IP Library Granted Patent US 11,419,878
Granted Patent B2
US 11,419,878 · App. 16/089,274 · Granted Aug 23, 2022

Medicine obtained by combining FXR agonist and ARB

Inventors: Tadashi Namisaki (Nara, JP); Hitoshi Yoshiji (Nara, JP)
Assignee: Intercept Pharmaceuticals, Inc.
A61K31/575A61K31/41A61K31/4178A61K31/4184A61K31/42A61K31/4245A61K31/454A61K45/06A61P1/16
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Quick Facts
Patent No.
US 11,419,878
App. No.
16/089,274
Granted
Aug 23, 2022
Kind
B2
Abstract

The present invention provides an NASH therapeutic agent including: an FXR agonist, preferably obeticholic acid or a pharmaceutically acceptable salt thereof; and an ARB or a pharmaceutically acceptable salt thereof.

Claims (5)

1. A pharmaceutical composition comprising a combination of obeticholic acid or a pharmaceutically acceptable salt thereof in the amount of 2 mg-100 mg and losartan or a pharmaceutically acceptable salt thereof in the amount of 5 mg-100 mg, wherein the obeticholic acid or pharmaceutically acceptable salt thereof and losartan or pharmaceutically acceptable salt thereof are the only active pharmaceutical ingredients present in the composition.

2. The pharmaceutical composition of claim 1 , comprising one or more pharmaceutically acceptable carriers or excipients.

3. The pharmaceutical composition of claim 1 , comprising obeticholic acid or a pharmaceutically acceptable salt thereof in the amount of 5 mg-50 mg.

4. The pharmaceutical composition of claim 1 , comprising losartan or a pharmaceutically acceptable salt thereof in the amount of 10 mg-50 mg.

5. The pharmaceutical composition of claim 1 , comprising obeticholic acid or a pharmaceutically acceptable salt thereof in the amount of 5 mg-50 mg and losartan or a pharmaceutically acceptable salt thereof in the amount of 10 mg-50 mg.

Assignments (4)
RELEASE OF SECURITY INTEREST Recorded Jan 4, 2024
From: U.S. BANK TRUST COMPANY, NATIONAL ASSOCIATION
To: INTERCEPT PHARMACEUTICALS, INC.
Reel/Frame 066662/0210 →
CHANGE OF ADDRESS Recorded Aug 22, 2022
From: INTERCEPT PHARMACEUTICALS, INC.
To: INTERCEPT PHARMACEUTICALS, INC.
Reel/Frame 061297/0990 →
SECURITY INTEREST Recorded Aug 18, 2021
From: INTERCEPT PHARMACEUTICALS, INC.
To: U.S. BANK NATIONAL ASSOCIATION
Reel/Frame 057650/0772 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 3, 2019
From: NAMISAKI, TADASHI; YOSHIJI, HITOSHI
To: NARA MEDICAL UNIVERSITY
Reel/Frame 050615/0642 →
Priority Claims (1)
JP JP2016-064475 · Mar 28, 2016 · national
Continuity (1)
Related Publication 20190247404A1 · Aug 15, 2019