IP Library Granted Patent US 10,383,868
Granted Patent B2
US 10,383,868 · App. 15/361,485 · Granted Aug 20, 2019

Quinoline containing compounds and their use for treating endoplasmic reticulum stress-related diseases

Inventor: Russell Dahl (Saint John, IN)
A61K31/4709A61K31/47
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Quick Facts
Patent No.
US 10,383,868
App. No.
15/361,485
Granted
Aug 20, 2019
Kind
B2
Abstract

Provided herein are quinoline, pharmaceutical compositions thereof, and methods of their use for treating, preventing, or ameliorating one or more symptoms of an endoplasmic reticulum stress-caused disease. Also provided herein are methods of their use for reducing endoplasmic reticulum stress and modulating the activity of a sarcoplasmic/endoplasmic reticulum Ca 2+ ATPase.

Claims (4)

1. A method for treating or ameliorating one or more symptoms of type 2 diabetes in a subject in need thereof, comprising administering to the subject an effective amount of a compound, wherein the compound is selected from the group consisting of:

or an isotope variant thereof, or a pharmaceutically acceptable salt, solvate, or hydrate thereof.

2. The method of claim 1 , wherein the method comprises administering to the subject a second therapeutic agent, in combination or alternation.

3. The method of claim 1 , wherein the subject is a human.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 13, 2021
From: DAHL, RUSSELL, DR
To: NEURODON CORPORATION
Reel/Frame 055251/0757 →
Continuity (2)
Provisional Application 62260513 · Nov 28, 2015
Related Publication 20170231973A1 · Aug 17, 2017