IP Library Granted Patent US 10,624,869
Granted Patent B2
US 10,624,869 · App. 15/589,887 · Granted Apr 21, 2020

Methods for the treatment of recurrent glioblastoma (RGBM)

Inventor: Stanislaw R. Burzynski (Houston, TX)
A61K31/198A61K31/192A61K31/197A61K31/436A61K31/44A61K31/506A61K39/3955A61K45/06A61P35/00C07K16/22A61K2039/545A61K2300/00
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Quick Facts
Patent No.
US 10,624,869
App. No.
15/589,887
Granted
Apr 21, 2020
Kind
B2
Abstract

Methods for the treatment of cancer, including glioblastoma multiforme (GBM) and recurrent glioblastoma multiforme (RGBM). The method includes administering to a patient a plurality of extraneous antineoplastons and a plurality of targeted agents. The plurality of extraneous antineoplastons may include two or more antineoplastons selected from phenylacetylglutaminate sodium (PG), phenylacetylisoglutaminate sodium (iso-PG), and phenylacetate (PN). The plurality of targeted agents may include two or more agents selected from bevacizumab, pazopanib, sorafenib, dasatinib, and everolimus.

Claims (21)

1. A method for treating recurrent glioblastoma multiforme (RGBM) in a patient in need thereof, the method consisting of:

(a) intravenously administering to a patient a plurality of extraneous antineoplastons consisting of about a 4:1 ratio of phenylacetate (PN) and phenylacetylglutaminate sodium (PG) at a dosage of from about 0.08 g/kg/day to about 0.6 g/kg/day; and

(b) administering to the patient a plurality of targeted agents consisting of pazopanib administered orally at a dose of from about 1 mg/kg/day to about 12 mg/kg/day,

dasatinib administered orally at a dose of from about 0.3 mg/kg/day to about 2.0 mg/kg/day,

everolimus administered orally at a dose of from about 0.03 mg/kg/day to about 0.15 mg/kg/day, and

bevacizumab administered intravenously every 1 to 3 weeks at a dose of from about 2 mg/kg/day to about 15 mg/kg/day.

2. The method of claim 1 , wherein the plurality of extraneous antineoplastons consists of about a 4:1 ratio of PN and PG in the following amounts:

from about 0.064 g/kg/day to about 0.48 g/kg/day PN and

from about 0.016 g/kg/day to about 0.12 g/kg/day PG.

3. The method of claim 1 , wherein the plurality of extraneous antineoplastons and the pazopanib, dasatinib, and everolimus are administered daily for at least 8 weeks and the bevacizumab is administered intravenously every 1 to 3 weeks for at least 8 weeks.

4. The method of claim 1 , wherein the patient failed to achieve an objective response as a result of at least one radiation treatment and/or at least chemotherapy treatment comprising temozolomide (TMZ) and/or bevacizumab (BVZ), prior to the administration of the plurality of extraneous antineoplastons and the plurality of targeted agents.

5. The method of claim 1 , wherein the patient has undergone a resection of a glioma prior to the administration of the plurality of extraneous antineoplastons and the plurality of targeted agents.

6. A method for treating recurrent glioblastoma multiforme (RGBM) in a patient in need thereof, the method consisting of concurrently administering to a patient:

(a) intravenously, a plurality of extraneous antineoplastons consisting of about a 4:1 ratio of phenylacetate (PN) and phenylacetylglutaminate sodium (PG) at a dosage of from about 0.08 g/kg/day to about 0.6 g/kg/day;

(b) orally, pazopanib at a dose of from about 1 mg/kg/day to about 12 mg/kg/day, dasatinib at a dose of from about 0.3 mg/kg/day to about 2.0 mg/kg/day, and everolimus at a dose of from about 0.03 mg/kg/day to about 0.15 mg/kg/day; and

(c) intravenously, bevacizumab every 1 to 3 weeks at a dose of from about 2 mg/kg/day to about 15 mg/kg/day.

7. The method of claim 6 , wherein the plurality of extraneous antineoplastons consists of about a 4:1 ratio of PN and PG in the following amounts:

from about 0.064 g/kg/day to about 0.48 g/kg/day PN; and

from about 0.016 g/kg/day to about 0.12 g/kg/day PG.

8. The method of claim 1 , wherein the about a 4:1 ratio of phenylacetate (PN) and phenylacetylglutaminate sodium (PG) is intravenously administered at a dosage of from about 0.2 g/kg/day to about 0.4 g/kg/day.

9. The method of claim 6 , wherein the about a 4:1 ratio of phenylacetate (PN) and phenylacetylglutaminate sodium (PG) is intravenously administered at a dosage of from about 0.2 g/kg/day to about 0.4 g/kg/day.

Continuity (1)
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Cited By (1)
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