IP Library Granted Patent US 10,143,665
Granted Patent B2
US 10,143,665 · App. 15/238,037 · Granted Dec 4, 2018

Methods for storing cysteamine formulations and related methods of treatment

Inventors: Michael DesJardin (Aptos, CA); Mark Johnson (Fort Collins, CO)
Assignee: Horizon Orphan LLC
A61K31/145A61K9/5026
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Quick Facts
Patent No.
US 10,143,665
App. No.
15/238,037
Granted
Dec 4, 2018
Kind
B2
Abstract

Methods of storing and methods of stabilizing pharmaceutical compositions comprising cysteamine, or a pharmaceutically acceptable salt thereof, are provided. Methods of distributing pharmaceutical compositions comprising cysteamine, or a pharmaceutically acceptable salt thereof, and methods of treating cystinosis also are provided.

Claims (8)

1. A method of treating cystinosis in a subject in need thereof, comprising administering twice daily to the subject an oral pharmaceutical composition comprising cysteamine bitartrate, wherein the oral pharmaceutical composition contains 2-hydroxythiomorpholine in an amount less than 0.5% relative to the amount of cysteamine bitartrate, and wherein the oral pharmaceutical composition is stored at a temperature of between about 2° C. and about 8° C. prior to administration.

2. The method according to claim 1 , wherein the oral pharmaceutical composition further comprises an enteric coating wherein the enteric coating comprises poly(methacrylic acid co-ethyl acrylate) 1:1.

3. A method of treating cystinosis in a subject in need thereof, comprising administering twice daily to the subject an oral pharmaceutical composition comprising cysteamine bitartrate, wherein the oral pharmaceutical composition contains cystamine in an amount less than 4% relative to the amount of cysteamine bitartrate, and wherein the oral pharmaceutical composition is stored at a temperature of between about 2° C. and about 8° C. prior to administration.

4. The method according to claim 3 , wherein the oral pharmaceutical composition further comprises an enteric coating, wherein the enteric coating comprises poly(methacrylic acid co-ethyl acrylate) 1:1.

5. A method of treating cystinosis in a subject in need thereof, comprising administering twice daily to the subject an oral pharmaceutical composition comprising cysteamine bitartrate, wherein the oral pharmaceutical composition contains cystamine tartrate amide in an amount less than 0.5% relative to the amount of cysteamine bitartrate, and wherein the oral pharmaceutical composition is stored at a temperature of between about 2° C. and about 8° C. prior to administration.

6. The method according to claim 5 , wherein the oral pharmaceutical composition further comprises an enteric coating, wherein the enteric coating comprises poly(methacrylic acid co-ethyl acrylate) 1:1.

7. A method of treating cystinosis in a subject in need thereof, comprising administering twice daily to the subject an oral pharmaceutical composition comprising cysteamine bitartrate, wherein the oral pharmaceutical composition contains 2-hydroxymethylthiazolidine in an amount less than 0.05% relative to the amount of cysteamine bitartrate, and wherein the oral pharmaceutical composition is stored at a temperature of between about 2° C. and about 8° C. prior to administration.

8. The method according to claim 7 , wherein the oral pharmaceutical composition further comprises an enteric coating, wherein the enteric coating comprises poly(methacrylic acid co-ethyl acrylate) 1:1.

Assignments (6)
MERGER AND CHANGE OF NAME Recorded Sep 19, 2025
From: HORIZON THERAPEUTICS, LLC; HORIZON ORPHAN LLC
To: HORIZON THERAPEUTICS U.S. HOLDING LLC
Reel/Frame 072311/0255 →
RELEASE OF SECURITY INTEREST Recorded Oct 6, 2023
From: CITIBANK, N.A.
To: HORIZON THERAPEUTICS U.S. HOLDING LLC (FKA RAPTOR PHARMACEUTICALS INC.)
Reel/Frame 065178/0955 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Aug 21, 2018
From: JOHNSON, MARK
To: HORIZON ORPHAN LLC
Reel/Frame 046651/0208 →
CHANGE OF NAME Recorded Dec 20, 2016
From: RAPTOR PHARMACEUTICALS INC.
To: HORIZON ORPHAN LLC
Reel/Frame 041034/0782 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Nov 3, 2016
From: DESJARDIN, MICHAEL
To: RAPTOR PHARMACEUTICALS INC.
Reel/Frame 040556/0045 →
SECURITY AGREEMENT Recorded Oct 26, 2016
From: RAPTOR PHARMACEUTICALS INC.
To: CITIBANK, N.A., AS COLLATERAL AGENT
Reel/Frame 040479/0578 →
Continuity (2)
Provisional Application 62256613 · Nov 17, 2015
Related Publication 20170135968A1 · May 18, 2017