IP Library Granted Patent US 9,789,110
Granted Patent B2
US 9,789,110 · App. 15/193,440 · Granted Oct 17, 2017

Diacylglycerol acyltransferase 2 inhibitors

Inventor: Kentaro Futatsugi (Quincy, MA)
Assignee: Pfizer Inc.
A61K31/506A61K31/4545A61K31/5377A61K31/606A61K45/06C07D401/04C07D401/14C07D413/14C07D487/02C07D487/04C07D491/08
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Quick Facts
Patent No.
US 9,789,110
App. No.
15/193,440
Granted
Oct 17, 2017
Kind
B2
Abstract

Compounds of Formula I that inhibit the activity of the diacylglycerol acyltransferase 2 (DGAT2) and their uses in the treatment of diseases linked thereto in animals are described herein.

Claims (5)

1. A method for treating non-alcoholic steatohepatitis (NASH) in humans comprising the step of administering to a human in need of such treatment a therapeutically effective amount of a compound having the structure:

or a pharmaceutically acceptable salt thereof.

2. A method for treating non-alcoholic steatohepatitis (NASH) in humans comprising the step of administering to a human in need of such treatment a therapeutically effective amount of a compound comprising 3-((2-(3-(2-ethoxyphenoxy)piperidin-1-yl)pyrimidine-5-carboxamido)methyl)benzoic acid or (R)-3-((2-(3-(2-ethoxyphenoxy)piperidin-1-yl)pyrimidine-5-carboxamido)methyl)benzoic acid or a pharmaceutically acceptable salt thereof.

3. The method according to claim 1 wherein said compound or pharmaceutically acceptable salt thereof is in admixture with at least one pharmaceutically acceptable excipient.

4. The method according to claim 2 wherein said compound or pharmaceutically acceptable salt thereof is in admixture with at least one pharmaceutically acceptable excipient.

Assignments (1)
ASSIGNEE ADDRESS CORRECTION Recorded Mar 20, 2023
From: PFIZER INC.
To: PFIZER INC.
Reel/Frame 063119/0087 →
Continuity (3)
Division 14643210 · Mar 10, 2015
Provisional Application 61954351 · Mar 17, 2014
Related Publication 20160303125A1 · Oct 20, 2016