IP Library Granted Patent US 11,337,917
Granted Patent B2
US 11,337,917 · App. 15/634,924 · Granted May 24, 2022

Soft chewable pharmaceutical products

Inventors: Rainer Roepke (Schwabenheim, DE); Carsten Schmidt (Mainz, DE); Susi Alteheld (Bad Kreuznach, DE); Carina Hang (Grolsheim, DE)
Assignee: INTERVET INC.
A61K9/0056A61K9/145A61K9/1617A61K9/2013A61K9/282A61K9/4858A61K9/5015A61K9/5123A61K31/35A61K31/365A61K31/42A61K31/422A61K31/7048A61K45/06A61K47/10A61K47/12A61K47/16A61K47/18A61K47/20A61K47/22A61K47/26A61K47/36A61K47/38A61K47/42A61K47/44A61P33/00A61P33/14A61P43/00
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Quick Facts
Patent No.
US 11,337,917
App. No.
15/634,924
Granted
May 24, 2022
Kind
B2
Abstract

A soft chewable pharmaceutical product for delivery of a pharmaceutically acceptable active ingredient to an animal comprising pamoic acid or a pharmaceutically acceptable salt and a process for the manufacture of such soft chewable pharmaceutical product.

Claims (31)

1. A solid soft chewable veterinary composition effective for treating and/or controlling flea or tick infestation in an animal comprising:

a) an isoxazoline active ingredient of 4-[5-(3,5-Dichlorophenyl)-5-trifluoromethyl-4,5-dihydroisoxazol-3-yl]-2-methyl-N-[(2,2,2-trifluoro-ethylcarbamoyl) -methyl]-benzamide or a pharmaceutically acceptable salt thereof at a concentration between 5% and 20% by weight;

b) a forming agent, a surfactant, a filler and a humectant, wherein the forming agent is PEG 3350; the surfactant is sodium lauryl sulfate at a concentration of 2% (w/w); the filler is corn starch and the humectant is glycerol at a concentration of about 2.9% to 4% (w/w).;

c) wherein the effect is achieved at a dosage based upon the weight and type of animal; and

d) wherein the composition is effective for fleas or ticks by administration to the animal every 2 or 3 months.

2. The solid soft chewable veterinary composition of claim 1 , wherein the composition further comprises soybean oil.

3. The solid soft chewable veterinary composition of claim 1 , wherein the carrier further comprises a lubricant agent which is magnesium stearate.

4. The solid soft chewable veterinary composition of claim 1 , wherein the composition further comprises a flavoring which is pork or liver.

5. The solid soft chewable veterinary composition of claim 4 , wherein the flavoring is present in a concentration of about 10% to about 20% (w/w).

6. The solid soft chewable veterinary composition of claim 1 , wherein the filler is present in a concentration of about 10% to about 20% (w/w).

7. The solid soft chewable veterinary composition of claim 1 , wherein the forming agent is present at a concentration of about 1% to 40% (w/w).

8. The solid soft chewable veterinary composition of claim 1 , wherein the composition comprises a pharmaceutically acceptable salt of the isoxazoline active ingredient.

9. A solid soft chewable veterinary composition effective for treating and/or controlling flea or tick infestation in an animal comprising:

a) an isoxazoline active ingredient of 4[5-(3,5-Dichlorophenyl)-5-trifluoromethyl-4,5-dihydroisoxazol-3-yl]-2-methyl-N- [2,2,2-trifluoro-ethylcarbamoyl) -methyl]-benzamide or a pharmaceutically acceptable salt thereof at a concentration of about 9% to about 14% by weight;

b) a forming agent, a surfactant, a filler and a humectant, wherein the forming agent is PEG 3350; the surfactant is sodium lauryl sulfate at a concentration of 2% (w/w); the filler is corn starch and the humectant is glycerol at a concentration of about 2.9% to 4% (w/w);

c) wherein the effect is achieved at a dosage based upon the weight and type of animal; and

d) wherein the composition is effective for fleas or ticks by administration to the animal every 2 or 3 months.

10. A solid soft chewable veterinary composition effective for treating and/or controlling flea or tick infestation in an animal comprising:

a) an isoxazoline active ingredient of 4-[5-3,5 -Dichlorophenyl)-5-trifluoromethyl-4,5-dihydroisoxazol-3-yl]-2-methyl-N- [(2,2,2-trifluoro-ethylcarbamoyl) -methyl]-benzamide or a pharmaceutically acceptable salt thereof at a concentration from about 0.1% to 40% by weight;

b) a forming agent, a surfactant, a filler and a humectant, wherein the forming agent is PEG 3350; the surfactant is sodium lauryl sulfate at a concentration of 2% (w/w); the filler is corn starch and the humectant is glycerol at a concentration of about 2.9% to 4% (w/w);

c) wherein the effect is achieved at a dosage dependent upon the weight and type of animal; and

d) wherein the composition is effective for fleas or ticks by administration to the animal every 3 months.

11. The solid soft chewable veterinary composition of claim 1 , wherein the effect is about 100% against ticks about 48 hours after administration to the animal.

12. The solid soft chewable veterinary composition of claim 8 , wherein the effect is about 100% against ticks about 48 hours after administration to the animal.

13. The solid soft chewable veterinary composition of claim 9 , wherein the effect is about 100% against ticks about 48 hours after administration to the animal.

14. The solid soft chewable veterinary composition of claim 1 , wherein the effect is achieved at a dosage of about 8 mg/kg - 20 mg/kg of isoxazoline active ingredient.

15. The solid soft chewable veterinary composition of claim 8 , wherein the effect is achieved at a dosage of about 8 mg/kg - 20 mg/kg of isoxazoline active ingredient.

16. The solid soft chewable veterinary composition of claim 9 , wherein the effect is achieved at a dosage of about 8 mg/kg - 20 mg/kg of isoxazoline active ingredient.

17. The solid soft chewable veterinary composition of claim 1 , wherein the composition is effective against ticks for at least 58 days after administration to the animal.

18. The solid soft chewable veterinary composition of claim 8 , wherein the composition is effective against ticks for at least 58 days after administration to the animal.

19. The solid soft chewable veterinary composition of claim 9 , wherein the composition is effective against ticks for at least 58 days after administration to the animal.

Assignments (4)
CHANGE OF ADDRESS Recorded Sep 26, 2023
From: INTERVET INC.
To: INTERVET INC.
Reel/Frame 065028/0818 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Nov 28, 2017
From: ROEPKE, RAINER
To: INTERVET INC.
Reel/Frame 044237/0290 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Nov 28, 2017
From: SCHMIDT, CARSTEN
To: INTERVET INC.
Reel/Frame 044237/0460 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Nov 28, 2017
From: ALTEHELD, SUSI; HANG, CARINA
To: INTERVET INC.
Reel/Frame 044237/0779 →
Priority Claims (1)
EP 12163198 · Apr 4, 2012 · regional
Continuity (4)
Continuation 15390244 · Dec 23, 2016
Continuation 14390040
Provisional Application 61782434 · Mar 14, 2013
Related Publication 20170290766A1 · Oct 12, 2017
Cited By (3)
US 12,304,903 US 12,544,336 US 12,655,138