IP Library Granted Patent US 9,844,559
Granted Patent B2
US 9,844,559 · App. 15/454,874 · Granted Dec 19, 2017

Neridronic acid for treating bone marrow lesions

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Quick Facts
Patent No.
US 9,844,559
App. No.
15/454,874
Granted
Dec 19, 2017
Kind
B2
Abstract

Oral dosage forms of osteoclast inhibitors, such as zoledronic acid, in an acid or a salt form can be used to treat or alleviate pain or related conditions, such as bone marrow lesions.

Claims (29)

1. A method of treating a bone marrow lesion comprising:

selecting a patient having 1) a bone marrow lesion and 2) an OARSI Grade 0 or Kellgren and Lawrence Grade 0 or Grade 1 of joint space narrowing, and intravenously administering neridronic acid to the patient at least two times, for the treatment of the bone marrow lesion.

2. The method of claim 1 , wherein the neridronic acid is administered daily.

3. The method of claim 1 , wherein the neridronic acid is administered weekly.

4. The method of claim 1 , wherein the neridronic acid is administered monthly.

5. The method of claim 1 , wherein the patient is suffering from complex regional pain syndrome.

6. The method of claim 5 , wherein a fracture is an inciting event for the complex regional pain syndrome.

7. The method of claim 6 , wherein about 50 mg to about 600 mg of the neridronic acid is administered within a period of about one month.

8. The method of claim 1 , wherein administering the neridronic acid results in a reduction in size of the bone marrow lesion of at least about 20% relative to the baseline before administration of the neridronic acid.

9. The method of claim 1 , further comprising administration of a steroid.

10. The method of claim 9 , wherein about 200 mg to about 400 mg of the neridronic acid is administered within a period of about one month.

11. The method of claim 9 , wherein about 300 mg to about 600 mg of the neridronic acid is administered within a period of about one month.

12. The method of claim 10 , wherein the neridronic acid is administered in two doses.

13. The method of claim 11 , wherein the neridronic acid is administered in two doses.

14. The method of claim 1 , wherein the neridronic acid is in an acid form.

15. The method of claim 1 , wherein the neridronic acid is in a salt form.

16. A method of treating a bone marrow edema comprising: selecting a patient having 1) a bone marrow edema and 2) an OARSI Grade 0 or Kellgren and Lawrence Grade 0 or Grade 1 of joint space narrowing, and orally administering neridronic acid to the patient for the treatment of the bone marrow edema.

17. The method of claim 16 , wherein the neridronic acid is administered daily.

18. The method of claim 16 , wherein the neridronic acid is administered weekly.

19. The method of claim 16 , wherein the neridronic acid is administered monthly.

20. The method of claim 16 , wherein the patient is suffering from complex regional pain syndrome.

21. The method of claim 20 , wherein a fracture is an inciting event for the complex regional pain syndrome.

22. The method of claim 21 , wherein about 50 mg to about 600 mg of the neridronic acid is administered within a period of about one month.

23. The method of claim 16 , wherein about 200 mg to about 400 mg of the neridronic acid is administered within a period of about one month.

24. The method of claim 16 , wherein about 300 mg to about 600 mg of the neridronic acid is administered within a period of about one month.

25. The method of claim 23 , wherein the neridronic acid is administered in at least two doses.

26. The method of claim 24 , wherein the neridronic acid is administered in at least two doses.

27. The method of claim 16 , wherein the neridronic acid is in an acid form.

28. The method of claim 16 , wherein the neridronic acid is in a salt form.

Assignments (3)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 10, 2018
From: TABUTEAU, HERRIOT
To: ANTECIP BIOVENTURES II LLC
Reel/Frame 045034/0542 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Dec 8, 2017
From: TABUTEAU, HERRIOT
To: ANTECIP BIOVENTURES II LLC
Reel/Frame 044777/0488 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 9, 2017
From: TABUTEAU, HERRIOT
To: ANTECIP BIOVENTURES II LLC
Reel/Frame 041532/0597 →