IP Library Granted Patent US 10,058,574
Granted Patent B2
US 10,058,574 · App. 15/592,178 · Granted Aug 28, 2018

Compositions comprising bacterial strains

Inventors: George Grant (Aberdeen, GB); Angela Margaret Patterson (Norwich, GB); Imke Mulder (Aberdeen, GB); Seanin McCluskey (Aberdeen, GB); Emma Raftis (Leeds, GB)
Assignee: 4D Pharma Research Limited
A61K35/74A23C9/12A23L33/135A61K9/19A61K39/0216C12R1/01A23V2002/00A61K2039/52A61K2039/545A61K2039/58
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Quick Facts
Patent No.
US 10,058,574
App. No.
15/592,178
Granted
Aug 28, 2018
Kind
B2
Abstract

The invention provides compositions comprising bacterial strains for treating and preventing inflammatory and autoimmune diseases.

Claims (45)

1. A pharmaceutical composition that comprises a therapeutically effective amount of a bacteria strain of the genus Bacteroides;

wherein the bacteria strain is lyophilized;

wherein the pharmaceutical composition optionally further comprises a pharmaceutically acceptable excipient, diluent, or carrier;

wherein the therapeutically effective amount of the bacteria strain comprises from about 1×10 3 to about 1×10 11 CFU/g of the bacteria strain with respect to total weight of the pharmaceutical composition; and

wherein the bacteria strain comprises a polynucleotide sequence of a 16S rRNA gene that has at least 95% sequence identity to the polynucleotide sequence of SEQ ID NO:4, as determined by a Smith-Waterman homology search algorithm using an affine gap search with a gap open penalty of 12, a gap extension penalty of 2, and a Blocks Substitution Matrix (BLOSUM) of 62.

2. The pharmaceutical composition of claim 1 , wherein the bacteria strain comprises the polynucleotide sequence of SEQ ID NO:4.

3. The pharmaceutical composition of claim 1 , wherein the pharmaceutical composition is effective to reduce a level of at least one pro-inflammatory cytokine.

4. The pharmaceutical composition of claim 3 , wherein the at least one pro-inflammatory cytokine comprises an IL-17 cytokine selected from the group consisting of: IL-17A, IL-17B, IL-17C, IL-17D, IL-17E, and IL-17F.

5. The pharmaceutical composition of claim 3 , wherein the at least one pro-inflammatory cytokine comprises a cytokine selected from the group consisting of: IFN-γ, IL-1β, RANTES, MIP-1α, IL-8, and IL-6.

6. The pharmaceutical composition of claim 1 , wherein the pharmaceutical composition contains a single bacteria strain.

7. The pharmaceutical composition of claim 1 , wherein the bacteria strain is viable and capable of at least partially colonizing an intestine of a human subject.

8. The pharmaceutical composition of claim 1 , wherein at least 50% of the bacteria strain as measured by an amount of CFU, remains viable after about 1 year of storage when the pharmaceutical composition is stored in a closed container at 25° C. at 95% relative humidity.

9. The pharmaceutical composition of claim 1 , wherein the pharmaceutical composition is a lyophilized composition.

10. The pharmaceutical composition of claim 1 , wherein the pharmaceutical composition comprises a lyoprotectant which is the pharmaceutically acceptable excipient, diluent, or carrier.

11. The pharmaceutical composition of claim 1 , wherein the pharmaceutical composition comprises a prebiotic compound selected from the group consisting of: a fructo-oligosaccharide, a short-chain fructo-oligosaccharide, inulin, an isomalt-oligosaccharide, a transgalacto-oligosaccharide, a pectin, a xylo-oligosaccharide, a chitosan-oligosaccharide, a beta-glucan, an arable gum modified starch, a polydextrose, a D-tagatose, an acacia fiber, carob, an oat, and a citrus fiber.

12. A method of treating a condition mediated by the Th17 pathway in a subject in need thereof, comprising administering to the subject a therapeutically effective amount of a pharmaceutical composition that comprises a bacteria strain of the genus Bacteroides;

wherein the administering is effective to produce a decrease in production of at least one pro-inflammatory cytokine in the subject, thereby treating the condition mediated by the Th17 pathway in the subject; and

wherein the bacteria strain is lyophilized;

wherein the pharmaceutical composition optionally further comprises a pharmaceutically acceptable excipient, diluent, or carrier;

wherein the therapeutically effective amount of the bacteria strain comprises from about 1×10 3 to about 1×10 11 CFU/g of the bacteria strain with respect to total weight of the pharmaceutical composition; and

wherein the bacteria strain comprises a polynucleotide sequence of a 16S rRNA gene that has at least 95% sequence identity to the polynucleotide sequence of SEQ ID NO:4, as determined by a Smith-Waterman homology search algorithm using an affine gap search with a gap open penalty of 12, a gap extension penalty of 2, and a Blocks Substitution Matrix (BLOSUM) of 62.

13. The method of claim 12 , wherein the pharmaceutical composition comprises a single bacteria strain.

14. The method of claim 12 , wherein the at least one pro-inflammatory cytokine comprises a cytokine of the Th17 pathway.

15. The method of claim 12 , wherein the at least one pro-inflammatory cytokine comprises an IL-17 cytokine selected from the group consisting of: IL-17A, IL-17B, IL-17C, IL-17D, IL-17E, and IL-17F.

16. The method of claim 12 , wherein the at least one pro-inflammatory cytokine comprises a cytokine selected from the group consisting of: IFN-γ, IL-1β, RANTES, MIP-1α, IL-8, and IL-6.

17. The method of claim 12 , wherein the condition mediated by the Th17 pathway is selected from the group consisting of: uveitis; a cancer; multiple sclerosis; an arthritis; neuromyelitis optica; psoriasis; systemic lupus erythematosus; an inflammatory bowel disease; celiac disease; an asthma; allergic asthma; neutrophilic asthma; chronic obstructive pulmonary disease (COPD); scleritis; vasculitis; Behcet's disease; atherosclerosis; atopic dermatitis; emphysema; periodontitis; allergic rhinitis; and allograft rejection.

18. The method of claim 17 , wherein the condition mediated by the Th17 pathway is an asthma; and wherein the treating comprises reducing neutrophilia or eosinophilia.

19. The method of claim 17 , wherein the condition mediated by the Th17 pathway is an arthritis selected from the group consisting of rheumatoid arthritis, osteoarthritis, psoriatic arthritis, spondyloarthritis, ankylosing spondylitis, and juvenile idiopathic arthritis; and wherein the method reduces joint swelling.

20. The method of claim 12 , wherein the bacteria strain comprises the polynucleotide sequence of SEQ ID NO:4.

21. The method of claim 12 , wherein the subject has the condition, or has been identified as being at risk of the condition.

22. The method of claim 12 , further comprising administering an additional therapeutic agent to the subject.

23. The method of claim 12 , wherein the administering of the pharmaceutical composition comprises oral, rectal, nasal, buccal, sublingual, intraperitoneal, or subcutaneous administration.

24. The method of claim 12 , wherein the administering comprises providing one or more doses of 1 g, 3 g, 5 g, or 10 g of the pharmaceutical composition.

25. The pharmaceutical composition of claim 1 , wherein the bacteria strain is non-spore forming.

26. The pharmaceutical composition of claim 1 , wherein the polynucleotide sequence of the 16S rRNA gene has at least 98% sequence identity to the polynucleotide sequence of SEQ ID NO:4, as determined by the Smith-Waterman homology search algorithm using the affine gap search with the gap open penalty of 12, the gap extension penalty of 2, and the BLOSUM of 62.

27. The method of claim 12 , wherein the polynucleotide sequence of the 16S rRNA gene has at least 98% sequence identity to the polynucleotide sequence of SEQ ID NO:4, as determined by the Smith-Waterman homology search algorithm using the affine gap search with the gap open penalty of 12, the gap extension penalty of 2, and the BLOSUM of 62.

28. The pharmaceutical composition of claim 1 , wherein the bacteria strain is strain 675 deposited under accession number NCIMB 42408.

29. The pharmaceutical composition of claim 1 , wherein the polynucleotide sequence of the 16S rRNA gene has at least 99% sequence identity to the polynucleotide sequence of SEQ ID NO:4, as determined by the Smith-Waterman homology search algorithm using the affine gap search with the gap open penalty of 12, the gap extension penalty of 2, and the BLOSUM of 62.

30. The pharmaceutical composition of claim 1 , wherein the bacteria strain is of the species Bacteroides coprocola.

31. The pharmaceutical composition of claim 1 , wherein the pharmaceutical composition is comprised in a capsule.

32. The method of claim 12 , wherein the polynucleotide sequence of the 16S rRNA gene has at least 99% sequence identity to the polynucleotide sequence of SEQ ID NO:4, as determined by the Smith-Waterman homology search algorithm using the affine gap search with the gap open penalty of 12, the gap extension penalty of 2, and the BLOSUM of 62.

33. The method of claim 12 , wherein the bacteria strain is of the species Bacteroides coprocola.

34. The method of claim 12 , wherein the bacteria strain is strain 675 deposited under accession number NCIMB 42408.

35. The method of claim 12 , wherein the pharmaceutical composition is comprised in a capsule.

36. The method of claim 12 , wherein the pharmaceutical composition comprises a lyoprotectant which is the pharmaceutically acceptable excipient, diluent, or carrier.

Assignments (7)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jun 14, 2023
From: 4D PHARMA PLC; 4D PHARMA RESEARCH LIMITED
To: CJ BIOSCIENCE, INC.
Reel/Frame 063992/0427 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 31, 2022
From: OXFORD FINANCE LUXEMBOURG S.A R.L.
To: ARMISTICE CAPITAL MASTER FUND LTD.
Reel/Frame 061806/0371 →
INTELECTUAL PROPERTY SECURITY AGREEMENT Recorded Jul 30, 2021
From: 4D PHARMA PLC; 4D PHARMA RESEARCH LIMITED; 4D PHARMA CORK LIMITED; 4D PHARMA DELAWARE INC.
To: OXFORD FINANCE LUXEMBOURG S.A R.L.
Reel/Frame 057042/0715 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 24, 2018
From: GRANT, GEORGE
To: 4D PHARMA RESEARCH LIMITED
Reel/Frame 044711/0304 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 24, 2018
From: MCCLUSKEY, SEANIN
To: 4D PHARMA RESEARCH LIMITED
Reel/Frame 044711/0429 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 24, 2018
From: MULDER, IMKE; RAFTIS, EMMA
To: 4D PHARMA RESEARCH LIMITED
Reel/Frame 044711/0611 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 24, 2018
From: PATTERSON, ANGELA M.
To: 4D PHARMA RESEARCH LIMITED
Reel/Frame 044711/0661 →
Priority Claims (3)
GB 1510470.6 · Jun 15, 2015 · national
GB 1520510.7 · Nov 20, 2015 · national
GB 1603786.3 · Mar 4, 2016 · national
Continuity (2)
Continuation PCTGB2016051768 · Jun 15, 2016
Related Publication 20170319634A1 · Nov 9, 2017
Cited By (1)
US 12,421,518