IP Library Granted Patent US 10,851,171
Granted Patent B2
US 10,851,171 · App. 15/945,554 · Granted Dec 1, 2020

Method for the selection of antibodies against BCMA

Inventors: Minh Diem Vu (Wollerau, CH); Klaus Strein (Weinheim, DE); Ekkehard Moessner (Kreuzlingen, CH); Ralf Hosse (Cham, CH); Oliver Ast (Bassersdorf, CH); Anne Freimoser-Grundschober (Zurich, CH); Marina Bacac (Zurich, CH); Tanja Fauti (Zurich, CH); Christian Klein (Bonstetten, CH); Pablo Umana (Wollerau, CH); Samuel Moser (Rotkreuz, CH)
Assignee: ENGMAB SARL
C07K16/2878A61K39/395A61K39/3955C07K16/3061G01N33/6863A61K2039/505C07K16/28C07K16/2809C07K16/2863C07K2317/31C07K2317/33C07K2317/56C07K2317/565C07K2317/66C07K2317/71C07K2317/732C07K2317/76C07K2317/92C12N5/06C12N15/63G01N2333/7151G01N2500/04
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Quick Facts
Patent No.
US 10,851,171
App. No.
15/945,554
Granted
Dec 1, 2020
Kind
B2
Abstract

An antibody specifically binding to human BCMA, characterized in that the binding of said antibody is not reduced by APRIL and not reduced by BAFF, said antibody does not alter APRIL-dependent NF-κB activation, BAFF-dependent NF-κB activation, and does not alter NF-κB activation without BAFF and APRIL is useful as a therapeutic agent.

Claims (4)

1. A bispecific antibody specifically binding to human B cell maturation factor (BCMA) and CD3, comprising variable heavy and light chains of anti-CD3ε antibody SP34, wherein said bispecific antibody further comprises variable heavy and light chains of an antibody specifically binding to BCMA wherein variable domain VH comprises a CDR1H of SEQ ID NO:39, a CDR2H of SEQ ID NO:49 and a CDR3H of SEQ ID NO:59 and variable domain VL comprises a CDR1L of SEQ ID NO:69, a CDR2L of SEQ ID NO:79 and a CDR3L of SEQ ID NO:89.

2. A bispecific antibody according to claim 1 wherein the bispecific antibody binds BCMA extracellular domain with a dissociation constant (Kd) of 10 −8 M or less.

3. A bispecific antibody according to claim 1 wherein the bispecific antibody binds specifically to cynomolgus BCMA.

4. A pharmaceutical composition comprising an antibody according to claim 1 and a pharmaceutically acceptable excipient.

Assignments (13)
NUNC PRO TUNC ASSIGNMENT Recorded Apr 17, 2023
From: ENGMAB BETA HOLDINGS LLC
To: BRISTOL-MYERS SQUIBB COMPANY
Reel/Frame 063353/0610 →
NUNC PRO TUNC ASSIGNMENT Recorded Apr 17, 2023
From: ENGMAB SÀRL
To: ENGMAB BETA HOLDINGS LLC
Reel/Frame 063353/0350 →
CHANGE OF NAME Recorded Mar 29, 2021
From: ENGMAB AG
To: ENGMAB SÀRL
Reel/Frame 055747/0027 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 26, 2021
From: ROCHE GLYCART AG
To: F. HOFFMANN-LA ROCHE AG
Reel/Frame 055731/0228 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 26, 2021
From: F. HOFFMANN-LA ROCHE AG
To: ENGMAB AG
Reel/Frame 055731/0551 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 26, 2021
From: VU, MINH DIEM; STREIN, KLAUS
To: ENGMAB AG
Reel/Frame 055728/0025 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 26, 2021
From: MOESSNER, EKKEHARD; HOSSE, RALF; AST, OLIVER; FREIMOSER-GRUNDSCHOBER, ANNE; BACAC, MARINA; FAUTI, TANJA; KLEIN, CHRISTIAN; UMANA, PABLO; MOSER, SAMUEL
To: ROCHE GLYCART AG
Reel/Frame 055728/0454 →
CHANGE OF NAME Recorded Oct 22, 2020
From: ENGMAB AG
To: ENGMAB SÀRL
Reel/Frame 054137/0728 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded May 16, 2019
From: VU, MINH DIEM; STREIN, KLAUS
To: ENGMAB AG
Reel/Frame 049204/0608 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded May 16, 2019
From: AST, OLIVER; FAUTI, TANJA; FREIMOSER-GRUNDSCHOBER, ANNE; HOSSE, RALF; KLEIN, CHRISTIAN; MOESSNER, EKKEHARD; MOSER, SAMUEL; MURR, RAMONA; UMANA, PABLO
To: ROCHE GLYART AG
Reel/Frame 049204/0667 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded May 16, 2019
From: JUNG-IMHOF, SABINE; KLOSTERMANN, STEFAN; MOLHOJ, MICHAEL; REGULA, JOERG THOMAS; SCHAEFER, WOLFGANG
To: ROCHE DIAGNOSTICS GMBH
Reel/Frame 049204/0685 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded May 16, 2019
From: ROCHE GLYCART AG
To: F. HOFFMANN-LA ROCHE AG
Reel/Frame 049204/0710 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded May 16, 2019
From: F. HOFFMANN-LA ROCHE AG
To: ENGMAB AG
Reel/Frame 049204/0734 →
Priority Claims (2)
EP 13000570 · Feb 5, 2013 · regional
EP 13000571 · Feb 5, 2013 · regional
Continuity (2)
Division 14764967
Related Publication 20180222991A1 · Aug 9, 2018
Cited By (1)
US 12,637,522