IP Library Granted Patent US 10,711,060
Granted Patent B2
US 10,711,060 · App. 15/829,284 · Granted Jul 14, 2020

Antibody molecules to LAG-3 and uses thereof

Inventors: Frédéric Triebel (Versailles, FR); Chrystelle Brignone (Chatenay-Malabry, FR); Walter A. Blattler (Brookline, MA); Jennifer Marie Mataraza (Cambridge, MA); Catherine Anne Sabatos-Peyton (Cambridge, MA); Hwai Wen Chang (Cambridge, MA); Gerhard Johann Frey (San Diego, CA)
Assignees: NOVARTIS AG; Immutep S.A.S.
C07K16/2803A61K39/39558A61K45/06C07K2317/24C07K2317/51C07K2317/515C07K2317/56C07K2317/565C07K2317/70C07K2317/76G01N2333/70596
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Quick Facts
Patent No.
US 10,711,060
App. No.
15/829,284
Granted
Jul 14, 2020
Kind
B2
Abstract

Antibody molecules that specifically bind to LAG-3 are disclosed. The anti-LAG-3 antibody molecules can be used to treat, prevent and/or diagnose cancerous or infectious disorders.

Claims (9)

1. An isolated nucleic acid molecule comprising a first nucleotide sequence that encodes a VH and a second nucleotide sequence that encodes a VL of an antibody molecule that binds to human LAG-3, wherein the antibody molecule comprises:

(a) a heavy chain variable region (VH) comprising a VHCDR1 amino acid sequence of SEQ ID NO: 4, a VHCDR2 amino acid sequence of SEQ ID NO: 5, and a VHCDR3 amino acid sequence of SEQ ID NO: 3; and a light chain variable region (VL) comprising a VLCDR1 amino acid sequence of SEQ ID NO: 13, a VLCDR2 amino acid sequence of SEQ ID NO: 14, and a VLCDR3 amino acid sequence of SEQ ID NO: 15;

(b) a VH comprising a VHCDR1 amino acid sequence of SEQ ID NO: 1; a VHCDR2 amino acid sequence of SEQ ID NO: 2; and a VHCDR3 amino acid sequence of SEQ ID NO: 3; and a VL comprising a VLCDR1 amino acid sequence of SEQ ID NO: 10, a VLCDR2 amino acid sequence of SEQ ID NO: 11, and a VLCDR3 amino acid sequence of SEQ ID NO: 12;

(c) a VH comprising a VHCDR1 amino acid sequence of SEQ ID NO: 286, a VHCDR2 amino acid sequence of SEQ ID NO: 5, and a VHCDR3 amino acid sequence of SEQ ID NO: 3; and a VL comprising a VLCDR1 amino acid sequence of SEQ ID NO: 13, a VLCDR2 amino acid sequence of SEQ ID NO: 14, and a VLCDR3 amino acid sequence of SEQ ID NO: 15; or

(d) a VH comprising a VHCDR1 amino acid sequence of SEQ ID NO: 286; a VHCDR2 amino acid sequence of SEQ ID NO: 2; and a VHCDR3 amino acid sequence of SEQ ID NO: 3; and a VL comprising a VLCDR1 amino acid sequence of SEQ ID NO: 10, a VLCDR2 amino acid sequence of SEQ ID NO: 11, and a VLCDR3 amino acid sequence of SEQ ID NO: 12.

2. An expression vector comprising the nucleic acid molecule of claim 1 .

3. An isolated host cell comprising the nucleic acid molecule of claim 1 .

4. A method of producing an antibody molecule, comprising culturing the host cell of claim 3 under conditions suitable for gene expression, wherein upon gene expression the antibody molecule is produced.

5. The method of claim 4 , further comprising isolating the antibody molecule.

Assignments (6)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded May 3, 2018
From: TRIEBEL, FRÉDÉRIC; BRIGNONE, CHRYSTELLE
To: IMMUTEP S.A.
Reel/Frame 045703/0723 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded May 3, 2018
From: CHANG, HWAI WEN; FREY, GERHARD JOHANN
To: BIOATLA, LLC
Reel/Frame 045703/0750 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded May 3, 2018
From: BLATTLER, WALTER A.; MATARAZA, JENNIFER MARIE; SABATOS-PEYTON, CATHERINE ANNE
To: COSTIM PHARMACEUTICALS INC.
Reel/Frame 045703/0784 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded May 3, 2018
From: BIOATLA, LLC
To: COSTIM PHARMACEUTICALS INC.
Reel/Frame 045703/0797 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded May 3, 2018
From: COSTIM PHARMACEUTICALS INC.
To: NOVARTIS AG
Reel/Frame 045703/0805 →
CHANGE OF NAME Recorded May 3, 2018
From: IMMUTEP S.A.
To: IMMUTEP S.A.S.
Reel/Frame 046061/0526 →
Continuity (5)
Division 14657260 · Mar 13, 2015
Provisional Application 62094889 · Dec 19, 2014
Provisional Application 62059690 · Oct 3, 2014
Provisional Application 61953536 · Mar 14, 2014
Related Publication 20180086830A1 · Mar 29, 2018
Cited By (4)
US 12,252,535 US 12,582,713 US 12,600,777 US 12,630,633