IP Library Granted Patent US 9,889,111
Granted Patent B2
US 9,889,111 · App. 15/339,196 · Granted Feb 13, 2018

Pharmaceutical composition comprising omega-(arylsulfonyl)alkylnitrile

Inventors: Joseph St. Laurent (Lakeville, MA); Gerald S. Jones (Norwood, MA); David M. Bresse (Middleboro, MA)
Assignee: OLATEC THERAPEUTICS LLC
A61K31/277A61K9/0014A61K9/0053A61K9/06A61K47/10A61K47/14A61K47/32A61K47/34
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Quick Facts
Patent No.
US 9,889,111
App. No.
15/339,196
Granted
Feb 13, 2018
Kind
B2
Abstract

The present invention is directed to a pharmaceutical composition comprising a pharmaceutically acceptable carrier and a ω-(arylsulfonyl)alkylnitrile compound, or a pharmaceutically acceptable salt thereof. The present invention is also directed to a method for treating inflammation, inflammatory-related disorders, or pain, by administering an ω-(arylsulfonyl)alkylnitrile compound or a pharmaceutically acceptable salt or solvate thereof to a subject in need thereof.

Claims (12)

1. A pharmaceutical composition comprising a pharmaceutically acceptable carrier and a compound of C, or a pharmaceutically acceptable salt thereof:

2. The pharmaceutical composition according to claim 1 , wherein the compound has at least 90% (w/w) purity, and the composition is in a topical form of gels, creams, lotions, ointments, or patches.

3. The pharmaceutical composition according to claim 2 , wherein the pharmaceutically acceptable carrier is an emollient selected from the group consisting of: lauryl lactate, diethylene glycol monoethyl ether, caprylic/capric triglyceride, octisalate, silicone fluid, squalene, and sunflower oil.

4. The pharmaceutical composition according to claim 2 , wherein the pharmaceutically acceptable carrier is a permeation enhancer selected from the group consisting of lactate esters and diethylene glycol monoethyl ether.

5. The pharmaceutical composition according to claim 4 , further comprising acrylates/C10-30 alkyl and tris(2-hydroxyethyl)amine.

6. The pharmaceutical composition according to claim 1 , wherein the compound has at least 90% (w/w) purity, and the composition is in an oral form of tablets or capsules.

7. A method of treating inflammation, comprising the steps of:

identifying a subject suffering from inflammation, and

administering to the subject the pharmaceutical composition of claim 1 , in an amount effective to treat inflammation.

8. The method according to claim 7 , wherein said method reduces or alleviates the symptoms of localized manifestations of inflammation characterized by acute or chronic swelling, pain, or redness.

9. The method according to claim 7 , wherein said compound is administered by local administration or systemic administration.

10. The method according to claim 7 , wherein said compound is administered by topical administration.

Assignments (3)
CHANGE OF NAME Recorded Nov 7, 2023
From: OLATEC THERAPEUTICS LLC
To: OLATEC THERAPEUTICS, INC.
Reel/Frame 065489/0809 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Nov 3, 2016
From: ST. LAURENT, JOSEPH; JONES, GERALD S.; BRESSE, DAVID M.
To: OLATEC INDUSTRIES LLC
Reel/Frame 040219/0003 →
CHANGE OF NAME Recorded Nov 3, 2016
From: OLATEC INDUSTRIES LLC
To: OLATEC THERAPEUTICS LLC
Reel/Frame 040562/0388 →
Continuity (5)
Continuation 14554848 · Nov 26, 2014
Continuation In Part 13909957 · Jun 4, 2013
Provisional Application 61655916 · Jun 5, 2012
Provisional Application 61909762 · Nov 27, 2013
Related Publication 20170105962A1 · Apr 20, 2017