IP Library Granted Patent US 10,188,653
Granted Patent B2
US 10,188,653 · App. 15/693,785 · Granted Jan 29, 2019

Diacylglycerol acyltransferase 2 inhibitors

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Quick Facts
Patent No.
US 10,188,653
App. No.
15/693,785
Granted
Jan 29, 2019
Kind
B2
Abstract

Compounds of Formula I that inhibit the activity of the diacylglycerol acyltransferase 2 (DGAT2) and their uses in the treatment of diseases linked thereto in animals are described herein.

Claims (5)

1. A method for treating non-alcoholic fatty liver disease (NAFLD) in humans comprising the step of administering to a human in need of such treatment a therapeutically effective amount of a compound having the structure:

or a pharmaceutically acceptable salt thereof.

2. A method for treating non-alcoholic fatty liver disease (NAFLD), in humans comprising the step of administering to a human in need of such treatment a therapeutically effective amount of a compound comprising 3-((2-(3-(2-ethoxyphenoxy)piperidin-1-yl)pyrimidine-5-carboxamido)methyl)benzoic acid or (R)-3-((2-(3-(2-ethoxyphenoxy)piperidin-1-yl)pyrimidine-5-carboxamido)methyl)benzoic acid or a pharmaceutically acceptable salt thereof.

3. The method according to claim 1 wherein said compound or pharmaceutically acceptable salt thereof is in admixture with at least one pharmaceutically acceptable excipient.

4. The method according to claim 2 wherein said compound or pharmaceutically acceptable salt thereof is in admixture with at least one pharmaceutically acceptable excipient.

Assignments (1)
ASSIGNEE ADDRESS CORRECTION Recorded Mar 20, 2023
From: PFIZER INC.
To: PFIZER INC.
Reel/Frame 063119/0087 →