IP Library Granted Patent US 10,016,421
Granted Patent B2
US 10,016,421 · App. 15/120,053 · Granted Jul 10, 2018

Histone deacetylase 6 inhibition for enhancing T-cell function during anti-tumor response and tumor-peptide vaccination

Inventors: Eduardo M. Sotomayor (Tampa, FL); Alejandro V. Villagra (Tampa, FL)
Assignee: H. Lee Moffitt Cancer Center and Research Institute, Inc.
A61K31/505A61K31/17A61K31/416A61K31/422A61K31/437A61K31/454A61K31/69A61K39/0011A61K39/3955A61K45/06C12N5/0636C12N5/0638A61K2039/5158A61K2039/545A61K2039/55511A61K2039/57A61K2039/585C12N2501/065C12N2501/2302
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Quick Facts
Patent No.
US 10,016,421
App. No.
15/120,053
Granted
Jul 10, 2018
Kind
B2
Abstract

Disclosed are methods whereby an effective amount of a HDAC6 inhibitor is used to activate a subjects T-cell response to tumor or tumor vaccine. Methods of using HDAC6 inhibitors to increase a subjects anti-tumor immune response, alone or in conjunction with other tumor treatments, are also disclosed.

Claims (14)

1. A method of increasing expression of CD69 in a subject's T-cells, comprising: administering to a subject having melanoma, ovarian cancer, breast cancer, or colorectal cancer an amount of a HDAC6 inhibitor effective to increase expression of CD69 in the subject's T-cells, wherein the HDAC6 inhibitor is selected from the group consisting of ACY1215, Tubstatin A, Tubacin, and any combination thereof.

2. The method of claim 1 , wherein the inhibitor is ACY1215.

3. The method of claim 1 , wherein the inhibitor is Tubstatin A, Tubacin, or any combination thereof.

4. The method of claim 1 , wherein the subject is also administered ipilimumab, revlimid, velcade, vemurafenib, or any combination thereof.

5. A method for ex vivo expanding tumor-infiltrating lymphocytes for use in adoptive cell therapy, comprising: culturing tumor fragments from the subject in a culture medium comprising IL-2 and an HDAC6 inhibitor selected from the group consisting of ACY1215, Tubstatin A, Tubacin, and any combination thereof in an amount effective to expand tumor-infiltrating lymphocytes with enriched tumor-reactivity and specificity.

6. A method for treating melanoma, ovarian cancer, breast cancer, or colorectal cancer in a subject, comprising: expanding tumor-infiltrating lymphocytes from a tumor fragment from the subject by culturing the tumor fragments in a culture medium comprising IL-2 and an HDAC6 inhibitor selected from the group consisting of ACY1215, Tubstatin A, Tubacin, and any combination thereof in an amount effective to expand tumor-infiltrating lymphocytes with enriched tumor-reactivity and specificity; treating the subject with nonmyeloablative lymphodepleting chemotherapy; and administering the tumor-infiltrating lymphocytes to the subject.

7. The method of claim 1 , wherein the oncological disorder is metastatic.

8. The method of claim 1 , wherein the oncological disorder is recurrent.

9. The method of claim 1 , wherein the subject is a human.

10. The method of claim 6 , wherein the inhibitor is ACY1215.

11. The method of claim 6 , wherein the inhibitor is Tubstatin A, Tubacin, or any combination thereof.

12. A method of increasing T-cell activation and response against peptide vaccine, comprising: administering to a subject an effective amount of an HDAC6 inhibitor selected from the group consisting of ACY1215, Tubstatin A, Tubacin, and any combination thereof to increase T-cell activation and response against tumor or peptide vaccine in the subject.

13. The method of claim 12 , wherein the HDAC6 inhibitor is administered with the peptide vaccine.

14. The method of claim 12 , wherein the HDAC6 inhibitor is administered within a week after the subject has been administered a peptide vaccine.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Nov 17, 2016
From: SOTOMAYOR, EDUARDO M.; VILLAGRA, ALEJANDRO V.
To: H. LEE MOFFITT CANCER CENTER AND RESEARCH INSTITUTE, INC.
Reel/Frame 040355/0286 →
Continuity (3)
Provisional Application 62085878 · Dec 1, 2014
Provisional Application 61975811 · Apr 5, 2014
Related Publication 20170056402A1 · Mar 2, 2017
Cited By (4)
US 12,201,617 US 12,280,111 US 12,312,345 US 12,365,871