IP Library Granted Patent US 11,911,361
Granted Patent B2
US 11,911,361 · App. 15/712,515 · Granted Feb 27, 2024

Stable cannabinoid formulations

Inventors: Kiran Kumar Vangara (Phoenix, AZ); Huaguang Li (Chandler, AZ); Ningxin Yan (Chandler, AZ); Hung Q. Nguyen (Chandler, AZ); Venkat R. Goskonda (Phoenix, AZ)
Assignee: RADIUS PHARMACEUTICALS, INC.
A61K31/352A61K9/0095A61K9/08A61K31/05A61K31/355A61K31/365A61K47/10A61K47/14A61K47/22A61K47/26A61K47/44A61P25/08A61P25/28
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Quick Facts
Patent No.
US 11,911,361
App. No.
15/712,515
Granted
Feb 27, 2024
Kind
B2
Abstract

The present invention is generally directed to substantially pure cannabidiol, stable cannabinoid pharmaceutical formulations, and methods of their use.

Claims (25)

1. A method of treating Prader-Willi syndrome in a subject in need of such treatment, comprising administering to the subject an effective amount of an oral pharmaceutical formulation consisting of:

from about 8% to about 32% w/w cannabidiol;

caprylic/capric triglyceride at a concentration of 58 to 90% w/w;

alpha tocopherol at a concentration of from 0.01 to 1% w/w;

a sweetener at a concentration of 0.01 to 2% w/w; and

a flavoring agent at a concentration of 0.01 to about 1% w/w,

wherein w/w denotes weight by weight of the formulation, and wherein the effective amount results in administration of from about 20 to about 40 milligrams of cannabidiol per kilogram body weight of the subject per day, and wherein the subject is a human subject.

2. The method of claim 1 , wherein the method involves treating one or more symptoms of Prader-Willi syndrome.

3. The method of claim 2 , wherein the one or more symptoms of Prader-Willi syndrome is hyperphagia.

4. The method of claim 1 , wherein the human subject is a pediatric subject.

5. The method of claim 1 , wherein the dose of the cannabidiol is about 40 milligrams of cannabidiol per kilogram body weight of the subject per day.

6. The method of claim 1 , wherein the cannabidiol is greater than 98% pure.

7. The method of claim 1 , wherein the cannabidiol is synthetic cannabidiol.

8. The method of claim 1 , wherein the oral pharmaceutical formulation consists of:

10.53% w/w of cannabidiol;

88.945% w/w of caprylic/capric triglyceride;

0.2% w/w of alpha tocopherol;

0.025% w/w of sweetener; and

0.3% w/w of flavoring agent.

9. The method of claim 1 , wherein the oral pharmaceutical formulation consists of:

31.09% w/w of cannabidiol;

68.385% w/w of caprylic/capric triglyceride;

0.2% w/w of alpha tocopherol;

0.025% w/w of sweetener; and

0.3% w/w of flavoring agent.

Assignments (16)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Sep 10, 2024
From: RADIUS PHARMACEUTICALS, INC.
To: FRESH CUT DEVELOPMENT, LLC
Reel/Frame 068543/0020 →
RELEASE OF SECURITY INTEREST Recorded Jul 23, 2024
From: WILMINGTON TRUST, NATIONAL ASSOCIATION
To: RADIUS HEALTH, INC.
Reel/Frame 068051/0671 →
SECURITY INTEREST Recorded Aug 16, 2022
From: RADIUS HEALTH, INC.
To: WILMINGTON TRUST, NATIONAL ASSOCIATION
Reel/Frame 061179/0001 →
RELEASE OF SECURITY INTEREST Recorded Aug 15, 2022
From: MIDCAP FUNDING IV TRUST
To: RADIUS HEALTH, INC.; RADIUS PHARMACEUTICALS, INC.
Reel/Frame 061176/0914 →
RELEASE OF SECURITY INTEREST Recorded Aug 15, 2022
From: MIDCAP FINANCIAL TRUST
To: RADIUS HEALTH, INC.; RADIUS PHARMACEUTICALS, INC.
Reel/Frame 061176/0938 →
CHANGE OF ADDRESS Recorded Jun 23, 2021
From: RADIUS PHARMACEUTICALS, INC.
To: RADIUS PHARMACEUTICALS, INC.
Reel/Frame 056650/0050 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded May 18, 2021
From: VANGARA, KIRAN KUMAR; LI, HUAGUANG; YAN, NINGXIN; NGUYEN, HUNG Q.; GOSKONDA, VENKAT R.
To: INSYS DEVELOPMENT COMPANY, INC.
Reel/Frame 056270/0534 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 20, 2021
From: FRESH CUT DEVELOPMENT, LLC
To: RADIUS PHARMACEUTICALS, INC.
Reel/Frame 055979/0946 →
SECURITY AGREEMENT SUPPLEMENT (REVOLVING) Recorded Mar 17, 2021
From: RADIUS HEALTH, INC.; RADIUS PHARMACEUTICALS, INC.
To: MIDCAP FUNDING IV TRUST, AS AGENT
Reel/Frame 055632/0634 →
REAFFIRMATION, JOINDER & AMENDMENT TO SECURITY AGREEMENT (TERM) Recorded Mar 17, 2021
From: RADIUS HEALTH, INC.; RADIUS PHARMACEUTICALS, INC.; RADIUS HEALTH VENTURES, INC.
To: MIDCAP FINANCIAL TRUST, AS AGENT
Reel/Frame 055632/0017 →
REAFFIRMATION, JOINDER & AMENDMENT TO SECURITY AGREEMENT (REVOLVING) Recorded Mar 17, 2021
From: RADIUS HEALTH, INC.; RADIUS PHARMACEUTICALS, INC.; RADIUS HEALTH VENTURES, INC.
To: MIDCAP FUNDING IV TRUST, AS AGENT
Reel/Frame 055632/0316 →
SECURITY AGREEMENT SUPPLEMENT (TERM) Recorded Mar 17, 2021
From: RADIUS HEALTH, INC.; RADIUS PHARMACEUTICALS, INC.
To: MIDCAP FINANCIAL TRUST, AS AGENT
Reel/Frame 055632/0653 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Dec 19, 2019
From: BENUVIA THERAPEUTICS INC.
To: FRESH CUT DEVELOPMENT, LLC
Reel/Frame 051381/0283 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Dec 2, 2019
From: INSYS THERAPEUTICS, INC; INSYS PHARMA, INC.; INSYS DEVELOPMENT COMPANY, INC.
To: FRESH CUT DEVELOPMENT, LLC
Reel/Frame 051151/0685 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Dec 2, 2019
From: FRESH CUT DEVELOPMENT, LLC
To: BENUVIA THERAPEUTICS INC.
Reel/Frame 051151/0852 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Sep 6, 2019
From: VANGARA, KIRAN KUMAR; YAN, NINGXIN; NGUYEN, HUNG Q.; GOSKONDA, VENKAT R.
To: INSYS DEVELOPMENT COMPANY, INC.
Reel/Frame 050297/0201 →
Continuity (8)
Continuation In Part 15499178 · Apr 27, 2017
Continuation In Part 15253010 · Aug 31, 2016
Continuation In Part 15166476 · May 27, 2016
Continuation In Part 14815936 · Jul 31, 2015
Continuation In Part 14724351 · May 28, 2015
Provisional Application 62154660 · Apr 29, 2015
Provisional Application 62004495 · May 29, 2014
Related Publication 20180028489A1 · Feb 1, 2018