IP Library Granted Patent US 10,973,796
Granted Patent B2
US 10,973,796 · App. 15/791,885 · Granted Apr 13, 2021

Compositions and methods for lowering levels of high-sensitivity C-reactive protein (hs-CRP) in a subject

Inventors: Mehar Manku (Birmingham, GB); Ian Osterloh (Kent, GB); Pierre Wicker (Mystic, CT); Rene Braeckman (Richboro, PA); Paresh Soni (Mystic, CT)
Assignee: Amarin Pharmaceuticals Ireland Limited
A61K31/232A61K9/48A61K9/4866A61K31/202A61K31/366A61K31/40A61K31/505
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Quick Facts
Patent No.
US 10,973,796
App. No.
15/791,885
Granted
Apr 13, 2021
Kind
B2
Abstract

The present disclosure provides methods for treating and/or preventing cardiovascular-related disease and, in particular, a method of blood lipid therapy comprising administering to a subject in need thereof a pharmaceutical composition comprising eicosapentaenoic acid or a derivative thereof. In some embodiments, the method comprises lowering high sensitivity CRP (hs-CRP) levels in a subject including, for example, a subject with a HbA 1c value of about 5.00%-8.50% or at least about 6.8%.

Claims (7)

1. A method of reducing a high sensitivity C-reactive protein (hsCRP) level in a diabetic subject in need thereof, the method comprising: (a) identifying the diabetic subject having a fasting baseline triglyceride level of about 200 mg/dl to about 1500 mg/dl and an hsCRP level of about 0.1 mg/L to about 10 mg/L, and (b) administering to the diabetic subject about 2 g to about 4 g per day of a pharmaceutical composition comprising at least about 90%, by weight of all fatty acids present, ethyl eicosapentaenoate, for a period effective to reduce the hsCRP level in the diabetic subject.

2. The method of claim 1 wherein the composition is administered to the diabetic subject 1 to 4 times per day.

3. The method of claim 1 wherein the composition is present in a capsule.

4. The method of claim 1 wherein the diabetic subject is not on concomitant lipid-altering therapy.

5. The method of claim 1 further comprising a step of measuring a baseline lipid profile in the diabetic subject prior to administering the pharmaceutical composition to said diabetic subject.

6. The method of claim 1 , wherein the period is about 12 weeks and is effective to: (a) reduce triglyceride levels compared to baseline; (b) reduce ICAM-1 level compared to baseline; (c) reduce ox-LDL level compared to baseline; (d) reduce IL-6 level compared to baseline; and/or (e) reduce hsCRP level compared to baseline.

7. The method of claim 1 wherein the diabetic subject exhibits one or more of: (a) a placebo-adjusted reduction in triglyceride level of at least about 5% as compared to baseline; (b) a placebo-adjusted increase in ICAM-1 level of less than 10% or a placebo-adjusted reduction in ICAM-1 level of at least about 1% as compared to baseline; (c) a placebo-adjusted increase in ox-LDL level of less than 10% or a placebo-adjusted reduction in ox-LDL level of at least about 1% as compared to baseline; (d) a placebo-adjusted increase in Lp-PLA 2 level of less than 10% or a placebo-adjusted reduction in Lp-PLA 2 level of at least 1% as compared to baseline; (e) a placebo-adjusted increase in IL-6 level of less than 15% or a placebo-adjusted reduction in IL-6 level of at least 1% as compared to baseline; and/or (f) a placebo-adjusted reduction in hsCRP level of at least 5% as compared to baseline.

Assignments (4)
RELEASE OF SECURITY INTEREST Recorded Nov 19, 2020
From: CPPIB CREDIT EUROPE S.À R.L.
To: AMARIN PHARMACEUTICALS IRELAND LIMITED
Reel/Frame 054484/0552 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 25, 2018
From: MANKU, MEHAR; OSTERLOH, IAN; WICKER, PIERRE; BRAECKMAN, RENE; SONI, PARESH
To: AMARIN PHARMACEUTICALS IRELAND LIMITED
Reel/Frame 045141/0898 →
SECURITY INTEREST Recorded Dec 21, 2017
From: AMARIN PHARMACEUTICALS IRELAND LIMITED
To: CPPIB CREDIT EUROPE S.À R.L.
Reel/Frame 044938/0257 →
PATENT SECURITY ASSIGNMENT AND ASSUMPTION AGREEMENT Recorded Dec 20, 2017
From: BIOPHARMA SECURED DEBT FUND II HOLDINGS CAYMAN LP
To: CPPIB CREDIT EUROPE S.À R.L.
Reel/Frame 044956/0395 →
Continuity (5)
Division 13735660 · Jan 7, 2013
Provisional Application 61670408 · Jul 11, 2012
Provisional Application 61656347 · Jun 6, 2012
Provisional Application 61584013 · Jan 6, 2012
Related Publication 20180042883A1 · Feb 15, 2018