IP Library Granted Patent US 11,395,796
Granted Patent B2
US 11,395,796 · App. 16/170,160 · Granted Jul 26, 2022

Anti-CD37 immunoconjugate and anti-CD20 antibody combinations

Inventors: Angela Romanelli (Lexington, MA); Rodrigo R. Ruiz-Soto (Boston, MA); Jose Ponte (Weymouth, MA); Jutta Deckert (Lexington, MA); Jan Pinkas (Belmont, MA)
Assignee: Debiopharm International, S.A.
A61K9/0019A61K47/6801A61K47/6803A61K47/6849A61K47/6867A61P35/02C07K16/2887C07K16/2896A61K2039/507A61K2039/545C07K2317/24
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Quick Facts
Patent No.
US 11,395,796
App. No.
16/170,160
Granted
Jul 26, 2022
Kind
B2
Abstract

Methods of administering immunoconjugates that bind to CD37 (e.g., IMGN529) in combination with antibodies that bind to CD20 are provided. The methods comprise administering an anti-CD37 immunoconjugate (e.g., IMGN529) and an anti-CD20 antibody to a person in need thereof, for example, a cancer patient.

Claims (10)

1. A method for treating a human patient having a B-cell cancer comprising administering to said patient in need thereof (i) an immunoconjugate that binds to CD37 comprising a DM1 maytansinoid, an SMCC linker, and an antibody that binds to CD37 comprising the heavy chain sequence set forth in SEQ ID NO:18 and the light chain sequence set forth in SEQ ID NO: 21; and (ii) rituximab, wherein said immunoconjugate that binds to CD37 is administered at a dose of 0.7 mg/kg once every three weeks and wherein the rituximab is administered at a dose of about 375 mg/m2 on week 1, day 1 of a three week schedule.

2. The method of claim 1 , wherein the immunoconjugate that binds to CD37 and the rituximab produce a synergistic effect, with a Synergy Score of at least 4 in vitro.

3. The method of claim 1 , wherein the immunoconjugate that binds to CD37 and the rituximab have a combination index value of less than 0.5.

4. The method of claim 1 , wherein the cancer is leukemia or lymphoma.

5. The method of claim 1 , wherein the cancer is selected from the group consisting of NHL, precursor B-cell lymphoblastic leukemia/lymphoma, B-cell chronic lymphocytic leukemia (CLL)/small lymphocytic lymphoma (SLL), B-cell prolymphocytic leukemia, lymphoplasmacytic lymphoma, mantle cell lymphoma (MCL), follicular lymphoma (FL), cutaneous follicle center lymphoma, marginal zone B-cell lymphoma, hairy cell leukemia, diffuse large B-cell lymphoma (DLBCL), Burkitt's lymphoma, plasmacytoma, plasma cell myeloma, post-transplant lymphoproliferative disorder, Waldenstrom's macroglobulinemia, acute lymphoblastic leukemia (ALL), and anaplastic large-cell lymphoma (ALCL).

6. The method of claim 1 , wherein the cancer overexpresses MYC and/or BCL2.

7. The method of claim 1 , wherein the immunoconjugate that binds to CD37 and the rituximab are administered intravenously.

8. The method of claim 1 , further comprising administering a corticosteroid to the patient.

9. The method of claim 1 , further comprising administering a growth factor to the patient.

10. The method of claim 1 , wherein the human patient has relapsed diffuse large B-cell lymphoma (DLBCL).

Assignments (2)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 26, 2018
From: ROMANELLI, ANGELA; RUIZ-SOTO, RODRIGO R.; PONTE, JOSE; DECKERT, JUTTA; PINKAS, JAN
To: IMMUNOGEN, INC.
Reel/Frame 047326/0384 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 26, 2018
From: IMMUNOGEN, INC.
To: DEBIOPHARM INTERNATIONAL, S.A.
Reel/Frame 047326/0399 →
Continuity (4)
Continuation 15171732 · Jun 2, 2016
Provisional Application 62263449 · Dec 4, 2015
Provisional Application 62172672 · Jun 8, 2015
Related Publication 20190183788A1 · Jun 20, 2019
Cited By (5)
US 12,227,567 US 12,239,732 US 12,281,166 US 12,497,458 US 12,559,566