IP Library Granted Patent US 10,815,300
Granted Patent B2
US 10,815,300 · App. 16/168,060 · Granted Oct 27, 2020

Methods for treating vascular leak syndrome and cancer

Inventors: Kevin Peters (Cincinnati, OH); Robert Shalwitz (Bexley, OH)
Assignee: AERPIO PHARMACEUTICALS, INC.
C07K16/28C07K16/40A61K38/2013A61K2039/505A61P27/02A61P35/00C07K14/55
View Patent ↗
Loading inventors, assignments & file history…
Monitor This Case
Get email alerts when status or documents change.
Order Certified Copies
Most orders are placed with the USPTO same day — all within 24 business hours.
Order via The Patent Place →
Pre-filled with this patent's details
Quick Facts
Patent No.
US 10,815,300
App. No.
16/168,060
Granted
Oct 27, 2020
Kind
B2
Abstract

Disclosed are methods for treating Vascular Leak Syndrome and preventing cancer metastasis. Further disclosed are methods for treating vascular leakage due to inflammatory diseases, sepsis, cancer or the presence of pathogens.

Claims (11)

1. A method for reducing vascular leak syndrome in an eye of a human having vascular leak in the eye, comprising administering to the human a composition comprising a therapeutically-effective amount of an HPTPβ-ECD binding agent, wherein the HPTPβ-ECD binding agent is R15E6 or a humanized form thereof, wherein vascular leak syndrome is reduced by a reduction in neovascularization, wherein the therapeutically-effective amount of the HPTPβ-ECD binding agent is from about 0.01 mg/kg to about 10 mg/kg by weight of the human.

2. The method of claim 1 , wherein the reduction in neovascularization is a reduction in choroidal neovascularization.

3. The method of claim 1 , wherein the reduction in neovascularization is a reduction in retinal neovascularization.

4. The method of claim 1 , wherein the human suffers from an inflammatory disease or condition.

5. The method of claim 1 , wherein the human has a cancer.

6. The method of claim 1 , wherein the HPTPβ-ECD binding agent inhibits HPTPβ.

7. The method of claim 1 , wherein the administering is by intravenous injection.

8. The method of claim 1 , wherein the administering is by subcutaneous injection.

9. The method of claim 1 , wherein the administering is by intraocular injection.

10. The method of claim 1 , wherein the HPTPβ-ECD binding agent is conjugated to a vehicle, wherein the vehicle is PEG.

11. A method for reducing vascular leak syndrome in an eye of a human having vascular leak in the eye, comprising administering to the human a composition comprising a therapeutically-effective amount of an HPTPβ-ECD binding agent, wherein the HPTPβ-ECD binding agent is R15E6 or a humanized form thereof, wherein vascular leak syndrome is reduced by a reduction in neovascularization, wherein the administering is by intraocular injection.

Assignments (4)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Sep 9, 2021
From: AERPIO PHARMACEUTICALS, INC.
To: EYEPOINT PHARMACEUTICALS, INC.
Reel/Frame 057448/0033 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 17, 2020
From: AERPIO THERAPEUTICS LLC
To: AERPIO PHARMACEUTICALS, INC.
Reel/Frame 052432/0789 →
CHANGE OF NAME Recorded Jul 31, 2019
From: AERPIO THERAPEUTICS, INC.
To: AERPIO THERAPEUTICS LLC
Reel/Frame 049918/0806 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 27, 2019
From: PETERS, KEVIN; SHALWITZ, ROBERT
To: AERPIO THERAPEUTICS, INC.
Reel/Frame 048457/0591 →