLO, INC.
To: GILEAD APOLLO, LLC
Reel/Frame 040209/0033 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jul 29, 2016
From: HARRIMAN, GERALDINE C.; MASSE, CRAIG E.; HARWOOD, JAMES; BHAT, SATHESH; GREENWOOD, JEREMY ROBERT
To: NIMBUS APOLLO, INC.
Reel/Frame 039294/0712 →
MERGER AND CHANGE OF NAME Recorded Jul 27, 2016
From: NIMBUS APOLLO, INC.; GILEAD APOLLO, INC.
To: GILEAD APOLLO, INC.
Reel/Frame 039490/0648 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 5, 2016
From: MASSE, CRAIG E.
To: NIMBUS DISCOVERY, INC.
Reel/Frame 038191/0089 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 5, 2016
From: NIMBUS DISCOVERY, INC.
To: NIMBUS APOLLO, INC.
Reel/Frame 038191/0098 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 5, 2016
From: SCHRÖDINGER, L.L.C.
To: NIMBUS DISCOVERY, INC.
Reel/Frame 038353/0704 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 5, 2016
From: SCHRÖDINGER, INC.
To: SCHRÖDINGER, L.L.C.
Reel/Frame 038353/0874 →
EMPLOYMENT AGREEMENT Recorded Apr 5, 2016
From: GREENWOOD, JEREMY ROBERT
To: SCHRÖDINGER, INC.
Reel/Frame 038403/0642 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 5, 2016
From: HARRIMAN, GERALDINE C.
To: NIMBUS DISCOVERY, INC.
Reel/Frame 038191/0056 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 5, 2016
From: BHAT, SATHESH
To: SCHRÖDINGER, INC.
Reel/Frame 038191/0025 →
Continuity (7)
Continuation 14604497 · Jan 23, 2015
Continuation 13673610 · Nov 9, 2012
Provisional Application 61675513 · Jul 25, 2012
Provisional Application 61651878 · May 25, 2012
Provisional Application 61615092 · Mar 23, 2012
Provisional Application 61559023 · Nov 11, 2011
Related Publication 20160297834A1 · Oct 13, 2016