IP Library Granted Patent US 10,407,502
Granted Patent B2
US 10,407,502 · App. 15/111,102 · Granted Sep 10, 2019

Immunomodulatory agents

Inventors: Samuel D. Waksal (New York, NY); Zhenping Zhu (Woodcliff Lake, NJ); Yan Wu (Doylestown, PA); Stella Martomo (Edgewater, NJ); Zhaojing Zhong (Bronx, NY); Dan Lu (Montvale, NJ)
Assignee: KADMON CORPORATION, LLC
C07K16/2827A61K47/6849C07K14/5443C07K14/7155A61K2039/505C07K2317/31C07K2317/55C07K2317/74C07K2317/76C07K2317/92C07K2319/00
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Quick Facts
Patent No.
US 10,407,502
App. No.
15/111,102
Granted
Sep 10, 2019
Kind
B2
Abstract

The invention provides antibodies that specifically bind to PD-L1 and fusion molecules comprising PD-L1 binding proteins constructed with an IL15 receptor-binding domain, nucleic acid molecules encoding the same, and therapeutic compositions thereof. The agents inhibit PD-L1-mediated immunosuppression and enhance cell and cytokine mediated immunity for the treatment of neoplastic and infectious diseases.

Claims (7)

1. A PD-L1 binding protein comprising a heavy chain CDR-1H comprising SEQ ID NO:121; a heavy chain CDR-2H comprising SEQ ID NO:123; a heavy chain CDR-3H comprising SEQ ID NO:125; a light chain CDR-1L comprising SEQ ID NO:127; a light chain CDR-2L comprising SEQ ID NO:128; and a light chain CDR-3L comprising SEQ ID NO:129.

2. The PD-L1 binding protein of claim 1 , comprising a heavy chain variable domain comprising SEQ ID NO:126 or a sequence that is at least 85% identical to SEQ ID NO:126.

3. The PD-L1 binding protein of claim 1 , comprising a light chain variable domain comprising SEQ ID NO:130 or a sequence that is at least 85% identical to SEQ ID NO:130.

4. The PD-L1 binding protein of claim 1 , further comprising (i) an IL-15 receptor (M-15R) alpha sushi domain comprising amino acids 1-61 of SEQ ID NO:261; and (ii) IL-15 comprising amino acids 96-209 of SEQ ID NO:261, an amino acid sequence at least 95% identical to IL-15, or an IL-15R binding fragment thereof.

5. The PD-L1 binding protein of claim 4 , further comprises a flexible linker joining the IL-15R alpha sushi domain to the IL-15 or IL-15R-binding fragment thereof.

6. The PD-L1 binding protein of claim 5 , wherein the flexible linker comprises 15-20 amino acids which are predominantly serine and glycine.

7. The PD-L1 binding protein of claim 1 , further comprising SEQ ID NO: 261.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Nov 20, 2018
From: WAKSAL, SAMUEL D.; ZHU, ZHENPING; WU, YAN; MARTOMO, STELLA A.; ZHONG, ZHAOJING; LU, DAN
To: KADMON CORPORATION, LLC
Reel/Frame 047552/0781 →
Cited By (1)
US 12,384,846