IP Library Granted Patent US 11,065,277
Granted Patent B2
US 11,065,277 · App. 15/774,763 · Granted Jul 20, 2021

Method of ameliorating side effects of sickle cell disease treatments

Inventors: Craig Branch (Cornwall, NY); Seetharama Acharya (Cresskill, NJ)
Assignee: Albert Einstein College of Medicine
A61K35/14A61K9/0053A61K31/17A61K31/192A61K31/341A61K31/352A61K31/353A61K31/437A61K31/7048A61K38/38A61K38/42A61K45/06A61K47/60A61P7/00
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Quick Facts
Patent No.
US 11,065,277
App. No.
15/774,763
Granted
Jul 20, 2021
Kind
B2
Abstract

A method of reducing a cerebral tissue pathology associated with a sickle cell disease therapy in a subject is provided using (i) a synthetic high-oxygen affinity hemoglobin-containing molecule or (ii) synthetically treated high-oxygen affinity blood.

Claims (13)

1. A method of reducing cell sickling and preventing a cerebral tissue pathology in a subject having a sickle cell disease with vaso-occlusion comprising:

administering a 10% top-load of a pegylated hemoglobin (PEG-Hb) molecule having a higher oxygen affinity than hemoglobin in red blood cells to the subject, wherein the PEG-Hb molecule reduces cell sickling and is sufficient to protect against a cerebral tissue pathology caused by a reduced cerebral blood flow (CBF) that results from administering the 10% top-load to treat the sickle cell disease with vaso-occlusion in the subject; and

administering an amount of 5-hydroxyl methyl furfural or a composition comprising red blood cells ex vivo treated with 5-hydroxyl methyl furfural to the subject.

2. The method of claim 1 , wherein the cerebral tissue pathology is cerebral hypoxic insult.

3. The method of claim 1 , wherein the PEG-Hb molecule comprises a hemoglobin molecule having 6 molecules of 3,000 mw polyethylene glycol (PEG) attached thereto (P3K6 Hb).

4. The method of claim 3 , wherein the P3K6 Hb is extension arm facilitated P3K6 Hb (EAF P3K6 Hb).

5. The method of claim 3 , wherein the P3K6 Hb is an antioxidant adduct of EAF P3K6 Hb.

6. The method of claim 5 , wherein the antioxidant is a flavonoid.

7. The method of claim 1 , further comprising administering a pegylated albumin (PEG-Alb) molecule.

8. The method of claim 1 , further comprising administering an amount of a quercetin to the subject.

9. The method of claim 5 , further comprising orally administering an amount of hydroxyl urea to the subject.

10. A method of reducing cell sickling and preventing a cerebral tissue pathology in a subject having a sickle cell disease with vaso-occlusion comprising:

administering a 10% top-load of an EAF P3K6-Hb molecule to the subject, wherein the PEG-Hb molecule reduces cell sickling and is sufficient to protect against a cerebral tissue pathology caused by a reduced cerebral blood flow (CBF) that results from administering the 10% top-load to treat the sickle cell disease with vaso-occlusion in the subject.

Assignments (3)
MERGER AND CHANGE OF NAME Recorded Aug 21, 2019
From: ALBERT EINSTEIN COLLEGE OF MEDICINE, INC.; ALBERT EINSTEIN COLLEGE OF MEDICINE
To: ALBERT EINSTEIN COLLEGE OF MEDICINE
Reel/Frame 050130/0432 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Aug 15, 2019
From: BRANCH, CRAIG; ACHARYA, SEETHARAMA
To: ALBERT EINSTEIN COLLEGE OF MEDICINE, INC.
Reel/Frame 050068/0659 →
MERGER AND CHANGE OF NAME Recorded Feb 26, 2019
From: ALBERT EINSTEIN COLLEGE OF MEDICINE, INC.; ALBERT EINSTEIN COLLEGE OF MEDICINE
To: ALBERT EINSTEIN COLLEGE OF MEDICINE
Reel/Frame 048438/0275 →