IP Library Patent Application 15540566
Patent Application
App. No. 15/540,566

USE OF PICOLINAMIDES AS FUNGICIDES

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Quick Facts
Patent No.
US None
App. No.
15/540,566
Abstract

This disclosure relates to picolinamides of Formula I and their use as fungicides.

Claims (46)

1 . A composition for the control of a fungal pathogen including mixtures of at least one of the compounds of Formula 1

wherein

X is hydrogen or C(O)R 5 ;

Y is hydrogen, C(O)R 5 , or Q;

Q is

R 1 and R 11 are independently chosen from hydrogen or alkyl, optionally substituted with 0, 1 or multiple R 8 ; Alternatively, R 1 and R 11 may be taken together to form a 3-6 membered saturated or partially saturated carbocycle or heterocycle, optionally substituted with 0, 1 or multiple R 8 ;

R 2 and R 12 are independently chosen from hydrogen or methyl;

R 3 is chosen from aryl or heteroaryl, each optionally substituted with 0, 1 or multiple R 8 ;

R 4 is chosen from alkyl, aryl, or acyl, each optionally substituted with 0, 1 or multiple R 8 ;

R 5 is chosen from alkoxy or benzyloxy, each optionally substituted with 0, 1, or multiple R 8 ;

R 6 is chosen from hydrogen, alkoxy, or halo, each optionally substituted with 0, 1, or multiple R 8 ;

R 7 is chosen from hydrogen, —C(O)R 9 , or —CH 2 OC(O)R 9 ;

R 8 is chosen from hydrogen, alkyl, aryl, acyl, halo, alkenyl, alkoxy, or heterocyclyl, each optionally substituted with 0, 1, or multiple R 10 ;

R 9 is chosen from alkyl, alkoxy, or aryl, each optionally substituted with 0, 1, or multiple R 8 ; and

R 10 is chosen from hydrogen, alkyl, aryl, acyl, halo, alkenyl, alkoxy, or heterocyclyl.

2 . A composition according to claim 1 , wherein X is hydrogen and Y is Q.

3 . A composition according to claim 2 , wherein R 6 is alkoxy.

4 . A composition according to claim 3 , wherein R 7 is hydrogen.

5 . A composition according to claim 4 , wherein R 1 and R 11 are independently chosen from hydrogen or alkyl.

6 . (canceled)

7 . A composition according to claim 4 , wherein R 3 is aryl, optionally substituted with 0, 1 or multiple R 8 .

8 . A composition according to claim 4 , wherein R 4 is chosen from alkyl or aryl, each optionally substituted with 0, 1 or multiple R 8 .

9 . A composition according to claim 4 , wherein R 1 and R 11 are independently chosen from hydrogen or alkyl, optionally substituted with 0, 1 or multiple R 8 , and R 4 is chosen from alkyl or aryl, each optionally substituted with 0, 1 or multiple R 8 .

10 . A composition according to claim 3 , wherein R 7 is chosen from —C(O)R 9 , or —CH 2 OC(O)R 9 .

11 . A composition according to claim 10 , wherein R 9 is alkyl, optionally substituted with 0, 1 or multiple R 8 .

12 . A composition according to claim 11 , wherein R 1 and R 11 are independently chosen from hydrogen or alkyl.

13 . (canceled)

14 . A composition according to claim 11 , wherein R 3 is aryl, optionally substituted with 0, 1 or multiple R 8 .

15 . A composition according to claim 11 , wherein R 4 is chosen from alkyl or aryl, each optionally substituted with 0, 1 or multiple R 8 .

16 . A composition according to claim 11 , wherein R 1 and R 11 are independently chosen from hydrogen or alkyl, R 3 is aryl, optionally substituted with 0, 1 or multiple R 8 , and R 4 is chosen from alkyl or aryl, each optionally substituted with 0, 1 or multiple R 8 .

17 . A composition according to claim 16 , wherein R 9 is chosen from —CH 3 , —CH 2 OCH 2 CH 3 , —CH 2 CH 2 OCH 3 , —CH(CH 3 ) 2 , —CH 2 CH 2 CH 2 CH 3 , or -cyclopropyl.

18 . A composition for the control of a fungal pathogen including at least one of the compositions of claim 9 and a phytologically acceptable carrier material.

19 . A composition for the control of a fungal pathogen including at least one of the compositions of claim 16 and a phytologically acceptable carrier material.

20 . (canceled)

21 . A composition for the control of a fungal pathogen including mixtures of at least one of the compositions of claim 9 and another pesticide including fungicides, insecticides, nematocides, miticides, arthropodicides, bactericides and combinations thereof.

22 . A composition for the control of a fungal pathogen including mixtures of at least one of the compositions of claim 16 and another pesticide including fungicides, insecticides, nematocides, miticides, arthropodicides, bactericides and combinations thereof.

23 . (canceled)

24 . (canceled)

25 . (canceled)

26 . (canceled)

27 . (canceled)

28 . A method for the control and prevention of fungal attack on a plant, the method including the step of: Applying a fungicidally effective amount of at least one of the compositions of claim 9 to at least one of the plant, an area adjacent to the plant, soil adapted to support growth of the plant, a root of the plant, and foliage of the plant.

29 . A method for the control and prevention of fungal attack on a plant, the method including the step of: Applying a fungicidally effective amount of at least one of the compositions of claim 16 to at least one of the plant, an area adjacent to the plant, soil adapted to support growth of the plant, a root of the plant, and foliage of the plant.

30 . (canceled)

31 . (canceled)

32 . (canceled)

Assignments (1)
CHANGE OF NAME Recorded Nov 8, 2021
From: DOW AGROSCIENCES LLC
To: CORTEVA AGRISCIENCE LLC
Reel/Frame 058044/0184 →