IP Library Granted Patent US 10,329,357
Granted Patent B2
US 10,329,357 · App. 15/463,340 · Granted Jun 25, 2019

Treatment of ocular disease

View Patent ↗
Loading inventors, assignments & file history…
Monitor This Case
Get email alerts when status or documents change.
Order Certified Copies
Most orders are placed with the USPTO same day — all within 24 business hours.
Order via The Patent Place →
Pre-filled with this patent's details
Quick Facts
Patent No.
US 10,329,357
App. No.
15/463,340
Granted
Jun 25, 2019
Kind
B2
Abstract

Disclosed are methods for treating eye diseases or conditions characterized by vascular instability, vascular leakage and neovacularization such as diabetic macular edema, age-related macular edema, choroidal neovascularization, diabetic retinopathy, trauma, ocular ischemia, retinal angiomatous proliferation, macular telangiectasia and uveitis.

Claims (11)

1. A method for reducing retinal neovascularization in a human in need thereof, the method comprising administering to the human a therapeutically-effective amount of an intact monoclonal antibody, wherein the intact monoclonal antibody is R15E6 or a humanized form thereof, wherein the human has diabetic macular edema, wherein the antibody R15E6 is produced by a hybridoma deposited under the accession number ATCC PTA-7580.

2. The method of claim 1 , wherein the intact monoclonal antibody inhibits a tyrosine phosphatase.

3. The method of claim 1 , wherein the intact monoclonal antibody inhibits human protein tyrosine phosphatase beta (HPTP-β).

4. The method of claim 1 , wherein the intact monoclonal antibody is administered by intraocular injection.

5. The method of claim 1 , wherein the intact monoclonal antibody is administered by subcutaneous injection.

6. The method of claim 1 , wherein the intact monoclonal antibody is administered by intravenous injection.

7. The method of claim 1 , wherein the therapeutically-effective amount is from about 0.01 mg/kg to about 10 mg/kg by weight of the human.

8. The method of claim 1 , wherein the intact monoclonal antibody binds an FN3 repeat of HPTP-β.

9. The method of claim 1 , wherein the intact monoclonal antibody binds a first FN3 repeat of HPTP-β.

10. The method of claim 1 , wherein the intact monoclonal antibody binds to SEQ ID NO: 4.

11. The method of claim 1 , wherein the intact monoclonal antibody enhances Tie2 receptor activation.

Assignments (4)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Sep 9, 2021
From: AERPIO PHARMACEUTICALS, INC.
To: EYEPOINT PHARMACEUTICALS, INC.
Reel/Frame 057448/0033 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 17, 2020
From: AERPIO THERAPEUTICS LLC
To: AERPIO PHARMACEUTICALS, INC.
Reel/Frame 052432/0789 →
CHANGE OF NAME Recorded Jul 31, 2019
From: AERPIO THERAPEUTICS, INC.
To: AERPIO THERAPEUTICS LLC
Reel/Frame 049924/0512 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 5, 2017
From: PETERS, KEVIN; SHALWITZ, ROBERT
To: AERPIO THERAPEUTICS, INC.
Reel/Frame 041853/0119 →
Cited By (1)
US 12,398,204