IP Library Granted Patent US 10,383,864
Granted Patent B2
US 10,383,864 · App. 15/974,217 · Granted Aug 20, 2019

Methods for treatment of Fabry disease

Inventors: David J. Lockhart (Emerald Hills, CA); Jeff Castelli (New Hope, PA)
Assignee: Amicus Therapeutics, Inc.
A61K31/445A61K9/0053A61K9/48A61K31/45A61K45/06C07D211/46G01N33/5094G01N2333/924G01N2333/94G01N2800/04G01N2800/52
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Quick Facts
Patent No.
US 10,383,864
App. No.
15/974,217
Granted
Aug 20, 2019
Kind
B2
Abstract

Provided are in vitro and in vivo methods for determining whether a patient with Fabry disease will respond to treatment with a specific pharmacological chaperone.

Claims (20)

1. A method for treatment of Fabry disease in a human patient in need thereof, the method comprising administering to the patient about 50 to about 250 mg of 1-deoxygalactonojirimycin or a salt thereof every other day.

2. The method of claim 1 , wherein the 1-deoxygalactonojirimycin or salt thereof is administered as an oral dosage form.

3. The method of claim 2 , wherein the oral dosage form comprises a tablet, a capsule or a solution.

4. The method of claim 1 , wherein the patient does not eat food from about 2 hours before to about 2 hours after administering the 1-deoxygalactonojirimycin or salt thereof.

5. The method of claim 1 , wherein the 1-deoxygalactonojirimycin or salt thereof enhances α-galactosidase A activity.

6. The method of claim 1 , wherein the patient is male.

7. The method of claim 1 , wherein the patient is female.

8. The method of claim 1 , wherein the patient is administered about 50 to about 150 mg of the 1-deoxygalactonojirimycin or salt thereof every other day.

9. The method of claim 1 , wherein the patient is administered about 150 to about 250 mg of the 1-deoxygalactonojirimycin or salt thereof every other day.

10. A method for treatment of Fabry disease in a human patient in need thereof, the method comprising administering to the patient about 50 to about 250 mg of migalastat hydrochloride every other day.

11. The method of claim 10 , wherein the migalastat hydrochloride is administered as an oral dosage form.

12. The method of claim 11 , wherein the oral dosage form comprises a tablet, a capsule or a solution.

13. The method of claim 10 , wherein the patient does not eat food from about 2 hours before to about 2 hours after administering the migalastat hydrochloride.

14. The method of claim 10 , wherein the migalastat hydrochloride enhances α-galactosidase A activity.

15. The method of claim 10 , wherein the patient is male.

16. The method of claim 10 , wherein the patient is female.

17. The method of claim 10 , wherein the patient is administered about 50 to about 150 mg of the migalastat hydrochloride every other day.

18. The method of claim 10 , wherein the patient is administered about 150 to about 250 mg of migalastat hydrochloride every other day.

19. A method for treatment of Fabry disease in a human patient in need thereof, the method comprising administering to the patient a therapeutically effective dose of 1-deoxygalactonojirimycin or a salt thereof every other day, wherein the patient does not eat food from about 2 hours before to about 2 hours after administering the 1-deoxygalactonojirimycin or salt thereof.

20. The method of claim 19 , wherein the patient is administered about 150 mg of the 1-deoxygalactonojirimycin or salt thereof every other day.

Assignments (10)
SECURITY INTEREST Recorded Apr 27, 2026
From: BIOMARIN PHARMACEUTICAL INC.; AMICUS THERAPEUTICS, INC.
To: CITIBANK, N.A., AS COLLATERAL AGENT
Reel/Frame 075493/0968 →
RELEASE OF SECURITY INTEREST Recorded Apr 27, 2026
From: WILMINGTON TRUST, NATIONAL ASSOCIATION
To: AMICUS THERAPEUTICS, INC.
Reel/Frame 075494/0030 →
SECURITY INTEREST Recorded Oct 6, 2023
From: AMICUS THERAPEUTICS, INC.
To: WILMINGTON TRUST, NATIONAL ASSOCIATION
Reel/Frame 065177/0196 →
RELEASE OF SECURITY INTEREST Recorded Oct 6, 2023
From: HAYFIN SERVICES LLP
To: AMICUS THERAPEUTICS, INC.
Reel/Frame 065164/0945 →
SECURITY INTEREST Recorded Jul 30, 2020
From: AMICUS THERAPEUTICS, INC.
To: HAYFIN SERVICES LLP, AS AGENT
Reel/Frame 053365/0342 →
RELEASE OF SECURITY INTEREST Recorded Jul 30, 2020
From: BPCR LIMITED PARTNERSHIP
To: AMICUS THERAPEUTICS, INC.
Reel/Frame 053360/0659 →
OMNIBUS CONFIRMATION OF ASSIGNMENT AGREEMENT Recorded May 21, 2020
From: BIOPHARMA CREDIT PLC
To: BPCR LIMITED PARTNERSHIP
Reel/Frame 052741/0173 →
SECURITY INTEREST Recorded May 11, 2020
From: AMICUS THERAPEUTICS, INC.
To: BIOPHARMA CREDIT PLC
Reel/Frame 052625/0916 →
SECURITY INTEREST Recorded Sep 28, 2018
From: AMICUS THERAPEUTICS, INC.
To: BIOPHARMA CREDIT PLC
Reel/Frame 047004/0208 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Sep 6, 2018
From: LOCKHART, DAVID J.; CASTELLI, JEFF
To: AMICUS THERAPEUTICS, INC.
Reel/Frame 046799/0464 →
Continuity (8)
Continuation 15338923 · Oct 31, 2016
Continuation 14641707 · Mar 9, 2015
Continuation 13445338 · Apr 12, 2012
Continuation 12966904 · Dec 13, 2010
Division 11749512 · May 16, 2007
Provisional Application 60853631 · Oct 23, 2006
Provisional Application 60801089 · May 16, 2006
Related Publication 20180325881A1 · Nov 15, 2018
Cited By (2)
US 12,280,042 US 12,594,268