IP Library Granted Patent US 10,864,175
Granted Patent B2
US 10,864,175 · App. 16/140,090 · Granted Dec 15, 2020

Eutectic formulations of cyclobenzaprine hydrochloride and amitriptyline hydrochloride

Inventors: Marino Nebuloni (Rho, IT); Patrizia Colombo (Trezzano sul Naviglio, IT)
Assignee: Tonix Pharma Holdings Limited
A61K31/135A61K9/145A61K9/1623A61K9/1688A61K9/1694A61K31/047A61K31/137A61K47/02A61K47/10A61K47/12A61K47/26A61K31/55
View Patent ↗
Loading inventors, assignments & file history…
Monitor This Case
Get email alerts when status or documents change.
Order Certified Copies
Most orders are placed with the USPTO same day — all within 24 business hours.
Order via The Patent Place →
Pre-filled with this patent's details
Quick Facts
Patent No.
US 10,864,175
App. No.
16/140,090
Granted
Dec 15, 2020
Kind
B2
Abstract

The present invention relates to pharmaceutical compositions and methods of manufacturing the same, comprising a eutectic of Cyclobenzaprine HCl and mannitol or Amitriptyline HCl and mannitol.

Claims (4)

1. A eutectic of Cyclobenzaprine HCl and β-mannitol comprising 75%±2% cyclobenzaprine HCl and 25%±2% β-mannitol by weight.

2. The eutectic of claim 1 , wherein the Cyclobenzaprine HCl:β-mannitol molar ratio is 1.76±0.1.

3. The eutectic of claim 1 or 2 , wherein the Cyclobenzaprine HCl is micronized Cyclobenzaprine HCl.

4. The eutectic of any one of claim 1 - 3 , wherein the eutectic melts at 143.6±3° C.

Assignments (5)
NOVATION AGREEMENT Recorded Jul 8, 2024
From: TONIX PHARMA HOLDINGS LIMITED
To: TONIX PHARMA LIMITED
Reel/Frame 068217/0592 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 25, 2020
From: TONIX PHARMACEUTICALS, INC.
To: TONIX PHARMA HOLDINGS LIMITED
Reel/Frame 052010/0959 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Sep 24, 2018
From: NEBULONI, MARINO; COLOMBO, PATRIZIA
To: REDOX SRL
Reel/Frame 046954/0489 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Sep 24, 2018
From: REDOX SRL
To: TONIX PHARMACEUTICALS, INC.
Reel/Frame 046954/0510 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Sep 24, 2018
From: TONIX PHARMACEUTICALS, INC.
To: TONIX PHARMA HOLDINGS LIMITED
Reel/Frame 046954/0517 →
Continuity (3)
Continuation 14776624
Provisional Application 61792757 · Mar 15, 2013
Related Publication 20190022030A1 · Jan 24, 2019