IP Library Granted Patent US 10,605,808
Granted Patent B2
US 10,605,808 · App. 15/140,321 · Granted Mar 31, 2020

Antibody producing non-human animals

Inventors: Ton Logtenberg (Utrecht, NL); Mark Throsby (Utrecht, NL); Robert A. Kramer (Utrecht, NL); Rui Daniel Pinto (Utrecht, NL); Cornelis A. Dekruif (De Bilt, NL); Erwin Houtzager (Zeist, NL)
Assignee: Merus N.V.
G01N33/56966C07K16/00C07K16/005C07K16/10C07K16/22C07K16/248C07K16/2863C07K16/32C07K2317/10C07K2317/14C07K2317/21C07K2317/24C07K2317/31C07K2317/34C07K2317/51C07K2317/515C07K2317/52C07K2317/55C07K2317/56C07K2317/622C07K2317/64C07K2317/76C07K2317/94C07K2319/00
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Quick Facts
Patent No.
US 10,605,808
App. No.
15/140,321
Granted
Mar 31, 2020
Kind
B2
Abstract

Described are transgenic, non-human animals comprising a nucleic acid encoding an immunoglobulin light chain, whereby the immunoglobulin light chain is a common human, human-like, or humanized light chain. Further provided is methods for producing an immunoglobulin from the transgenic, non-human animal.

Claims (18)

1. A method for selecting a single recombinant cell that produces a heterogeneous combination of monospecific and bispecific antibodies, or antibody fragments thereof, wherein the heterogeneous combination of antibodies has specific affinity for two target epitopes, the method comprising:

providing three different variable regions consisting of at least two different heavy chain regions and one light chain variable region from recombinant cells, wherein the sequence of the antigen binding parts of the variable regions originate from a single species and wherein one variable region is able to functionally pair with more than one other variable region, and under conditions allowing for pairing of variable regions and secretion of the paired regions from the recombinant cells resulting in the production of said heterogeneous combination,

providing two target epitopes, and

selecting a single recombinant cell from the recombinant cells that produces a heterogeneous combination that binds the two target epitopes,

wherein the one light chain variable region comprises a rearranged human immunoglobulin light chain variable region consisting of a V and a J and is encoded by a human immunoglobulin light chain V gene segment joined to a human immunoglobulin light chain J gene segment,

wherein the at least two different heavy chain variable regions are each encoded by nucleic acid sequences obtained from a transgenic mouse,

wherein a first of the at least two different heavy chain variable regions encoded by nucleic acid sequences obtained from a transgenic mouse is produced by recombination of a heavy chain gene in a first transgenic mouse in response to challenge with a first antigen comprising at least one of the two target epitopes and wherein a second of the at least two different heavy chain variable regions encoded by nucleic acid sequences obtained from a transgenic mouse is produced by recombination of a heavy chain gene in a second transgenic mouse in response to challenge with a second antigen comprising at least one of the two target epitopes, wherein the first transgenic mouse and second transgenic mouse may be the same mouse or two different mice; and

wherein the genome of each transgenic mouse comprises a transgene comprising the human immunoglobulin light chain V gene segment joined to the human immunoglobulin light chain J gene segment and wherein that mouse further comprises a human VH locus.

2. The method according to claim 1 , wherein said two target epitopes are associated with a disease and/or disorder.

3. The method according to claim 2 , further comprising:

subjecting a heterogeneous combination to a biological assay indicative of an effect of the combination on the disease and/or disorder.

4. The method according to claim 1 , wherein the one variable region able to functionally pair with more than one other variable region does not significantly contribute to the resulting binding specificity of the resulting paired regions.

5. The method according to claim 1 , wherein the combination comprises two monospecific antibodies produced in the single recombinant cell.

6. The method according to claim 1 , wherein the human immunoglobulin light chain V gene segment joined to the human immunoglobulin light chain J gene segment is obtained from a transgenic mouse.

7. The method according to claim 1 , wherein the transgenic mouse, in response to the two target epitopes, produces antibodies with immunoglobulin light chains comprising the rearranged human light chain variable region and murine light chain constant region, paired with a diversity of immunoglobulin heavy chains which bind the two target epitopes.

8. The method according to claim 1 , wherein a first heavy chain of the two heavy chain regions is obtained by immunizing a first mouse with a first target epitope of the two target epitopes and wherein a second heavy chain of the two heavy chain regions is obtained by immunizing a second mouse with a second target epitope of the two target epitopes.

9. The method according to claim 1 , further comprising:

isolating from the set of recombinant cells a single recombinant cell that produces the single heterogeneous combination.

Assignments (6)
NOTICE OF GRANT OF SECURITY INTEREST IN PATENTS Recorded Jan 30, 2026
From: MERUS B.V.
To: WILMINGTON TRUST, NATIONAL ASSOCIATION
Reel/Frame 074562/0322 →
SECURITY INTEREST Recorded Jan 29, 2026
From: MERUS B.V.
To: MORGAN STANLEY SENIOR FUNDING, INC.
Reel/Frame 074532/0434 →
CORRECTIVE ASSIGNMENT TO CORRECT THE ASSIGNEE ADDRESS PREVIOUSLY RECORDED AT REEL: 041675 FRAME: 0842. ASSIGNOR(S) HEREBY CONFIRMS THE CHANGE ADDRESS. Recorded Apr 4, 2017
From: MERUS N.V.
To: MERUS N.V.
Reel/Frame 042322/0304 →
CHANGE OF ADDRESS Recorded Feb 10, 2017
From: MERUS N.V.
To: MERUS N.V.
Reel/Frame 041675/0842 →
CHANGE OF NAME Recorded Jun 1, 2016
From: MERUS B.V.
To: MERUS N.V.
Reel/Frame 038853/0599 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded May 12, 2016
From: HOOGENBOOM, HENDRICUS RENERUS; LOGTENBERG, TON; THROSBY, MARK; KRAMER, ROBERT A; PINTO, RUI DANIEL; DE KRUIF, CORNELIS A.; HOUTZAGER, ERWIN
To: MERUS B.V.
Reel/Frame 038693/0257 →
Continuity (4)
Continuation 12589181 · Oct 19, 2009
Continuation 12459285 · Jun 29, 2009
Provisional Application 61133274 · Jun 27, 2008
Related Publication 20160238600A1 · Aug 18, 2016
Cited By (2)
US 12,291,798 US 12,696,885