IP Library Granted Patent US 10,196,353
Granted Patent B2
US 10,196,353 · App. 15/358,458 · Granted Feb 5, 2019

Chemical compounds

Inventors: Philip Stewart Turnbull (Research Triangle Park, NC); Rodolfo Cadilla (Research Triangle Park, NC)
Assignee: GlaxoSmithKline Intellectual Property (No 2) Limited
C07D209/14A61K31/404C07D209/08C07D209/10C07D209/42C07D401/06
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Quick Facts
Patent No.
US 10,196,353
App. No.
15/358,458
Granted
Feb 5, 2019
Kind
B2
Abstract

This invention relates to non-steroidal compounds that are modulators of androgen receptor, and also to the methods for the making and use of such compounds.

Claims (12)

1. A pharmaceutically acceptable salt of the compound:

2. A pharmaceutical composition comprising a pharmaceutically acceptable salt of the compound according to claim 1 and one or more pharmaceutically acceptable excipients.

3. A method of treating muscle wasting associated with chronic obstructive pulmonary disease (COPD), wherein said method comprises administering a pharmaceutically acceptable salt of the compound according to claim 1 to a human subject in need thereof.

4. A method of treating muscle wasting associated with chronic kidney disease (CKD), wherein said method comprises administering a pharmaceutically acceptable salt of the compound according to claim 1 to a human subject in need thereof.

5. A method of treating muscle wasting associated with chronic heart failure (CHF), wherein said method comprises administering a pharmaceutically acceptable salt of the compound according to claim 1 to a human subject in need thereof.

6. A method of treating urinary incontinence, wherein said method comprises administering a pharmaceutically acceptable salt of the compound according to claim 1 to a human subject in need thereof.

7. A method of accelerating hip fracture repair and healing, wherein said method comprises administering a pharmaceutically acceptable salt of the compound according to claim 1 to a human subject in need thereof.

8. The method according to claim 3 , wherein 0.1-50 mgs of a pharmaceutically acceptable salt of the compound is administered.

9. The method according to claim 4 , wherein 0.1-50 mgs of a pharmaceutically acceptable salt of the compound is administered.

10. The method according to claim 5 , wherein 0.1-50 mgs of a pharmaceutically acceptable salt of the compound is administered.

11. The method according to claim 6 , wherein 0.1-50 mgs of a pharmaceutically acceptable salt of the compound is administered.

12. The method according to claim 7 , wherein 0.1-50 mgs of a pharmaceutically acceptable salt of the compound is administered.

Assignments (2)
CHANGE OF ADDRESS Recorded Apr 16, 2025
From: GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO.2) LIMITED
To: GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO.2) LIMITED
Reel/Frame 070854/0469 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Dec 19, 2018
From: TURNBULL, PHILIP STEWART; CADILLA, RODOLFO
To: GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO.2) LIMITED
Reel/Frame 047817/0269 →
Continuity (5)
Continuation 14549034 · Nov 20, 2014
Continuation 13941911 · Jul 15, 2013
Provisional Application 61748874 · Jan 4, 2013
Provisional Application 61672455 · Jul 17, 2012
Related Publication 20170073309A1 · Mar 16, 2017