IP Library Granted Patent US 10,272,097
Granted Patent B2
US 10,272,097 · App. 15/106,883 · Granted Apr 30, 2019

Uses of oxygenated cholesterol sulfates (OCS)

Inventors: Shunlin Ren (Richmond, VA); Felix Theeuwes (Los Altos Hills, CA); James E. Brown (Los Gatos, CA); WeiQi Lin (Emerald Hills, CA)
Assignees: Virginia Commonwealth University; Durect Corporation
A61K31/575A01N1/0226A61K31/568A61K35/12
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Quick Facts
Patent No.
US 10,272,097
App. No.
15/106,883
Granted
Apr 30, 2019
Kind
B2
Abstract

Methods of preventing and/or treating ischemia, organ dysfunction and/or organ failure, including multiple organ dysfunction syndrome (MODS), and necrosis and apoptosis associated with organ dysfunction/failure, are provided. For instance, the methods involve contacting organ(s) with an oxygenated cholesterol sulfate (OCS), e.g. 5-cholesten-3,25-diol, 3-sulfate (25HC3S). The organ(s) may be in vivo (e.g. in a patient that is treated with the OCS) or ex vivo (e.g. an organ that has been harvested from a donor and is to be transplanted).

Claims (19)

1. A method of treating acute kidney dysfunction or acute kidney failure in a subject in need thereof, comprising

administering to the subject an amount of 5-cholesten-3,25-diol, 3-sulfate (25HC3S) or pharmaceutically acceptable salt thereof that is sufficient to treat the acute kidney dysfunction or acute kidney failure, wherein the subject does not have hyperlipidemia.

2. The method of claim 1 , wherein the 25HC3S or pharmaceutically acceptable salt thereof is administered at a dose ranging from about 0.001 mg/kg to about 100 mg/kg.

3. The method of claim 1 , wherein the administering is performed orally or by injection.

4. The method of claim 1 , wherein the administering is performed orally.

5. The method of claim 1 , wherein the administering is performed by injection.

6. The method of claim 1 , wherein the administering is performed orally, parenterally, intravenously, intramuscularly, subcutaneously, by intradermal injection, by intraperitoneal injection, transdermally, sublingually, rectally, by buccal delivery, by inhalation of an aerosol, intravaginally, intranasally, or topically.

7. The method of claim 1 , wherein the 25HC3S or pharmaceutically acceptable salt thereof is administered in a formulation further comprising a pharmaceutically acceptable carrier.

8. The method of claim 1 , wherein the 25HC3S or pharmaceutically acceptable salt thereof comprises a pharmaceutically acceptable salt of 25HC3S.

9. The method of claim 2 , wherein the 25HC3S or pharmaceutically acceptable salt thereof comprises a pharmaceutically acceptable salt of 25HC3S.

10. The method of claim 3 , wherein the 25HC3S or pharmaceutically acceptable salt thereof comprises a pharmaceutically acceptable salt of 25HC3S.

11. The method of claim 4 , wherein the 25HC3S or pharmaceutically acceptable salt thereof comprises a pharmaceutically acceptable salt of 25HC3S.

12. The method of claim 5 , wherein the 25HC3S or pharmaceutically acceptable salt thereof comprises a pharmaceutically acceptable salt of 25HC3S.

13. The method of claim 6 , wherein the 25HC3S or pharmaceutically acceptable salt thereof comprises a pharmaceutically acceptable salt of 25HC3S.

14. The method of claim 7 , wherein the 25HC3S or pharmaceutically acceptable salt thereof comprises a pharmaceutically acceptable salt of 25HC3S.

15. The method of claim 4 , wherein the 25HC3S or pharmaceutically acceptable salt thereof is administered at a dose ranging from about 0.001 mg/kg to about 100 mg/kg.

16. The method of claim 5 , wherein the 25HC3S or pharmaceutically acceptable salt thereof is administered at a dose ranging from about 0.001 mg/kg to about 100 mg/kg.

17. The method of claim 1 , wherein the 25HC3S or pharmaceutically acceptable salt thereof is administered at a dose ranging from about 0.1 mg/kg to about 10 mg/kg.

18. The method of claim 1 , wherein the administering occurs for not more than 14 days.

Assignments (6)
SECURITY INTEREST Recorded Mar 30, 2026
From: BAUSCH HEALTH IRELAND LIMITED; MEDICIS PHARMACEUTICAL CORPORATION; SALIX PHARMACEUTICALS, INC.; SOLTA MEDICAL IRELAND LIMITED
To: THE BANK OF NEW YORK MELLON
Reel/Frame 074223/0753 →
SECURITY INTEREST Recorded Mar 30, 2026
From: MEDICIS PHARMACEUTICAL CORPORATION
To: JPMORGAN CHASE BANK, N.A.
Reel/Frame 074227/0509 →
MERGER Recorded Feb 25, 2026
From: DURECT CORPORATION
To: MEDICIS PHARMACEUTICAL CORPORATION
Reel/Frame 073889/0196 →
MERGER Recorded Feb 19, 2026
From: DURECT CORPORATION
To: MEDICIS PHARMACEUTICAL CORPORATION
Reel/Frame 073837/0231 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 9, 2023
From: VIRGINIA COMMONWEALTH UNIVERSITY
To: THE UNITED STATES GOVERNMENT AS REPRESENTED BY THE DEPARTMENT OF VETERANS AFFAIRS; VIRGINIA COMMONWEALTH UNIVERSITY
Reel/Frame 062318/0868 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jun 21, 2016
From: REN, SHUNLIN; THEEUWES, FELIX; BROWN, JAMES E.; LIN, WEIQI
To: VIRGINIA COMMONWEALTH UNIVERSITY; DURECT CORPORATION
Reel/Frame 038971/0172 →
Continuity (2)
Provisional Application 61920617 · Dec 24, 2013
Related Publication 20170014429A1 · Jan 19, 2017
Cited By (3)
US 12,226,423 US 12,642,805 US 12,692,288