IP Library Granted Patent US 10,858,339
Granted Patent B2
US 10,858,339 · App. 15/941,993 · Granted Dec 8, 2020

Aryl cyclopropyl-amino-isoquinolinyl amide compounds

Inventors: Mitchell A. deLong (Chapel Hill, NC); Jill M. Sturdivant (Chapel Hill, NC); Cynthia L. Lichorowic (Raleigh, NC); Andriy Kornilov (Ypsilanti, MI)
Assignee: Aerie Pharmaceuticals, Inc.
C07D401/12A61P27/06C07C69/76C07D217/02C07D217/22C07D217/24C07D401/04C07D401/14C07D405/12C07D405/14C07D409/12C07D417/12C07C2601/02
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Quick Facts
Patent No.
US 10,858,339
App. No.
15/941,993
Granted
Dec 8, 2020
Kind
B2
Abstract

Provided herein are arylcyclopropyl amino-isoquinoline amide compounds. In particular, the disclosure provides compounds that affect the function of kinases in a cell and that are useful as therapeutic agents or with therapeutic agents. The compounds of the disclosure are useful in the treatment of a variety of diseases and conditions including eye diseases such as glaucoma, cardiovascular diseases, diseases characterized by abnormal growth, such as cancers, and inflammatory diseases. The disclosure further provides compositions containing isoquinoline amide compounds.

Claims (4)

1. A compound, wherein the compound is:

or a pharmaceutically acceptable salt thereof.

2. A composition, comprising the compound of claim 1 .

3. A pharmaceutical composition, comprising the compound of claim 1 and a pharmaceutically acceptable carrier.

Assignments (5)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jun 24, 2024
From: AERIE PHARMACEUTICALS, INC.
To: ALCON INC.
Reel/Frame 067822/0168 →
RELEASE OF SECURITY INTEREST Recorded Sep 5, 2019
From: DEERFIELD PRIVATE DESIGN FUND III, L.P.
To: AERIE PHARMACEUTICALS, INC.
Reel/Frame 050276/0807 →
SECURITY INTEREST Recorded Jul 23, 2018
From: AERIE PHARMACEUTICALS, INC.
To: DEERFIELD PRIVATE DESIGN FUND III, L.P.
Reel/Frame 046432/0307 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 30, 2018
From: DELONG, MITCHELL A.; STURDIVANT, JILL M.; LICHOROWIC, CYNTHIA L.
To: AERIE PHARMACEUTICALS, INC.
Reel/Frame 045401/0393 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 30, 2018
From: DELONG, MITCHELL A.; STURDIVANT, JILL M.; LICHOROWIC, CYNTHIA L.; KORNILOV, ANDRIY
To: AERIE PHARMACEUTICALS, INC.
Reel/Frame 045401/0511 →
Continuity (3)
Provisional Application 62643131 · Mar 14, 2018
Provisional Application 62480239 · Mar 31, 2017
Related Publication 20180327381A1 · Nov 15, 2018
Cited By (1)
US 12,458,620