IP Library Granted Patent US 10,363,307
Granted Patent B2
US 10,363,307 · App. 15/654,854 · Granted Jul 30, 2019

Methods of treating psoriatic arthritis using IL-17 antagonists

Inventors: Shephard Mpofu (Oberwil, CH); Hanno Richards (Therwil, CH); Karthinathan Thangavelu (Geneva, CH); Matthias Machacek (Allschwil, CH)
Assignee: Novartis AG
A61K39/3955A61K31/519A61K45/06C07K16/244A61K2039/505A61K2039/545A61K2039/55C07K2317/21C07K2317/34C07K2317/76C07K2317/90
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Quick Facts
Patent No.
US 10,363,307
App. No.
15/654,854
Granted
Jul 30, 2019
Kind
B2
Abstract

The disclosure relates to novel regimens for treating an inflammatory arthritis, e.g., psoriatic arthritis, which employ a therapeutically effective amount of an IL-17 antagonist, e.g., IL-17 binding molecule (e.g., IL-17 antibody or antigen binding fragment thereof, e.g., secukinumab) or IL-17 receptor binding molecule (e.g., IL-17 antibody or antigen binding fragment thereof).

Claims (31)

1. A method of treating Psoriatic Arthritis (PsA), comprising:

a) subcutaneously administering to a patient having PsA five doses of about 150 mg-about 300 mg of an IL-17 antibody, each of the five doses being delivered weekly; and

b) thereafter, subcutaneously administering to the patient a dose of about 150 mg-about 300 mg of the IL-17 antibody every month, wherein the IL-17 antibody comprises:

i) an immunoglobulin V H domain comprising the amino acid sequence set forth as SEQ ID NO:8 and an immunoglobulin V L domain comprising the amino acid sequence set forth as SEQ ID NO:10;

ii) an immunoglobulin V H domain comprising the hypervariable regions comprising the amino acid sequences set forth as SEQ ID NOs:1-3, respectively, and an immunoglobulin V L domain comprising the hypervariable regions comprising the amino acid sequences set forth as SEQ ID NOs:4-6, respectively; or

iii) an immunoglobulin V H domain comprising the hypervariable regions comprising the amino acid sequences set forth as SEQ ID NOs:11-13, respectively, and an immunoglobulin V L domain comprising the hypervariable regions comprising the amino acid sequences set forth as SEQ ID NOs:4-6, respectively.

2. The method according to claim 1 , wherein the IL-17 antibody is secukinumab.

3. The method according to claim 1 , wherein, prior to treatment with the IL-17 antibody, the patient had an inadequate response to, had failure to, or was intolerant to treatment with a TNF alpha antagonist.

4. The method according to claim 1 , wherein the patient has co-existing moderate to severe plaque psoriasis.

5. The method according to claim 1 , further comprising administering a DMARD to the patient.

6. The method according to claim 5 , wherein the DMARD is methotrexate.

7. A method of treating PsA in a patient, comprising administering about 150 mg—about 300 mg of secukinumab by subcutaneous injection to the patient at weeks 0, 1, 2, 3 and 4, followed by about 150 mg—about 300 mg of secukinumab every 4 weeks.

8. The method according to claim 7 , wherein the patient has active PsA.

9. The method according to claim 7 , wherein, prior to treatment with secukinumab, the patient had an inadequate response to, had failure to, or was intolerant to treatment with a TNF alpha antagonist.

10. The method according to claim 7 , wherein the patient has co-existing moderate to severe plaque psoriasis.

11. The method according to claim 7 , further comprising administering a DMARD to the patient.

12. The method according to claim 11 , wherein the DMARD is methotrexate.

13. The method according to claim 7 , comprising administering about 300 mg of secukinumab by subcutaneous injection to the patient at weeks 0, 1, 2, 3 and 4, followed by 300 mg of secukinumab every 4 weeks.

14. The method according to claim 13 , wherein the patient has active PsA.

15. The method according to claim 13 , wherein, prior to treatment with secukinumab, the patient responded inadequately to treatment with at least one DMARD.

16. The method according to claim 13 , wherein, prior to treatment with secukinumab, the patient had an inadequate response to, had failure to, or was intolerant to treatment with a TNF alpha antagonist.

17. The method according to claim 13 , wherein the patient has co-existing moderate to severe plaque psoriasis.

18. The method according to claim 13 , further comprising administering a DMARD to the patient.

19. The method according to claim 18 , wherein the DMARD is methotrexate.

20. The method according to claim 7 , comprising administering about 150 mg of secukinumab by subcutaneous injection to the patient at weeks 0, 1, 2, 3 and 4, followed by 150 mg of secukinumab every 4 weeks.

21. The method according to claim 20 , wherein the patient has active PsA.

22. The method according to claim 20 , wherein, prior to treatment with secukinumab, the patient responded inadequately to treatment with at least one DMARD.

23. The method according to claim 20 , wherein, prior to treatment with secukinumab, the patient had an inadequate response to, had failure to, or was intolerant to treatment with a TNF alpha antagonist.

24. The method according to claim 20 , wherein the patient has co-existing moderate to severe plaque psoriasis.

25. The method according to claim 20 , further comprising administering a DMARD to the patient.

26. The method according to claim 25 , wherein the DMARD is methotrexate.

Assignments (3)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Dec 18, 2018
From: MACHACEK, MATTHIAS
To: NOVARTIS PHARMA AG
Reel/Frame 047802/0666 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Dec 18, 2018
From: MPOFU, SHEPHARD; RICHARDS, HANNO; THANGAVELU, KARTHINATHAN
To: NOVARTIS AG
Reel/Frame 047802/0777 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Dec 18, 2018
From: NOVARTIS PHARMA AG
To: NOVARTIS AG
Reel/Frame 047802/0828 →
Continuity (3)
Division 13877585
Provisional Application 61410533 · Nov 5, 2010
Related Publication 20180008706A1 · Jan 11, 2018