IP Library Granted Patent US 11,351,183
Granted Patent B2
US 11,351,183 · App. 16/095,228 · Granted Jun 7, 2022

Use of thyroid beta-agonists

Inventors: Brian Lian (San Diego, CA); Rochelle Hanley (Ann Arbor, MI); Misha Dinerman (Cincinnati, OH); Mark Erion (Brookline, MA); Serge Boyer (San Diego, CA); Hongjian Jiang (Shanghai, CN)
Assignees: Viking Therapeutics, Inc.; Metabasis Therapeutics, Inc.
A61K31/662
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Quick Facts
Patent No.
US 11,351,183
App. No.
16/095,228
Granted
Jun 7, 2022
Kind
B2
Abstract

Methods useful for treating X-linked adrenoleukodystrophy are provided.

Claims (23)

1. A method of therapeutic treatment for X-linked adrenoleukodystrophy, comprising administering to a subject a compound having the structure

or a salt, ester, or prodrug thereof.

2. The method of claim 1 , wherein the compound is

or a salt, ester, or prodrug thereof.

3. The method of claim 2 , wherein the compound is

4. The method of claim 1 , wherein the compound is

or a salt, ester, or prodrug thereof.

5. The method of claim 4 , wherein the compound is

6. The method of claim 1 , wherein the compound is administered at a dose of between about 1_mg and about 100 mg per day.

7. The method of claim 1 , wherein the compound is administered daily, every other day, or intermittently for three months followed by a period of time from about 2 months to about 1 week when the compound is not administered.

8. The method of claim 6 , wherein the compound is administered at a dose of between about 1_mg and about 50 mg per day.

9. The method of claim 8 , wherein the compound is administered at a dose of between about 1_mg and about 25 mg per day.

10. The method of claim 1 , wherein the compound is administered at a dose of 100 mg/day, 50 mg/day, 25 mg/day, 20 mg/day, 15 mg/day, 10 mg/day, 5 mg/day, or 1 mg/day.

11. The method of claim 10 , wherein the compound is administered at a dose of 5 mg/day, 10 mg/day, or 15 mg/day.

12. The method of claim 10 , wherein the compound is administered at a dose of 5 mg/day.

13. The method of claim 10 , wherein the compound is administered at a dose of 10 mg/day.

14. The method of claim 1 , wherein the compound is administered at a dose of between about 1 mg and about 100 mg every other day.

15. The method of claim 14 , wherein the compound is administered at a dose of between about 1 mg and about 50 mg every other day.

16. The method of claim 14 , wherein the compound is administered at a dose of between about 1 mg and about 25 mg every other day.

17. The method of claim 1 , wherein the compound is administered at a dose of 10 mg every other day or 15 mg every other day.

18. The method of claim 1 , wherein the compound is administered daily, every other day, or intermittently for three months followed by a period of time of one month when the thyroid hormone receptor beta agonist is not administered.

19. The method of claim 1 , wherein the compound is administered daily, every other day, or intermittently for three months followed by a period of time of 14 days when the thyroid hormone receptor beta agonist is not administered.

20. The method of claim 1 , wherein the compound is administered daily, every other day, or intermittently for two months followed by a period of time of one month when the thyroid hormone receptor beta agonist is not administered.

Assignments (4)
SECURITY INTEREST Recorded Oct 18, 2023
From: CYDEX PHARMACEUTICALS, INC.; LIGAND PHARMACEUTICALS INCORPORATED; METABASIS THERAPEUTICS, INC.; PFENEX INC.
To: CITIBANK, N.A., AS ADMINISTRATIVE AGENT
Reel/Frame 065271/0025 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Nov 30, 2018
From: JIANG, HONGJIAN
To: METABASIS THERAPEUTICS INC.
Reel/Frame 047643/0946 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Nov 15, 2018
From: ERION, MARK; BOYER, SERGE
To: METABASIS THERAPEUTICS, INC.
Reel/Frame 047517/0859 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Nov 15, 2018
From: LIAN, BRIAN; HANLEY, ROCHELLE; DINERMAN, MISHA
To: VIKING THERAPEUTICS, INC.
Reel/Frame 047517/0930 →
Cited By (1)
US 12,678,430