IP Library Granted Patent US 10,456,442
Granted Patent B2
US 10,456,442 · App. 15/579,988 · Granted Oct 29, 2019

FGF receptor ligands for treating diabetes and obesity

Inventor: Streamson Chua, Jr. (Dobbs Ferry, NY)
Assignee: Albert Einstein College of Medicine
A61K38/10A61K9/0043A61P3/04A61P3/10
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Quick Facts
Patent No.
US 10,456,442
App. No.
15/579,988
Granted
Oct 29, 2019
Kind
B2
Abstract

Methods for treating diabetes or obesity are provided comprising administering to the subject an amount of an agent that binds a central nervous system FGF receptor homodimer.

Claims (7)

1. A method of treating diabetes or obesity in a subject comprising administering to the subject a peptide consisting of the sequence X1-X2-F-X3-X4-X5-V-X6-X7-Q-X8-X9-X10, wherein F is a phenylalanine, V is a valine, Q is glutamine, X1 is the amino acid P or V, X2 is the amino acid N or D, X3 is the amino acid T, N or R, X4 is the amino acid Q or I, X5 is the amino acid H or Y, X6 is the amino acid R or E, X7 is the amino acid E, D or N, X8 is the amino acid S, G or T, X9 is the amino acid L, A or R, and X10 is the amino acid V, M or A (SEQ ID NO:1) in an amount effective to treat diabetes or obesity in the subject.

2. The method of claim 1 , wherein X1 is P, X2 is N, X4 is Q, and X6 is R (SEQ ID NO:2).

3. The method of claim 2 , wherein X3 is T or N, X7 is E or D, X8 is S or G, X9 is L or A, and X10 is V or M (SEQ ID NO:3).

4. The method of claim 1 , wherein the peptide consists of the sequence PNFTQHVREQSLV (SEQ ID NO:4).

5. The method of claim 1 , wherein the peptide consists of the sequence PNFNQYVRDQGAM (SEQ ID NO:5).

6. The method of claim 1 , wherein the peptide consists of the sequence VDFRIHVENQTRA (SEQ ID NO:6).

7. The method of claim 1 , wherein the diabetes is type II diabetes.

Assignments (1)
MERGER AND CHANGE OF NAME Recorded Feb 26, 2019
From: ALBERT EINSTEIN COLLEGE OF MEDICINE, INC.; ALBERT EINSTEIN COLLEGE OF MEDICINE
To: ALBERT EINSTEIN COLLEGE OF MEDICINE
Reel/Frame 048438/0275 →
Continuity (2)
Provisional Application 62181413 · Jun 18, 2015
Related Publication 20180169181A1 · Jun 21, 2018