IP Library Granted Patent US 10,675,255
Granted Patent B2
US 10,675,255 · App. 16/017,303 · Granted Jun 9, 2020

Sphingosine pathway modulating compounds for the treatment of cancers

Inventors: Elazar Rabbani (New York, NY); James J. Donegan (Long Beach, NY)
Assignee: Enzo Bochem, Inc.
A61K31/137A61K31/135A61K31/4245A61K45/06A61P35/00A61P35/02A61K2300/00
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Quick Facts
Patent No.
US 10,675,255
App. No.
16/017,303
Granted
Jun 9, 2020
Kind
B2
Abstract

The invention provides methods and compositions for treating cancers and myeloproliferative disorders using sphingosine kinase-1 inhibitors, such as SK1-I, and selective sphingosine-1-phosphate receptor agonists, such as ozanimod.

Claims (15)

1. A method for treating hepatocellular carcinoma (HCC) in a mammalian subject, consisting of the step of:

administering to a mammalian subject in need of treatment for hepatocellular carcinoma, an effective amount of the compound

or a pharmaceutically acceptable salt thereof.

2. The method of claim 1 , wherein the mammalian subject is a human subject.

3. A method for inducing apoptosis of mammalian hepatocellular carcinoma (HCC) cells, consisting of the step of:

contacting the mammalian hepatocellular carcinoma cells with an effective amount of the compound

or a pharmaceutically acceptable salt thereof,

thereby inducing apoptosis of said cells.

4. The method of claim 3 , wherein the mammalian hepatocellular carcinoma cells are human hepatocellular carcinoma cells.

5. A method for treating hepatocellular carcinoma (HCC) in a mammalian subject, consisting of the step of:

administering to a mammalian subject in need of treatment for hepatocellular carcinoma, a pharmaceutical composition consisting of:

(i) an effective amount of the compound

or a pharmaceutically acceptable salt thereof, and

(ii) at least one pharmaceutically acceptable excipient.

6. The method of claim 5 , wherein the mammalian subject is a human subject.

Assignments (4)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jul 9, 2026
From: ENZO BIOCHEM, INC.; ENZO LIFE SCIENCES, INC.; ENZO THERAPEUTICS, INC.
To: SERAPH BIOTECH CONSULTING, LLC
Reel/Frame 075219/0465 →
RELEASE OF SECURITY INTEREST Recorded Jul 24, 2023
From: GEMINO HEALTHCARE FINANCE, LLC D/B/A SLR HEALTHCARE ABL
To: ENZO BIOCHEM, INC.; ENZO CLINICAL LABS, INC.; ENZO LIFE SCIENCES U.S. HOLDING CORP; ENZO LIFE SCIENCES, INC.
Reel/Frame 064369/0031 →
SECURITY INTEREST Recorded Apr 3, 2023
From: ENZO LIFE SCIENCES, INC.; ENZO CLINICAL LABS, INC.; ENZO BIOCHEM, INC.; ENZO LIFE SCIENCES U.S. HOLDING CORP
To: GEMINO HEALTHCARE FINANCE, LLC D/B/A SLR HEALTHCARE ABL
Reel/Frame 063239/0103 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jul 17, 2018
From: RABBANI, ELAZAR; DONEGAN, JAMES J.; DIAMOND, PAUL
To: ENZO BIOCHEM, INC.
Reel/Frame 046367/0073 →
Continuity (2)
Provisional Application 62524221 · Jun 23, 2017
Related Publication 20180369169A1 · Dec 27, 2018