IP Library Granted Patent US 10,703,748
Granted Patent B2
US 10,703,748 · App. 16/177,149 · Granted Jul 7, 2020

Diazanaphthalen-3-yl carboxamides and preparation and use thereof

Inventors: Sunil Kumar Kc (San Diego, CA); Chi Ching Mak (San Diego, CA); Jianguo Cao (San Diego, CA); Venkataiah Bollu (San Diego, CA); Chandramouli Chiruta (San Diego, CA); Gopi Kumar Mittapalli (San Diego, CA); Brian Walter Eastman (San Diego, CA); Brian Joseph Hofilena (San Diego, CA)
Assignee: Samumed, LLC
C07D471/04A61P25/00A61P25/28A61P29/00A61P35/00C07D401/14C07D417/14C07D487/04
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Quick Facts
Patent No.
US 10,703,748
App. No.
16/177,149
Granted
Jul 7, 2020
Kind
B2
Abstract

Diazanaphthalene compounds for treating various diseases and pathologies are disclosed. More particularly, the present disclosure concerns the use of a diazanaphthalene compound or analogs thereof, in the treatment of disorders characterized by the activation of Wnt pathway signaling (e.g., cancer, abnormal cellular proliferation, angiogenesis, Alzheimer's disease, lung disease, inflammation, auto-immune diseases and osteoarthritis), the modulation of cellular events mediated by Wnt pathway signaling, as well as neurological conditions/disorders/diseases linked to overexpression of DYRK1A.

Claims (4722)

1. A compound, or a pharmaceutically acceptable salt thereof, of Formula I:

wherein:

R 1 , R 2 , R 4 , and R 5 are independently absent or selected from the group consisting of H, halide, unsubstituted —(C 1-3 haloalkyl), and unsubstituted —(C 1-3 alkyl);

R 3 is selected from the group consisting of -aryl optionally substituted with 1-5 R 7 and -heteroaryl optionally substituted with 1-4 R 8 ;

R 6 is selected from the group consisting of —(C 1-4 alkylene) p aryl substituted with 1-5 R 9 , —(C 2-4 alkenylene) p aryl substituted with 1-5 R 9 , —(C 1-4 alkylene) p heteroaryl optionally substituted with 1-6 R 10 ; —(C 1-4 alkylene) p heterocyclyl optionally substituted with 1-10 R 11 , —(C 1-4 alkylene) p carbocyclyl optionally substituted with 1-12 R 12 , —(C 1-4 alkylene)N(R 13 )(R 14 ), —N(R 15 )(R 16 ), —CF(C 1-9 alkyl) 2 , —(C 1-4 alkylene) p O(C 3-9 alkyl), and —(C 2-9 alkynyl) optionally substituted with one or more halides; wherein each alkyl of —CF(C 1-9 alkyl) 2 is, independently, optionally substituted with one or more halides; wherein each —(C 1-4 alkylene) is, independently, optionally substituted with one or more substituents; wherein —(C 1-4 alkenylene) is, optionally substituted with one or more substituents;

R 7 is selected from the group consisting of halide and —N(R 17 ) 2 ;

each R 8 is independently selected from the group consisting of H, halide, unsubstituted —(C 1-9 alkyl), unsubstituted —(C 2-9 alkenyl), unsubstituted —(C 2-9 alkynyl), unsubstituted —(C 1-9 haloalkyl), —CN, —N(R 15 )(R 18 ), —(C 1-4 alkylene) p XR 19 , —C(═O)N(R 5 ) 2 , —(C 1-4 alkylene) p heterocyclyl optionally substituted with 1-10 R 20 , and -carbocyclyl optionally substituted with 1-12 R 21 ; wherein each —(C 1-4 alkylene) is, independently, optionally substituted with one or more substituents;

alternatively, two adjacent R 8 are taken together to form a ring which is selected from the group consisting of -heterocyclyl optionally substituted with 1-10 R 22 and -carbocyclyl optionally substituted with 1-12 R 21 ;

each R 9 is independently selected from the group consisting of halide, unsubstituted —(C 1-9 alkyl), unsubstituted —(C 2-9 alkenyl), unsubstituted —(C 2-9 alkynyl), unsubstituted —(C 1-9 haloalkyl), —XR 23 , C(═O)N(R 5 ) 2 , —(C 1-4 alkylene) p N(R 24 ) 2 , —(C 1-4 alkylene) p heterocyclyl optionally substituted with 1-10 R 22 , and —(C 1-4 alkylene) p carbocyclyl optionally substituted with 1-12 R 21 ; wherein each —(C 1-4 alkylene) is, independently, optionally substituted with one or more substituents;

with the proviso that when Y 2 is N then R 9 is not —OMe or

each R 10 is independently selected from the group consisting of halide, unsubstituted —(C 1-9 alkyl), unsubstituted —(C 2-9 alkenyl), unsubstituted —(C 2-9 alkynyl), unsubstituted —(C 1-9 haloalkyl), —CN, —XR 23 , —C(═O)N(R 15 ) 2 , —(C 1-4 alkylene) p N(R 24 ) 2 , —(C 1-4 alkylene) p heterocyclyl optionally substituted with 1-10 R 22 , and —(C 1-4 alkylene) p carbocyclyl optionally substituted with 1-12 R 21 ; wherein each —(C 1-4 alkylene) is, independently, optionally substituted with one or more substituents;

each R 11 is independently selected from the group consisting of halide, unsubstituted —(C 1-9 alkyl), unsubstituted —(C 2-9 alkenyl), unsubstituted —(C 2-9 alkynyl), unsubstituted —(C 1-9 haloalkyl), —(C 1-4 alkylene) p OR 19 , —(C 1-4 alkylene) p heterocyclyl optionally substituted with 1-10 R 22 , —(C 1-4 alkylene) p carbocyclyl optionally substituted with 1-12 R 21 , —N(R 15 )(R 25 ), —C(═O)(R 26 ), —(C 1-4 alkylene)C(═O)OR 27 , —(C 1-4 alkylene)aryl optionally substituted with one or more halides, —(C 1-4 alkylene) p heteroaryl optionally substituted with one or more halides, and —SO 2 (R 28 ); wherein each —(C 1-4 alkylene) is, independently, optionally substituted with one or more substituents;

alternatively, two R 11 attached to the same carbon atom can together represent ═O to form a carbonyl group;

each R 12 is independently selected from the group consisting of halide, unsubstituted —(C 1-9 alkyl), unsubstituted —(C 2-9 alkenyl), unsubstituted —(C 2-9 alkynyl), unsubstituted —(C 1-9 haloalkyl), —(C 1-4 alkylene) p OR 19 , —N(R 15 )(R 29 ), —C(═O)(R 26 ), —C(═O)OR 27 , —(C 1-4 alkylene) p heterocyclyl optionally substituted with 1-10 R 22 , and —(C 1-4 alkylene) p carbocyclyl optionally substituted with 1-12 R 21 ; wherein each —(C 1-4 alkylene) is, independently, optionally substituted with one or more substituents;

R 13 is selected from the group consisting of H, unsubstituted —(C 1-9 alkyl), unsubstituted —(C 2-9 alkenyl), unsubstituted —(C 2-9 alkynyl), unsubstituted —(C 1-9 haloalkyl), —(C 1-4 alkylene) p heterocyclyl optionally substituted with 1-10 R 20 , and -carbocyclyl optionally substituted with 1-12 R 21 ; wherein —(C 1-4 alkylene) is, optionally substituted with one or more substituents;

R 14 is selected from the group consisting of unsubstituted —(C 1-9 alkyl), unsubstituted —(C 2-9 alkenyl), unsubstituted —(C 2-9 alkynyl), unsubstituted —(C 1-9 haloalkyl), —(C 1-4 alkylene) p heterocyclyl optionally substituted with 1-10 R 20 , and -carbocyclyl optionally substituted with 1-12 R 21 ; wherein —(C 1-4 alkylene) is, optionally substituted with one or more substituents;

each R 15 is selected from the group consisting of H, unsubstituted —(C 1-s alkyl), unsubstituted —(C 2-5 alkenyl), unsubstituted —(C 2-5 alkynyl), and unsubstituted —(C 1-5 haloalkyl);

R 16 is selected from the group consisting of —(C 1-4 alkylene) p heterocyclyl optionally substituted with 1-10 R 20 , and —(C 1-4 alkylene) p carbocyclyl optionally substituted with 1-12 R 21 ; wherein each —(C 1-4 alkylene) is, independently, optionally substituted with one or more substituents;

R 17 is independently selected from the group consisting of H, unsubstituted —(C 1-5 alkyl), unsubstituted —(C 2-5 alkenyl), unsubstituted —(C 2-5 alkynyl), and unsubstituted —(C 1-5 haloalkyl);

alternatively, two adjacent R 17 are taken together to form a -heterocyclyl ring optionally substituted with 1-10 R 22 ;

R 18 is independently selected from the group consisting of H, unsubstituted —(C 1-5 alkyl), unsubstituted —(C 2-5 alkenyl), unsubstituted —(C 2-5 alkynyl), unsubstituted —(C 1-5 haloalkyl), —(C═O)R 5 , and —(C 1-4 alkylene) p heterocyclyl optionally substituted with one or more halides or one or more unsubstituted —(C 1-5 alkyl); wherein —(C 1-4 alkylene) is, independently, optionally substituted with one or more substituents;

each R 19 is independently selected from the group consisting of H, unsubstituted —(C 1-s alkyl), unsubstituted —(C 2-5 alkenyl), unsubstituted —(C 2-5 alkynyl), unsubstituted —(C 1-5 haloalkyl), —(C 1-4 alkylene) p heterocyclyl optionally substituted with one or more halides or one or more unsubstituted —(C 1-5 alkyl), and —(C 1-4 alkylene) p carbocyclyl optionally substituted with 1-12 R 21 ; wherein each —(C 1-4 alkylene) is, independently, optionally substituted with one or more substituents;

each R 20 independently is selected from the group consisting of halide, unsubstituted —(C 1-5 alkyl), unsubstituted —(C 2-5 alkenyl), unsubstituted —(C 2-5 alkynyl), unsubstituted —(C 1-5 haloalkyl), —CN, —OH, —N(R 5 ) 2 , and —(C 1-4 alkylene) p carbocyclyl optionally substituted with 1-12 R 21 ; wherein each —(C 1-4 alkylene) is, independently, optionally substituted with one or more substituents;

each R 21 is independently selected from the group consisting of halide, unsubstituted —(C 1-5 alkyl), unsubstituted —(C 2-5 alkenyl), unsubstituted —(C 2-5 alkynyl), unsubstituted —(C 1-5 haloalkyl), and —CN;

each R 22 is independently selected from the group consisting of halide, unsubstituted —(C 1-5 alkyl), unsubstituted —(C 2-5 alkenyl), unsubstituted —(C 2-5 alkynyl), unsubstituted —(C 1-5 haloalkyl), —CN, —OH, —N(R 15 ) 2 , —C(═O)R 34 , and —(C 1-4 alkylene) p carbocyclyl optionally substituted with 1-12 R 21 ; wherein each —(C 1-4 alkylene) is, independently, optionally substituted with one or more substituents;

each R 23 is independently selected from the group consisting of H, unsubstituted —(C 1-5 alkyl), unsubstituted —(C 2-5 alkenyl), unsubstituted —(C 2-5 alkynyl), unsubstituted —(C 1-5 haloalkyl), —(C 1-4 alkylene)N(R 15 ) 2 , —(C 1-4 alkylene) p aryl optionally substituted with 1-10 R 30 , —(C 1-4 alkylene) p heterocyclyl optionally substituted with 1-12 R 31 , and —(C 1-4 alkylene) p carbocyclyl optionally substituted with 1-12 R 21 ; wherein each —(C 1-4 alkylene) is, independently, optionally substituted with one or more substituents;

each R 24 is independently selected from the group consisting of H, unsubstituted —(C 1-5 alkyl), unsubstituted —(C 2-5 alkenyl), unsubstituted —(C 2-5 alkynyl), unsubstituted —(C 1-5 haloalkyl), —(C 1-4 alkylene) p heterocyclyl optionally substituted with one or more halides or one or more unsubstituted —(C 1-5 alkyl), and —(C 1-4 alkylene)N(R 15 ) 2 ; wherein each —(C 1-4 alkylene) is, independently, optionally substituted with one or more substituents;

each R 25 is selected from the group consisting of H, unsubstituted —(C 1-5 alkyl), unsubstituted —(C 2-5 alkenyl), unsubstituted —(C 2-5 alkynyl), unsubstituted —(C 1-5 haloalkyl), —(C 1-4 alkylene) p heterocyclyl optionally substituted with 1-10 R 32 , —(C 1-4 alkylene) p carbocyclyl optionally substituted with 1-12 R 21 , —(C 1-4 alkylene)OR 33 ; wherein each —(C 1-4 alkylene) is, independently, optionally substituted with one or more substituents;

R 26 is selected from the group consisting of H, unsubstituted —(C 3-5 alkyl), unsubstituted —(C 2-5 alkenyl), unsubstituted —(C 2-5 alkynyl), unsubstituted —(C 1-5 haloalkyl), —(C 1-4 alkylene) p aryl optionally substituted with one or more halides or unsubstituted —(C 1-5 alkyl), —(C 1-4 alkylene) p heteroaryl optionally substituted with one or more halides or one or more unsubstituted —(C 1-5 alkyl), and —(C 1-4 alkylene) p heterocyclyl optionally substituted with one or more halides or one or more unsubstituted —(C 1-5 alkyl); wherein each —(C 1-4 alkylene) is, independently, optionally substituted with one or more substituents;

R 27 is selected from the group consisting of H, unsubstituted —(C 1-5 alkyl), unsubstituted —(C 2-5 alkenyl), unsubstituted —(C 2-5 alkynyl), unsubstituted —(C 1-5 haloalkyl), —(C 1-4 alkylene) p aryl optionally substituted with one or more halides or one or more unsubstituted —(C 1-5 alkyl), —(C 1-4 alkylene) p heteroaryl optionally substituted with one or more halides or unsubstituted —(C 1-5 alkyl), and —(C 1-4 alkylene) p heterocyclyl optionally substituted with one or more halides or one or more unsubstituted —(C 1-5 alkyl); wherein each —(C 1-4 alkylene) is, independently, optionally substituted with one or more substituents;

R 28 is selected from the group consisting of unsubstituted —(C 1-5 alkyl), unsubstituted —(C 2-5 alkenyl), unsubstituted —(C 2-5 alkynyl), unsubstituted —(C 1-5 haloalkyl), —(C 1-4 alkylene) p aryl optionally substituted with one or more halides or one or more unsubstituted —(C 1-5 alkyl), —(C 1-4 alkylene) p heteroaryl optionally substituted with one or more halides or one or more unsubstituted —(C 1-5 alkyl), and —(C 1-4 alkylene) p heterocyclyl optionally substituted with one or more halides or one or more unsubstituted —(C 1-5 alkyl); wherein —(C 1-4 alkylene) is, optionally substituted with one or more substituents;

each R 29 is selected from the group consisting of H, unsubstituted —(C 1-s alkyl), unsubstituted —(C 2 -5 alkenyl), unsubstituted —(C 2-5 alkynyl), unsubstituted —(C 1-5 haloalkyl), —(C 1-4 alkylene) p heterocyclyl optionally substituted with 1-10 R 32 , —(C 1-4 alkylene) p carbocyclyl optionally substituted with 1-12 R 21 , —(C 1-4 alkylene)OR 33 , and —C(═O)O(C 1-5 alkyl); wherein each —(C 1-4 alkylene) is, independently, optionally substituted with one or more substituents;

each R 30 is independently selected from the group consisting of halide, unsubstituted —(C 1-5 alkyl), unsubstituted —(C 2-5 alkenyl), unsubstituted —(C 2-5 alkynyl), unsubstituted —(C 1-5 haloalkyl), and —CN;

each R 31 is independently selected from the group consisting of halide, unsubstituted —(C 1-5 alkyl), unsubstituted —(C 2-5 alkenyl), unsubstituted —(C 2-5 alkynyl), unsubstituted —(C 1-5 haloalkyl), —CN, —OH, —C(═O)R 34 , —N(R 24 ) 2 , and —(C 1-4 alkylene) p carbocyclyl optionally substituted with 1-12 R 21 ; wherein each —(C 1-4 alkylene) is, independently, optionally substituted with one or more substituents;

each R 32 is independently selected from the group consisting of halide and unsubstituted —(C 1-5 alkyl);

each R 33 is independently selected from the group consisting of H and unsubstituted —(C 1-5 alkyl);

each R 34 is independently selected from the group consisting of —O(C 15 alkyl) and a heteroaryl optionally substituted with 1-6 R 35 ;

each R 35 is a -heterocyclyl optionally substituted with one or more halides or one or more unsubstituted —(C 1-5 alkyl);

each X is selected from the group consisting of O and S;

Y 3 is CH or nitrogen;

Y 1 , Y 2 , Y 4 , and Y 5 are independently selected from the group consisting of carbon and nitrogen;

wherein

if Y 1 is nitrogen then Y 2 , Y 4 , and Y 5 are carbon, Y 3 is CH, and R 4 is absent;

if Y 2 is nitrogen then Y 1 , Y 4 , and Y 5 are carbon, Y 3 is CH, and R 5 is absent;

if Y 3 is nitrogen then Y 1 , Y 2 , Y 4 , and Y 5 are carbon;

if Y 4 is nitrogen then Y 1 , Y 2 , and Y 5 are carbon, Y 3 is CH, and R 1 is absent;

if Y 5 is nitrogen then Y 1 , Y 2 , and Y 4 are carbon, Y 3 is CH, and R 2 is absent;

each p is independently 0 or 1; and

wherein the compound of Formula I is selected from the group consisting of

or a pharmaceutically acceptable salt thereof.

2. The compound of claim 1 , wherein R 1 , R 2 , R 4 , and R 5 are H.

3. The compound of claim 1 , wherein R 3 is selected from the group consisting of pyrazolyl, imidazolyl, triazolyl, thiadiazolyl, and oxazolyl, each optionally substituted with 1-4 R 8 .

4. The compound of claim 3 , wherein R 3 is a pyrazol-4-yl, substituted with one —(C 1-3 alkyl).

5. The compound of claim 3 , wherein R 3 is a imidazol-5-yl, substituted with one —(C 1-3 alkyl).

6. The compound of claim 3 , wherein R 3 is a imidazol-5-yl, substituted with two —(C 1-3 alkyl).

7. The compound of claim 3 , wherein R 3 is a 1,2,3-triazol-4-yl, substituted with one —(C 1-3 alkyl).

8. The compound of claim 3 , wherein R 3 is a thiadiazol-2-yl, substituted with one —(C 1-3 alkyl).

9. The compound of claim 3 , wherein R 3 is a oxazol-5-yl, substituted with one —(C 1-3 alkyl).

10. The compound of claim 3 , wherein R 6 is -heterocyclyl, optionally substituted with 1-2 R 11 .

11. The compound of claim 3 , wherein R 6 is a —CH 2 heterocyclyl optionally substituted with 1-2 R 11 .

12. The compound of claim 1 , wherein the compound of Formula I is selected from the group consisting of:

N-(2-(1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-1-isobutylpiperidine-4-carboxamide [1];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)cyclopropanecarboxamide [2];

4,4-difluoro-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)cyclohexane-1-carboxamide [3];

trans-4-methoxy-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)cyclohexane-1-carboxamide [4];

trans-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-4-morpholinocyclohexane-1-carboxamide [5];

trans-4-((3-fluoroazetidin-1-yl)methyl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl) cyclohexane-1-carboxamide [6];

trans-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-4-((4-methylpiperazin-1-yl) methyl)cyclohexane-1-carboxamide [7];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(pyrrolidin-1-yl)acetamide [8];

(S)-2-(3-fluoropyrrolidin-1-yl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl) acetamide [9];

(S)—N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)tetrahydrofuran-2-carboxamide [10];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [11];

1-methyl-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [12];

1-isopropyl-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [13];

1-(tert-butyl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [14];

1-cyclopropyl-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [15];

1-isobutyl-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [16];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-1-neopentylpiperidine-4-carboxamide [17];

1-(2-fluoroethyl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [18];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [19];

1-butyl-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [20];

1-benzoyl-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [21];

1-(2,2-difluoropropyl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [22];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)azetidine-3-carboxamide [23];

1-(2,2-difluoroethyl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [24];

1-(2-fluoro-2-methylpropyl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [25];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-1-(oxetan-3-yl)piperidine-4-carboxamide [26];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-1-((3-methyloxetan-3-yl)methyl) piperidine-4-carboxamide [27];

1-(2-methoxyethyl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [28];

1-(2-isopropoxyethyl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [29];

1,1-diisobutyl-4-((2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)carbamoyl)piperidin-1-ium [30];

4-fluoro-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [31];

4-fluoro-1-methyl-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [32];

4-fluoro-1-isobutyl-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [33];

(S)—N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)piperidine-3-carboxamide [34];

(R)—N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)piperidine-3-carboxamide [35];

(S)-1-isobutyl-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)piperidine-3-carboxamide [36];

(R)-1-isobutyl-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)piperidine-3-carboxamide [37];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)tetrahydro-2H-pyran-4-carboxamide [38];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(piperidin-1-yl)acetamide [39];

2-(4-fluoropiperidin-1-yl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)acetamide [40];

trans-4-amino-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)cyclohexane-1-carboxamide [41];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl)acetamide [42];

(S)—N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)piperidine-2-carboxamide [43];

2-(4-isobutylpiperazin-1-yl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)acetamide [44];

2-(3,3-dimethylazetidin-1-yl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)acetamide [45];

(R)-2-(3-fluoropyrrolidin-1-yl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl) acetamide [46];

(S)—N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(2-methylpyrrolidin-1-yl) acetamide [47];

2-(3-azabicyclo[3.1.0]hexan-3-yl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl) acetamide [48];

2-(7-azabicyclo[2.2.1]heptan-7-yl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl) acetamide [49];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperidin-1-yl)acetamide [50];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(4-(trifluoromethyl)piperidin-1-yl) acetamide [51];

2-(4-(difluoromethyl)piperidin-1-yl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl) acetamide [52];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(6-azaspiro[2.5]octan-6-yl)acetamide [53];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(pyrrolidin-1-yl)propanamide [54];

(R)—N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(2-methylpyrrolidin-1-yl) acetamide [55];

2-(cyclobutyl(methyl)amino)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)acetamide [56];

2-(diethylamino)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)acetamide [57];

7-(2-fluoroethyl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-7-azaspiro[3.5]nonane-2-carboxamide [58];

4-methyl-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)piperazine-1-carboxamide [59];

(S)—N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(pyrrolidin-1-yl)propanamide [60];

(R)—N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(pyrrolidin-1-yl)propanamide [61];

(R)—N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)pyrrolidine-2-carboxamide [62];

2-methyl-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-azaspiro[3.3]heptane-6-carboxamide [63];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(2,2,2-trifluoroacetyl)-2-azaspiro[3.3]heptane-6-carboxamide [64];

2-(2-fluoroethyl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-azaspiro[3.3]heptane-6-carboxamide [65];

trans-4-(dimethylamino)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)cyclohexane-1-carboxamide [66];

1-acetyl-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [67];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-1-((1-(trifluoromethyl)cyclopropyl) methyl)piperidine-4-carboxamide [68];

(S)-1-(2-fluoropropyl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [69];

(R)-1-(2-fluoropropyl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [70];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-1-(methylsulfonyl)piperidine-4-carboxamide [71];

1′-methyl-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-[1,4′-bipiperidine]-4-carboxamide [72];

trans-4-(hydroxymethyl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)cyclohexane-1-carboxamide [73];

methyl 2-(4-((2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)carbamoyl)piperidin-1-yl) acetate [74];

1-benzyl-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [75];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-1-(2-(pyrrolidin-1-yl)acetyl)piperidine-4-carboxamide [76];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-morpholinoacetamide [77];

(S)—N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(3-methylmorpholino)acetamide [78];

(R)—N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(3-methylmorpholino)acetamide [79];

(S)—N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(2-methylmorpholino)acetamide [80];

2-((2R,6S)-2,6-dimethylmorpholino)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl) acetamide [81];

2-((1S,4S)-2-oxa-5-azabicyclo[2.2.1]heptan-5-yl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)acetamide [82];

2-((1R,4R)-2-oxa-5-azabicyclo[2.2.1]heptan-5-yl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)acetamide [83];

2-(3-oxa-8-azabicyclo[3.2.1]octan-8-yl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl) acetamide [84];

(S)—N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-morpholinopropanamide [85];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(morpholin-2-yl)acetamide [86];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(4-methylmorpholin-2-yl)acetamide [87];

2-(4-ethylpiperazin-1-yl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)acetamide [88];

2-(4-isopropylpiperazin-1-yl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)acetamide [89];

2-(4-cyclopropylpiperazin-1-yl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl) acetamide [90];

2-(4-(2-fluoroethyl)piperazin-1-yl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl) acetamide [91];

(S)-2-(2,4-dimethylpiperazin-1-yl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl) acetamide [92];

1-(2-hydroxyethyl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [93];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-1-(pyridin-2-ylmethyl)piperidine-4-carboxamide [94];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-1-(oxazol-2-ylmethyl)piperidine-4-carboxamide [95];

(R)—N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-1-oxotetrahydro-1H-pyrrolo[1,2-c]imidazole-2(3H)-carboxamide [96];

(R)-1-methyl-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)pyrrolidine-2-carboxamide [97];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-1-(tetrahydro-2H-pyran-4-yl)piperidine-4-carboxamide [98];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-1-(pyrimidin-2-ylmethyl)piperidine-4-carboxamide [99];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-1-(pyrazin-2-ylmethyl)piperidine-4-carboxamide [100];

1-((5-methyl-1,2,4-oxadiazol-3-yl)methyl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [101];

1-(2-hydroxy-2-methylpropyl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl) piperidine-4-carboxamide [102];

tert-butyl 2-(4-((2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)carbamoyl)piperidin-1-yl)acetate [103];

2-(4-((2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)carbamoyl)piperidin-1-yl)acetic acid [104];

2-(4-methyl-1,4-diazepan-1-yl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl) acetamide [105];

tert-butyl (2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)carbamate [106];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)but-2-ynamide [107];

trans-4-((2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)carbamoyl)cyclohexane-1-carboxylic acid [108];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-3-morpholinopropanamide [109];

trans-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-3-morpholinocyclobutane-1-carboxamide [110];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)quinuclidine-4-carboxamide [111];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(piperidin-1-yl)propanamide [112];

1-isobutyl-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)azepane-4-carboxamide [113];

2-(4-methoxypiperidin-1-yl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)acetamide [114];

2-(4-hydroxypiperidin-1-yl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)acetamide [115];

3-(hydroxymethyl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)bicyclo[1.1.1]pentane-1-carboxamide [116];

1-methyl-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)azepane-4-carboxamide [117];

trans-4-(dimethylamino)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)cyclohexane-1-carboxamide [118];

trans-4-(bis(methyl-d 3 )amino)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl) cyclohexane-1-carboxamide [119];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-3-((4-methylpiperazin-1-yl)methyl) bicyclo[1.1.1]pentane-1-carboxamide [120];

methyl trans-4-((2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)carbamoyl)cyclohexane-1-carboxylate [121];

2-(1-isobutylpyrrolidin-3-yl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)acetamide [122];

trans-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-4-(4-methylpiperazine-1-carbonyl)cyclohexane-1-carboxamide [123];

1-isobutyl-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [124];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-1-(phenylsulfonyl)piperidine-4-carboxamide [125];

8-methyl-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-3,8-diazabicyclo[3.2.1]octane-3-carboxamide [126];

3-methyl-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-3,8-diazabicyclo[3.2.1]octane-8-carboxamide [127];

(1R,3s,5S)-3-amino-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-8-azabicyclo[3.2.1] octane-8-carboxamide [128];

(1R,3s,5S)—N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-3-((3,3,3-trifluoropropyl) amino)-8-azabicyclo[3.2.1]octane-8-carboxamide [129];

(1R,3s,5S)-3-((1,3-difluoropropan-2-yl)amino)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-8-azabicyclo[3.2.1]octane-8-carboxamide [130];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)morpholine-4-carboxamide [131];

4-(dimethylamino)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)piperidine-1-carboxamide [132];

(S)-2,4-dimethyl-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)piperazine-1-carboxamide [133];

1-methyl-3-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-1-(1-methylpiperidin-4-yl)urea [134];

1-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-3-(1-methylpiperidin-4-yl)urea [135];

4-isopropyl-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)piperazine-1-carboxamide [136];

(R)-3,4-dimethyl-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)piperazine-1-carboxamide [137];

N-(2-(1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [138];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-3-(piperazin-1-yl)benzamide [139];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-3-(4-methylpiperazin-1-yl)benzamide [140];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-3-(pyrrolidin-1-ylmethyl)benzamide [141];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-3-(piperidin-4-yloxy)benzamide [142];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-3-((1-methylpiperidin-4-yl)oxy) benzamide [143];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-4-(piperidin-4-yloxy)benzamide [144];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-4-((1-methylpiperidin-4-yl)oxy) benzamide [145];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(piperazin-1-yl)isonicotinamide [146];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [147];

2-(4-isopropylpiperazin-1-yl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl) isonicotinamide [148];

2-(4-cyclopropylpiperazin-1-yl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl) isonicotinamide [149];

2-(4-(2-fluoroethyl)piperazin-1-yl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl) isonicotinamide [150];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-6-(4-methylpiperazin-1-yl)nicotinamide [151];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-5-(piperidin-4-yloxy)nicotinamide [152];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(piperidin-4-yloxy)isonicotinamide [153];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-((1-methylpiperidin-4-yl)oxy) isonicotinamide [154];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-5-(piperidin-4-ylamino)nicotinamide [155];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-5-((1-methylpiperidin-4-yl)amino) nicotinamide [156];

2-(4-aminopiperidin-1-yl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl) isonicotinamide [157];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(4-(methylamino)piperidin-1-yl) isonicotinamide [158];

2-(4-(dimethylamino)piperidin-1-yl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl) isonicotinamide [159];

2-((1-isopropylpiperidin-4-yl)oxy)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl) isonicotinamide [160];

2-(3-aminoazetidin-1-yl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl) isonicotinamide [161];

2-(3-(dimethylamino)azetidin-1-yl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl) isonicotinamide [162];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-morpholinoisonicotinamide [163];

2-((2-(dimethylamino)ethyl)amino)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl) isonicotinamide [164];

2-(2-(dimethylamino)ethoxy)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl) isonicotinamide [165];

2-(4-isobutylpiperazin-1-yl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl) isonicotinamide [166];

2-(azetidin-3-yloxy)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)isonicotinamide [167];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-((1-methylazetidin-3-yl)oxy) isonicotinamide [168];

2-(4-ethylpiperazin-1-yl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl) isonicotinamide [169];

4-((dimethylamino)methyl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)benzamide [170];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-3-(1-methylpiperidin-4-yl)benzamide [171];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-3-((4-methylpiperazin-1-yl)methyl) benzamide [172];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)isonicotinamide [173];

2-hydroxy-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)isonicotinamide [174];

2-isopropoxy-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)isonicotinamide [175];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(1-methylpiperidin-4-yl) isonicotinamide [176];

1′-methyl-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-1′,2′,3′,6′-tetrahydro-[2,4′-bipyridine]-4-carboxamide [177];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(4-(6-(4-methylpiperazin-1-yl) nicotinoyl)piperazin-1-yl)isonicotinamide [178];

2-(4-hydroxy-4-methyl-4λ 4 -piperazin-1-yl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)isonicotinamide [179];

2-methyl-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-6-(4-methylpiperazin-1-yl) isonicotinamide [180];

3-methyl-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [181];

2-(4-methyl-1,4-diazepan-1-yl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl) isonicotinamide [182];

2-((2S,6R)-2,6-dimethylmorpholino)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl) isonicotinamide [183];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(2,7-diazaspiro[3.5]nonan-2-yl) isonicotinamide [184];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(7-methyl-2,7-diazaspiro[3.5]nonan-2-yl)isonicotinamide [185];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(2,7-diazaspiro[3.5]nonan-7-yl) isonicotinamide [186];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(2-methyl-2,7-diazaspiro[3.5]nonan-7-yl)isonicotinamide [187];

2-(methyl(1-methylpiperidin-4-yl)amino)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)isonicotinamide [188];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-((1-methylpiperidin-4-yl)thio) isonicotinamide [189];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl)pyrimidine-4-carboxamide [190];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-6-(4-methylpiperazin-1-yl)pyridazine-4-carboxamide [191];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-6-(4-methylpiperazin-1-yl)pyrimidine-4-carboxamide [192];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-phenylacetamide [193];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-3-phenylpropanamide [194];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(pyridin-3-yl)acetamide [195];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-3-(pyridin-3-yl)propanamide [196];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(pyridin-4-yl)acetamide [197];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-3-(pyridin-4-yl)propanamide [198];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)isoindoline-5-carboxamide [199];

2-methyl-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)isoindoline-5-carboxamide [200];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-1,2,3,4-tetrahydroisoquinoline-7-carboxamide [201];

2-methyl-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-1,2,3,4-tetrahydroisoquinoline-7-carboxamide [202];

2-methyl-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-1,2,3,4-tetrahydroisoquinoline-6-carboxamide [203];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-1,2,3,4-tetrahydroisoquinoline-6-carboxamide [204];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-1H-indole-5-carboxamide [205];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)benzofuran-5-carboxamide [206];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)furo[2,3-c]pyridine-5-carboxamide [207];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)benzo[b]thiophene-5-carboxamide [208];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)benzofuran-6-carboxamide [209];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)benzo[d]oxazole-6-carboxamide [210];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)benzo[d]thiazole-6-carboxamide [211];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)benzo[d]oxazole-5-carboxamide [212];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)benzo[d]thiazole-5-carboxamide [213];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)quinoline-3-carboxamide [214];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)quinoline-6-carboxamide [215];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)quinoxaline-6-carboxamide [216];

5-chloro-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [217];

3-chloro-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [218];

2-(2,5-diazabicyclo [2.2.1]heptan-2-yl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)isonicotinamide [219];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(5-methyl-2,5-diazabicyclo[2.2.1] heptan-2-yl)isonicotinamide [220];

3-fluoro-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [221];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-((4-methylpiperazin-1-yl)methyl) isonicotinamide [222];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(morpholinomethyl)isonicotinamide [223];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(pyrrolidin-1-ylmethyl) isonicotinamide [224];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(2-(4-methylpiperazin-1-yl)pyridin-4-yl)acetamide [225];

1-methyl-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-1H-indazole-5-carboxamide [226];

1-methyl-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-1H-benzo[d]imidazole-5-carboxamide [227];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-1-(piperidin-4-yl)-1H-pyrazole-4-carboxamide [228];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-1-(1-methylpiperidin-4-yl)-1H-pyrazole-4-carboxamide [229];

1-(1-ethylpiperidin-4-yl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-1H-pyrazole-4-carboxamide [230];

1-(1-(2-fluoroethyl)piperidin-4-yl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-1H-pyrazole-4-carboxamide [231];

1-(1-isopropylpiperidin-4-yl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-1H-pyrazole-4-carboxamide [232];

1-(1-cyclopropylpiperidin-4-yl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-1H-pyrazole-4-carboxamide [233];

isopropyl 4-(4-((2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)carbamoyl)-1H-pyrazol-1-yl)piperidine-1-carboxylate [234];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-1-(piperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide [235];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-1-(1-methylpiperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide [236];

1-(1-(2-fluoroethyl)piperidin-4-yl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-1H-1,2,3-triazole-4-carboxamide [237];

1-(1-isopropylpiperidin-4-yl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-1H-1,2,3-triazole-4-carboxamide [238];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl)oxazole-5-carboxamide [239];

2-(3-(dimethylamino)azetidin-1-yl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl) oxazole-4-carboxamide [240];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(piperidin-4-yl)oxazole-4-carboxamide [241];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(1-methylpiperidin-4-yl)oxazole-4-carboxamide [242];

2-(1-(2-fluoroethyl)piperidin-4-yl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl) oxazole-4-carboxamide [243];

2-(1-isopropylpiperidin-4-yl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)oxazole-4-carboxamide [244];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl)oxazole-4-carboxamide [245];

2-(3-(dimethylamino)azetidin-1-yl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl) thiazole-5-carboxamide [246];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(piperidin-4-yl)thiazole-4-carboxamide [247];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl)thiazole-4-carboxamide [248];

2-(1-(2-fluoroethyl)piperidin-4-yl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl) thiazole-4-carboxamide [249];

2-(1-isopropylpiperidin-4-yl)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)thiazole-4-carboxamide [250];

1-methyl-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl-8-d)piperidine-4-carboxamide [251];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-1-(2-(methyl-d 3 )propyl-1,1,2,3,3,3-d 6 ) piperidine-4-carboxamide [252];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(pyrrolidin-1-yl-2,2,5,5-d 4 )acetamide [253];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(4-(methyl-d 3 )piperazin-1-yl) acetamide [254];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(morpholino-d 8 )acetamide [255];

(S)—N-(2-(1-(methyl-d 3 )-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(pyrrolidin-1-yl)propanamide [256];

1-isobutyl-N-(2-(1-(methyl-d 3 )-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [257];

N-(2-(1-(methyl-d 3 )-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl) acetamide [258];

N-(2-(1-(methyl-d 3 )-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(pyrrolidin-1-yl)acetamide [259];

N-(2-(1-(methyl-d 3 )-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(piperidin-1-yl)acetamide [260];

N-(2-(1-(methyl-d 3 )-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [261];

N-(2-(1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(4-(methyl-d 3 )piperazin-1-yl)isonicotinamide [262];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(4-(methyl-d 3 )piperazin-1-yl) isonicotinamide [263];

N-(2-(1-(methyl-d 3 )-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [264];

N-(2-(1-(methyl-d 3 )-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(4-(methyl-d 3 )piperazin-1-yl) isonicotinamide [265];

N-(2-(1-(methyl-d 3 )-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-1-(piperidin-4-yl)-1H-pyrazole-4-carboxamide [266];

N-(2-(1-(methyl-d 3 )-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-1-(1-methylpiperidin-4-yl)-1H-pyrazole-4-carboxamide [267];

N-(2-(1-(methyl-d 3 )-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(piperidin-4-yl)oxazole-4-carboxamide [268];

N-(2-(1-(methyl-d 3 )-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(1-methylpiperidin-4-yl)oxazole-4-carboxamide [269];

N-(2-(1-ethyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(pyrrolidin-1-yl)acetamide [270];

N-(2-(1-cyclopropyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(pyrrolidin-1-yl)acetamide [271];

N-(2-(1-cyclopropyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [272];

N-(2-(1-(1-methylpiperidin-4-yl)-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl) cyclohexanecarboxamide [273];

2-(pyrrolidin-1-yl)-N-(2-(5-(trifluoromethyl)-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)acetamide [274];

N-(2-(5-(hydroxymethyl)-1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-1-methylpiperidine-4-carboxamide [275];

N-(2-(5-(hydroxymethyl)-1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)tetrahydro-2H-pyran-4-carboxamide [276];

N-(2-(1-isopropyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-3-(piperidin-4-yloxy)benzamide [294];

N-(2-(1-isopropyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-3-((1-methylpiperidin-4-yl)oxy) benzamide [295];

N-(2-(1-isopropyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-4-(piperidin-4-yloxy)benzamide [296];

N-(2-(1-cyclopropyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [297];

4-fluoro-N-(2-(1-(1-methylpiperidin-4-yl)-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)benzamide [298];

4-(difluoromethoxy)-N-(2-(1-(1-methylpiperidin-4-yl)-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl) benzamide [299];

5-fluoro-N-(2-(1-(1-methylpiperidin-4-yl)-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)nicotinamide [300];

N 2 -methyl-N 5 -(2-(1-(1-methylpiperidin-4-yl)-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)pyridine-2,5-dicarboxamide [301];

1-isopropyl-N-(2-(1-(1-methylpiperidin-4-yl)-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-1H-pyrazole-4-carboxamide [302];

2-methyl-N-(2-(1-(1-methylpiperidin-4-yl)-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)thiazole-5-carboxamide [303];

N-(2-(5-amino-1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [304];

4-(difluoromethoxy)-N-(2-(5-(hydroxymethyl)-1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl) benzamide [305];

N-(2-(5-(hydroxymethyl)-1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [306];

N-(2-(5-(hydroxymethyl)-1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(7-methyl-2,7-diazaspiro[3.5]nonan-2-yl)isonicotinamide [307];

4-fluoro-N-(2-(1-methyl-5-(pyrrolidin-1-ylmethyl)-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl) benzamide [308];

4-fluoro-N-(2-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl) benzamide [309];

4-(difluoromethoxy)-N-(2-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)benzamide [310];

N-(2-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-3-(pyrrolidin-1-ylmethyl)benzamide [311];

N-(2-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(7-methyl-2,7-diazaspiro[3.5]nonan-2-yl)isonicotinamide [312];

N-(2-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-morpholinoisonicotinamide [313];

N-(2-(1-methyl-5-(morpholinomethyl)-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-morpholinoisonicotinamide [314];

N-(2-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)-1,6-naphthyridin-7-yl)-1-((1-(trifluoromethyl)cyclopropyl)methyl)piperidine-4-carboxamide [315];

3,3-difluoro-N-(2-(5-methyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)-1,6-naphthyridin-7-yl)cyclobutane-1-carboxamide [316];

N-((4,4-difluorocyclohexyl)methyl)-2-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a] pyrazin-3-yl)-1,6-naphthyridin-7-amine [317];

N-(2-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)-1,6-naphthyridin-7-yl)-1-((1-(trifluoromethyl)cyclopropyl)methyl)piperidine-4-carboxamide [318];

N-(2-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)-1,6-naphthyridin-7-yl)-2-(pyrrolidin-1-yl)acetamide [319];

2-(7-azabicyclo[2.2.1]heptan-7-yl)-N-(2-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)-1,6-naphthyridin-7-yl)acetamide [320];

(R)—N-(2-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)-1,6-naphthyridin-7-yl)-1-isobutylpiperidine-3-carboxamide [321];

N-(2-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)-1,6-naphthyridin-7-yl) piperidine-4-carboxamide [322];

4-fluoro-N-(2-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)-1,6-naphthyridin-7-yl)-1-isobutylpiperidine-4-carboxamide [323];

N-(2-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl)acetamide [324];

4-fluoro-N-(2-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)-1,6-naphthyridin-7-yl)benzamide [325];

N-(2-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)-1,6-naphthyridin-7-yl)-3-(4-methylpiperazin-1-yl)benzamide [326];

N 5 -(2-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)-1,6-naphthyridin-7-yl)-N 2 -methylpyridine-2,5-dicarboxamide [327];

N-(2-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)-1,6-naphthyridin-7-yl)-6-(4-methylpiperazin-1-yl)nicotinamide [328];

2-(azetidin-3-yloxy)-N-(2-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-1,6-naphthyridin-7-yl)isonicotinamide [329];

N-(2-(1-methyl-1H-pyrazol-5-yl)-1,6-naphthyridin-7-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [330];

1-methyl-N-(2-(1-methyl-1H-pyrazol-3-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [331];

N-(2-(1-methyl-1H-pyrazol-3-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [332];

2-fluoro-2-methyl-N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)propanamide [333];

2,2,3,3-tetramethyl-N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)cyclopropane-1-carboxamide [334];

trans-N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)-4-(pyrrolidin-1-yl) cyclohexane-1-carboxamide [335];

trans-N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)-4-morpholinocyclohexane-1-carboxamide [336];

N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)-2-(piperidin-1-yl)acetamide [337];

1-ethyl-4-fluoro-N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [338];

4-fluoro-1-isobutyl-N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [339];

N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [340];

N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)cyclopropanecarboxamide [341];

4,4-difluoro-N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)cyclohexane-1-carboxamide [342];

trans-4-(dimethylamino)-N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl) cyclohexane-1-carboxamide [343];

trans-N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)-4-((4-methylpiperazin-1-yl) methyl)cyclohexane-1-carboxamide [344];

N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [345];

1-isobutyl-N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [346];

N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)-1-((1-(trifluoromethyl)cyclopropyl) methyl)piperidine-4-carboxamide [347];

N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)-1-((3-methyloxetan-3-yl)methyl) piperidine-4-carboxamide [348];

N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)-1-(2-(pyrrolidin-1-yl)acetyl) piperidine-4-carboxamide [349];

1′-methyl-N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)-[1,4′-bipiperidine]-4-carboxamide [350];

(R)—N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)piperidine-3-carboxamide [351];

(R)-1-isobutyl-N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)piperidine-3-carboxamide [352];

N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)-2-(pyrrolidin-1-yl)acetamide [353];

N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl) acetamide [354];

2-(7-azabicyclo[2.2.1]heptan-7-yl)-N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl) acetamide [355];

1-(2-hydroxy-2-methylpropyl)-N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl) piperidine-4-carboxamide [356];

N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)-2-morpholinoacetamide [357];

2-(4-methoxypiperidin-1-yl)-N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl) acetamide [358];

N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)morpholine-4-carboxamide [359];

N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)-1-(piperidin-4-yl)-1H-pyrazole-4-carboxamide [360];

N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)-1-(1-methylpiperidin-4-yl)-1H-pyrazole-4-carboxamide [361];

1-(1-ethylpiperidin-4-yl)-N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)-1H-pyrazole-4-carboxamide [362];

1-(1-isopropylpiperidin-4-yl)-N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)-1H-pyrazole-4-carboxamide [363];

N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)-1H-1,2,3-triazole-4-carboxamide [364];

1-(1-(2-fluoroethyl)piperidin-4-yl)-N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)-1H-1,2,3-triazole-4-carboxamide [365];

1-(1-isopropylpiperidin-4-yl)-N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)-1H-1,2,3-triazole-4-carboxamide [366];

N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)-2-(piperidin-4-yl)oxazole-4-carboxamide [367];

N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)-2-(1-methylpiperidin-4-yl)oxazole-4-carboxamide [368];

2-(1-isopropylpiperidin-4-yl)-N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl) oxazole-4-carboxamide [369];

2-fluoro-N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)benzamide [370];

N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)-3-((1-methylpiperidin-4-yl)oxy) benzamide [371];

N 2 -methyl-N 5 -(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)pyridine-2,5-dicarboxamide [372];

N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)-6-(4-methylpiperazin-1-yl) nicotinamide [373];

2-(3-(dimethylamino)azetidin-1-yl)-N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl) isonicotinamide [374];

N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)-2-(1-methylpiperidin-4-yl) isonicotinamide [375];

2-(4-(dimethylamino)piperidin-1-yl)-N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)isonicotinamide [376];

N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)-2-morpholinoisonicotinamide [377];

N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [378];

2-(4-methyl-1,4-diazepan-1-yl)-N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl) isonicotinamide [379];

2-(4-isopropylpiperazin-1-yl)-N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl) isonicotinamide [380];

N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)-2-(piperidin-4-ylamino) isonicotinamide [381];

2-(methyl(1-methylpiperidin-4-yl)amino)-N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)isonicotinamide [382];

N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)-2-((1-methylpiperidin-4-yl)thio) isonicotinamide [383];

2-methyl-N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)-1,2,3,4-tetrahydroisoquinoline-6-carboxamide [384];

N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)-2-(piperazin-1-yl)isonicotinamide [385];

N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)-2-(2-(4-methylpiperazin-1-yl) pyridin-4-yl)acetamide [386];

1,1-bis(methyl-d 3 )-4-(4-((2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)carbamoyl) pyridin-2-yl)piperazin-1-ium [387];

N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)-2-(4-(methyl-d3)piperazin-1-yl) isonicotinamide [388];

N-(2-(1-methyl-1H-1,2,3-triazol-5-yl)-1,6-naphthyridin-7-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [389];

N-(2-(4-methyl-4H-1,2,4-triazol-3-yl)-1,6-naphthyridin-7-yl)-2-morpholinoacetamide [390];

N-(2-(4-methyl-4H-1,2,4-triazol-3-yl)-1,6-naphthyridin-7-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [391];

4-fluoro-1-isobutyl-N-(2-(4-methyl-4H-1,2,4-triazol-3-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [392];

N-(2-(4,5-dimethyl-4H-1,2,4-triazol-3-yl)-1,6-naphthyridin-7-yl)-2-morpholinoacetamide [393];

N-(2-(4,5-dimethyl-4H-1,2,4-triazol-3-yl)-1,6-naphthyridin-7-yl)-1-(3,3,3-trifluoropropyl) piperidine-4-carboxamide [394];

N-(2-(1H-1,2,3-triazol-1-yl)-1,6-naphthyridin-7-yl)-4-fluoro-1-isobutylpiperidine-4-carboxamide [395];

N-(2-(2H-1,2,3-triazol-2-yl)-1,6-naphthyridin-7-yl)-4-fluoro-1-isobutylpiperidine-4-carboxamide [396];

N-(2-(1H-1,2,4-triazol-1-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [397];

1-isobutyl-N-(2-(1-methyl-1H-tetrazol-5-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [398];

2,2,3,3-tetramethyl-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)cyclopropane-1-carboxamide [399];

4,4-difluoro-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)cyclohexane-1-carboxamide [400];

N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-2-(piperidin-1-yl)acetamide [401];

2-fluoro-2-methyl-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)propanamide [402];

1-fluoro-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)cyclopropane-1-carboxamide [403];

2-methyl-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-2-azaspiro [3.3]heptane-6-carboxamide [404];

1-fluoro-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)cyclohexane-1-carboxamide [405];

trans-4-methoxy-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)cyclohexane-1-carboxamide [406];

trans-4-(hydroxymethyl)-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)cyclohexane-1-carboxamide [407];

N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)azetidine-3-carboxamide [408];

(R)—N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)tetrahydrofuran-2-carboxamide [409];

1-(2-methoxyethyl)-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [410];

N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [411];

1-isobutyl-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [412];

N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-1-(methylsulfonyl)piperidine-4-carboxamide [413];

N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-2-(pyrrolidin-1-yl)propanamide [414];

2-isopropoxy-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)acetamide [415];

3-isopropoxy-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)propanamide [416];

N-(2-(1,2-dimethyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)cyclopropanecarboxamide [417];

N-(2-(1,2-dimethyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)cyclohexanecarboxamide [418];

N-(2-(1,2-dimethyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-4,4-difluorocyclohexane-1-carboxamide [419];

(S)—N-(2-(1,2-dimethyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)tetrahydrofuran-2-carboxamide [420];

N-(2-(1,2-dimethyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-3,3-difluorocyclobutane-1-carboxamide [421];

N-(2-(1,2-dimethyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-1-fluorocyclopropane-1-carboxamide [422];

N-(2-(1,2-dimethyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)morpholine-4-carboxamide [423];

N-(2-(1,2-dimethyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)morpholine-d 8 -4-carboxamide [424];

1-methyl-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-1H-pyrazole-4-carboxamide [425];

1-ethyl-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-1H-pyrazole-4-carboxamide [426];

1-isopropyl-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-1H-pyrazole-4-carboxamide [427];

1-cyclopropyl-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-1H-pyrazole-4-carboxamide [428];

N-(2-(5-(azetidin-1-ylmethyl)-1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-4,4-difluorocyclohexane-1-carboxamide [277];

4,4-difluoro-N-(2-(1-methyl-5-(pyrrolidin-1-ylmethyl)-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl) cyclohexane-1-carboxamide [278];

4,4-difluoro-N-(2-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl) cyclohexane-1-carboxamide [279];

2-(2-fluoroethyl)-N-(2-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-azaspiro[3.3]]heptane-6-carboxamide [280];

tert-butyl 6-((2-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)carbamoyl)-2-azaspiro[3.3]heptane-2-carboxylate [281];

2-fluoro-2-methyl-N-(2-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)propanamide [282];

2-(diethylamino)-N-(2-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)acetamide [283];

trans-4-methoxy-N-(2-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)cyclohexane-1-carboxamide [284];

trans-4-(hydroxymethyl)-N-(2-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)cyclohexane-1-carboxamide [285];

(R)—N-(2-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)pyrrolidine-2-carboxamide [286];

1-isobutyl-N-(2-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl) piperidine-4-carboxamide [287];

N-(2-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-1-(oxetan-3-yl)piperidine-4-carboxamide [288];

1-benzoyl-N-(2-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl) piperidine-4-carboxamide [289];

N-(2-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)tetrahydro-2H-pyran-4-carboxamide [290];

N-(2-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperidin-1-yl)acetamide [291];

N-(2-(1-(difluoromethyl)-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [292];

N-(2-(1-ethyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [293];

1-isobutyl-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-1H-pyrazole-4-carboxamide [429];

1-methyl-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-1H-pyrazole-3-carboxamide [430];

N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-2-(1-methyl-1H-pyrazol-4-yl) acetamide [431];

1-methyl-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-1H-imidazole-4-carboxamide [432];

1-isopropyl-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-1H-imidazole-4-carboxamide [433];

N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-1-(tetrahydro-2H-pyran-4-yl)-1H-imidazole-4-carboxamide [434];

1,2-dimethyl-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-1H-imidazole-5-carboxamide [435];

1-methyl-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-1H-1,2,4-triazole-3-carboxamide [436];

2-methyl-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)oxazole-4-carboxamide [437];

2-isopropyl-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)oxazole-4-carboxamide [438];

4-methyl-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)oxazole-2-carboxamide [439];

4-methyl-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)thiazole-2-carboxamide [440];

2-methyl-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)thiazole-4-carboxamide [441];

5-methyl-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-1,3,4-oxadiazole-2-carboxamide [442];

5-methyl-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-1,3,4-thiadiazole-2-carboxamide [443];

1-isopropyl-N-(2-(1-isopropyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-1H-pyrazole-4-carboxamide [444];

N-(2-(1,2-dimethyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-1-methyl-1H-pyrazole-4-carboxamide [445];

N-(2-(1,2-dimethyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-1-isopropyl-1H-pyrazole-4-carboxamide [446];

N-(2-(1,2-dimethyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-2-methylthiazole-5-carboxamide [447];

4-fluoro-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)benzamide [448];

4-(difluoromethoxy)-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)benzamide [449];

N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-3-(pyrrolidin-1-ylmethyl)benzamide [450];

2-fluoro-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)benzamide-3,4,5,6-d 4 [451];

4-fluoro-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)benzamide-2,3,5,6-d 4 [452];

2-chloro-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)benzamide-3,4,5,6-d 4 [453];

4-chloro-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)benzamide-2,3,5,6-d 4 [454];

4-(methyl-d 3 )—N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)benzamide [455];

4-methyl-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)benzamide-2,3,5,6-d 4 [456];

4-(methyl-d 3 )—N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)benzamide-2,3,5,6-d 4 [257];

4-(methoxy-d 3 )—N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)benzamide [458];

4-(methoxy-d 3 )—N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)benzamide-2,3,5,6-d 4 [459];

4-methoxy-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)benzamide-2,3,5,6-d 4 [460];

(E)-N-(2-(1,2-dimethyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-3-(phenyl-2,3,4,5,6-d 5 ) acrylamide [461];

(E)-N-(2-(1,2-dimethyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-3-(phenyl-2,3,4,5,6-d 5 ) acrylamide-2,3-d 2 [462];

N-(2-(1,2-dimethyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-2-(4-fluorophenyl)acetamide-2,2-d 2 [463];

(E)-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-3-(phenyl-2,3,4,5,6-d 5 )acrylamide [464];

(E)-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-3-(phenyl-2,3,4,5,6-d 5 )acrylamide-2,3-d 2 [465];

2-(4-fluorophenyl)-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)acetamide-2,2-d 2 [466];

N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [467];

2-(dimethylamino)-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)isonicotinamide [468];

2-(3-aminoazetidin-1-yl)-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl) isonicotinamide [469];

N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-2-(pyrrolidin-1-yl)isonicotinamide [470];

N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-2-(piperidin-1-yl)isonicotinamide [471];

N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-2-morpholinoisonicotinamide [472];

2-(4-isopropylpiperazin-1-yl)-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl) isonicotinamide [473];

2-(4-cyclopropylpiperazin-1-yl)-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl) isonicotinamide [474];

N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-2-(2,7-diazaspiro[3.5]nonan-2-yl) isonicotinamide [475];

N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-2-(7-methyl-2,7-diazaspiro[3.5]nonan-2-yl)isonicotinamide [476];

N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)isoindoline-5-carboxamide [477];

2-methyl-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)isoindoline-5-carboxamide [478];

2-(azetidin-1-yl)-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)isonicotinamide [479];

2-methoxy-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)isonicotinamide [480];

2-methyl-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)isonicotinamide [481];

2-cyano-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)isonicotinamide [482];

2-(3,3-difluoroazetidin-1-yl)-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl) isonicotinamide [483];

2-(4,4-difluoropiperidin-1-yl)-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl) isonicotinamide [484];

2-isopropoxy-N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)isonicotinamide [485];

N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-2-(pyrrolidin-1-yl-2,2,5,5-d 4 ) isonicotinamide [486];

N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-2-(pyrrolidin-1-yl-d 8 )isonicotinamide [487];

N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-2-(piperidin-1-yl-d 10 )isonicotinamide [488];

N-(2-(1-methyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-2-(morpholino-d 8 )isonicotinamide [489];

N-(2-(1,2-dimethyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-4-isopropoxybenzamide [490];

N-(2-(1,2-dimethyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-4-(piperidin-4-yloxy)benzamide [491];

4-(benzyloxy)-N-(2-(1,2-dimethyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)benzamide [492];

N-(2-(1,2-dimethyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-2-fluorobenzamide-3,4,5,6-d 4 [493];

N-(2-(1,2-dimethyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-4-fluorobenzamide-2,3,5,6-d 4 [494];

2-chloro-N-(2-(1,2-dimethyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)benzamide-3,4,5,6-d 4 [495];

4-chloro-N-(2-(1,2-dimethyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)benzamide-2,3,5,6-d 4 [496];

N-(2-(1,2-dimethyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-4-(methyl-d 3 )benzamide [497];

N-(2-(1,2-dimethyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-4-methylbenzamide-2,3,5,6-d 4 [498];

N-(2-(1,2-dimethyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-4-(methyl-d 3 )benzamide-2,3,5,6-d 4 [499];

N-(2-(1,2-dimethyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-4-(methoxy-d 3 )benzamide [500];

N-(2-(1,2-dimethyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-4-(methoxy-d 3 )benzamide-2,3,5,6-d 4 [501];

N-(2-(1,2-dimethyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-4-methoxybenzamide-2,3,5,6-d 4 [502];

N-(2-(1,2-dimethyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [503];

N-(2-(1,2-dimethyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-2-morpholinoisonicotinamide [504];

N-(2-(1,2-dimethyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-2-(pyrrolidin-1-yl)isonicotinamide [505];

N-(2-(1,2-dimethyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-2-(dimethylamino)isonicotinamide [506];

N-(2-(1,2-dimethyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-2-(pyrrolidin-1-yl-2,2,5,5-d 4 ) isonicotinamide [507];

N-(2-(1,2-dimethyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-2-(pyrrolidin-1-yl-d 8 ) isonicotinamide [508];

N-(2-(1,2-dimethyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-2-(piperidin-1-yl-d 10 ) isonicotinamide [509];

N-(2-(1,2-dimethyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-2-(morpholino-d 8 )isonicotinamide [510];

N-(2-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-1,6-naphthyridin-7-yl) cyclopropanecarboxamide [511];

N-(2-(7-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-1,6-naphthyridin-7-yl) cyclopropanecarboxamide [512];

3,3-difluoro-N-(2-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-1,6-naphthyridin-7-yl) cyclobutane-1-carboxamide [513];

(R)—N-(2-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-1,6-naphthyridin-7-yl)pyrrolidine-2-carboxamide [514];

(R)—N-(2-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-1,6-naphthyridin-7-yl)piperidine-3-carboxamide [515];

1-methyl-N-(2-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [516];

N-(2-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-1,6-naphthyridin-7-yl)-1-((1-(trifluoromethyl)cyclopropyl)methyl)piperidine-4-carboxamide [517];

1-benzoyl-N-(2-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [518];

4-fluoro-1-isobutyl-N-(2-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-1,6-naphthyridin-7-yl) piperidine-4-carboxamide [519];

(R)-2-(2-methylpyrrolidin-1-yl)-N-(2-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-1,6-naphthyridin-7-yl)acetamide [520];

2-(cyclobutyl(methyl)amino)-N-(2-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-1,6-naphthyridin-7-yl)acetamide [521];

4-fluoro-N-(2-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-1,6-naphthyridin-7-yl)benzamide [522];

4-isopropoxy-N-(2-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-1,6-naphthyridin-7-yl) benzamide [523];

4-(difluoromethoxy)-N-(2-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-1,6-naphthyridin-7-yl) benzamide [524];

2-((2-(dimethylamino)ethyl)amino)-N-(2-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-1,6-naphthyridin-7-yl)isonicotinamide [525];

2-((1-isopropylpiperidin-4-yl)oxy)-N-(2-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-1,6-naphthyridin-7-yl)isonicotinamide [526];

N-(2-(oxazol-5-yl)-1,6-naphthyridin-7-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [527];

N-(2-(oxazol-5-yl)-1,6-naphthyridin-7-yl)cyclopropanecarboxamide [528];

(R)—N-(2-(oxazol-5-yl)-1,6-naphthyridin-7-yl)tetrahydrofuran-2-carboxamide [529];

(R)—N-(2-(oxazol-5-yl)-1,6-naphthyridin-7-yl)piperidine-3-carboxamide [530];

N-(2-(oxazol-5-yl)-1,6-naphthyridin-7-yl)tetrahydro-2H-pyran-4-carboxamide [531];

N-(2-(oxazol-5-yl)-1,6-naphthyridin-7-yl)-1-(2-(pyrrolidin-1-yl)acetyl)piperidine-4-carboxamide [532];

1′-methyl-N-(2-(oxazol-5-yl)-1,6-naphthyridin-7-yl)-[1,4′-bipiperidine]-4-carboxamide [533];

cis-4-morpholino-N-(2-(oxazol-5-yl)-1,6-naphthyridin-7-yl)cyclohexane-1-carboxamide [534];

2-(cyclobutyl(methyl)amino)-N-(2-(oxazol-5-yl)-1,6-naphthyridin-7-yl)acetamide [535];

N-(2-(oxazol-5-yl)-1,6-naphthyridin-7-yl)-2-(pyrrolidin-1-yl)acetamide [536];

(R)-2-(2-methylpyrrolidin-1-yl)-N-(2-(oxazol-5-yl)-1,6-naphthyridin-7-yl)acetamide [537];

2-(4-methylpiperazin-1-yl)-N-(2-(oxazol-5-yl)-1,6-naphthyridin-7-yl)acetamide [538];

trans-4-((4-methylpiperazin-1-yl)methyl)-N-(2-(oxazol-5-yl)-1,6-naphthyridin-7-yl)cyclohexane-1-carboxamide [539];

1-(2,2-difluoropropyl)-N-(2-(oxazol-5-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [540];

trans-4-(hydroxymethyl)-N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl)cyclohexane-1-carboxamide [541];

trans-4-(methylamino)-N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl)cyclohexane-1-carboxamide [542];

trans-4-((1,3-difluoropropan-2-yl)amino)-N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl) cyclohexane-1-carboxamide [543];

trans-N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl)-4-((propan-2-yl-1,1,1,3,3,3-d 6 )amino) cyclohexane-1-carboxamide [544];

trans-4-((2,2-difluoroethyl)amino)-N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl) cyclohexane-1-carboxamide [545];

trans-N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl)-4-((3,3,3-trifluoropropyl)amino) cyclohexane-1-carboxamide [546];

trans-4-((2-methoxyethyl)amino)-N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl) cyclohexane-1-carboxamide [547];

trans-4-(dimethylamino)-N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl)cyclohexane-1-carboxamide [548];

trans-4-(bis(methyl-d 3 )amino)-N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl)cyclohexane-1-carboxamide [549];

cis-4-(dimethylamino)-N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl)cyclohexane-1-carboxamide [550];

trans-4-((2,2-difluoroethyl)(methyl)amino)-N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl) cyclohexane-1-carboxamide [551];

trans-4-(methyl(oxetan-3-yl)amino)-N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl) cyclohexane-1-carboxamide [552];

trans-4-((2-fluoroethyl)amino)-N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl)cyclohexane-1-carboxamide [553];

trans-4-(2-(fluoromethyl)aziridin-1-yl)-N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl) cyclohexane-1-carboxamide [554];

trans-4-((3-fluoroazetidin-1-yl)methyl)-N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl) cyclohexane-1-carboxamide [555];

trans-N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl)-3-morpholinocyclobutane-1-carboxamide [556];

trans-N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl)-4-morpholinocyclohexane-1-carboxamide [557];

N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl)-2-(piperidin-1-yl)acetamide [558];

2-(4-methoxypiperidin-1-yl)-N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl)acetamide [559];

N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl)acetamide [560];

N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl)morpholine-4-carboxamide [561];

N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl)-2-morpholinoacetamide [562];

N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl)-3-morpholinopropanamide [563];

1-methyl-N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [564];

1-(2,2-difluoropropyl)-N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [565];

N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl)-4-morpholinopiperidine-1-carboxamide [566];

4-((1,3-difluoropropan-2-yl)amino)-N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl) piperidine-1-carboxamide [567];

(1R,3s,5S)-3-((1,3-difluoropropan-2-yl)amino)-N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl)-8-azabicyclo[3.2.1]octane-8-carboxamide [568];

(1R,3s,5S)-3-((1,3-difluoropropan-2-yl)amino)-N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl)-8-azabicyclo[3.2.1]octane-8-carboxamide [569];

4-(dimethylamino)-N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl)piperidine-1-carboxamide [570];

4-((2,2-difluoroethyl)(methyl)amino)-N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl) piperidine-1-carboxamide [571];

(3S,4S)-4-amino-3-fluoro-N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl)piperidine-1-carboxamide [572];

(3S,4S)-3-fluoro-4-(methylamino)-N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl)piperidine-1-carboxamide [573];

(3R,4R)-4-amino-3-fluoro-N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl)piperidine-1-carboxamide [574];

(3R,4R)-3-fluoro-4-(methylamino)-N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl)piperidine-1-carboxamide [575];

4-((2-fluoroethyl)amino)-N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl)piperidine-1-carboxamide [576];

4-((2,2-difluoroethyl)amino)-N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl)piperidine-1-carboxamide [577];

(1R,3s,5S)-3-amino-N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl)-8-azabicyclo[3.2.1] octane-8-carboxamide [578];

(1R,3r,5S)-3-amino-N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl)-8-azabicyclo[3.2.1] octane-8-carboxamide [579];

(1R,3r,5S)-3-((2-fluoroethyl)amino)-N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl)-8-azabicyclo[3.2.1]octane-8-carboxamide [580];

(1R,3r,5S)-3-((2,2-difluoroethyl)amino)-N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl)-8-azabicyclo[3.2.1]octane-8-carboxamide [581];

(1R,3s,5S)—N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl)-3-((3,3,3-trifluoropropyl)amino)-8-azabicyclo[3.2.1]octane-8-carboxamide [582];

(3S,4S)-3-fluoro-4-(isopropylamino)-N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl) piperidine-1-carboxamide [583];

N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl)-5,6-dihydroimidazo[1,2-a]pyrazine-7(8H)-carboxamide [584];

2-methyl-N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl)-5,6-dihydroimidazo[1,2-a]pyrazine-7(8H)-carboxamide [585];

N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl)-2-(morpholino-d 8 )acetamide [586];

trans-N-(2-(2-methyloxazol-4-yl)-1,6-naphthyridin-7-yl)-4-(4-methylpiperazin-1-yl)cyclohexane-1-carboxamide [587];

N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl)-1-(1-methylpiperidin-4-yl)-1H-pyrazole-4-carboxamide [588];

2-(1H-imidazol-1-yl)-N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl)acetamide [589];

4-(difluoromethoxy)-N-(2-(oxazol-5-yl)-1,6-naphthyridin-7-yl)benzamide [590];

3-((1-methylpiperidin-4-yl)oxy)-N-(2-(oxazol-5-yl)-1,6-naphthyridin-7-yl)benzamide [591];

N-(2-(oxazol-5-yl)-1,6-naphthyridin-7-yl)isonicotinamide [592];

2-(3-aminoazetidin-1-yl)-N-(2-(oxazol-5-yl)-1,6-naphthyridin-7-yl)isonicotinamide [593];

2-(1-methylpiperidin-4-yl)-N-(2-(oxazol-5-yl)-1,6-naphthyridin-7-yl)isonicotinamide [594];

1′-methyl-N-(2-(oxazol-5-yl)-1,6-naphthyridin-7-yl)-1′,2′,3′,6′-tetrahydro-[2,4′-bipyridine]-4-carboxamide [595];

2-(4-methylpiperazin-1-yl)-N-(2-(oxazol-5-yl)-1,6-naphthyridin-7-yl)isonicotinamide [596];

2-(7-methyl-2,7-diazaspiro[3.5]nonan-2-yl)-N-(2-(oxazol-5-yl)-1,6-naphthyridin-7-yl) isonicotinamide [597];

N-(2-(oxazol-5-yl)-1,6-naphthyridin-7-yl)-2-(2,7-diazaspiro[3.5]nonan-7-yl)isonicotinamide [598];

N-(2-(oxazol-5-yl)-1,6-naphthyridin-7-yl)-2-(piperidin-4-ylamino)isonicotinamide [599];

2-methyl-N-(2-(oxazol-5-yl)-1,6-naphthyridin-7-yl)isoindoline-5-carboxamide [600];

N-(2-(oxazol-5-yl)-1,6-naphthyridin-7-yl)-1,2,3,4-tetrahydroisoquinoline-7-carboxamide [601];

N-(2-(2-methyloxazol-5-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [602];

N-(2-(3-methylisoxazol-5-yl)-1,6-naphthyridin-7-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [603];

4-fluoro-1-isobutyl-N-(2-(5-methyl-1,3,4-oxadiazol-2-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [604];

1-isobutyl-N-(2-(5-methyl-1,3,4-oxadiazol-2-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [605];

N-(2-(5-(dimethylamino)-1,3,4-oxadiazol-2-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [606];

N-(2-(5-(dimethylamino)-1,3,4-oxadiazol-2-yl)-1,6-naphthyridin-7-yl)-1-methylpiperidine-4-carboxamide [607];

N-(2-(5-methyl-1,3,4-oxadiazol-2-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [608];

3,3-difluoro-N-(2-(thiazol-5-yl)-1,6-naphthyridin-7-yl)cyclobutane-1-carboxamide [609];

2-methyl-N-(2-(thiazol-5-yl)-1,6-naphthyridin-7-yl)-2-azaspiro [3.3]heptane-6-carboxamide [610];

1-fluoro-N-(2-(thiazol-5-yl)-1,6-naphthyridin-7-yl)cyclohexane-1-carboxamide [611];

trans-4-(dimethylamino)-N-(2-(thiazol-5-yl)-1,6-naphthyridin-7-yl)cyclohexane-1-carboxamide [612];

trans-4-((3-fluoroazetidin-1-yl)methyl)-N-(2-(thiazol-5-yl)-1,6-naphthyridin-7-yl)cyclohexane-1-carboxamide [613];

N-(2-(thiazol-5-yl)-1,6-naphthyridin-7-yl)azetidine-3-carboxamide [614];

1-methyl-N-(2-(thiazol-5-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [615];

1-(2,2-difluoropropyl)-N-(2-(thiazol-5-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [616];

1-(oxetan-3-yl)-N-(2-(thiazol-5-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [617];

1-(2-(pyrrolidin-1-yl)acetyl)-N-(2-(thiazol-5-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [618];

1′-methyl-N-(2-(thiazol-5-yl)-1,6-naphthyridin-7-yl)-[1,4′-bipiperidine]-4-carboxamide [619];

2-(pyrrolidin-1-yl)-N-(2-(thiazol-5-yl)-1,6-naphthyridin-7-yl)propanamide [620];

2-(piperidin-1-yl)-N-(2-(thiazol-5-yl)-1,6-naphthyridin-7-yl)acetamide [621];

2-(4-methylpiperazin-1-yl)-N-(2-(thiazol-5-yl)-1,6-naphthyridin-7-yl)acetamide [622];

2-morpholino-N-(2-(thiazol-5-yl)-1,6-naphthyridin-7-yl)acetamide [623];

4-(piperidin-4-yloxy)-N-(2-(thiazol-5-yl)-1,6-naphthyridin-7-yl)benzamide [624];

N-(2-(thiazol-5-yl)-1,6-naphthyridin-7-yl)isonicotinamide [625];

6-(4-methylpiperazin-1-yl)-N-(2-(thiazol-5-yl)-1,6-naphthyridin-7-yl)nicotinamide [626];

1′-methyl-N-(2-(thiazol-5-yl)-1,6-naphthyridin-7-yl)-1′,2′,3′,6′-tetrahydro-[2,4′-bipyridine]-4-carboxamide [627];

2-(3-(dimethylamino)azetidin-1-yl)-N-(2-(thiazol-5-yl)-1,6-naphthyridin-7-yl)isonicotinamide [628];

2-(4-(dimethylamino)piperidin-1-yl)-N-(2-(thiazol-5-yl)-1,6-naphthyridin-7-yl)isonicotinamide [629];

2-(4-methylpiperazin-1-yl)-N-(2-(thiazol-5-yl)-1,6-naphthyridin-7-yl)isonicotinamide [630];

2-((1-methylpiperidin-4-yl)thio)-N-(2-(thiazol-5-yl)-1,6-naphthyridin-7-yl)isonicotinamide [631];

N-(2-(thiazol-5-yl)-1,6-naphthyridin-7-yl)-1,2,3,4-tetrahydroisoquinoline-7-carboxamide [632];

trans-4-((1,3-difluoropropan-2-yl)amino)-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)cyclohexane-1-carboxamide [633];

N-(2-(2-methylthiazol-5-yl)-1,6-naphthyridin-7-yl)morpholine-4-carboxamide [634];

N-(2-(2-methylthiazol-5-yl)-1,6-naphthyridin-7-yl)-2-(pyrrolidin-1-yl)acetamide [635];

2-((1R,4R)-2-oxa-5-azabicyclo [2.2.1]heptan-5-yl)-N-(2-(2-methylthiazol-5-yl)-1,6-naphthyridin-7-yl)acetamide [636];

N-(2-(2-methylthiazol-5-yl)-1,6-naphthyridin-7-yl)-2-morpholinoacetamide [637];

N-(2-(2-methylthiazol-5-yl)-1,6-naphthyridin-7-yl)-2-(morpholino-d 8 )acetamide [638];

2-(4-methylpiperazin-1-yl)-N-(2-(2-methylthiazol-5-yl)-1,6-naphthyridin-7-yl)acetamide [639];

1-methyl-N-(2-(2-methylthiazol-5-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [640];

N-(2-(2-methylthiazol-5-yl)-1,6-naphthyridin-7-yl)isonicotinamide [641];

N-(2-(2-methylthiazol-5-yl)-1,6-naphthyridin-7-yl)nicotinamide [642];

2-(4-methylpiperazin-1-yl)-N-(2-(2-methylthiazol-5-yl)-1,6-naphthyridin-7-yl)isonicotinamide [643];

trans-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-4-morpholinocyclohexane-1-carboxamide [644];

trans-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-4-(4-methylpiperazin-1-yl) cyclohexane-1-carboxamide [645];

4-isopropyl-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)piperazine-1-carboxamide [646];

4-((2-methoxyethyl)(methyl)amino)-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl) piperidine-1-carboxamide [647];

4-((1,3-difluoropropan-2-yl)amino)-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl) piperidine-1-carboxamide [648];

N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-4-((3,3,3-trifluoropropyl)amino) piperidine-1-carboxamide [649];

4-((2-fluoroethyl)amino)-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)piperidine-1-carboxamide [650];

(3R,4S)-4-amino-3-fluoro-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl) piperidine-1-carboxamide [651];

(3R,4R)-4-amino-3-fluoro-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl) piperidine-1-carboxamide [652];

(3S,4S)-3-fluoro-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-4-(methylamino) piperidine-1-carboxamide [653];

(3R,4R)-3-fluoro-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-4-(methylamino) piperidine-1-carboxamide [654];

4-amino-3,3-difluoro-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)piperidine-1-carboxamide [655];

(3R,4R)-3-fluoro-4-(isopropylamino)-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)piperidine-1-carboxamide [656];

(3R,4S)-3-fluoro-4-(isopropylamino)-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)piperidine-1-carboxamide [657];

3,3-difluoro-4-(isopropylamino)-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl) piperidine-1-carboxamide [658];

(3S,4S)-3-fluoro-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-4-((propan-2-yl-1,1,1,3,3,3-d 6 )amino)piperidine-1-carboxamide [659];

(1R,3s,5S)-3-((1,3-difluoropropan-2-yl)amino)-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-8-azabicyclo[3.2.1]octane-8-carboxamide [660];

(1R,3s,5S)-3-((1,3-difluoropropan-2-yl)amino)-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-8-azabicyclo[3.2.1]octane-8-carboxamide [661];

4-(dimethylamino)-N-(2-(2-methylthiazol-5-yl)-1,6-naphthyridin-7-yl)piperidine-1-carboxamide [662];

4-((2,2-difluoroethyl)amino)-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl) piperidine-1-carboxamide [663];

4-((2,2-difluoroethyl)(methyl-d 3 )amino)-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)piperidine-1-carboxamide [664];

N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-4-morpholinopiperidine-1-carboxamide [665];

N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-4-(4-methylpiperazin-1-yl) piperidine-1-carboxamide [666];

(R)-3,4-dimethyl-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)piperazine-1-carboxamide [667];

(S)-3,4-dimethyl-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)piperazine-1-carboxamide [668];

(1R,3r,5S)-3-((2-fluoroethyl)amino)-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-8-azabicyclo[3.2.1]octane-8-carboxamide [669];

(1R,3r,5 S)-3-((2,2-difluoroethyl)amino)-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-8-azabicyclo[3.2.1]octane-8-carboxamide [670];

(1R,3r,5 S)-3-amino-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-8-azabicyclo [3.2.1]octane-8-carboxamide [671];

(1 S,4S)-5-methyl-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-2,5-diazabicyclo [2.2.1]heptane-2-carboxamide [672];

(1R,4R)-5-methyl-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-2,5-diazabicyclo [2.2.1]heptane-2-carboxamide [673];

8-methyl-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-3,8-diazabicyclo [3.2.1]octane-3-carboxamide [674];

3-methyl-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-3,8-diazabicyclo [3.2.1]octane-8-carboxamide [675];

N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-5,6-dihydroimidazo[1,2-a]pyrazine-7(8H)-carboxamide [676];

2-(4-methylpiperazin-1-yl)-N-(2-(5-methylthiazol-2-yl)-1,6-naphthyridin-7-yl)isonicotinamide [677];

2-(4-methylpiperazin-1-yl)-N-(2-(4-methylthiazol-2-yl)-1,6-naphthyridin-7-yl)isonicotinamide [678];

N-(2-(2-(methylamino)thiazol-5-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [679];

1-methyl-N-(2-(2-(methylamino)thiazol-5-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [680];

N-(2-(2-(diethylamino)thiazol-5-yl)-1,6-naphthyridin-7-yl)-2-(4-fluoropiperidin-1-yl)acetamide [681];

N-(2-(2-(diethylamino)thiazol-5-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl)acetamide [682];

N-(2-(2-aminothiazol-5-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [683];

N-(2-(2-(methylamino)thiazol-5-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [684];

N-(2-(2-(dimethylamino)thiazol-5-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [685];

2-(4-isopropylpiperazin-1-yl)-N-(2-(2-(methylamino)thiazol-5-yl)-1,6-naphthyridin-7-yl) isonicotinamide [686];

2-(3-(dimethylamino)azetidin-1-yl)-N-(2-(2-(methylamino)thiazol-5-yl)-1,6-naphthyridin-7-yl) isonicotinamide [687];

2-(3-(dimethylamino)azetidin-1-yl)-N-(2-(2-(dimethylamino)thiazol-5-yl)-1,6-naphthyridin-7-yl) isonicotinamide [688];

2-(3-aminoazetidin-1-yl)-N-(2-(2-(dimethylamino)thiazol-5-yl)-1,6-naphthyridin-7-yl) isonicotinamide [689];

N-(2-(5-chlorothiazol-2-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [690];

2-(7-(2-(4-methylpiperazin-1-yl)isonicotinamido)-1,6-naphthyridin-2-yl)thiazole-5-carboxamide [691];

N-(2-(isothiazol-4-yl)-1,6-naphthyridin-7-yl)-1-methylpiperidine-4-carboxamide [692];

N-(2-(1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-4-(difluoromethoxy)benzamide [693];

N-(2-(1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-4-(piperidin-4-yloxy)benzamide [694];

N-(2-(1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-4-((1-methylpiperidin-4-yl)oxy)benzamide [695];

N-(2-(1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-3-((1-methylpiperidin-4-yl)oxy)benzamide [696];

N 5 -(2-(1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-N 2 -methylpyridine-2,5-dicarboxamide [697];

N-(2-(1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-6-(4-methylpiperazin-1-yl)nicotinamide [698];

N-(2-(1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-1′-methyl-1′,2′,3′,6′-tetrahydro-[2,4′-bipyridine]-4-carboxamide [699];

N-(2-(1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-2-(3-(dimethylamino)azetidin-1-yl) isonicotinamide [700];

N-(2-(1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [701];

N-(2-(1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-2-(4-isopropylpiperazin-1-yl)isonicotinamide [702];

N-(2-(1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-2-morpholinoisonicotinamide [703];

1-fluoro-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)cyclohexane-1-carboxamide [704];

trans-4-methoxy-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)cyclohexane-1-carboxamide [705];

cis-4-methoxy-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)cyclohexane-1-carboxamide [706];

trans-4-amino-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)cyclohexane-1-carboxamide [707];

trans-4-(dimethylamino)-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl) cyclohexane-1-carboxamide [708];

trans-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-4-morpholinocyclohexane-1-carboxamide [709];

trans-4-(hydroxymethyl)-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)cyclohexane-1-carboxamide [710];

N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [711];

4-fluoro-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [712];

1-methyl-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [713];

4-fluoro-1-methyl-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [714];

1-(2-fluoroethyl)-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [715];

1-(2,2-difluoroethyl)-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [716];

N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [717];

1-(2,2-difluoropropyl)-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [718];

1-benzoyl-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [719];

N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-2-(pyrrolidin-1-yl)acetamide [720];

N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-2-(piperidin-1-yl)acetamide [721];

2-(4-methoxypiperidin-1-yl)-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl) acetamide [722];

N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl) acetamide [723];

N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-2-morpholinoacetamide [724];

(R)—N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-2-(3-methylmorpholino)acetamide [725];

2-(7-azabicyclo[2.2.1]heptan-7-yl)-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl) acetamide [726];

2-((1R,4R)-2-oxa-5-azabicyclo [2.2.1]heptan-5-yl)-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)acetamide [727];

2-(3-oxa-8-azabicyclo[3.2.1]octan-8-yl)-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)acetamide [728];

2-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)acetamide [729];

N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-2-(1,4-oxazepan-4-yl)acetamide [730];

N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-2-morpholinoacetamide-2,2-d 2 [731];

N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-2-(morpholino-d)acetamide [732];

1-methyl-3-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-1-(1-methylpiperidin-4-yl)urea [733];

(3S,4S)-4-amino-3-fluoro-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl) piperidine-1-carboxamide [734];

(3S,4S)-4-(dimethylamino)-3-fluoro-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)piperidine-1-carboxamide [735];

N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)morpholine-4-carboxamide [736];

N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-4-(methylamino)piperidine-1-carboxamide [737];

4-(dimethylamino)-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)piperidine-1-carboxamide [738];

4-((2,2-difluoroethyl)(methyl)amino)-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)piperidine-1-carboxamide [739];

(3S,4S)-3-fluoro-4-(isopropylamino)-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)piperidine-1-carboxamide [740];

2-methyl-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-5,6-dihydroimidazo[1,2-a]pyrazine-7(8H)-carboxamide [741];

4-methyl-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)piperazine-1-carboxamide [742];

N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-1-(1-methylpiperidin-4-yl)-1H-pyrazole-4-carboxamide [743];

1-(1-isopropylpiperidin-4-yl)-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-1H-pyrazole-4-carboxamide [744];

N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-1-(1-methylpiperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide [745];

N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-2-(piperidin-4-yl)oxazole-4-carboxamide [746];

N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-2-(1-methylpiperidin-4-yl)oxazole-4-carboxamide [747];

2-(3-(dimethylamino)azetidin-1-yl)-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl) isonicotinamide [748];

1′-methyl-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-1′,2′,3′,6′-tetrahydro-[2,4′-bipyridine]-4-carboxamide [749];

N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [750];

2-(methyl(1-methylpiperidin-4-yl)amino)-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)isonicotinamide [751];

2-(azetidin-3-yloxy)-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)isonicotinamide [752];

N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-3-((1-methylpiperidin-4-yl)oxy) benzamide [753];

N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-2-((1-methylpiperidin-4-yl)thio) isonicotinamide [754];

6-(4-methylpiperazin-1-yl)-N-(2-(5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)nicotinamide [755];

2-(4-methylpiperazin-1-yl)-N-(2-(5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)isonicotinamide [756];

N-(2-(5-amino-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [757];

N-(2-(5-(dimethylamino)-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [758];

N-(2-(3-amino-5-fluorophenyl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [759];

N-(2-(3-fluoro-5-(isopropylamino)phenyl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [760];

1-methyl-N-(2-(pyridin-2-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [761];

2-(4-methylpiperazin-1-yl)-N-(2-(pyridin-2-yl)-1,6-naphthyridin-7-yl)isonicotinamide [762];

2-(4-methylpiperazin-1-yl)-N-(2-(pyridin-4-yl)-1,6-naphthyridin-7-yl)isonicotinamide [763];

N-(2-(pyridin-3-yl)-1,6-naphthyridin-7-yl)cyclopropanecarboxamide [764];

N-(2-(pyridin-3-yl)-1,6-naphthyridin-7-yl)-2-(pyrrolidin-1-yl)acetamide [765];

1-methyl-N-(2-(pyridin-3-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [766];

N-(2-(pyridin-3-yl)-1,6-naphthyridin-7-yl)quinuclidine-4-carboxamide [767];

2-morpholino-N-(2-(pyridin-3-yl)-1,6-naphthyridin-7-yl)acetamide [768];

2-(morpholino-d 8 )—N-(2-(pyridin-3-yl)-1,6-naphthyridin-7-yl)acetamide [769];

2-(4-methylpiperazin-1-yl)-N-(2-(pyridin-3-yl)-1,6-naphthyridin-7-yl)acetamide [770];

2-(4-methyl-1,4-diazepan-1-yl)-N-(2-(pyridin-3-yl)-1,6-naphthyridin-7-yl)acetamide [771];

2-(4-methylpiperazin-1-yl)-N-(2-(pyridin-3-yl)-1,6-naphthyridin-7-yl)isonicotinamide [772];

2-(2-methyl-1H-imidazol-1-yl)-N-(2-(pyridin-3-yl)-1,6-naphthyridin-7-yl)acetamide [773];

2-(1H-imidazol-1-yl)-N-(2-(pyridin-3-yl)-1,6-naphthyridin-7-yl)acetamide [774];

2-(piperidin-4-yl)-N-(2-(pyridin-3-yl)-1,6-naphthyridin-7-yl)oxazole-4-carboxamide [775];

2-(1-methylpiperidin-4-yl)-N-(2-(pyridin-3-yl)-1,6-naphthyridin-7-yl)oxazole-4-carboxamide [776];

2-(1-isopropylpiperidin-4-yl)-N-(2-(pyridin-3-yl)-1,6-naphthyridin-7-yl)oxazole-4-carboxamide [777];

trans-N-(2-(5-fluoropyridin-3-yl)-1,6-naphthyridin-7-yl)-3-morpholinocyclobutane-1-carboxamide [778];

trans-N-(2-(5-fluoropyridin-3-yl)-1,6-naphthyridin-7-yl)-4-((4-methylpiperazin-1-yl)methyl) cyclohexane-1-carboxamide [779];

N-(2-(5-fluoropyridin-3-yl)-1,6-naphthyridin-7-yl)-2-(pyrrolidin-1-yl)acetamide [780];

N-(2-(5-fluoropyridin-3-yl)-1,6-naphthyridin-7-yl)-1-methylpiperidine-4-carboxamide [781];

N-(2-(5-fluoropyridin-3-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl)acetamide [782];

N-(2-(6-fluoropyridin-3-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl)acetamide [783];

N-(2-(5-fluoropyridin-3-yl)-1,6-naphthyridin-7-yl)-2-morpholinoacetamide [784];

N-(2-(5-fluoropyridin-3-yl)-1,6-naphthyridin-7-yl)-3-morpholinopropanamide [785];

N-(2-(5-fluoropyridin-3-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [786];

N-(2-(5-fluoropyridin-3-yl)-1,6-naphthyridin-7-yl)-2-(piperidin-4-yl)oxazole-4-carboxamide [787];

N-(2-(5-fluoropyridin-3-yl)-1,6-naphthyridin-7-yl)-2-(1-methylpiperidin-4-yl)oxazole-4-carboxamide [788];

N-(2-(5-fluoropyridin-3-yl)-1,6-naphthyridin-7-yl)-2-(1-isopropylpiperidin-4-yl)oxazole-4-carboxamide [789];

N-(2-(5-chloropyridin-3-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [790];

N-(2-(5-methylpyridin-3-yl)-1,6-naphthyridin-7-yl)-2-morpholinoacetamide [791];

N-(2-(5-(difluoromethyl)pyridin-3-yl)-1,6-naphthyridin-7-yl)-3-(piperidin-4-yl)benzamide [792];

N-(2-(5-(difluoromethyl)pyridin-3-yl)-1,6-naphthyridin-7-yl)-3-(1-methylpiperidin-4-yl) benzamide [793];

N-(2-(5-(difluoromethyl)pyridin-3-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [794];

2-(4-methylpiperazin-1-yl)-N-(2-(5-(trifluoromethyl)pyridin-3-yl)-1,6-naphthyridin-7-yl) acetamide [795];

2-(4-methylpiperazin-1-yl)-N-(2-(6-(trifluoromethyl)pyridin-3-yl)-1,6-naphthyridin-7-yl) acetamide [796];

N-(2-(5-(hydroxymethyl)pyridin-3-yl)-1,6-naphthyridin-7-yl)-1-methylpiperidine-4-carboxamide [797];

N-(2-(5-cyanopyridin-3-yl)-1,6-naphthyridin-7-yl)-1-methylpiperidine-4-carboxamide [798];

N-(2-(5-methoxypyridin-3-yl)-1,6-naphthyridin-7-yl)-1-methylpiperidine-4-carboxamide [799];

N-(2-(5-methoxypyridin-3-yl)-1,6-naphthyridin-7-yl)-2-morpholinoacetamide [800];

N-(2-(5-methoxypyridin-3-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [801];

4-fluoro-N-(2-(5-(piperidin-4-yloxy)pyridin-3-yl)-1,6-naphthyridin-7-yl)benzamide [802];

N-(2-(5-aminopyridin-3-yl)-1,6-naphthyridin-7-yl)-4-fluorobenzamide [803];

N-(2-(5-aminopyridin-3-yl)-1,6-naphthyridin-7-yl)-4-(piperidin-4-yloxy)benzamide [804];

N-(2-(5-aminopyridin-3-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [805];

N-(2-(5-aminopyridin-3-yl)-1,6-naphthyridin-7-yl)-2-(piperidin-4-yl)oxazole-4-carboxamide [806];

N-(2-(6-aminopyridin-3-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [807];

N-(2-(6-(methylamino)pyridin-3-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [808];

N-(2-(5-(isopropylamino)pyridin-3-yl)-1,6-naphthyridin-7-yl)-3-(piperidin-4-yl)benzamide [809];

N-(2-(5-(isopropylamino)pyridin-3-yl)-1,6-naphthyridin-7-yl)-3-(1-methylpiperidin-4-yl) benzamide [810];

N-(2-(5-(isopropylamino)pyridin-3-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [811];

N-(2-(5-(piperidin-4-ylamino)pyridin-3-yl)-1,6-naphthyridin-7-yl)cyclohexanecarboxamide [812];

4-fluoro-N-(2-(5-(piperidin-4-ylamino)pyridin-3-yl)-1,6-naphthyridin-7-yl)benzamide [813];

4-fluoro-N-(2-(5-((1-methylpiperidin-4-yl)amino)pyridin-3-yl)-1,6-naphthyridin-7-yl)benzamide [814];

N-(2-(5-acetamidopyridin-3-yl)-1,6-naphthyridin-7-yl)-1-methylpiperidine-4-carboxamide [815];

N-(2-(5-(dimethylamino)pyridin-3-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [816];

N-(2-(6-(dimethylamino)pyridin-3-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [817];

1-methyl-N-(2-(5-(pyrrolidin-1-yl)pyridin-3-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [818];

N-(2-(5-(pyrrolidin-1-ylmethyl)pyridin-3-yl)-1,6-naphthyridin-7-yl)cyclopropanecarboxamide [819];

4-fluoro-N-(2-(5-(pyrrolidin-1-ylmethyl)pyridin-3-yl)-1,6-naphthyridin-7-yl)benzamide [820];

N-(2-(5-((4-hydroxypiperidin-1-yl)methyl)pyridin-3-yl)-1,6-naphthyridin-7-yl) cyclopropanecarboxamide [821];

4-fluoro-N-(2-(5-((4-hydroxypiperidin-1-yl)methyl)pyridin-3-yl)-1,6-naphthyridin-7-yl) benzamide [822];

N-(2-(5-(piperazin-1-ylmethyl)pyridin-3-yl)-1,6-naphthyridin-7-yl)cyclopropanecarboxamide [823];

N-(2-(5-((4-methylpiperazin-1-yl)methyl)pyridin-3-yl)-1,6-naphthyridin-7-yl) cyclopropanecarboxamide [824];

N-(2-(5-(morpholinomethyl)pyridin-3-yl)-1,6-naphthyridin-7-yl)cyclopropanecarboxamide [825];

N-methyl-5-(7-(1-methylpiperidine-4-carboxamido)-1,6-naphthyridin-2-yl)nicotinamide [826];

N-methyl-5-(7-(2-(4-methylpiperazin-1-yl)isonicotinamido)-1,6-naphthyridin-2-yl)nicotinamide [827];

N-(2-(pyridin-3-yl-d 4 )-1,6-naphthyridin-7-yl)-2-(pyrrolidin-1-yl)acetamide [828];

2-(4-methylpiperazin-1-yl)-N-(2-(pyridin-3-yl-d 4 )-1,6-naphthyridin-7-yl)acetamide [829];

2-morpholino-N-(2-(pyridin-3-yl-d 4 )-1,6-naphthyridin-7-yl)acetamide [830];

1-methyl-N-(2-(2-methylpyrimidin-5-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [831];

2-(4-methylpiperazin-1-yl)-N-(2-(2-methylpyrimidin-5-yl)-1,6-naphthyridin-7-yl)isonicotinamide [832];

N-(2-(2-aminopyrimidin-5-yl)-1,6-naphthyridin-7-yl)-1-methylpiperidine-4-carboxamide [833];

2-morpholino-N-(2-(pyridazin-3-yl)-1,6-naphthyridin-7-yl)acetamide [834];

2-morpholino-N-(2-(pyridazin-4-yl)-1,6-naphthyridin-7-yl)acetamide [835];

N-(2-(pyridazin-4-yl)-1,6-naphthyridin-7-yl)-2-(pyrrolidin-1-yl)acetamide [836];

trans-3-morpholino-N-(2-(pyrazin-2-yl)-1,6-naphthyridin-7-yl)cyclobutane-1-carboxamide [837];

trans-4-(dimethylamino)-N-(2-(pyrazin-2-yl)-1,6-naphthyridin-7-yl)cyclohexane-1-carboxamide [838];

trans-4-morpholino-N-(2-(pyrazin-2-yl)-1,6-naphthyridin-7-yl)cyclohexane-1-carboxamide [839];

trans-4-((3-fluoroazetidin-1-yl)methyl)-N-(2-(pyrazin-2-yl)-1,6-naphthyridin-7-yl)cyclohexane-1-carboxamide [840];

trans-4-((4-methylpiperazin-1-yl)methyl)-N-(2-(pyrazin-2-yl)-1,6-naphthyridin-7-yl)cyclohexane-1-carboxamide [841];

N-(2-(pyrazin-2-yl)-1,6-naphthyridin-7-yl)-2-(pyrrolidin-1-yl)acetamide [842];

1-methyl-N-(2-(pyrazin-2-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [843];

4-fluoro-1-methyl-N-(2-(pyrazin-2-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [844];

1-(2-fluoroethyl)-N-(2-(pyrazin-2-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [845];

1-(oxetan-3-yl)-N-(2-(pyrazin-2-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [846];

2-morpholino-N-(2-(pyrazin-2-yl)-1,6-naphthyridin-7-yl)acetamide [847];

1-methyl-N-(2-(pyrazin-2-yl)-1,6-naphthyridin-7-yl)azepane-4-carboxamide [848];

1-isobutyl-N-(2-(pyrazin-2-yl)-1,6-naphthyridin-7-yl)azepane-4-carboxamide [849];

1-(2-hydroxy-2-methylpropyl)-N-(2-(pyrazin-2-yl)-1,6-naphthyridin-7-yl)azepane-4-carboxamide [850];

4-(morpholinomethyl)-N-(2-(pyrazin-2-yl)-1,6-naphthyridin-7-yl)benzamide [851];

2-(4-methylpiperazin-1-yl)-N-(2-(pyrazin-2-yl)-1,6-naphthyridin-7-yl)isonicotinamide [852];

N-(2-(6-(methylamino)pyrazin-2-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [853];

N-(2-(6-(isopropylamino)pyrazin-2-yl)-1,6-naphthyridin-7-yl)azetidine-3-carboxamide [854];

N-(2-(6-(isopropylamino)pyrazin-2-yl)-1,6-naphthyridin-7-yl)-1-methylpiperidine-4-carboxamide [855];

N-(2-(6-(isopropylamino)pyrazin-2-yl)-1,6-naphthyridin-7-yl)-1-methylpiperidine-4-carboxamide [856];

1-(2-fluoroethyl)-N-(2-(6-(isopropylamino)pyrazin-2-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [857];

1-isopropyl-N-(2-(6-(isopropylamino)pyrazin-2-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [858];

1-isopentyl-N-(2-(6-(isopropylamino)pyrazin-2-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [859];

N-(2-(6-(isopropylamino)pyrazin-2-yl)-1,6-naphthyridin-7-yl)-3-(piperidin-4-yl)benzamide [860];

N-(2-(6-(isopropylamino)pyrazin-2-yl)-1,6-naphthyridin-7-yl)-3-(1-methylpiperidin-4-yl) benzamide [861];

N-(2-(6-(isopropylamino)pyrazin-2-yl)-1,6-naphthyridin-7-yl)-1-(piperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide [862];

1-(1-(2-fluoroethyl)piperidin-4-yl)-N-(2-(6-(isopropylamino)pyrazin-2-yl)-1,6-naphthyridin-7-yl)-1H-1,2,3-triazole-4-carboxamide [863];

N-(2-(6-(isopropylamino)pyrazin-2-yl)-1,6-naphthyridin-7-yl)-1-(1-isopropylpiperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide [864];

N-(2-(6-(isopropylamino)pyrazin-2-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [865];

N-(2-(6-(tert-butylamino)pyrazin-2-yl)-1,6-naphthyridin-7-yl)-2-(3-(dimethylamino)azetidin-1-yl)isonicotinamide [866];

N-(2-(6-(tert-butylamino)pyrazin-2-yl)-1,6-naphthyridin-7-yl)-1′-methyl-1′,2′,3′,6′-tetrahydro-[2,4′-bipyridine]-4-carboxamide [867];

N-(2-(6-(tert-butylamino)pyrazin-2-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [868];

N-(2-(6-(tert-butylamino)pyrazin-2-yl)-1,6-naphthyridin-7-yl)-2-(4-isopropylpiperazin-1-yl) isonicotinamide [869];

N-(2-(6-(tert-butylamino)pyrazin-2-yl)-1,6-naphthyridin-7-yl)-2-morpholinoisonicotinamide [870];

N-(2-(6-(((3-fluoroazetidin-3-yl)methyl)amino)pyrazin-2-yl)-1,6-naphthyridin-7-yl) cyclopropanecarboxamide [871];

4-fluoro-N-(2-(6-(((3-fluoroazetidin-3-yl)methyl)amino)pyrazin-2-yl)-1,6-naphthyridin-7-yl) benzamide [872];

N-(2-(6-(piperidin-4-ylamino)pyrazin-2-yl)-1,6-naphthyridin-7-yl)cyclobutanecarboxamide [873];

3,3-difluoro-N-(2-(6-(piperidin-4-ylamino)pyrazin-2-yl)-1,6-naphthyridin-7-yl)cyclobutane-1-carboxamide [874];

N-(2-(6-(piperidin-4-ylamino)pyrazin-2-yl)-1,6-naphthyridin-7-yl)cyclopentanecarboxamide [875];

4,4-difluoro-N-(2-(6-(piperidin-4-ylamino)pyrazin-2-yl)-1,6-naphthyridin-7-yl)cyclohexane-1-carboxamide [876];

N-(2-(6-(piperidin-4-ylamino)pyrazin-2-yl)-1,6-naphthyridin-7-yl)tetrahydro-2H-pyran-4-carboxamide [877];

4-fluoro-N-(2-(6-(piperidin-4-ylamino)pyrazin-2-yl)-1,6-naphthyridin-7-yl)benzamide [878];

N-(2-(6-(((3S,4S)-3-fluoropiperidin-4-yl)amino)pyrazin-2-yl)-1,6-naphthyridin-7-yl) cyclopropanecarboxamide [879];

4-fluoro-N-(2-(6-(((3S,4S)-3-fluoropiperidin-4-yl)amino)pyrazin-2-yl)-1,6-naphthyridin-7-yl) benzamide [880];

N-(2-(6-((1-methylpiperidin-4-yl)amino)pyrazin-2-yl)-1,6-naphthyridin-7-yl) cyclobutanecarboxamide [881];

N-(2-(6-((1-methylpiperidin-4-yl)amino)pyrazin-2-yl)-1,6-naphthyridin-7-yl) cyclopentanecarboxamide [882];

4-fluoro-N-(2-(6-((1-methylpiperidin-4-yl)amino)pyrazin-2-yl)-1,6-naphthyridin-7-yl)benzamide [883];

N-(2-(6-((1-isopropylpiperidin-4-yl)amino)pyrazin-2-yl)-1,6-naphthyridin-7-yl) cyclopropanecarboxamide [884];

3,3-difluoro-N-(2-(6-((1-isopropylpiperidin-4-yl)amino)pyrazin-2-yl)-1,6-naphthyridin-7-yl) cyclobutane-1-carboxamide [885];

N-(2-(6-((1-isopropylpiperidin-4-yl)amino)pyrazin-2-yl)-1,6-naphthyridin-7-yl) cyclopentanecarboxamide [886];

4-fluoro-N-(2-(6-((1-isopropylpiperidin-4-yl)amino)pyrazin-2-yl)-1,6-naphthyridin-7-yl) benzamide [887];

N-(2-(6-(dimethylamino)pyrazin-2-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [888];

N-(2-(6-(diethylamino)pyrazin-2-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [889];

N-(2-(6-(3-aminoazetidin-1-yl)pyrazin-2-yl)-1,6-naphthyridin-7-yl)-4-fluorobenzamide [890];

2-(4-methylpiperazin-1-yl)-N-(2-(6-(pyrrolidin-1-yl)pyrazin-2-yl)-1,6-naphthyridin-7-yl) isonicotinamide [891];

N-(2-(6-(azetidin-3-ylmethoxy)pyrazin-2-yl)-1,6-naphthyridin-7-yl)-4-fluorobenzamide [892];

N-(2-(6-(azetidin-3-yloxy)pyrazin-2-yl)-1,6-naphthyridin-7-yl)-4-fluorobenzamide [893];

N-(2-(1H-pyrrolo[2,3-b]pyridin-5-yl)-1,6-naphthyridin-7-yl)-1-(1-methylpiperidin-4-yl)-1H-pyrazole-4-carboxamide [894];

N-(2-(1H-pyrrolo[3,2-b]pyridin-6-yl)-1,6-naphthyridin-7-yl)-1-(1-methylpiperidin-4-yl)-1H-pyrazole-4-carboxamide [895];

N-(2-(1H-pyrrolo[2,3-c]pyridin-4-yl)-1,6-naphthyridin-7-yl)-1-(1-methylpiperidin-4-yl)-1H-pyrazole-4-carboxamide [896];

N-(2-(1H-pyrrolo[2,3-b]pyridin-5-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [897];

N-(2-(1H-pyrrolo[3,2-b]pyridin-6-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [898];

N-(2-(1H-pyrrolo[2,3-c]pyridin-4-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [899];

2-(4-methylpiperazin-1-yl)-N-(2-(oxazolo[5,4-b]pyridin-6-yl)-1,6-naphthyridin-7-yl) isonicotinamide [900];

N-(2-(2-methyl-1H-pyrrolo[2,3-b]pyridin-5-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [901];

N-(2-(3-methyl-1H-pyrrolo[2,3-b]pyridin-5-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [902];

N-(2-(2-methyl-1H-pyrrolo[3,2-b]pyridin-6-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [903];

N-(2-(5H-pyrrolo[2,3-b]pyrazin-2-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [904];

N-(2-(5H-pyrrolo[2,3-b]pyrazin-3-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [905];

1-isopropyl-N-(2-(6-(piperidin-4-ylamino)pyrazin-2-yl)-1,6-naphthyridin-7-yl)-1H-pyrazole-4-carboxamide [906];

1-isopropyl-N-(2-(6-((1-methylpiperidin-4-yl)amino)pyrazin-2-yl)-1,6-naphthyridin-7-yl)-1H-pyrazole-4-carboxamide [907];

trans-4-((2-fluoroethyl)amino)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl) cyclohexane-1-carboxamide [4535];

trans-4-((2-methoxyethyl)amino)-N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl) cyclohexane-1-carboxamide [4536];

tert-butyl (trans-4-((2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)carbamoyl)cyclohexyl) carbamate [4537];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-((1-methylpiperidin-4-yl)amino) isonicotinamide [4538];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl)thiazole-5-carboxamide [4539];

N-(2-(1-methyl-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(4-methylpiperazin-1-yl)thiazole-5-carboxamide [4540];

N-(2-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-1,6-naphthyridin-7-yl)-2-(2,7-diazaspiro[3.5]nonan-2-yl)isonicotinamide [4541];

N-(2-(1-methyl-1H-1,2,3-triazol-4-yl)-1,6-naphthyridin-7-yl)-4-(piperidin-4-yloxy)benzamide [4542];

N-(2-(1-methyl-1H-tetrazol-5-yl)-1,6-naphthyridin-7-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [4543];

N-(2-(1,2-dimethyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-2-(pyrrolidin-1-yl)propanamide [4544];

N-(2-(1,2-dimethyl-1H-imidazol-5-yl)-1,6-naphthyridin-7-yl)-2-(piperidin-1-yl)propanamide [4545];

4-isopropoxy-N-(2-(7-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-1,6-naphthyridin-7-yl)benzamide [4546];

trans-3-morpholino-N-(2-(oxazol-5-yl)-1,6-naphthyridin-7-yl)cyclobutane-1-carboxamide [4547];

trans-4-(hydroxymethyl)-N-(2-(oxazol-5-yl)-1,6-naphthyridin-7-yl)cyclohexane-1-carboxamide [4548];

N-(2-(oxazol-5-yl)-1,6-naphthyridin-7-yl)piperidine-4-carboxamide [4549];

4-morpholino-N-(2-(oxazol-5-yl)-1,6-naphthyridin-7-yl)piperidine-1-carboxamide [4550];

N-(2-(oxazol-5-yl)-1,6-naphthyridin-7-yl)-4-(piperidin-4-yloxy)benzamide [4551];

N-(2-(oxazol-5-yl)-1,6-naphthyridin-7-yl)-3-(piperidin-4-yloxy)benzamide [4552];

2-methyl-N-(2-(oxazol-5-yl)-1,6-naphthyridin-7-yl)-5,6-dihydroimidazo[1,2-a]pyrazine-7(8H)-carboxamide [4553];

2-(1H-imidazol-1-yl)-N-(2-(oxazol-5-yl)-1,6-naphthyridin-7-yl)acetamide [4554];

trans-4-(hydroxymethyl)-N-(2-(thiazol-5-yl)-1,6-naphthyridin-7-yl)cyclohexane-1-carboxamide [4555];

trans-4-(dimethylamino)-N-(2-(thiazol-5-yl)-1,6-naphthyridin-7-yl)cyclohexane-1-carboxamide [4556];

N-(2-(thiazol-5-yl)-1,6-naphthyridin-7-yl)-1-((1-(trifluoromethyl)cyclopropyl)methyl)piperidine-4-carboxamide [4557];

trans-4-(hydroxymethyl)-N-(2-(2-methylthiazol-5-yl)-1,6-naphthyridin-7-yl)cyclohexane-1-carboxamide [4558];

trans-4-(dimethylamino)-N-(2-(2-methylthiazol-5-yl)-1,6-naphthyridin-7-yl)cyclohexane-1-carboxamide [4559];

N-(2-(2-methylthiazol-5-yl)-1,6-naphthyridin-7-yl)-1-(oxetan-3-yl)piperidine-4-carboxamide [4560];

N-(2-(2-methylthiazol-5-yl)-1,6-naphthyridin-7-yl)-1-(2-(pyrrolidin-1-yl)acetyl)piperidine-4-carboxamide [4561];

2-((1S,4S)-2-oxa-5-azabicyclo [2.2.1]heptan-5-yl)-N-(2-(5-methyl-1,3,4-thiadiazol-2-yl)-1,6-naphthyridin-7-yl)acetamide [4562];

N-(2-(5-(cyano(4-hydroxypiperidin-1-yl)methyl)pyridin-3-yl)-1,6-naphthyridin-7-yl) cyclopropanecarboxamide [4563];

4-fluoro-N-(2-(6-((1-methylazetidin-3-yl)methoxy)pyrazin-2-yl)-1,6-naphthyridin-7-yl) benzamide [4564];

1-isopropyl-N-(2-(6-((1-methylpiperidin-4-yl)amino)pyrazin-2-yl)-1,6-naphthyridin-7-yl)-1H-pyrazole-4-carboxamide [4565]; or a pharmaceutically acceptable salt thereof.

13. The compound of claim 1 , wherein the compound of Formula I is selected from the group consisting of:

N-(7-(1H-pyrazol-4-yl)quinazolin-2-yl)-1-isobutylpiperidine-4-carboxamide [908];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)cyclopropanecarboxamide [909];

4,4-difluoro-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)cyclohexane-1-carboxamide [910];

trans-4-methoxy-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)cyclohexane-1-carboxamide [911];

trans-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-4-morpholinocyclohexane-1-carboxamide [912];

trans-4-((3-fluoroazetidin-1-yl)methyl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl) cyclohexane-1-carboxamide [913];

trans-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-4-((4-methylpiperazin-1-yl)methyl) cyclohexane-1-carboxamide [914];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(pyrrolidin-1-yl)acetamide [915];

(S)-2-(3-fluoropyrrolidin-1-yl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)acetamide [916];

(S)—N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)tetrahydrofuran-2-carboxamide [917];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)piperidine-4-carboxamide [918];

1-methyl-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)piperidine-4-carboxamide [919];

1-isopropyl-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)piperidine-4-carboxamide [920];

1-(tert-butyl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)piperidine-4-carboxamide [921];

1-cyclopropyl-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)piperidine-4-carboxamide [922];

1-isobutyl-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)piperidine-4-carboxamide [923];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-1-neopentylpiperidine-4-carboxamide [924];

1-(2-fluoroethyl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)piperidine-4-carboxamide [925];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [926];

1-butyl-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)piperidine-4-carboxamide [927];

1-benzoyl-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)piperidine-4-carboxamide [928];

1-(2,2-difluoropropyl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)piperidine-4-carboxamide [929];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)azetidine-3-carboxamide [930];

1-(2,2-difluoroethyl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)piperidine-4-carboxamide [931];

1-(2-fluoro-2-methylpropyl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)piperidine-4-carboxamide [932];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-1-(oxetan-3-yl)piperidine-4-carboxamide [933];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-1-((3-methyloxetan-3-yl)methyl)piperidine-4-carboxamide [934];

1-(2-methoxyethyl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)piperidine-4-carboxamide [935];

1-(2-isopropoxyethyl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)piperidine-4-carboxamide [936];

1,1-diisobutyl-4-((7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)carbamoyl)piperidin-1-ium [937];

4-fluoro-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)piperidine-4-carboxamide [938];

4-fluoro-1-methyl-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)piperidine-4-carboxamide [939];

4-fluoro-1-isobutyl-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)piperidine-4-carboxamide [940];

(S)—N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)piperidine-3-carboxamide [941];

(R)—N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)piperidine-3-carboxamide [942];

(S)-1-isobutyl-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)piperidine-3-carboxamide [943];

(R)-1-isobutyl-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)piperidine-3-carboxamide [944];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)tetrahydro-2H-pyran-4-carboxamide [945];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(piperidin-1-yl)acetamide [946];

2-(4-fluoropiperidin-1-yl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)acetamide [947];

trans-4-amino-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)cyclohexane-1-carboxamide [948];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)acetamide [949];

(S)—N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)piperidine-2-carboxamide [950];

2-(4-isobutylpiperazin-1-yl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)acetamide [951];

2-(3,3-dimethylazetidin-1-yl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)acetamide [952];

(R)-2-(3-fluoropyrrolidin-1-yl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)acetamide [953];

(S)—N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(2-methylpyrrolidin-1-yl)acetamide [954];

2-(3-azabicyclo[3.1.0]hexan-3-yl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)acetamide [955];

2-(7-azabicyclo[2.2.1]heptan-7-yl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)acetamide [956];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(4-methylpiperidin-1-yl)acetamide [957];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(4-(trifluoromethyl)piperidin-1-yl)acetamide [958];

2-(4-(difluoromethyl)piperidin-1-yl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)acetamide [959];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(6-azaspiro[2.5]octan-6-yl)acetamide [960];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(pyrrolidin-1-yl)propanamide [961];

(R)—N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(2-methylpyrrolidin-1-yl)acetamide [962];

2-(cyclobutyl(methyl)amino)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)acetamide [963];

2-(diethylamino)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)acetamide [964];

7-(2-fluoroethyl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-7-azaspiro[3.5]nonane-2-carboxamide [965];

4-methyl-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)piperazine-1-carboxamide [966];

(S)—N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(pyrrolidin-1-yl)propanamide [967];

(R)—N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(pyrrolidin-1-yl)propanamide [968];

(R)—N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)pyrrolidine-2-carboxamide [969];

2-methyl-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-azaspiro[3.3]heptane-6-carboxamide [970];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(2,2,2-trifluoroacetyl)-2-azaspiro [3.3] heptane-6-carboxamide [971];

2-(2-fluoroethyl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-azaspiro [3.3]heptane-6-carboxamide [972];

trans-4-(dimethylamino)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)cyclohexane-1-carboxamide [973];

1-acetyl-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)piperidine-4-carboxamide [974];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-1-((1-(trifluoromethyl)cyclopropyl)methyl) piperidine-4-carboxamide [975];

(S)-1-(2-fluoropropyl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)piperidine-4-carboxamide [976];

(R)-1-(2-fluoropropyl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)piperidine-4-carboxamide [977];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(piperidin-1-yl)propanamide [978];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-1-(methylsulfonyl)piperidine-4-carboxamide [979];

1′-methyl-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-[1,4′-bipiperidine]-4-carboxamide [980];

trans-4-(hydroxymethyl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)cyclohexane-1-carboxamide [981];

methyl 2-(4-((7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)carbamoyl)piperidin-1-yl)acetate [982];

1-benzyl-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)piperidine-4-carboxamide [983];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-1-(2-(pyrrolidin-1-yl)acetyl)piperidine-4-carboxamide [984];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-morpholinoacetamide [985];

(S)—N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(3-methylmorpholino)acetamide [986];

(R)—N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(3-methylmorpholino)acetamide [987];

(S)—N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(2-methylmorpholino)acetamide [988];

2-((2R,6S)-2,6-dimethylmorpholino)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)acetamide [989];

2-((1S,4S)-2-oxa-5-azabicyclo [2.2.1]heptan-5-yl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)acetamide [990];

2-((1R,4R)-2-oxa-5-azabicyclo [2.2.1]heptan-5-yl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)acetamide [991];

2-(3-oxa-8-azabicyclo[3.2.1]octan-8-yl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl) acetamide [992];

(S)—N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-morpholinopropanamide [993];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(morpholin-2-yl)acetamide [994];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(4-methylmorpholin-2-yl)acetamide [995];

2-(4-ethylpiperazin-1-yl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)acetamide [996];

2-(4-isopropylpiperazin-1-yl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)acetamide [997];

2-(4-cyclopropylpiperazin-1-yl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)acetamide [998];

2-(4-(2-fluoroethyl)piperazin-1-yl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)acetamide [999];

(S)-2-(2,4-dimethylpiperazin-1-yl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)acetamide [1000];

1-(2-hydroxyethyl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)piperidine-4-carboxamide [1001];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-1-(pyridin-2-ylmethyl)piperidine-4-carboxamide [1002];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-1-(oxazol-2-ylmethyl)piperidine-4-carboxamide [1003];

(R)—N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-1-oxotetrahydro-1H-pyrrolo[1,2-c] imidazole-2(3H)-carboxamide [1004];

(R)-1-methyl-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)pyrrolidine-2-carboxamide [1005];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-1-(tetrahydro-2H-pyran-4-yl)piperidine-4-carboxamide [1006];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-1-(pyrimidin-2-ylmethyl)piperidine-4-carboxamide [1007];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-1-(pyrazin-2-ylmethyl)piperidine-4-carboxamide [1008];

1-((5-methyl-1,2,4-oxadiazol-3-yl)methyl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)piperidine-4-carboxamide [1009];

1-(2-hydroxy-2-methylpropyl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)piperidine-4-carboxamide [1010];

tert-butyl 2-(4-((7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)carbamoyl)piperidin-1-yl)acetate [1011];

2-(4-((7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)carbamoyl)piperidin-1-yl)acetic acid [1012];

2-(4-methyl-1,4-diazepan-1-yl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)acetamide [1013];

tert-butyl (7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)carbamate [1014];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)but-2-ynamide [1015];

trans-4-((7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)carbamoyl)cyclohexane-1-carboxylic acid [1016];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-3-morpholinopropanamide [1017];

trans-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-3-morpholinocyclobutane-1-carboxamide [1018];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)quinuclidine-4-carboxamide [1019];

1-isobutyl-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)azepane-4-carboxamide [1020];

2-(4-methoxypiperidin-1-yl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)acetamide [1021];

2-(4-hydroxypiperidin-1-yl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)acetamide [1022];

3-(hydroxymethyl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)bicyclo[1.1.1]pentane-1-carboxamide [1023];

1-methyl-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)azepane-4-carboxamide [1024];

trans-4-(dimethylamino)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)cyclohexane-1-carboxamide [1025];

trans-4-(bis(methyl-d 3 )amino)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)cyclohexane-1-carboxamide [1026];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-3-((4-methylpiperazin-1-yl)methyl)bicyclo [1.1.1]pentane-1-carboxamide [1027];

methyl trans-4-((7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)carbamoyl)cyclohexane-1-carboxylate [1028];

2-(1-isobutylpyrrolidin-3-yl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)acetamide [1029];

trans-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-4-(4-methylpiperazine-1-carbonyl) cyclohexane-1-carboxamide [1030];

1-isobutyl-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)piperidine-4-carboxamide [1031];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-1-(phenylsulfonyl)piperidine-4-carboxamide [1032];

8-methyl-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-3,8-diazabicyclo[3.2.1]octane-3-carboxamide [1033];

3-methyl-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-3,8-diazabicyclo[3.2.1]octane-8-carboxamide [1034];

(1R,3 s,5 S)-3-amino-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-8-azabicyclo [3.2.1]octane-8-carboxamide [1035];

(1R,3s,5S)—N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-3-((3,3,3-trifluoropropyl)amino)-8-azabicyclo[3.2.1]octane-8-carboxamide [1036];

(1R,3s,5S)-3-((1,3-difluoropropan-2-yl)amino)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-8-azabicyclo[3.2.1]octane-8-carboxamide [1037];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)morpholine-4-carboxamide [1038];

4-(dimethylamino)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)piperidine-1-carboxamide [1039];

(S)-2,4-dimethyl-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)piperazine-1-carboxamide [1040];

1-methyl-3-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-1-(1-methylpiperidin-4-yl)urea [1041];

1-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-3-(1-methylpiperidin-4-yl)urea [1042];

4-isopropyl-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)piperazine-1-carboxamide [1043];

(R)-3,4-dimethyl-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)piperazine-1-carboxamide [1044];

N-(7-(1H-pyrazol-4-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [1045];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-3-(piperazin-1-yl)benzamide [1046];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-3-(4-methylpiperazin-1-yl)benzamide [1047];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-3-(pyrrolidin-1-ylmethyl)benzamide [1048];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-3-(piperidin-4-yloxy)benzamide [1049];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-3-((1-methylpiperidin-4-yl)oxy)benzamide [1050];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-4-(piperidin-4-yloxy)benzamide [1051];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-4-((1-methylpiperidin-4-yl)oxy)benzamide [1052];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(piperazin-1-yl)isonicotinamide [1053];

[1054];

2-(4-isopropylpiperazin-1-yl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)isonicotinamide [1055];

2-(4-cyclopropylpiperazin-1-yl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl) isonicotinamide [1056];

2-(4-(2-fluoroethyl)piperazin-1-yl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl) isonicotinamide [1057];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-6-(4-methylpiperazin-1-yl)nicotinamide [1058];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-5-(piperidin-4-yloxy)nicotinamide [1059];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(piperidin-4-yloxy)isonicotinamide [1060];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-((1-methylpiperidin-4-yl)oxy) isonicotinamide [1061];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-5-(piperidin-4-ylamino)nicotinamide [1062];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-5-((1-methylpiperidin-4-yl)amino)nicotinamide [1063];

2-(4-aminopiperidin-1-yl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)isonicotinamide [1064];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(4-(methylamino)piperidin-1-yl) isonicotinamide [1065];

2-(4-(dimethylamino)piperidin-1-yl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl) isonicotinamide [1066];

2-((1-isopropylpiperidin-4-yl)oxy)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl) isonicotinamide [1067];

2-(3-aminoazetidin-1-yl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)isonicotinamide [1068];

2-(3-(dimethylamino)azetidin-1-yl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl) isonicotinamide [1069];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-morpholinoisonicotinamide [1070];

2-((2-(dimethylamino)ethyl)amino)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl) isonicotinamide [1071];

2-(2-(dimethylamino)ethoxy)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)isonicotinamide [1072];

2-(4-isobutylpiperazin-1-yl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)isonicotinamide [1073];

2-(azetidin-3-yloxy)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)isonicotinamide [1074];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-((1-methylazetidin-3-yl)oxy)isonicotinamide [1075];

2-(4-ethylpiperazin-1-yl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)isonicotinamide [1076];

4-((dimethylamino)methyl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)benzamide [1077];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-3-(1-methylpiperidin-4-yl)benzamide [1078];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-3-((4-methylpiperazin-1-yl)methyl)benzamide [1079];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)isonicotinamide [1080];

2-hydroxy-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)isonicotinamide [1081];

2-isopropoxy-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)isonicotinamide [1082];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(1-methylpiperidin-4-yl)isonicotinamide [1083];

1′-methyl-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-1′,2′,3′,6′-tetrahydro-[2,4′-bipyridine]-4-carboxamide [1084];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(4-(6-(4-methylpiperazin-1-yl) nicotinoyl)piperazin-1-yl)isonicotinamide [1085];

2-(4-hydroxy-4-methyl-4λ 4 -piperazin-1-yl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl) isonicotinamide [1086];

2-methyl-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-6-(4-methylpiperazin-1-yl) isonicotinamide [1087];

3-methyl-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [1088];

2-(4-methyl-1,4-diazepan-1-yl)-N-(7-(-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)isonicotinamide [1089];

2-((2S,6R)-2,6-dimethylmorpholino)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl) isonicotinamide [1090];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(2,7-diazaspiro[3.5]nonan-2-yl) isonicotinamide [1091];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(7-methyl-2,7-diazaspiro[3.5]nonan-2-yl) isonicotinamide [1092];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(2,7-diazaspiro[3.5]nonan-7-yl) isonicotinamide [1093];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(2-methyl-2,7-diazaspiro[3.5]nonan-7-yl) isonicotinamide [1094];

2-(methyl(1-methylpiperidin-4-yl)amino)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl) isonicotinamide [1095];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-((1-methylpiperidin-4-yl)thio) isonicotinamide [1096];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)pyrimidine-4-carboxamide [1097];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-6-(4-methylpiperazin-1-yl)pyridazine-4-carboxamide [1098];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-6-(4-methylpiperazin-1-yl)pyrimidine-4-carboxamide [1099];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-phenylacetamide [1100];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-3-phenylpropanamide [1101];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(pyridin-3-yl)acetamide [1102];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-3-(pyridin-3-yl)propanamide [1103];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(pyridin-4-yl)acetamide [1104];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-3-(pyridin-4-yl)propanamide [1105];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)isoindoline-5-carboxamide [1106];

2-methyl-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)isoindoline-5-carboxamide [1107];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-1,2,3,4-tetrahydroisoquinoline-7-carboxamide [1108];

2-methyl-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-1,2,3,4-tetrahydroisoquinoline-7-carboxamide [1109];

2-methyl-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-1,2,3,4-tetrahydroisoquinoline-6-carboxamide [1110];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-1,2,3,4-tetrahydroisoquinoline-6-carboxamide [1111];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-1H-indole-5-carboxamide [1112];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)benzofuran-5-carboxamide [1113];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)furo[2,3-c]pyridine-5-carboxamide [1114];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)benzo[b]thiophene-5-carboxamide [1115];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)benzofuran-6-carboxamide [1116];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)benzo[d]oxazole-6-carboxamide [1117];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)benzo[d]thiazole-6-carboxamide [1118];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)benzo[d]oxazole-5-carboxamide [1119];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)benzo[d]thiazole-5-carboxamide [1120];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)quinoline-3-carboxamide [1121];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)quinoline-6-carboxamide [1122];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)quinoxaline-6-carboxamide [1123];

5-chloro-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [1124];

3-chloro-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [1125];

2-(2,5-diazabicyclo[2.2.1]heptan-2-yl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl) isonicotinamide [1126];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(5-methyl-2,5-diazabicyclo [2.2.1]heptan-2-yl)isonicotinamide [1127];

3-fluoro-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [1128];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-((4-methylpiperazin-1-yl)methyl) isonicotinamide [1129];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(morpholinomethyl)isonicotinamide [1130];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(pyrrolidin-1-ylmethyl)isonicotinamide [1131];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(2-(4-methylpiperazin-1-yl)pyridin-4-yl) acetamide [1132];

1-methyl-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-1H-indazole-5-carboxamide [1133];

1-methyl-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-1H-benzo[d]imidazole-5-carboxamide [1134];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-1-(piperidin-4-yl)-1H-pyrazole-4-carboxamide [1135];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-1-(1-methylpiperidin-4-yl)-1H-pyrazole-4-carboxamide [1136];

1-(1-ethylpiperidin-4-yl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-1H-pyrazole-4-carboxamide [1137];

1-(1-(2-fluoroethyl)piperidin-4-yl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-1H-pyrazole-4-carboxamide [1138];

1-(1-isopropylpiperidin-4-yl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-1H-pyrazole-4-carboxamide [1139];

1-(1-cyclopropylpiperidin-4-yl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-1H-pyrazole-4-carboxamide [1140];

isopropyl 4-(4-((7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)carbamoyl)-1H-pyrazol-1-yl)piperidine-1-carboxylate [1141];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-1-(piperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide [1142];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-1-(1-methylpiperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide [1143];

1-(1-(2-fluoroethyl)piperidin-4-yl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-1H-1,2,3-triazole-4-carboxamide [1144];

1-(1-isopropylpiperidin-4-yl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-1H-1,2,3-triazole-4-carboxamide [1145];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)oxazole-5-carboxamide [1146];

2-(3-(dimethylamino)azetidin-1-yl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)oxazole-4-carboxamide [1147];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(piperidin-4-yl)oxazole-4-carboxamide [1148];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(1-methylpiperidin-4-yl)oxazole-4-carboxamide [1149];

2-(1-(2-fluoroethyl)piperidin-4-yl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)oxazole-4-carboxamide [1150];

2-(1-isopropylpiperidin-4-yl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)oxazole-4-carboxamide [1151];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)oxazole-4-carboxamide [1152];

2-(3-(dimethylamino)azetidin-1-yl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)thiazole-5-carboxamide [1153];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(piperidin-4-yl)thiazole-4-carboxamide [1154];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)thiazole-4-carboxamide [1155];

2-(1-(2-fluoroethyl)piperidin-4-yl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)thiazole-4-carboxamide [1156];

2-(1-isopropylpiperidin-4-yl)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)thiazole-4-carboxamide [1157];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-1-(2-(methyl-d 3 )propyl-1,1,2,3,3,3-d 6 ) piperidine-4-carboxamide [1158];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(pyrrolidin-1-yl-2,2,5,5-d 4 )acetamide [1159];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(4-(methyl-d 3 )piperazin-1-yl)acetamide [1160];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(morpholino-d 8 )acetamide [1161];

(S)—N-(7-(1-(methyl-d 3 )-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(pyrrolidin-1-yl)propanamide [1162];

1-isobutyl-N-(7-(1-(methyl-d 3 )-1H-pyrazol-4-yl)quinazolin-2-yl)piperidine-4-carboxamide [1163];

N-(7-(1-(methyl-d 3 )-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)acetamide [1164];

N-(7-(1-(methyl-d 3 )-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(pyrrolidin-1-yl)acetamide [1165];

N-(7-(1-(methyl-d 3 )-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(piperidin-1-yl)acetamide [1166];

N-(7-(1-(methyl-d 3 )-1H-pyrazol-4-yl)quinazolin-2-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [1167];

N-(7-(1H-pyrazol-4-yl)quinazolin-2-yl)-2-(4-(methyl-d 3 )piperazin-1-yl)isonicotinamide [1168];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(4-(methyl-d 3 )piperazin-1-yl)isonicotinamide [1169];

N-(7-(1-(methyl-d 3 )-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [1170];

N-(7-(1-(methyl-d 3 )-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(4-(methyl-d 3 )piperazin-1-yl) isonicotinamide [1171];

N-(7-(1-(methyl-d 3 )-1H-pyrazol-4-yl)quinazolin-2-yl)-1-(piperidin-4-yl)-1H-pyrazole-4-carboxamide [1172];

N-(7-(1-(methyl-d 3 )-1H-pyrazol-4-yl)quinazolin-2-yl)-1-(1-methylpiperidin-4-yl)-1H-pyrazole-4-carboxamide [1173];

N-(7-(1-(methyl-d 3 )-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(piperidin-4-yl)oxazole-4-carboxamide [1174];

N-(7-(1-(methyl-d 3 )-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(1-methylpiperidin-4-yl)oxazole-4-carboxamide [1175];

N-(7-(1-ethyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(pyrrolidin-1-yl)acetamide [1176];

N-(7-(1-cyclopropyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(pyrrolidin-1-yl)acetamide [1177];

N-(7-(1-cyclopropyl-1H-pyrazol-4-yl)quinazolin-2-yl)-1-(3,3-trifluoropropyl)piperidine-4-carboxamide [1178];

N-(7-(1-(1-methylpiperidin-4-yl)-1H-pyrazol-4-yl)quinazolin-2-yl)cyclohexanecarboxamide [1179];

2-(pyrrolidin-1-yl)-N-(7-(5-(trifluoromethyl)-1H-pyrazol-4-yl)quinazolin-2-yl)acetamide [1180];

N-(7-(5-(hydroxymethyl)-1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-1-methylpiperidine-4-carboxamide [1181];

N-(7-(5-(hydroxymethyl)-1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)tetrahydro-2H-pyran-4-carboxamide [1182];

N-(7-(5-(azetidin-1-ylmethyl)-1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-4,4-difluorocyclohexane-1-carboxamide [1183];

4,4-difluoro-N-(7-(1-methyl-5-(pyrrolidin-1-ylmethyl)-1H-pyrazol-4-yl)quinazolin-2-yl) cyclohexane-1-carboxamide [1184];

4,4-difluoro-N-(7-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)quinazolin-2-yl) cyclohexane-1-carboxamide [1185];

2-(2-fluoroethyl)-N-(7-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)quinazolin-2-yl)-2-azaspiro[3.3]heptane-6-carboxamide [1186];

tert-butyl 6-((7-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)quinazolin-2-yl)carbamoyl)-2-azaspiro[3.3]heptane-2-carboxylate [1187];

2-fluoro-2-methyl-N-(7-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)quinazolin-2-yl) propanamide [1188];

2-(diethylamino)-N-(7-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)quinazolin-2-yl) acetamide [1189];

trans-4-methoxy-N-(7-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)quinazolin-2-yl) cyclohexane-1-carboxamide [1190];

trans-4-(hydroxymethyl)-N-(7-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)quinazolin-2-yl)cyclohexane-1-carboxamide [1191];

(R)—N-(7-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)quinazolin-2-yl)pyrrolidine-2-carboxamide [1192];

1-isobutyl-N-(7-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)quinazolin-2-yl)piperidine-4-carboxamide [1193];

N-(7-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)quinazolin-2-yl)-1-(oxetan-3-yl) piperidine-4-carboxamide [1194];

1-benzoyl-N-(7-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)quinazolin-2-yl)piperidine-4-carboxamide [1195];

N-(7-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)quinazolin-2-yl)tetrahydro-2H-pyran-4-carboxamide [1196];

N-(7-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(4-methylpiperidin-1-yl)acetamide [1197];

N-(7-(1-(difluoromethyl)-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [1198];

N-(7-(1-ethyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [1199];

N-(7-(1-isopropyl-1H-pyrazol-4-yl)quinazolin-2-yl)-3-(piperidin-4-yloxy)benzamide [1200];

N-(7-(1-isopropyl-1H-pyrazol-4-yl)quinazolin-2-yl)-3-((1-methylpiperidin-4-yl)oxy)benzamide [1201];

N-(7-(1-isopropyl-1H-pyrazol-4-yl)quinazolin-2-yl)-4-(piperidin-4-yloxy)benzamide [1202];

N-(7-(1-cyclopropyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [1203];

4-fluoro-N-(7-(1-(1-methylpiperidin-4-yl)-1H-pyrazol-4-yl)quinazolin-2-yl)benzamide [1204];

4-(difluoromethoxy)-N-(7-(1-(1-methylpiperidin-4-yl)-1H-pyrazol-4-yl)quinazolin-2-yl) benzamide [1205];

5-fluoro-N-(7-(1-(1-methylpiperidin-4-yl)-1H-pyrazol-4-yl)quinazolin-2-yl)nicotinamide [1206];

N 2 -methyl-N 5 -(7-(1-(1-methylpiperidin-4-yl)-1H-pyrazol-4-yl)quinazolin-2-yl)pyridine-2,5-dicarboxamide [1207];

1-isopropyl-N-(7-(1-(1-methylpiperidin-4-yl)-1H-pyrazol-4-yl)quinazolin-2-yl)-1H-pyrazole-4-carboxamide [1208];

2-methyl-N-(7-(1-(1-methylpiperidin-4-yl)-1H-pyrazol-4-yl)quinazolin-2-yl)thiazole-5-carboxamide [1209];

N-(7-(5-amino-1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [1210];

4-(difluoromethoxy)-N-(7-(5-(hydroxymethyl)-1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl) benzamide [1211];

N-(7-(5-(hydroxymethyl)-1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [1212];

N-(7-(5-(hydroxymethyl)-1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(7-methyl-2,7-diazaspiro [3.5]nonan-2-yl)isonicotinamide [1213];

4-fluoro-N-(7-(1-methyl-5-(pyrrolidin-1-ylmethyl)-1H-pyrazol-4-yl)quinazolin-2-yl)benzamide [1214];

4-fluoro-N-(7-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)quinazolin-2-yl)benzamide [1215];

4-(difluoromethoxy)-N-(7-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)quinazolin-2-yl) benzamide [1216];

N-(7-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)quinazolin-2-yl)-3-(pyrrolidin-1-ylmethyl)benzamide [1217];

N-(7-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(7-methyl-2,7-diazaspiro[3.5]nonan-2-yl)isonicotinamide [1218];

N-(7-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)quinazolin-2-yl)-2-morpholinoisonicotinamide [1219];

N-(7-(1-methyl-5-(morpholinomethyl)-1H-pyrazol-4-yl)quinazolin-2-yl)-2-morpholinoisonicotinamide [1220];

N-(7-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)quinazolin-2-yl)-1-((1-(trifluoromethyl) cyclopropyl)methyl)piperidine-4-carboxamide [1221];

3,3-difluoro-N-(7-(5-methyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)quinazolin-2-yl) cyclobutane-1-carboxamide [1222];

N-((4,4-difluorocyclohexyl)methyl)-7-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a] pyrazin-3-yl)quinazolin-2-amine [1223];

N-(7-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)quinazolin-2-yl)-1-((1-(trifluoromethyl)cyclopropyl)methyl)piperidine-4-carboxamide [1224];

N-(7-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)quinazolin-2-yl)-2-(pyrrolidin-1-yl)acetamide [1225];

2-(7-azabicyclo[2.2.1]heptan-7-yl)-N-(7-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)quinazolin-2-yl)acetamide [1226];

(R)—N-(7-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)quinazolin-2-yl)-1-isobutylpiperidine-3-carboxamide [1227];

N-(7-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)quinazolin-2-yl)piperidine-4-carboxamide [1228];

4-fluoro-N-(7-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)quinazolin-2-yl)-1-isobutylpiperidine-4-carboxamide [1229];

N-(7-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)acetamide [1230];

4-fluoro-N-(7-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)quinazolin-2-yl)benzamide [1231];

N-(7-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)quinazolin-2-yl)-3-(4-methylpiperazin-1-yl)benzamide [1232];

N 5 -(7-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)quinazolin-2-yl)-N 2 methylpyridine-2,5-dicarboxamide [1233];

N-(7-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)quinazolin-2-yl)-6-(4-methylpiperazin-1-yl)nicotinamide [1234];

2-(azetidin-3-yloxy)-N-(7-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl) quinazolin-2-yl)isonicotinamide [1235];

N-(7-(1-methyl-1H-pyrazol-5-yl)quinazolin-2-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [1236];

1-methyl-N-(7-(1-methyl-1H-pyrazol-3-yl)quinazolin-2-yl)piperidine-4-carboxamide [1237];

N-(7-(1-methyl-1H-pyrazol-3-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [1238];

2-fluoro-2-methyl-N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)propanamide [1239];

2,2,3,3-tetramethyl-N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)cyclopropane-1-carboxamide [1240];

trans-N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)-4-(pyrrolidin-1-yl)cyclohexane-1-carboxamide [1241];

trans-N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)-4-morpholinocyclohexane-1-carboxamide [1242];

N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)-2-(piperidin-1-yl)acetamide [1243];

1-ethyl-4-fluoro-N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)piperidine-4-carboxamide [1244];

4-fluoro-1-isobutyl-N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)piperidine-4-carboxamide [1245];

N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [1246];

N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)cyclopropanecarboxamide [1247];

4,4-difluoro-N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)cyclohexane-1-carboxamide [1248];

trans-4-(dimethylamino)-N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)cyclohexane-1-carboxamide [1249];

trans-N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)-4-((4-methylpiperazin-1-yl)methyl) cyclohexane-1-carboxamide [1250];

N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)piperidine-4-carboxamide [1251];

1-isobutyl-N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)piperidine-4-carboxamide [1252];

N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)-1-((1-(trifluoromethyl)cyclopropyl) methyl)piperidine-4-carboxamide [1253];

N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)-1-((3-methyloxetan-3-yl)methyl) piperidine-4-carboxamide [1254];

N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)-1-(2-(pyrrolidin-1-yl)acetyl)piperidine-4-carboxamide [1255];

1′-methyl-N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)-[1,4′-bipiperidine]-4-carboxamide [1256];

(R)—N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)piperidine-3-carboxamide [1257];

(R)-1-isobutyl-N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)piperidine-3-carboxamide [1258];

N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)-2-(pyrrolidin-1-yl)acetamide [1259];

N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)acetamide [1260];

2-(7-azabicyclo[2.2.1]heptan-7-yl)-N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl) acetamide [1261];

1-(2-hydroxy-2-methylpropyl)-N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)piperidine-4-carboxamide [1262];

N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)-2-morpholinoacetamide [1263];

2-(4-methoxypiperidin-1-yl)-N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)acetamide [1264];

N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)morpholine-4-carboxamide [1265];

N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)-1-(piperidin-4-yl)-1H-pyrazole-4-carboxamide [1266];

N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)-1-(1-methylpiperidin-4-yl)-1H-pyrazole-4-carboxamide [1267];

1-(1-ethylpiperidin-4-yl)-N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)-1H-pyrazole-4-carboxamide [1268];

1-(1-isopropylpiperidin-4-yl)-N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)-1H-pyrazole-4-carboxamide [1269];

N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)-1-(piperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide [1270];

1-(1-(2-fluoroethyl)piperidin-4-yl)-N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)-1H-1,2,3-triazole-4-carboxamide [1271];

1-(1-isopropylpiperidin-4-yl)-N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)-1H-1,2,3-triazole-4-carboxamide [1272];

N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)-2-(piperidin-4-yl)oxazole-4-carboxamide [1273];

N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)-2-(1-methylpiperidin-4-yl)oxazole-4-carboxamide [1274];

2-(1-isopropylpiperidin-4-yl)-N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)oxazole-4-carboxamide [1275];

2-fluoro-N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)benzamide [1276];

N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)-3-((1-methylpiperidin-4-yl)oxy)benzamide [1277];

N 2 -methyl-N 5 -(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)pyridine-2,5-dicarboxamide [1278];

N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)-6-(4-methylpiperazin-1-yl)nicotinamide [1279];

2-(3-(dimethylamino)azetidin-1-yl)-N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl) isonicotinamide [1280];

N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)-2-(1-methylpiperidin-4-yl)isonicotinamide [1281];

2-(4-(dimethylamino)piperidin-1-yl)-N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl) isonicotinamide [1282];

N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)-2-morpholinoisonicotinamide [1283];

N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [1284];

2-(4-methyl-1,4-diazepan-1-yl)-N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl) isonicotinamide [1285];

2-(4-isopropylpiperazin-1-yl)-N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl) isonicotinamide [1286];

N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)-2-(piperidin-4-ylamino)isonicotinamide [1287];

2-(methyl(1-methylpiperidin-4-yl)amino)-N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl) isonicotinamide [1288];

N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)-2-((1-methylpiperidin-4-yl)thio) isonicotinamide [1289];

2-methyl-N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)-1,2,3,4-tetrahydroisoquinoline-6-carboxamide [1290];

N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)-2-(piperazin-1-yl)isonicotinamide [1291];

N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)-2-(2-(4-methylpiperazin-1-yl)pyridin-4-yl) acetamide [1292];

1,1-bis(methyl-d 3 )-4-(4-((7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)carbamoyl)pyridin-2-yl)piperazin-1-ium [1293];

N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)-2-(4-(methyl-d 3 )piperazin-1-yl) isonicotinamide [1294];

N-(7-(1-methyl-1H-1,2,3-triazol-5-yl)quinazolin-2-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [1295];

N-(7-(4-methyl-4H-1,2,4-triazol-3-yl)quinazolin-2-yl)-2-morpholinoacetamide [1296];

N-(7-(4-methyl-4H-1,2,4-triazol-3-yl)quinazolin-2-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [1297];

4-fluoro-1-isobutyl-N-(7-(4-methyl-4H-1,2,4-triazol-3-yl)quinazolin-2-yl)piperidine-4-carboxamide [1298];

N-(7-(4,5-dimethyl-4H-1,2,4-triazol-3-yl)quinazolin-2-yl)-2-morpholinoacetamide [1299];

N-(7-(4,5-dimethyl-4H-1,2,4-triazol-3-yl)quinazolin-2-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [1300];

N-(7-(1H-1,2,3-triazol-1-yl)quinazolin-2-yl)-4-fluoro-1-isobutylpiperidine-4-carboxamide [1301];

N-(7-(2H-1,2,3-triazol-2-yl)quinazolin-2-yl)-4-fluoro-1-isobutylpiperidine-4-carboxamide [1302];

N-(7-(1H-1,2,4-triazol-1-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [1303];

1-isobutyl-N-(7-(1-methyl-1H-tetrazol-5-yl)quinazolin-2-yl)piperidine-4-carboxamide [1304];

2,2,3,3-tetramethyl-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)cyclopropane-1-carboxamide [1305];

4,4-difluoro-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)cyclohexane-1-carboxamide [1306];

N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)-2-(piperidin-1-yl)acetamide [1307];

2-fluoro-2-methyl-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)propanamide [1308];

1-fluoro-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)cyclopropane-1-carboxamide [1309];

2-methyl-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)-2-azaspiro[3.3]heptane-6-carboxamide [1310];

1-fluoro-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)cyclohexane-1-carboxamide [1311];

trans-4-methoxy-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)cyclohexane-1-carboxamide [1312];

trans-4-(hydroxymethyl)-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)cyclohexane-1-carboxamide [1313];

N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)azetidine-3-carboxamide [1314];

(R)—N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)tetrahydrofuran-2-carboxamide [1315];

1-(2-methoxyethyl)-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)piperidine-4-carboxamide [1316];

N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [1317];

1-isobutyl-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)piperidine-4-carboxamide [1318];

N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)-1-(methylsulfonyl)piperidine-4-carboxamide [1319];

N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)-2-(pyrrolidin-1-yl)propanamide [1320];

2-isopropoxy-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)acetamide [1321];

3-isopropoxy-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)propanamide [1322];

N-(7-(1,2-dimethyl-1H-imidazol-5-yl)quinazolin-2-yl)cyclopropanecarboxamide [1323];

N-(7-(1,2-dimethyl-1H-imidazol-5-yl)quinazolin-2-yl)cyclohexanecarboxamide [1324];

N-(7-(1,2-dimethyl-1H-imidazol-5-yl)quinazolin-2-yl)-4,4-difluorocyclohexane-1-carboxamide [1325];

(S)—N-(7-(1,2-dimethyl-1H-imidazol-5-yl)quinazolin-2-yl)tetrahydrofuran-2-carboxamide [1326];

N-(7-(1,2-dimethyl-1H-imidazol-5-yl)quinazolin-2-yl)-3,3-difluorocyclobutane-1-carboxamide [1327];

N-(7-(1,2-dimethyl-1H-imidazol-5-yl)quinazolin-2-yl)-1-fluorocyclopropane-1-carboxamide [1328];

N-(7-(1,2-dimethyl-1H-imidazol-5-yl)quinazolin-2-yl)morpholine-4-carboxamide [1329];

N-(7-(1,2-dimethyl-1H-imidazol-5-yl)quinazolin-2-yl)morpholine-d 8 -4-carboxamide [1330];

1-methyl-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)-1H-pyrazole-4-carboxamide [1331];

1-ethyl-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)-1H-pyrazole-4-carboxamide [1332];

1-isopropyl-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)-1H-pyrazole-4-carboxamide [1333];

1-cyclopropyl-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)-1H-pyrazole-4-carboxamide [1334];

1-isobutyl-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)-1H-pyrazole-4-carboxamide [1335];

1-methyl-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)-1H-pyrazole-3-carboxamide [1336];

N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)-2-(1-methyl-1H-pyrazol-4-yl)acetamide [1337];

1-methyl-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)-1H-imidazole-4-carboxamide [1338];

1-isopropyl-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)-1H-imidazole-4-carboxamide [1339];

N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)-1-(tetrahydro-2H-pyran-4-yl)-1H-imidazole-4-carboxamide [1340];

1,2-dimethyl-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)-1H-imidazole-5-carboxamide [1341];

1-methyl-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)-1H-1,2,4-triazole-3-carboxamide [1342];

2-methyl-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)oxazole-4-carboxamide [1343];

2-isopropyl-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)oxazole-4-carboxamide [1344];

4-methyl-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)oxazole-2-carboxamide [1345];

4-methyl-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)thiazole-2-carboxamide [1346];

2-methyl-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)thiazole-4-carboxamide [1347];

5-methyl-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)-1,3,4-oxadiazole-2-carboxamide [1348];

5-methyl-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)-1,3,4-thiadiazole-2-carboxamide [1349];

1-isopropyl-N-(7-(1-isopropyl-1H-imidazol-5-yl)quinazolin-2-yl)-1H-pyrazole-4-carboxamide [1350];

N-(7-(1,2-dimethyl-1H-imidazol-5-yl)quinazolin-2-yl)-1-methyl-1H-pyrazole-4-carboxamide [1351];

N-(7-(1,2-dimethyl-1H-imidazol-5-yl)quinazolin-2-yl)-1-isopropyl-1H-pyrazole-4-carboxamide [1352];

N-(7-(1,2-dimethyl-1H-imidazol-5-yl)quinazolin-2-yl)-2-methylthiazole-5-carboxamide [1353];

4-fluoro-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)benzamide [1354];

4-(difluoromethoxy)-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)benzamide [1355];

N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)-3-(pyrrolidin-1-ylmethyl)benzamide [1356];

2-fluoro-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)benzamide-3,4,5,6-d 4 [1357];

4-fluoro-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)benzamide-2,3,5,6-d 4 [1358];

2-chloro-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)benzamide-3,4,5,6-d 4 [1359];

4-chloro-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)benzamide-2,3,5,6-d 4 [1360];

4-(methyl-d 3 )—N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)benzamide [1361];

4-methyl-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)benzamide-2,3,5,6-d 4 [1362];

4-(methyl-d 3 )—N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)benzamide-2,3,5,6-d 4 [1363];

4-(methoxy-d 3 )—N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)benzamide [1364];

4-(methoxy-d 3 )—N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)benzamide-2,3,5,6-d 4 [1365];

4-methoxy-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)benzamide-2,3,5,6-d 4 [1366];

(E)-N-(7-(1,2-dimethyl-1H-imidazol-5-yl)quinazolin-2-yl)-3-(phenyl-2,3,4,5,6-d 5 )acrylamide [1367];

(E)-N-(7-(1,2-dimethyl-1H-imidazol-5-yl)quinazolin-2-yl)-3-(phenyl-2,3,4,5,6-d 5 )acrylamide-2,3-d 2 [1368];

N-(7-(1,2-dimethyl-1H-imidazol-5-yl)quinazolin-2-yl)-2-(4-fluorophenyl)acetamide-2,2-d 2 [1369];

(E)-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)-3-(phenyl-2,3,4,5,6-d 5 )acrylamide [1370];

(E)-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)-3-(phenyl-2,3,4,5,6-d 5 )acrylamide-2,3-d 2 [1371];

2-(4-fluorophenyl)-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)acetamide-2,2-d 2 [1372];

N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [1373];

2-(dimethylamino)-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)isonicotinamide [1374];

2-(3-aminoazetidin-1-yl)-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)isonicotinamide [1375];

N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)-2-(pyrrolidin-1-yl)isonicotinamide [1376];

N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)-2-(piperidin-1-yl)isonicotinamide [1377];

N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)-2-morpholinoisonicotinamide [1378];

2-(4-isopropylpiperazin-1-yl)-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)isonicotinamide [1379];

2-(4-cyclopropylpiperazin-1-yl)-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl) isonicotinamide [1380];

N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)-2-(2,7-diazaspiro[3.5]nonan-2-yl) isonicotinamide [1381];

N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)-2-(7-methyl-2,7-diazaspiro[3.5]nonan-2-yl) isonicotinamide [1382];

N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)isoindoline-5-carboxamide [1383];

2-methyl-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)isoindoline-5-carboxamide [1384];

2-(azetidin-1-yl)-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)isonicotinamide [1385];

2-methoxy-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)isonicotinamide [1386];

2-methyl-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)isonicotinamide [1387];

2-cyano-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)isonicotinamide [1388];

2-(3,3-difluoroazetidin-1-yl)-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)isonicotinamide [1389];

2-(4,4-difluoropiperidin-1-yl)-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)isonicotinamide [1390];

2-isopropoxy-N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)isonicotinamide [1391];

N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)-2-(pyrrolidin-1-yl-2,2,5,5-d 4 )isonicotinamide [1392];

N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)-2-(pyrrolidin-1-yl-d 8 )isonicotinamide [1393];

N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)-2-(piperidin-1-yl-d 10 )isonicotinamide [1394];

N-(7-(1-methyl-1H-imidazol-5-yl)quinazolin-2-yl)-2-(morpholino-d 8 )isonicotinamide [1395];

N-(7-(1,2-dimethyl-1H-imidazol-5-yl)quinazolin-2-yl)-4-isopropoxybenzamide [1396];

N-(7-(1,2-dimethyl-1H-imidazol-5-yl)quinazolin-2-yl)-4-(piperidin-4-yloxy)benzamide [1397];

4-(benzyloxy)-N-(7-(1,2-dimethyl-1H-imidazol-5-yl)quinazolin-2-yl)benzamide [1398];

N-(7-(1,2-dimethyl-1H-imidazol-5-yl)quinazolin-2-yl)-2-fluorobenzamide-3,4,5,6-d 4 [1399];

N-(7-(1,2-dimethyl-1H-imidazol-5-yl)quinazolin-2-yl)-4-fluorobenzamide-2,3,5,6-d 4 [1400];

2-chloro-N-(7-(1,2-dimethyl-1H-imidazol-5-yl)quinazolin-2-yl)benzamide-3,4,5,6-d 4 [1401];

4-chloro-N-(7-(1,2-dimethyl-1H-imidazol-5-yl)quinazolin-2-yl)benzamide-2,3,5,6-d 4 [1402];

N-(7-(1,2-dimethyl-1H-imidazol-5-yl)quinazolin-2-yl)-4-(methyl-d 3 )benzamide [1403];

N-(7-(1,2-dimethyl-1H-imidazol-5-yl)quinazolin-2-yl)-4-methylbenzamide-2,3,5,6-d 4 [1404];

N-(7-(1,2-dimethyl-1H-imidazol-5-yl)quinazolin-2-yl)-4-(methyl-d 3 )benzamide-2,3,5,6-d 4 [1405];

N-(7-(1,2-dimethyl-1H-imidazol-5-yl)quinazolin-2-yl)-4-(methoxy-d 3 )benzamide [1406];

N-(7-(1,2-dimethyl-1H-imidazol-5-yl)quinazolin-2-yl)-4-(methoxy-d 3 )benzamide-2,3,5,6-d 4 [1407];

N-(7-(1,2-dimethyl-1H-imidazol-5-yl)quinazolin-2-yl)-4-methoxybenzamide-2,3,5,6-d 4 [1408];

N-(7-(1,2-dimethyl-1H-imidazol-5-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [1409];

N-(7-(1,2-dimethyl-1H-imidazol-5-yl)quinazolin-2-yl)-2-morpholinoisonicotinamide [1410];

N-(7-(1,2-dimethyl-1H-imidazol-5-yl)quinazolin-2-yl)-2-(pyrrolidin-1-yl)isonicotinamide [1411];

N-(7-(1,2-dimethyl-1H-imidazol-5-yl)quinazolin-2-yl)-2-(dimethylamino)isonicotinamide [1412];

N-(7-(1,2-dimethyl-1H-imidazol-5-yl)quinazolin-2-yl)-2-(pyrrolidin-1-yl-2,2,5,5-d 4 ) isonicotinamide [1413];

N-(7-(1,2-dimethyl-1H-imidazol-5-yl)quinazolin-2-yl)-2-(pyrrolidin-1-yl-d 8 )isonicotinamide [1414];

N-(7-(1,2-dimethyl-1H-imidazol-5-yl)quinazolin-2-yl)-2-(piperidin-1-yl-d 10 )isonicotinamide [1415];

N-(7-(1,2-dimethyl-1H-imidazol-5-yl)quinazolin-2-yl)-2-(morpholino-d 8 )isonicotinamide [1416];

N-(7-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)quinazolin-2-yl)cyclopropanecarboxamide [1417];

N-(7-(7-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)quinazolin-2-yl) cyclopropanecarboxamide [1418];

3,3-difluoro-N-(7-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)quinazolin-2-yl)cyclobutane-1-carboxamide [1419];

(R)—N-(7-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)quinazolin-2-yl)pyrrolidine-2-carboxamide [1420];

(R)—N-(7-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)quinazolin-2-yl)piperidine-3-carboxamide [1421];

1-methyl-N-(7-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)quinazolin-2-yl)piperidine-4-carboxamide [1422];

N-(7-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)quinazolin-2-yl)-1-((1-(trifluoromethyl) cyclopropyl)methyl)piperidine-4-carboxamide [1423];

1-benzoyl-N-(7-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)quinazolin-2-yl)piperidine-4-carboxamide [1424];

4-fluoro-1-isobutyl-N-(7-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)quinazolin-2-yl) piperidine-4-carboxamide [1425];

(R)-2-(2-methylpyrrolidin-1-yl)-N-(7-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)quinazolin-2-yl)acetamide [1426];

2-(cyclobutyl(methyl)amino)-N-(7-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)quinazolin-2-yl)acetamide [1427];

4-fluoro-N-(7-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)quinazolin-2-yl)benzamide [1428];

4-isopropoxy-N-(7-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)quinazolin-2-yl)benzamide [1429];

4-(difluoromethoxy)-N-(7-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)quinazolin-2-yl) benzamide [1430];

2-((2-(dimethylamino)ethyl)amino)-N-(7-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl) quinazolin-2-yl)isonicotinamide [1431];

2-((1-isopropylpiperidin-4-yl)oxy)-N-(7-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl) quinazolin-2-yl)isonicotinamide [1432];

N-(7-(oxazol-5-yl)quinazolin-2-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [1433];

N-(7-(oxazol-5-yl)quinazolin-2-yl)cyclopropanecarboxamide [1434];

(R)—N-(7-(oxazol-5-yl)quinazolin-2-yl)tetrahydrofuran-2-carboxamide [1435];

(R)—N-(7-(oxazol-5-yl)quinazolin-2-yl)piperidine-3-carboxamide [1436];

N-(7-(oxazol-5-yl)quinazolin-2-yl)tetrahydro-2H-pyran-4-carboxamide [1437];

N-(7-(oxazol-5-yl)quinazolin-2-yl)-1-(2-(pyrrolidin-1-yl)acetyl)piperidine-4-carboxamide [1438];

1′-methyl-N-(7-(oxazol-5-yl)quinazolin-2-yl)-[1,4′-bipiperidine]-4-carboxamide [1439];

cis-4-morpholino-N-(7-(oxazol-5-yl)quinazolin-2-yl)cyclohexane-1-carboxamide [1440];

2-(cyclobutyl(methyl)amino)-N-(7-(oxazol-5-yl)quinazolin-2-yl)acetamide [1441];

N-(7-(oxazol-5-yl)quinazolin-2-yl)-2-(pyrrolidin-1-yl)acetamide [1442];

(R)-2-(2-methylpyrrolidin-1-yl)-N-(7-(oxazol-5-yl)quinazolin-2-yl)acetamide [1443];

2-(4-methylpiperazin-1-yl)-N-(7-(oxazol-5-yl)quinazolin-2-yl)acetamide [1444];

trans-4-((4-methylpiperazin-1-yl)methyl)-N-(7-(oxazol-5-yl)quinazolin-2-yl)cyclohexane-1-carboxamide [1445];

1-(2,2-difluoropropyl)-N-(7-(oxazol-5-yl)quinazolin-2-yl)piperidine-4-carboxamide [1446];

trans-4-(hydroxymethyl)-N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl)cyclohexane-1-carboxamide [1447];

trans-4-(methylamino)-N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl)cyclohexane-1-carboxamide [1448];

trans-4-((1,3-difluoropropan-2-yl)amino)-N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl) cyclohexane-1-carboxamide [1449];

trans-N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl)-4-((propan-2-yl-1,1,1,3,3,3-d 6 )amino) cyclohexane-1-carboxamide [1450];

trans-4-((2,2-difluoroethyl)amino)-N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl)cyclohexane-1-carboxamide [1451];

trans-N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl)-4-((3,3,3-trifluoropropyl)amino)cyclohexane-1-carboxamide [1452];

trans-4-((2-methoxyethyl)amino)-N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl)cyclohexane-1-carboxamide [1453];

trans-4-(dimethylamino)-N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl)cyclohexane-1-carboxamide [1454];

trans-4-(bis(methyl-d 3 )amino)-N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl)cyclohexane-1-carboxamide [1455];

cis-4-(dimethylamino)-N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl)cyclohexane-1-carboxamide [1456];

trans-4-((2,2-difluoroethyl)(methyl)amino)-N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl) cyclohexane-1-carboxamide [1457];

trans-4-(methyl(oxetan-3-yl)amino)-N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl)cyclohexane-1-carboxamide [1458];

trans-4-((2-fluoroethyl)amino)-N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl)cyclohexane-1-carboxamide [1459];

trans-4-(2-(fluoromethyl)aziridin-1-yl)-N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl)cyclohexane-1-carboxamide [1460];

trans-4-((3-fluoroazetidin-1-yl)methyl)-N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl)cyclohexane-1-carboxamide [1461];

trans-N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl)-3-morpholinocyclobutane-1-carboxamide [1462];

trans-N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl)-4-morpholinocyclohexane-1-carboxamide [1463];

N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl)-2-(piperidin-1-yl)acetamide [1464];

2-(4-methoxypiperidin-1-yl)-N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl)acetamide [1465];

N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)acetamide [1466];

N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl)morpholine-4-carboxamide [1467];

N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl)-2-morpholinoacetamide [1468];

N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl)-3-morpholinopropanamide [1469];

1-methyl-N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl)piperidine-4-carboxamide [1470];

1-(2,2-difluoropropyl)-N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl)piperidine-4-carboxamide [1471];

N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl)-4-morpholinopiperidine-1-carboxamide [1472];

4-((1,3-difluoropropan-2-yl)amino)-N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl)piperidine-1-carboxamide [1473];

(1R,3s,5S)-3-((1,3-difluoropropan-2-yl)amino)-N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl)-8-azabicyclo[3.2.1]octane-8-carboxamide [1474];

(1R,3s,5S)-3-((1,3-difluoropropan-2-yl)amino)-N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl)-8-azabicyclo[3.2.1]octane-8-carboxamide [1475];

4-(dimethylamino)-N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl)piperidine-1-carboxamide [1476];

4-((2,2-difluoroethyl)(methyl)amino)-N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl)piperidine-1-carboxamide [1477];

(3S,4S)-4-amino-3-fluoro-N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl)piperidine-1-carboxamide [1478];

(3S,4S)-3-fluoro-4-(methylamino)-N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl)piperidine-1-carboxamide [1479];

(3R,4R)-4-amino-3-fluoro-N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl)piperidine-1-carboxamide [1480];

(3R,4R)-3-fluoro-4-(methylamino)-N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl)piperidine-1-carboxamide [1481];

4-((2-fluoroethyl)amino)-N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl)piperidine-1-carboxamide [1482];

4-((2,2-difluoroethyl)amino)-N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl)piperidine-1-carboxamide [1483];

(1R,3s,5S)-3-amino-N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl)-8-azabicyclo [3.2.1]octane-8-carboxamide [1484];

(1R,3r,5S)-3-amino-N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl)-8-azabicyclo [3.2.1]octane-8-carboxamide [1485];

(1R,3r,5S)-3-((2-fluoroethyl)amino)-N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl)-8-azabicyclo [3.2.1]octane-8-carboxamide [1486];

(1R,3r,5S)-3-((2,2-difluoroethyl)amino)-N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl)-8-azabicyclo[3.2.1]octane-8-carboxamide [1487];

(1R,3s,5S)—N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl)-3-((3,3,3-trifluoropropyl)amino)-8-azabicyclo[3.2.1]octane-8-carboxamide [1488];

(3S,4S)-3-fluoro-4-(isopropylamino)-N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl)piperidine-1-carboxamide [1489];

N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl)-5,6-dihydroimidazo[1,2-a]pyrazine-7(8H)-carboxamide [1490];

2-methyl-N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl)-5,6-dihydroimidazo[1,2-a]pyrazine-7(8H)-carboxamide [1491];

N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl)-2-(morpholino-d 8 )acetamide [1492];

trans-N-(7-(2-methyloxazol-4-yl)quinazolin-2-yl)-4-(4-methylpiperazin-1-yl)cyclohexane-1-carboxamide [1493];

N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl)-1-(1-methylpiperidin-4-yl)-1H-pyrazole-4-carboxamide [1494];

2-(1H-imidazol-1-yl)-N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl)acetamide [1495];

4-(difluoromethoxy)-N-(7-(oxazol-5-yl)quinazolin-2-yl)benzamide [1496];

3-((1-methylpiperidin-4-yl)oxy)-N-(7-(oxazol-5-yl)quinazolin-2-yl)benzamide [1497];

N-(7-(oxazol-5-yl)quinazolin-2-yl)isonicotinamide [1498];

2-(3-aminoazetidin-1-yl)-N-(7-(oxazol-5-yl)quinazolin-2-yl)isonicotinamide [1499];

2-(1-methylpiperidin-4-yl)-N-(7-(oxazol-5-yl)quinazolin-2-yl)isonicotinamide [1500];

1′-methyl-N-(7-(oxazol-5-yl)quinazolin-2-yl)-1′,2′,3′,6′-tetrahydro-[2,4′-bipyridine]-4-carboxamide [1501];

2-(4-methylpiperazin-1-yl)-N-(7-(oxazol-5-yl)quinazolin-2-yl)isonicotinamide [1502];

2-(7-methyl-2,7-diazaspiro[3.5]nonan-2-yl)-N-(7-(oxazol-5-yl)quinazolin-2-yl)isonicotinamide [1503];

N-(7-(oxazol-5-yl)quinazolin-2-yl)-2-(2,7-diazaspiro[3.5]nonan-7-yl)isonicotinamide [1504];

N-(7-(oxazol-5-yl)quinazolin-2-yl)-2-(piperidin-4-ylamino)isonicotinamide [1505];

2-methyl-N-(7-(oxazol-5-yl)quinazolin-2-yl)isoindoline-5-carboxamide [1506];

N-(7-(oxazol-5-yl)quinazolin-2-yl)-1,2,3,4-tetrahydroisoquinoline-7-carboxamide [1507];

N-(7-(2-methyloxazol-5-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [1508];

N-(7-(3-methylisoxazol-5-yl)quinazolin-2-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [1509];

4-fluoro-1-isobutyl-N-(7-(5-methyl-1,3,4-oxadiazol-2-yl)quinazolin-2-yl)piperidine-4-carboxamide [1510];

1-isobutyl-N-(7-(5-methyl-1,3,4-oxadiazol-2-yl)quinazolin-2-yl)piperidine-4-carboxamide [1511];

N-(7-(5-(dimethylamino)-1,3,4-oxadiazol-2-yl)quinazolin-2-yl)piperidine-4-carboxamide [1512];

N-(7-(5-(dimethylamino)-1,3,4-oxadiazol-2-yl)quinazolin-2-yl)-1-methylpiperidine-4-carboxamide [1513];

N-(7-(5-methyl-1,3,4-oxadiazol-2-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [1514];

3,3-difluoro-N-(7-(thiazol-5-yl)quinazolin-2-yl)cyclobutane-1-carboxamide [1515];

2-methyl-N-(7-(thiazol-5-yl)quinazolin-2-yl)-2-azaspiro[3.3]heptane-6-carboxamide [1516];

1-fluoro-N-(7-(thiazol-5-yl)quinazolin-2-yl)cyclohexane-1-carboxamide [1517];

trans-4-(dimethylamino)-N-(7-(thiazol-5-yl)quinazolin-2-yl)cyclohexane-1-carboxamide [1518];

trans-4-((3-fluoroazetidin-1-yl)methyl)-N-(7-(thiazol-5-yl)quinazolin-2-yl)cyclohexane-1-carboxamide [1519];

N-(7-(thiazol-5-yl)quinazolin-2-yl)azetidine-3-carboxamide [1520];

1-methyl-N-(7-(thiazol-5-yl)quinazolin-2-yl)piperidine-4-carboxamide [1521];

1-(2,2-difluoropropyl)-N-(7-(thiazol-5-yl)quinazolin-2-yl)piperidine-4-carboxamide [1522];

1-(oxetan-3-yl)-N-(7-(thiazol-5-yl)quinazolin-2-yl)piperidine-4-carboxamide [1523];

1-(2-(pyrrolidin-1-yl)acetyl)-N-(7-(thiazol-5-yl)quinazolin-2-yl)piperidine-4-carboxamide [1524];

1′-methyl-N-(7-(thiazol-5-yl)quinazolin-2-yl)-[1,4′-bipiperidine]-4-carboxamide [1525];

2-(pyrrolidin-1-yl)-N-(7-(thiazol-5-yl)quinazolin-2-yl)propanamide [1526];

2-(piperidin-1-yl)-N-(7-(thiazol-5-yl)quinazolin-2-yl)acetamide [1527];

2-(4-methylpiperazin-1-yl)-N-(7-(thiazol-5-yl)quinazolin-2-yl)acetamide [1528];

2-morpholino-N-(7-(thiazol-5-yl)quinazolin-2-yl)acetamide [1529];

4-(piperidin-4-yloxy)-N-(7-(thiazol-5-yl)quinazolin-2-yl)benzamide [1530];

N-(7-(thiazol-5-yl)quinazolin-2-yl)isonicotinamide [1531];

6-(4-methylpiperazin-1-yl)-N-(7-(thiazol-5-yl)quinazolin-2-yl)nicotinamide [1532];

1′-methyl-N-(7-(thiazol-5-yl)quinazolin-2-yl)-1′,2′,3′,6′-tetrahydro-[2,4′-bipyridine]-4-carboxamide [1533];

2-(3-(dimethylamino)azetidin-1-yl)-N-(7-(thiazol-5-yl)quinazolin-2-yl)isonicotinamide [1534];

2-(4-(dimethylamino)piperidin-1-yl)-N-(7-(thiazol-5-yl)quinazolin-2-yl)isonicotinamide [1535];

2-(4-methylpiperazin-1-yl)-N-(7-(thiazol-5-yl)quinazolin-2-yl)isonicotinamide [1536];

2-((1-methylpiperidin-4-yl)thio)-N-(7-(thiazol-5-yl)quinazolin-2-yl)isonicotinamide [1537];

N-(7-(thiazol-5-yl)quinazolin-2-yl)-1,2,3,4-tetrahydroisoquinoline-7-carboxamide [1538];

trans-4-((1,3-difluoropropan-2-yl)amino)-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl) cyclohexane-1-carboxamide [1539];

N-(7-(2-methylthiazol-5-yl)quinazolin-2-yl)morpholine-4-carboxamide [1540];

N-(7-(2-methylthiazol-5-yl)quinazolin-2-yl)-2-(pyrrolidin-1-yl)acetamide [1541];

2-((1R,4R)-2-oxa-5-azabicyclo[2.2.1]heptan-5-yl)-N-(7-(2-methylthiazol-5-yl)quinazolin-2-yl) acetamide [1542];

N-(7-(2-methylthiazol-5-yl)quinazolin-2-yl)-2-morpholinoacetamide [1543];

N-(7-(2-methylthiazol-5-yl)quinazolin-2-yl)-2-(morpholino-d 8 )acetamide [1544];

2-(4-methylpiperazin-1-yl)-N-(7-(2-methylthiazol-5-yl)quinazolin-2-yl)acetamide [1545];

1-methyl-N-(7-(2-methylthiazol-5-yl)quinazolin-2-yl)piperidine-4-carboxamide [1546];

N-(7-(2-methylthiazol-5-yl)quinazolin-2-yl)isonicotinamide [1547];

N-(7-(2-methylthiazol-5-yl)quinazolin-2-yl)nicotinamide [1548];

2-(4-methylpiperazin-1-yl)-N-(7-(2-methylthiazol-5-yl)quinazolin-2-yl)isonicotinamide [1549];

trans-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-4-morpholinocyclohexane-1-carboxamide [1550];

trans-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-4-(4-methylpiperazin-1-yl) cyclohexane-1-carboxamide [1551];

4-isopropyl-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)piperazine-1-carboxamide [1552];

4-((2-methoxyethyl)(methyl)amino)-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl) piperidine-1-carboxamide [1553];

4-((1,3-difluoropropan-2-yl)amino)-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl) piperidine-1-carboxamide [1554];

N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-4-((3,3,3-trifluoropropyl)amino)piperidine-1-carboxamide [1555];

4-((2-fluoroethyl)amino)-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)piperidine-1-carboxamide [1556];

(3R,4S)-4-amino-3-fluoro-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)piperidine-1-carboxamide [1557];

(3R,4R)-4-amino-3-fluoro-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)piperidine-1-carboxamide [1558];

(3S,4S)-3-fluoro-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-4-(methylamino) piperidine-1-carboxamide [1559];

(3R,4R)-3-fluoro-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-4-(methylamino) piperidine-1-carboxamide [1560];

4-amino-3,3-difluoro-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)piperidine-1-carboxamide [1561];

(3R,4R)-3-fluoro-4-(isopropylamino)-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl) piperidine-1-carboxamide [1562];

(3R,4S)-3-fluoro-4-(isopropylamino)-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl) piperidine-1-carboxamide [1563];

3,3-difluoro-4-(isopropylamino)-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)piperidine-1-carboxamide [1564];

(3S,4S)-3-fluoro-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-4-((propan-2-yl-1,1,1,3,3,3-d 6 )amino)piperidine-1-carboxamide [1565];

(1R,3s,5S)-3-((1,3-difluoropropan-2-yl)amino)-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-8-azabicyclo[3.2.1]octane-8-carboxamide [1566];

(1R,3s,5S)-3-((1,3-difluoropropan-2-yl)amino)-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-8-azabicyclo[3.2.1]octane-8-carboxamide [1567];

4-(dimethylamino)-N-(7-(2-methylthiazol-5-yl)quinazolin-2-yl)piperidine-1-carboxamide [1568];

4-((2,2-difluoroethyl)amino)-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)piperidine-1-carboxamide [1569];

4-((2,2-difluoroethyl)(methyl-d 3 )amino)-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl) piperidine-1-carboxamide [1570];

N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-4-morpholinopiperidine-1-carboxamide [1571];

N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-4-(4-methylpiperazin-1-yl)piperidine-1-carboxamide [1572];

(R)-3,4-dimethyl-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)piperazine-1-carboxamide [1573];

(S)-3,4-dimethyl-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)piperazine-1-carboxamide [1574];

(1R,3r,5 S)-3-((2-fluoroethyl)amino)-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-8-azabicyclo[3.2.1]octane-8-carboxamide [1575];

(1R,3r,5S)-3-((2,2-difluoroethyl)amino)-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-8-azabicyclo[3.2.1]octane-8-carboxamide [1576];

(1R,3r,5S)-3-amino-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-8-azabicyclo[3.2.1] octane-8-carboxamide [1577];

(1S,4S)-5-methyl-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-2,5-diazabicyclo[2.2.1]heptane-2-carboxamide [1578];

(1R,4R)-5-methyl-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-2,5-diazabicyclo[2.2.1] heptane-2-carboxamide [1579];

8-methyl-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-3,8-diazabicyclo[3.2.1]octane-3-carboxamide [1580];

3-methyl-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-3,8-diazabicyclo[3.2.1]octane-8-carboxamide [1581];

N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-5,6-dihydroimidazo[1,2-a]pyrazine-7(8H)-carboxamide [1582];

2-(4-methylpiperazin-1-yl)-N-(7-(5-methylthiazol-2-yl)quinazolin-2-yl)isonicotinamide [1583];

2-(4-methylpiperazin-1-yl)-N-(7-(4-methylthiazol-2-yl)quinazolin-2-yl)isonicotinamide [1584];

N-(7-(2-(methylamino)thiazol-5-yl)quinazolin-2-yl)piperidine-4-carboxamide [1585];

1-methyl-N-(7-(2-(methylamino)thiazol-5-yl)quinazolin-2-yl)piperidine-4-carboxamide [1586];

N-(7-(2-(diethylamino)thiazol-5-yl)quinazolin-2-yl)-2-(4-fluoropiperidin-1-yl)acetamide [1587];

N-(7-(2-(diethylamino)thiazol-5-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)acetamide [1588];

N-(7-(2-aminothiazol-5-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [1589];

N-(7-(2-(methylamino)thiazol-5-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [1590];

N-(7-(2-(dimethylamino)thiazol-5-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [1591];

2-(4-isopropylpiperazin-1-yl)-N-(7-(2-(methylamino)thiazol-5-yl)quinazolin-2-yl) isonicotinamide [1592];

2-(3-(dimethylamino)azetidin-1-yl)-N-(7-(2-(methylamino)thiazol-5-yl)quinazolin-2-yl) isonicotinamide [1593];

2-(3-(dimethylamino)azetidin-1-yl)-N-(7-(2-(dimethylamino)thiazol-5-yl)quinazolin-2-yl) isonicotinamide [1594];

2-(3-aminoazetidin-1-yl)-N-(7-(2-(dimethylamino)thiazol-5-yl)quinazolin-2-yl)isonicotinamide [1595];

N-(7-(5-chlorothiazol-2-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [1596];

2-(2-(2-(4-methylpiperazin-1-yl)isonicotinamido)quinazolin-7-yl)thiazole-5-carboxamide [1597];

N-(7-(isothiazol-4-yl)quinazolin-2-yl)-1-methylpiperidine-4-carboxamide [1598];

N-(7-(1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-4-(difluoromethoxy)benzamide [1599];

N-(7-(1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-4-(piperidin-4-yloxy)benzamide [1600];

N-(7-(1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-4-((1-methylpiperidin-4-yl)oxy)benzamide [1601];

N-(7-(1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-3-((1-methylpiperidin-4-yl)oxy)benzamide [1602];

N 5 -(7-(1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-N 2 -methylpyridine-2,5-dicarboxamide [1603];

N-(7-(1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-6-(4-methylpiperazin-1-yl)nicotinamide [1604];

N-(7-(1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-1′-methyl-1′,2′,3′,6′-tetrahydro-[2,4′-bipyridine]-4-carboxamide [1605];

N-(7-(1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-2-(3-(dimethylamino)azetidin-1-yl)isonicotinamide [1606];

N-(7-(1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [1607];

N-(7-(1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-2-(4-isopropylpiperazin-1-yl)isonicotinamide [1608];

N-(7-(1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-2-morpholinoisonicotinamide [1609];

1-fluoro-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)cyclohexane-1-carboxamide [1610];

trans-4-methoxy-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)cyclohexane-1-carboxamide [1611];

cis-4-methoxy-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)cyclohexane-1-carboxamide [1612];

trans-4-amino-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)cyclohexane-1-carboxamide [1613];

trans-4-(dimethylamino)-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)cyclohexane-1-carboxamide [1614];

trans-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-4-morpholinocyclohexane-1-carboxamide [1615];

trans-4-(hydroxymethyl)-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)cyclohexane-1-carboxamide [1616];

N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)piperidine-4-carboxamide [1617];

4-fluoro-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)piperidine-4-carboxamide [1618];

1-methyl-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)piperidine-4-carboxamide [1619];

4-fluoro-1-methyl-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)piperidine-4-carboxamide [1620];

1-(2-fluoroethyl)-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)piperidine-4-carboxamide [1621];

1-(2,2-difluoroethyl)-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)piperidine-4-carboxamide [1622];

N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [1623];

1-(2,2-difluoropropyl)-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)piperidine-4-carboxamide [1624];

1-benzoyl-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)piperidine-4-carboxamide [1625];

N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-2-(pyrrolidin-1-yl)acetamide [1626];

N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-2-(piperidin-1-yl)acetamide [1627];

2-(4-methoxypiperidin-1-yl)-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)acetamide [1628];

N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)acetamide [1629];

N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-2-morpholinoacetamide [1630];

(R)—N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-2-(3-methylmorpholino)acetamide [1631];

2-(7-azabicyclo[2.2.1]heptan-7-yl)-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl) acetamide [1632];

2-((1R,4R)-2-oxa-5-azabicyclo[2.2.1]heptan-5-yl)-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl) quinazolin-2-yl)acetamide [1633];

2-(3-oxa-8-azabicyclo[3.2.1]octan-8-yl)-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl) acetamide [1634];

2-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl) acetamide [1635];

N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-2-(1,4-oxazepan-4-yl)acetamide [1636];

N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-2-morpholinoacetamide-2,2-d 2 [1637];

N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-2-(morpholino-d 8 )acetamide [1638];

1-methyl-3-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-1-(1-methylpiperidin-4-yl)urea [1639];

(3S,4S)-4-amino-3-fluoro-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)piperidine-1-carboxamide [1640];

(3S,4S)-4-(dimethylamino)-3-fluoro-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl) piperidine-1-carboxamide [1641];

N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)morpholine-4-carboxamide [1642];

N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-4-(methylamino)piperidine-1-carboxamide [1643];

4-(dimethylamino)-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)piperidine-1-carboxamide [1644];

4-((2,2-difluoroethyl)(methyl)amino)-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl) piperidine-1-carboxamide [1645];

(3S,4S)-3-fluoro-4-(isopropylamino)-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl) piperidine-1-carboxamide [1646];

2-methyl-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-5,6-dihydroimidazo[1,2-a] pyrazine-7(8H)-carboxamide [1647];

4-methyl-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)piperazine-1-carboxamide [1648];

N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-1-(1-methylpiperidin-4-yl)-1H-pyrazole-4-carboxamide [1649];

1-(1-isopropylpiperidin-4-yl)-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-1H-pyrazole-4-carboxamide [1650];

N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-1-(1-methylpiperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide [1651];

N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-2-(piperidin-4-yl)oxazole-4-carboxamide [1652];

N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-2-(1-methylpiperidin-4-yl)oxazole-4-carboxamide [1653];

2-(3-(dimethylamino)azetidin-1-yl)-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl) isonicotinamide [1654];

1′-methyl-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-1′,2′,3′,6′-tetrahydro-[2,4′-bipyridine]-4-carboxamide [1655];

N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [1656];

2-(methyl(1-methylpiperidin-4-yl)amino)-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl) isonicotinamide [1657];

2-(azetidin-3-yloxy)-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)isonicotinamide [1658];

N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-3-((1-methylpiperidin-4-yl)oxy)benzamide [1659];

N-(7-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-2-((1-methylpiperidin-4-yl)thio) isonicotinamide [1660];

6-(4-methylpiperazin-1-yl)-N-(7-(5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl)quinazolin-2-yl) nicotinamide [1661];

2-(4-methylpiperazin-1-yl)-N-(7-(5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl)quinazolin-2-yl) isonicotinamide [1662];

N-(7-(5-amino-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [1663];

N-(7-(5-(dimethylamino)-1,3,4-thiadiazol-2-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [1664];

N-(7-(3-amino-5-fluorophenyl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [1665];

N-(7-(3-fluoro-5-(isopropylamino)phenyl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [1666];

1-methyl-N-(7-(pyridin-2-yl)quinazolin-2-yl)piperidine-4-carboxamide [1667];

2-(4-methylpiperazin-1-yl)-N-(7-(pyridin-2-yl)quinazolin-2-yl)isonicotinamide [1668];

2-(4-methylpiperazin-1-yl)-N-(7-(pyridin-4-yl)quinazolin-2-yl)isonicotinamide [1669];

N-(7-(pyridin-3-yl)quinazolin-2-yl)cyclopropanecarboxamide [1670];

N-(7-(pyridin-3-yl)quinazolin-2-yl)-2-(pyrrolidin-1-yl)acetamide [1671];

1-methyl-N-(7-(pyridin-3-yl)quinazolin-2-yl)piperidine-4-carboxamide [1672];

N-(7-(pyridin-3-yl)quinazolin-2-yl)quinuclidine-4-carboxamide [1673];

2-morpholino-N-(7-(pyridin-3-yl)quinazolin-2-yl)acetamide [1674];

2-(morpholino-d 8 )—N-(7-(pyridin-3-yl)quinazolin-2-yl)acetamide [1675];

2-(4-methylpiperazin-1-yl)-N-(7-(pyridin-3-yl)quinazolin-2-yl)acetamide [1676];

2-(4-methyl-1,4-diazepan-1-yl)-N-(7-(pyridin-3-yl)quinazolin-2-yl)acetamide [1677];

2-(4-methylpiperazin-1-yl)-N-(7-(pyridin-3-yl)quinazolin-2-yl)isonicotinamide [1678];

2-(2-methyl-1H-imidazol-1-yl)-N-(7-(pyridin-3-yl)quinazolin-2-yl)acetamide [1679];

2-(1H-imidazol-1-yl)-N-(7-(pyridin-3-yl)quinazolin-2-yl)acetamide [1680];

2-(piperidin-4-yl)-N-(7-(pyridin-3-yl)quinazolin-2-yl)oxazole-4-carboxamide [1681];

2-(1-methylpiperidin-4-yl)-N-(7-(pyridin-3-yl)quinazolin-2-yl)oxazole-4-carboxamide [1682];

2-(1-isopropylpiperidin-4-yl)-N-(7-(pyridin-3-yl)quinazolin-2-yl)oxazole-4-carboxamide [1683];

trans-N-(7-(5-fluoropyridin-3-yl)quinazolin-2-yl)-3-morpholinocyclobutane-1-carboxamide [1684];

trans-N-(7-(5-fluoropyridin-3-yl)quinazolin-2-yl)-4-((4-methylpiperazin-1-yl)methyl) cyclohexane-1-carboxamide [1685];

N-(7-(5-fluoropyridin-3-yl)quinazolin-2-yl)-2-(pyrrolidin-1-yl)acetamide [1686];

N-(7-(5-fluoropyridin-3-yl)quinazolin-2-yl)-1-methylpiperidine-4-carboxamide [1687];

N-(7-(5-fluoropyridin-3-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)acetamide [1688];

N-(7-(6-fluoropyridin-3-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)acetamide [1689];

N-(7-(5-fluoropyridin-3-yl)quinazolin-2-yl)-2-morpholinoacetamide [1690];

N-(7-(5-fluoropyridin-3-yl)quinazolin-2-yl)-3-morpholinopropanamide [1691];

N-(7-(5-fluoropyridin-3-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [1692];

N-(7-(5-fluoropyridin-3-yl)quinazolin-2-yl)-2-(piperidin-4-yl)oxazole-4-carboxamide [1693];

N-(7-(5-fluoropyridin-3-yl)quinazolin-2-yl)-2-(1-methylpiperidin-4-yl)oxazole-4-carboxamide [1694];

N-(7-(5-fluoropyridin-3-yl)quinazolin-2-yl)-2-(1-isopropylpiperidin-4-yl)oxazole-4-carboxamide [1695];

N-(7-(5-chloropyridin-3-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [1696];

N-(7-(5-methylpyridin-3-yl)quinazolin-2-yl)-2-morpholinoacetamide [1697];

N-(7-(5-(difluoromethyl)pyridin-3-yl)quinazolin-2-yl)-3-(piperidin-4-yl)benzamide [1698];

N-(7-(5-(difluoromethyl)pyridin-3-yl)quinazolin-2-yl)-3-(1-methylpiperidin-4-yl)benzamide [1699];

N-(7-(5-(difluoromethyl)pyridin-3-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [1700];

2-(4-methylpiperazin-1-yl)-N-(7-(5-(trifluoromethyl)pyridin-3-yl)quinazolin-2-yl)acetamide [1701];

2-(4-methylpiperazin-1-yl)-N-(7-(6-(trifluoromethyl)pyridin-3-yl)quinazolin-2-yl)acetamide [1702];

N-(7-(5-(hydroxymethyl)pyridin-3-yl)quinazolin-2-yl)-1-methylpiperidine-4-carboxamide [1703];

N-(7-(5-cyanopyridin-3-yl)quinazolin-2-yl)-1-methylpiperidine-4-carboxamide [1704];

N-(7-(5-methoxypyridin-3-yl)quinazolin-2-yl)-1-methylpiperidine-4-carboxamide [1705];

N-(7-(5-methoxypyridin-3-yl)quinazolin-2-yl)-2-morpholinoacetamide [1706];

N-(7-(5-methoxypyridin-3-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [1707];

4-fluoro-N-(7-(5-(piperidin-4-yloxy)pyridin-3-yl)quinazolin-2-yl)benzamide [1708];

N-(7-(5-aminopyridin-3-yl)quinazolin-2-yl)-4-fluorobenzamide [1709];

N-(7-(5-aminopyridin-3-yl)quinazolin-2-yl)-4-(piperidin-4-yloxy)benzamide [1710];

N-(7-(5-aminopyridin-3-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [1711];

N-(7-(5-aminopyridin-3-yl)quinazolin-2-yl)-2-(piperidin-4-yl)oxazole-4-carboxamide [1712];

N-(7-(6-aminopyridin-3-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [1713];

N-(7-(6-(methylamino)pyridin-3-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [1714];

N-(7-(5-(isopropylamino)pyridin-3-yl)quinazolin-2-yl)-3-(piperidin-4-yl)benzamide [1715];

N-(7-(5-(isopropylamino)pyridin-3-yl)quinazolin-2-yl)-3-(1-methylpiperidin-4-yl)benzamide [1716];

N-(7-(5-(isopropylamino)pyridin-3-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1l-yl) isonicotinamide [1717];

N-(7-(5-(piperidin-4-ylamino)pyridin-3-yl)quinazolin-2-yl)cyclohexanecarboxamide [1718];

4-fluoro-N-(7-(5-(piperidin-4-ylamino)pyridin-3-yl)quinazolin-2-yl)benzamide [1719];

4-fluoro-N-(7-(5-((1-methylpiperidin-4-yl)amino)pyridin-3-yl)quinazolin-2-yl)benzamide [1720];

N-(7-(5-acetamidopyridin-3-yl)quinazolin-2-yl)-1-methylpiperidine-4-carboxamide [1721];

N-(7-(5-(dimethylamino)pyridin-3-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [1722];

N-(7-(6-(dimethylamino)pyridin-3-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [1723];

1-methyl-N-(7-(5-(pyrrolidin-1-yl)pyridin-3-yl)quinazolin-2-yl)piperidine-4-carboxamide [1724];

N-(7-(5-(pyrrolidin-1-ylmethyl)pyridin-3-yl)quinazolin-2-yl)cyclopropanecarboxamide [1725];

4-fluoro-N-(7-(5-(pyrrolidin-1-ylmethyl)pyridin-3-yl)quinazolin-2-yl)benzamide [1726];

N-(7-(5-((4-hydroxypiperidin-1-yl)methyl)pyridin-3-yl)quinazolin-2-yl) cyclopropanecarboxamide [1727];

4-fluoro-N-(7-(5-((4-hydroxypiperidin-1-yl)methyl)pyridin-3-yl)quinazolin-2-yl)benzamide [1728];

N-(7-(5-(piperazin-1-ylmethyl)pyridin-3-yl)quinazolin-2-yl)cyclopropanecarboxamide [1729];

N-(7-(5-((4-methylpiperazin-1-yl)methyl)pyridin-3-yl)quinazolin-2-yl)cyclopropanecarboxamide [1730];

N-(7-(5-(morpholinomethyl)pyridin-3-yl)quinazolin-2-yl)cyclopropanecarboxamide [1731];

N-methyl-5-(2-(1-methylpiperidine-4-carboxamido)quinazolin-7-yl)nicotinamide [1732];

N-methyl-5-(2-(2-(4-methylpiperazin-1-yl)isonicotinamido)quinazolin-7-yl)nicotinamide [1733];

N-(7-(pyridin-3-yl-d 4 )quinazolin-2-yl)-2-(pyrrolidin-1-yl)acetamide [1734];

2-(4-methylpiperazin-1-yl)-N-(7-(pyridin-3-yl-d 4 )quinazolin-2-yl)acetamide [1735];

2-morpholino-N-(7-(pyridin-3-yl-d 4 )quinazolin-2-yl)acetamide [1736];

1-methyl-N-(7-(2-methylpyrimidin-5-yl)quinazolin-2-yl)piperidine-4-carboxamide [1737];

2-(4-methylpiperazin-1-yl)-N-(7-(2-methylpyrimidin-5-yl)quinazolin-2-yl)isonicotinamide [1738];

N-(7-(2-aminopyrimidin-5-yl)quinazolin-2-yl)-1-methylpiperidine-4-carboxamide [1739];

2-morpholino-N-(7-(pyridazin-3-yl)quinazolin-2-yl)acetamide [1740];

2-morpholino-N-(7-(pyridazin-4-yl)quinazolin-2-yl)acetamide [1741];

N-(7-(pyridazin-4-yl)quinazolin-2-yl)-2-(pyrrolidin-1-yl)acetamide [1742];

trans-3-morpholino-N-(7-(pyrazin-2-yl)quinazolin-2-yl)cyclobutane-1-carboxamide [1743];

trans-4-(dimethylamino)-N-(7-(pyrazin-2-yl)quinazolin-2-yl)cyclohexane-1-carboxamide [1744];

trans-4-morpholino-N-(7-(pyrazin-2-yl)quinazolin-2-yl)cyclohexane-1-carboxamide [1745];

trans-4-((3-fluoroazetidin-1-yl)methyl)-N-(7-(pyrazin-2-yl)quinazolin-2-yl)cyclohexane-1-carboxamide [1746];

trans-4-((4-methylpiperazin-1-yl)methyl)-N-(7-(pyrazin-2-yl)quinazolin-2-yl)cyclohexane-1-carboxamide [1747];

N-(7-(pyrazin-2-yl)quinazolin-2-yl)-2-(pyrrolidin-1-yl)acetamide [1748];

1-methyl-N-(7-(pyrazin-2-yl)quinazolin-2-yl)piperidine-4-carboxamide [1749];

4-fluoro-1-methyl-N-(7-(pyrazin-2-yl)quinazolin-2-yl)piperidine-4-carboxamide [1750];

1-(2-fluoroethyl)-N-(7-(pyrazin-2-yl)quinazolin-2-yl)piperidine-4-carboxamide [1751];

1-(oxetan-3-yl)-N-(7-(pyrazin-2-yl)quinazolin-2-yl)piperidine-4-carboxamide [1752];

2-morpholino-N-(7-(pyrazin-2-yl)quinazolin-2-yl)acetamide [1753];

1-methyl-N-(7-(pyrazin-2-yl)quinazolin-2-yl)azepane-4-carboxamide [1754];

1-isobutyl-N-(7-(pyrazin-2-yl)quinazolin-2-yl)azepane-4-carboxamide [1755];

1-(2-hydroxy-2-methylpropyl)-N-(7-(pyrazin-2-yl)quinazolin-2-yl)azepane-4-carboxamide [1756];

4-(morpholinomethyl)-N-(7-(pyrazin-2-yl)quinazolin-2-yl)benzamide [1757];

2-(4-methylpiperazin-1-yl)-N-(7-(pyrazin-2-yl)quinazolin-2-yl)isonicotinamide [1758];

N-(7-(6-(methylamino)pyrazin-2-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [1759];

N-(7-(6-(isopropylamino)pyrazin-2-yl)quinazolin-2-yl)azetidine-3-carboxamide [1760];

N-(7-(6-(isopropylamino)pyrazin-2-yl)quinazolin-2-yl)piperidine-4-carboxamide [1761];

N-(7-(6-(isopropylamino)pyrazin-2-yl)quinazolin-2-yl)-1-methylpiperidine-4-carboxamide [1762];

1-(2-fluoroethyl)-N-(7-(6-(isopropylamino)pyrazin-2-yl)quinazolin-2-yl)piperidine-4-carboxamide [1763];

1-isopropyl-N-(7-(6-(isopropylamino)pyrazin-2-yl)quinazolin-2-yl)piperidine-4-carboxamide [1764];

1-isopentyl-N-(7-(6-(isopropylamino)pyrazin-2-yl)quinazolin-2-yl)piperidine-4-carboxamide [1765];

N-(7-(6-(isopropylamino)pyrazin-2-yl)quinazolin-2-yl)-3-(piperidin-4-yl)benzamide [1766];

N-(7-(6-(isopropylamino)pyrazin-2-yl)quinazolin-2-yl)-3-(1-methylpiperidin-4-yl)benzamide [1767];

N-(7-(6-(isopropylamino)pyrazin-2-yl)quinazolin-2-yl)-1-(piperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide [1768];

1-(1-(2-fluoroethyl)piperidin-4-yl)-N-(7-(6-(isopropylamino)pyrazin-2-yl)quinazolin-2-yl)-1H-1,2,3-triazole-4-carboxamide [1769];

N-(7-(6-(isopropylamino)pyrazin-2-yl)quinazolin-2-yl)-1-(1-isopropylpiperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide [1770];

N-(7-(6-(isopropylamino)pyrazin-2-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [1771];

N-(7-(6-(tert-butylamino)pyrazin-2-yl)quinazolin-2-yl)-2-(3-(dimethylamino)azetidin-1-yl) isonicotinamide [1772];

N-(7-(6-(tert-butylamino)pyrazin-2-yl)quinazolin-2-yl)-1′-methyl-1′,2′,3′,6′-tetrahydro-[2,4′-bipyridine]-4-carboxamide [1773];

N-(7-(6-(tert-butylamino)pyrazin-2-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [1774];

N-(7-(6-(tert-butylamino)pyrazin-2-yl)quinazolin-2-yl)-2-(4-isopropylpiperazin-1-yl) isonicotinamide [1775];

N-(7-(6-(tert-butylamino)pyrazin-2-yl)quinazolin-2-yl)-2-morpholinoisonicotinamide [1776];

N-(7-(6-(((3-fluoroazetidin-3-yl)methyl)amino)pyrazin-2-yl)quinazolin-2-yl) cyclopropanecarboxamide [1777];

4-fluoro-N-(7-(6-(((3-fluoroazetidin-3-yl)methyl)amino)pyrazin-2-yl)quinazolin-2-yl)benzamide [1778];

N-(7-(6-(piperidin-4-ylamino)pyrazin-2-yl)quinazolin-2-yl)cyclobutanecarboxamide [1779];

3,3-difluoro-N-(7-(6-(piperidin-4-ylamino)pyrazin-2-yl)quinazolin-2-yl)cyclobutane-1-carboxamide [1780];

N-(7-(6-(piperidin-4-ylamino)pyrazin-2-yl)quinazolin-2-yl)cyclopentanecarboxamide [1781];

4,4-difluoro-N-(7-(6-(piperidin-4-ylamino)pyrazin-2-yl)quinazolin-2-yl)cyclohexane-1-carboxamide [1782];

N-(7-(6-(piperidin-4-ylamino)pyrazin-2-yl)quinazolin-2-yl)tetrahydro-2H-pyran-4-carboxamide [1783];

4-fluoro-N-(7-(6-(piperidin-4-ylamino)pyrazin-2-yl)quinazolin-2-yl)benzamide [1784];

N-(7-(6-(((3 S,4S)-3-fluoropiperidin-4-yl)amino)pyrazin-2-yl)quinazolin-2-yl) cyclopropanecarboxamide [1785];

4-fluoro-N-(7-(6-(((3S,4S)-3-fluoropiperidin-4-yl)amino)pyrazin-2-yl)quinazolin-2-yl)benzamide [1786];

N-(7-(6-((1-methylpiperidin-4-yl)amino)pyrazin-2-yl)quinazolin-2-yl)cyclobutanecarboxamide [1787];

N-(7-(6-((1-methylpiperidin-4-yl)amino)pyrazin-2-yl)quinazolin-2-yl)cyclopentanecarboxamide [1788];

4-fluoro-N-(7-(6-((1-methylpiperidin-4-yl)amino)pyrazin-2-yl)quinazolin-2-yl)benzamide [1789];

N-(7-(6-((1-isopropylpiperidin-4-yl)amino)pyrazin-2-yl)quinazolin-2-yl) cyclopropanecarboxamide [1790];

3,3-difluoro-N-(7-(6-((1-isopropylpiperidin-4-yl)amino)pyrazin-2-yl)quinazolin-2-yl) cyclobutane-1-carboxamide [1791];

N-(7-(6-((1-isopropylpiperidin-4-yl)amino)pyrazin-2-yl)quinazolin-2-yl) cyclopentanecarboxamide [1792];

4-fluoro-N-(7-(6-((1-isopropylpiperidin-4-yl)amino)pyrazin-2-yl)quinazolin-2-yl)benzamide [1793];

N-(7-(6-(dimethylamino)pyrazin-2-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [1794];

N-(7-(6-(diethylamino)pyrazin-2-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [1795];

N-(7-(6-(3-aminoazetidin-1-yl)pyrazin-2-yl)quinazolin-2-yl)-4-fluorobenzamide [1796];

2-(4-methylpiperazin-1-yl)-N-(7-(6-(pyrrolidin-1-yl)pyrazin-2-yl)quinazolin-2-yl)isonicotinamide [1797];

N-(7-(6-(azetidin-3-ylmethoxy)pyrazin-2-yl)quinazolin-2-yl)-4-fluorobenzamide [1798];

N-(7-(6-(azetidin-3-yloxy)pyrazin-2-yl)quinazolin-2-yl)-4-fluorobenzamide [1799];

N-(7-(1H-pyrrolo[2,3-b]pyridin-5-yl)quinazolin-2-yl)-1-(1-methylpiperidin-4-yl)-1H-pyrazole-4-carboxamide [1800];

N-(7-(1H-pyrrolo[3,2-b]pyridin-6-yl)quinazolin-2-yl)-1-(1-methylpiperidin-4-yl)-1H-pyrazole-4-carboxamide [1801];

N-(7-(1H-pyrrolo[2,3-c]pyridin-4-yl)quinazolin-2-yl)-1-(1-methylpiperidin-4-yl)-1H-pyrazole-4-carboxamide [1802];

N-(7-(1H-pyrrolo[2,3-b]pyridin-5-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [1803];

N-(7-(1H-pyrrolo[3,2-b]pyridin-6-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [1804];

N-(7-(1H-pyrrolo[2,3-c]pyridin-4-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [1805];

2-(4-methylpiperazin-1-yl)-N-(7-(oxazolo[5,4-b]pyridin-6-yl)quinazolin-2-yl)isonicotinamide [1806];

N-(7-(2-methyl-1H-pyrrolo[2,3-b]pyridin-5-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [1807];

N-(7-(3-methyl-1H-pyrrolo[2,3-b]pyridin-5-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [1808];

N-(7-(2-methyl-1H-pyrrolo[3,2-b]pyridin-6-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [1809];

N-(7-(5H-pyrrolo[2,3-b]pyrazin-2-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [1810];

N-(7-(5H-pyrrolo[2,3-b]pyrazin-3-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [1811];

1-isopropyl-N-(7-(6-(piperidin-4-ylamino)pyrazin-2-yl)quinazolin-2-yl)-1H-pyrazole-4-carboxamide [1812];

1-isopropyl-N-(7-(6-((1-methylpiperidin-4-yl)amino)pyrazin-2-yl)quinazolin-2-yl)-1H-pyrazole-4-carboxamide [1813];

trans-4-((2-fluoroethyl)amino)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)cyclohexane-1-carboxamide [4566];

trans-4-((2-methoxyethyl)amino)-N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)cyclohexane-1-carboxamide [4567];

tert-butyl (trans-4-((7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)carbamoyl)cyclohexyl) carbamate [4568];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-((1-methylpiperidin-4-yl)amino) isonicotinamide [4569];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)thiazole-5-carboxamide [4570];

N-(7-(1-methyl-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(4-methylpiperazin-1-yl)thiazole-5-carboxamide [4571];

N-(7-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)quinazolin-2-yl)-2-(2,7-diazaspiro[3.5] nonan-2-yl)isonicotinamide [4572];

N-(7-(1-methyl-1H-1,2,3-triazol-4-yl)quinazolin-2-yl)-4-(piperidin-4-yloxy)benzamide [4573];

N-(7-(1-methyl-1H-tetrazol-5-yl)quinazolin-2-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [4574];

N-(7-(1,2-dimethyl-1H-imidazol-5-yl)quinazolin-2-yl)-2-(pyrrolidin-1-yl)propanamide [4575];

N-(7-(1,2-dimethyl-1H-imidazol-5-yl)quinazolin-2-yl)-2-(piperidin-1-yl)propanamide [4576];

4-isopropoxy-N-(7-(7-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)quinazolin-2-yl) benzamide [4577];

trans-3-morpholino-N-(7-(oxazol-5-yl)quinazolin-2-yl)cyclobutane-1-carboxamide [4578];

trans-4-(hydroxymethyl)-N-(7-(oxazol-5-yl)quinazolin-2-yl)cyclohexane-1-carboxamide [4579];

N-(7-(oxazol-5-yl)quinazolin-2-yl)piperidine-4-carboxamide [4580];

4-morpholino-N-(7-(oxazol-5-yl)quinazolin-2-yl)piperidine-1-carboxamide [4581];

N-(7-(oxazol-5-yl)quinazolin-2-yl)-4-(piperidin-4-yloxy)benzamide [4582];

N-(7-(oxazol-5-yl)quinazolin-2-yl)-3-(piperidin-4-yloxy)benzamide [4583];

2-methyl-N-(7-(oxazol-5-yl)quinazolin-2-yl)-5,6-dihydroimidazo[1,2-a]pyrazine-7(8H)-carboxamide [4584];

2-(1H-imidazol-1-yl)-N-(7-(oxazol-5-yl)quinazolin-2-yl)acetamide [4585];

trans-4-(hydroxymethyl)-N-(7-(thiazol-5-yl)quinazolin-2-yl)cyclohexane-1-carboxamide [4586];

trans-4-(dimethylamino)-N-(7-(thiazol-5-yl)quinazolin-2-yl)cyclohexane-1-carboxamide [4587];

N-(7-(thiazol-5-yl)quinazolin-2-yl)-1-((1-(trifluoromethyl)cyclopropyl)methyl)piperidine-4-carboxamide [4588];

trans-4-(hydroxymethyl)-N-(7-(2-methylthiazol-5-yl)quinazolin-2-yl)cyclohexane-1-carboxamide [4589];

trans-4-(dimethylamino)-N-(7-(2-methylthiazol-5-yl)quinazolin-2-yl)cyclohexane-1-carboxamide [4590];

N-(7-(2-methylthiazol-5-yl)quinazolin-2-yl)-1-(oxetan-3-yl)piperidine-4-carboxamide [4591];

N-(7-(2-methylthiazol-5-yl)quinazolin-2-yl)-1-(2-(pyrrolidin-1-yl)acetyl)piperidine-4-carboxamide [4592];

2-((1S,4S)-2-oxa-5-azabicyclo[2.2.1]heptan-5-yl)-N-(7-(5-methyl-1,3,4-thiadiazol-2-yl) quinazolin-2-yl)acetamide [4593];

N-(7-(5-(cyano(4-hydroxypiperidin-1-yl)methyl)pyridin-3-yl)quinazolin-2-yl) cyclopropanecarboxamide [4594];

4-fluoro-N-(7-(6-((1-methylazetidin-3-yl)methoxy)pyrazin-2-yl)quinazolin-2-yl)benzamide [4595];

1-isopropyl-N-(7-(6-((1-methylpiperidin-4-yl)amino)pyrazin-2-yl)quinazolin-2-yl)-1H-pyrazole-4-carboxamide [4596]; or a pharmaceutically acceptable salt thereof.

14. The compound of claim 1 , wherein the compound of Formula I is selected from the group consisting of:

N-(6-(1H-pyrazol-4-yl)cinnolin-3-yl)-1-isobutylpiperidine-4-carboxamide [1814];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)cyclopropanecarboxamide [1815];

4,4-difluoro-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)cyclohexane-1-carboxamide [1816];

trans-4-methoxy-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)cyclohexane-1-carboxamide [1817];

trans-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-4-morpholinocyclohexane-1-carboxamide [1818];

trans-4-((3-fluoroazetidin-1-yl)methyl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl) cyclohexane-1-carboxamide [1819];

trans-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-4-((4-methylpiperazin-1-yl)methyl) cyclohexane-1-carboxamide [1820];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(pyrrolidin-1-yl)acetamide [1821];

(S)-2-(3-fluoropyrrolidin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)acetamide [1822];

(S)—N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)tetrahydrofuran-2-carboxamide [1823];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)piperidine-4-carboxamide [1824];

1-methyl-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)piperidine-4-carboxamide [1825];

1-isopropyl-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)piperidine-4-carboxamide [1826];

1-(tert-butyl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)piperidine-4-carboxamide [1827];

1-cyclopropyl-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)piperidine-4-carboxamide [1828];

1-isobutyl-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)piperidine-4-carboxamide [1829];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-1-neopentylpiperidine-4-carboxamide [1830];

1-(2-fluoroethyl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)piperidine-4-carboxamide [1831];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [1832];

1-butyl-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)piperidine-4-carboxamide [1833];

1-benzoyl-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)piperidine-4-carboxamide [1834];

1-(2,2-difluoropropyl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)piperidine-4-carboxamide [1835];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)azetidine-3-carboxamide [1836];

1-(2,2-difluoroethyl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)piperidine-4-carboxamide [1837];

1-(2-fluoro-2-methylpropyl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)piperidine-4-carboxamide [1838];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-1-(oxetan-3-yl)piperidine-4-carboxamide [1839];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-1-((3-methyloxetan-3-yl)methyl)piperidine-4-carboxamide [1840];

1-(2-methoxyethyl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)piperidine-4-carboxamide [1841];

1-(2-isopropoxyethyl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)piperidine-4-carboxamide [1842];

1,1-diisobutyl-4-((6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)carbamoyl)piperidin-1-ium [1843];

4-fluoro-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)piperidine-4-carboxamide [1844];

4-fluoro-1-methyl-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)piperidine-4-carboxamide [1845];

4-fluoro-1-isobutyl-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)piperidine-4-carboxamide [1846];

(S)—N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)piperidine-3-carboxamide [1847];

(R)—N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)piperidine-3-carboxamide [1848];

(S)-1-isobutyl-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)piperidine-3-carboxamide [1849];

(R)-1-isobutyl-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)piperidine-3-carboxamide [1850];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)tetrahydro-2H-pyran-4-carboxamide [1851];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(piperidin-1-yl)acetamide [1852];

2-(4-fluoropiperidin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)acetamide [1853];

trans-4-amino-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)cyclohexane-1-carboxamide [1854];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)acetamide [1855];

(S)—N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)piperidine-2-carboxamide [1856];

2-(4-isobutylpiperazin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)acetamide [1857];

2-(3,3-dimethylazetidin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)acetamide [1858];

(R)-2-(3-fluoropyrrolidin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)acetamide [1859];

(S)—N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(2-methylpyrrolidin-1-yl)acetamide [1860];

2-(3-azabicyclo[3.1.0]hexan-3-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)acetamide [1861];

2-(7-azabicyclo[2.2.1]heptan-7-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)acetamide [1862];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(4-methylpiperidin-1-yl)acetamide [1863];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(4-(trifluoromethyl)piperidin-1-yl)acetamide [1864];

2-(4-(difluoromethyl)piperidin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)acetamide [1865];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(6-azaspiro[2.5]octan-6-yl)acetamide [1866];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(pyrrolidin-1-yl)propanamide [1867];

(R)—N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(2-methylpyrrolidin-1-yl)acetamide [1868];

2-(cyclobutyl(methyl)amino)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)acetamide [1869];

2-(diethylamino)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)acetamide [1870];

7-(2-fluoroethyl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-7-azaspiro[3.5]nonane-2-carboxamide [1871];

4-methyl-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)piperazine-1-carboxamide [1872];

(S)—N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(pyrrolidin-1-yl)propanamide [1873];

(R)—N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(pyrrolidin-1-yl)propanamide [1874];

(R)—N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)pyrrolidine-2-carboxamide [1875];

2-methyl-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-azaspiro[3.3]heptane-6-carboxamide [1876];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(2,2,2-trifluoroacetyl)-2-azaspiro[3.3]heptane-6-carboxamide [1877];

2-(2-fluoroethyl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-azaspiro[3.3]heptane-6-carboxamide [1878];

trans-4-(dimethylamino)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)cyclohexane-1-carboxamide [1879];

1-acetyl-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)piperidine-4-carboxamide [1880];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-1-((1-(trifluoromethyl)cyclopropyl)methyl) piperidine-4-carboxamide [1881];

(S)-1-(2-fluoropropyl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)piperidine-4-carboxamide [1882];

(R)-1-(2-fluoropropyl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)piperidine-4-carboxamide [1883];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(piperidin-1-yl)propanamide [1884];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-1-(methylsulfonyl)piperidine-4-carboxamide [1885];

1′-methyl-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-[1,4′-bipiperidine]-4-carboxamide [1886];

trans-4-(hydroxymethyl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)cyclohexane-1-carboxamide [1887];

methyl 2-(4-((6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)carbamoyl)piperidin-1-yl)acetate [1888];

1-benzyl-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)piperidine-4-carboxamide [1889];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-1-(2-(pyrrolidin-1-yl)acetyl)piperidine-4-carboxamide [1890];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-morpholinoacetamide [1891];

(S)—N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(3-methylmorpholino)acetamide [1892];

(R)—N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(3-methylmorpholino)acetamide [1893];

(S)—N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(2-methylmorpholino)acetamide [1894];

2-((2R,6S)-2,6-dimethylmorpholino)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)acetamide [1895];

2-((1S,4S)-2-oxa-5-azabicyclo [2.2.1]heptan-5-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)acetamide [1896];

2-((1R,4R)-2-oxa-5-azabicyclo[2.2.1]heptan-5-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)acetamide [1897];

2-(3-oxa-8-azabicyclo[3.2.1]octan-8-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)acetamide [1898];

(S)—N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-morpholinopropanamide [1899];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(morpholin-2-yl)acetamide [1900];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(4-methylmorpholin-2-yl)acetamide [1901];

2-(4-ethylpiperazin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)acetamide [1902];

2-(4-isopropylpiperazin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)acetamide [1903];

2-(4-cyclopropylpiperazin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)acetamide [1904];

2-(4-(2-fluoroethyl)piperazin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)acetamide [1905];

(S)-2-(2,4-dimethylpiperazin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)acetamide [1906];

1-(2-hydroxyethyl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)piperidine-4-carboxamide [1907];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-1-(pyridin-2-ylmethyl)piperidine-4-carboxamide [1908];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-1-(oxazol-2-ylmethyl)piperidine-4-carboxamide [1909];

(R)—N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-1-oxotetrahydro-1H-pyrrolo[1,2-c]imidazole-2(3H)-carboxamide [1910];

(R)-1-methyl-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)pyrrolidine-2-carboxamide [1911];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-1-(tetrahydro-2H-pyran-4-yl)piperidine-4-carboxamide [1912];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-1-(pyrimidin-2-ylmethyl)piperidine-4-carboxamide [1913];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-1-(pyrazin-2-ylmethyl)piperidine-4-carboxamide [1914];

1-((5-methyl-1,2,4-oxadiazol-3-yl)methyl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl) piperidine-4-carboxamide [1915];

1-(2-hydroxy-2-methylpropyl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)piperidine-4-carboxamide [1916];

tert-butyl 2-(4-((6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)carbamoyl)piperidin-1-yl)acetate [1917];

2-(4-((6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)carbamoyl)piperidin-1-yl)acetic acid [1918];

2-(4-methyl-1,4-diazepan-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)acetamide [1919];

tert-butyl (6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)carbamate [1920];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)but-2-ynamide [1921];

trans-4-((6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)carbamoyl)cyclohexane-1-carboxylic acid [1922];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-3-morpholinopropanamide [1923];

trans-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-3-morpholinocyclobutane-1-carboxamide [1924];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)quinuclidine-4-carboxamide [1925];

1-isobutyl-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)azepane-4-carboxamide [1926];

2-(4-methoxypiperidin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)acetamide [1927];

2-(4-hydroxypiperidin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)acetamide [1928];

3-(hydroxymethyl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)bicyclo[1.1.1]pentane-1-carboxamide [1929];

1-methyl-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)azepane-4-carboxamide [1930];

trans-4-(dimethylamino)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)cyclohexane-1-carboxamide [1931];

trans-4-(bis(methyl-d3)amino)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)cyclohexane-1-carboxamide [1932];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-3-((4-methylpiperazin-1-yl)methyl)bicyclo [1.1.1]pentane-1-carboxamide [1933];

methyl trans-4-((6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)carbamoyl)cyclohexane-1-carboxylate [1934];

2-(1-isobutylpyrrolidin-3-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)acetamide [1935];

trans-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-4-(4-methylpiperazine-1-carbonyl) cyclohexane-1-carboxamide [1936];

1-isobutyl-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)piperidine-4-carboxamide [1937];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-1-(phenylsulfonyl)piperidine-4-carboxamide [1938];

8-methyl-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-3,8-diazabicyclo[3.2.1]octane-3-carboxamide [1939];

3-methyl-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-3,8-diazabicyclo[3.2.1]octane-8-carboxamide [1940];

(1R,3 s,5 S)-3-amino-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-8-azabicyclo[3.2.1]octane-8-carboxamide [1941];

(1R,3s,5S)—N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-3-((3,3,3-trifluoropropyl)amino)-8-azabicyclo[3.2.1]octane-8-carboxamide [1942];

(1R,3s,5S)-3-((1,3-difluoropropan-2-yl)amino)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-8-azabicyclo[3.2.1]octane-8-carboxamide [1943];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)morpholine-4-carboxamide [1944];

4-(dimethylamino)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)piperidine-1-carboxamide [1945];

(S)-2,4-dimethyl-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)piperazine-1-carboxamide [1946];

1-methyl-3-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-1-(1-methylpiperidin-4-yl)urea [1947];

1-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-3-(1-methylpiperidin-4-yl)urea [1948];

4-isopropyl-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)piperazine-1-carboxamide [1949];

(R)-3,4-dimethyl-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)piperazine-1-carboxamide [1950];

N-(6-(1H-pyrazol-4-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [1951];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-3-(piperazin-1-yl)benzamide [1952];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-3-(4-methylpiperazin-1-yl)benzamide [1953];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-3-(pyrrolidin-1-ylmethyl)benzamide [1954];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-3-(piperidin-4-yloxy)benzamide [1955];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-3-((1-methylpiperidin-4-yl)oxy)benzamide [1956];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-4-(piperidin-4-yloxy)benzamide [1957];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-4-((1-methylpiperidin-4-yl)oxy)benzamide [1958];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(piperazin-1-yl)isonicotinamide [1959];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [1960];

2-(4-isopropylpiperazin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)isonicotinamide [1961];

2-(4-cyclopropylpiperazin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)isonicotinamide [1962];

2-(4-(2-fluoroethyl)piperazin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl) isonicotinamide [1963];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-6-(4-methylpiperazin-1-yl)nicotinamide [1964];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-5-(piperidin-4-yloxy)nicotinamide [1965];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(piperidin-4-yloxy)isonicotinamide [1966];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-((1-methylpiperidin-4-yl)oxy)isonicotinamide [1967];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-5-(piperidin-4-ylamino)nicotinamide [1968];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-5-((1-methylpiperidin-4-yl)amino)nicotinamide [1969];

2-(4-aminopiperidin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)isonicotinamide [1970];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(4-(methylamino)piperidin-1-yl) isonicotinamide [1971];

2-(4-(dimethylamino)piperidin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl) isonicotinamide [1972];

2-((1-isopropylpiperidin-4-yl)oxy)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl) isonicotinamide [1973];

2-(3-aminoazetidin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)isonicotinamide [1974];

2-(3-(dimethylamino)azetidin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl) isonicotinamide [1975];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-morpholinoisonicotinamide [1976];

2-((2-(dimethylamino)ethyl)amino)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl) isonicotinamide [1977];

2-(2-(dimethylamino)ethoxy)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)isonicotinamide [1978];

2-(4-isobutylpiperazin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)isonicotinamide [1979];

2-(azetidin-3-yloxy)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)isonicotinamide [1980];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-((1-methylazetidin-3-yl)oxy)isonicotinamide [1981];

2-(4-ethylpiperazin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)isonicotinamide [1982];

4-((dimethylamino)methyl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)benzamide [1983];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-3-(1-methylpiperidin-4-yl)benzamide [1984];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-3-((4-methylpiperazin-1-yl)methyl)benzamide [1985];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)isonicotinamide [1986];

2-hydroxy-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)isonicotinamide [1987];

2-isopropoxy-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)isonicotinamide [1988];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(1-methylpiperidin-4-yl)isonicotinamide [1989];

1′-methyl-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-1′,2′,3′,6′-tetrahydro-[2,4′-bipyridine]-4-carboxamide [1990];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(4-(6-(4-methylpiperazin-1-yl) nicotinoyl)piperazin-1-yl)isonicotinamide [1991];

2-(4-hydroxy-4-methyl-4λ 4 -piperazin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl) isonicotinamide [1992];

2-methyl-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-6-(4-methylpiperazin-1-yl) isonicotinamide [1993];

3-methyl-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [1994];

2-(4-methyl-1,4-diazepan-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)isonicotinamide [1995];

2-((2S,6R)-2,6-dimethylmorpholino)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl) isonicotinamide [1996];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(2,7-diazaspiro[3.5]nonan-2-yl)isonicotinamide [1997];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(7-methyl-2,7-diazaspiro[3.5]nonan-2-yl) isonicotinamide [1998];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(2,7-diazaspiro[3.5]nonan-7-yl)isonicotinamide [1999];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(2-methyl-2,7-diazaspiro[3.5]nonan-7-yl) isonicotinamide [2000];

2-(methyl(1-methylpiperidin-4-yl)amino)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl) isonicotinamide [2001];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-((1-methylpiperidin-4-yl)thio)isonicotinamide [2002];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)pyrimidine-4-carboxamide [2003];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-6-(4-methylpiperazin-1-yl)pyridazine-4-carboxamide [2004];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-6-(4-methylpiperazin-1-yl)pyrimidine-4-carboxamide [2005];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-phenylacetamide [2006];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-3-phenylpropanamide [2007];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(pyridin-3-yl)acetamide [2008];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-3-(pyridin-3-yl)propanamide [2009];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(pyridin-4-yl)acetamide [2010];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-3-(pyridin-4-yl)propanamide [2011];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)isoindoline-5-carboxamide [2012];

2-methyl-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)isoindoline-5-carboxamide [2013];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-1,2,3,4-tetrahydroisoquinoline-7-carboxamide [2014];

2-methyl-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-1,2,3,4-tetrahydroisoquinoline-7-carboxamide [2015];

2-methyl-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-1,2,3,4-tetrahydroisoquinoline-6-carboxamide [2016];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-1,2,3,4-tetrahydroisoquinoline-6-carboxamide [2017];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-1H-indole-5-carboxamide [2018];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)benzofuran-5-carboxamide [2019];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)furo[2,3-c]pyridine-5-carboxamide [2020];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)benzo[b]thiophene-5-carboxamide [2021];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)benzofuran-6-carboxamide [2022];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)benzo[d]oxazole-6-carboxamide [2023];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)benzo[d]thiazole-6-carboxamide [2024];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)benzo[d]oxazole-5-carboxamide [2025];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)benzo[d]thiazole-5-carboxamide [2026];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)quinoline-3-carboxamide [2027];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)quinoline-6-carboxamide [2028];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)quinoxaline-6-carboxamide [2029];

5-chloro-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [2030];

3-chloro-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [2031];

2-(2,5-diazabicyclo[2.2.1]heptan-2-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl) isonicotinamide [2032];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(5-methyl-2,5-diazabicyclo [2.2.1]heptan-2-yl)isonicotinamide [2033];

3-fluoro-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [2034];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-((4-methylpiperazin-1-yl)methyl) isonicotinamide [2035];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(morpholinomethyl)isonicotinamide [2036];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(pyrrolidin-1-ylmethyl)isonicotinamide [2037];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(2-(4-methylpiperazin-1-yl)pyridin-4-yl) acetamide [2038];

1-methyl-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-1H-indazole-5-carboxamide [2039];

1-methyl-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-1H-benzo[d]imidazole-5-carboxamide [2040];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-1-(piperidin-4-yl)-1H-pyrazole-4-carboxamide [2041];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-1-(1-methylpiperidin-4-yl)-1H-pyrazole-4-carboxamide [2042];

1-(1-ethylpiperidin-4-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-1H-pyrazole-4-carboxamide [2043];

1-(1-(2-fluoroethyl)piperidin-4-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-1H-pyrazole-4-carboxamide [2044];

1-(1-isopropylpiperidin-4-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-1H-pyrazole-4-carboxamide [2045];

1-(1-cyclopropylpiperidin-4-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-1H-pyrazole-4-carboxamide [2046];

isopropyl 4-(4-((6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)carbamoyl)-1H-pyrazol-1-yl) piperidine-1-carboxylate [2047];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-1-(piperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide [2048];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-1-(1-methylpiperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide [2049];

1-(1-(2-fluoroethyl)piperidin-4-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-1H-1,2,3-triazole-4-carboxamide [2050];

1-(1-isopropylpiperidin-4-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-1H-1,2,3-triazole-4-carboxamide [2051];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)oxazole-5-carboxamide [2052];

2-(3-(dimethylamino)azetidin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)oxazole-4-carboxamide [2053];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(piperidin-4-yl)oxazole-4-carboxamide [2054];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(1-methylpiperidin-4-yl)oxazole-4-carboxamide [2055];

2-(1-(2-fluoroethyl)piperidin-4-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)oxazole-4-carboxamide [2056];

2-(1-isopropylpiperidin-4-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)oxazole-4-carboxamide [2057];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)oxazole-4-carboxamide [2058];

2-(3-(dimethylamino)azetidin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)thiazole-5-carboxamide [2059];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(piperidin-4-yl)thiazole-4-carboxamide [2060];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)thiazole-4-carboxamide [2061];

2-(1-(2-fluoroethyl)piperidin-4-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)thiazole-4-carboxamide [2062];

2-(1-isopropylpiperidin-4-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)thiazole-4-carboxamide [2063];

1-methyl-N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl-4-d)piperidine-4-carboxamide [2064];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-1-(2-(methyl-d3)propyl-1,1,2,3,3,3-d 6 )piperidine-4-carboxamide [2065];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(pyrrolidin-1-yl-2,2,5,5-d 4 )acetamide [2066];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(4-(methyl-d 3 )piperazin-1-yl)acetamide [2067];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(morpholino-d 8 )acetamide [2068];

(S)—N-(6-(1-(methyl-d 3 )-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(pyrrolidin-1-yl)propanamide [2069];

1-isobutyl-N-(6-(1-(methyl-d 3 )-1H-pyrazol-4-yl)cinnolin-3-yl)piperidine-4-carboxamide [2070];

N-(6-(1-(methyl-d 3 )-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)acetamide [2071];

N-(6-(1-(methyl-d 3 )-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(pyrrolidin-1-yl)acetamide [2072];

N-(6-(1-(methyl-d 3 )-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(piperidin-1-yl)acetamide [2073];

N-(6-(1-(methyl-d 3 )-1H-pyrazol-4-yl)cinnolin-3-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [2074];

N-(6-(1H-pyrazol-4-yl)cinnolin-3-yl)-2-(4-(methyl-d 3 )piperazin-1-yl)isonicotinamide [2075];

N-(6-(1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(4-(methyl-d 3 )piperazin-1-yl)isonicotinamide [2076];

N-(6-(1-(methyl-d 3 )-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [2077];

N-(6-(1-(methyl-d 3 )-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(4-(methyl-d 3 )piperazin-1-yl) isonicotinamide [2078];

N-(6-(1-(methyl-d 3 )-1H-pyrazol-4-yl)cinnolin-3-yl)-1-(piperidin-4-yl)-1H-pyrazole-4-carboxamide [2079];

N-(6-(1-(methyl-d 3 )-1H-pyrazol-4-yl)cinnolin-3-yl)-1-(1-methylpiperidin-4-yl)-1H-pyrazole-4-carboxamide [2080];

N-(6-(1-(methyl-d 3 )-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(piperidin-4-yl)oxazole-4-carboxamide [2081];

N-(6-(1-(methyl-d 3 )-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(1-methylpiperidin-4-yl)oxazole-4-carboxamide [2082];

N-(6-(1-ethyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(pyrrolidin-1-yl)acetamide [2083];

N-(6-(1-cyclopropyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(pyrrolidin-1-yl)acetamide [2084];

N-(6-(1-cyclopropyl-1H-pyrazol-4-yl)cinnolin-3-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [2085];

N-(6-(1-(1-methylpiperidin-4-yl)-1H-pyrazol-4-yl)cinnolin-3-yl)cyclohexanecarboxamide [2086];

2-(pyrrolidin-1-yl)-N-(6-(5-(trifluoromethyl)-1H-pyrazol-4-yl)cinnolin-3-yl)acetamide [2087];

N-(6-(5-(hydroxymethyl)-1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-1-methylpiperidine-4-carboxamide [2088];

N-(6-(5-(hydroxymethyl)-1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)tetrahydro-2H-pyran-4-carboxamide [2089];

N-(6-(5-(azetidin-1-ylmethyl)-1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-4,4-difluorocyclohexane-1-carboxamide [2090];

4,4-difluoro-N-(6-(1-methyl-5-(pyrrolidin-1-ylmethyl)-1H-pyrazol-4-yl)cinnolin-3-yl) cyclohexane-1-carboxamide [2091];

4,4-difluoro-N-(6-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)cinnolin-3-yl) cyclohexane-1-carboxamide [2092];

2-(2-fluoroethyl)-N-(6-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)cinnolin-3-yl)-2-azaspiro[3.3]heptane-6-carboxamide [2093];

tert-butyl 6-((6-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)cinnolin-3-yl)carbamoyl)-2-azaspiro[3.3]heptane-2-carboxylate [2094];

2-fluoro-2-methyl-N-(6-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)cinnolin-3-yl) propanamide [2095];

2-(diethylamino)-N-(6-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)cinnolin-3-yl) acetamide [2096];

trans-4-methoxy-N-(6-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)cinnolin-3-yl) cyclohexane-1-carboxamide [2097];

trans-4-(hydroxymethyl)-N-(6-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)cinnolin-3-yl)cyclohexane-1-carboxamide [2098];

(R)—N-(6-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)cinnolin-3-yl)pyrrolidine-2-carboxamide [2099];

1-isobutyl-N-(6-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)cinnolin-3-yl)piperidine-4-carboxamide [2100];

N-(6-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)cinnolin-3-yl)-1-(oxetan-3-yl) piperidine-4-carboxamide [2101];

1-benzoyl-N-(6-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)cinnolin-3-yl)piperidine-4-carboxamide [2102];

N-(6-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)cinnolin-3-yl)tetrahydro-2H-pyran-4-carboxamide [2103];

N-(6-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(4-methylpiperidin-1-yl)acetamide [2104];

N-(6-(1-(difluoromethyl)-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [2105];

N-(6-(1-ethyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [2106];

N-(6-(1-isopropyl-1H-pyrazol-4-yl)cinnolin-3-yl)-3-(piperidin-4-yloxy)benzamide [2107];

N-(6-(1-isopropyl-1H-pyrazol-4-yl)cinnolin-3-yl)-3-((1-methylpiperidin-4-yl)oxy)benzamide [2108];

N-(6-(1-isopropyl-1H-pyrazol-4-yl)cinnolin-3-yl)-4-(piperidin-4-yloxy)benzamide [2109];

N-(6-(1-cyclopropyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [2110];

4-fluoro-N-(6-(1-(1-methylpiperidin-4-yl)-1H-pyrazol-4-yl)cinnolin-3-yl)benzamide [2111];

4-(difluoromethoxy)-N-(6-(1-(1-methylpiperidin-4-yl)-1H-pyrazol-4-yl)cinnolin-3-yl)benzamide [2112];

5-fluoro-N-(6-(1-(1-methylpiperidin-4-yl)-1H-pyrazol-4-yl)cinnolin-3-yl)nicotinamide [2113];

N 2 -methyl-N 5 -(6-(1-(1-methylpiperidin-4-yl)-1H-pyrazol-4-yl)cinnolin-3-yl)pyridine-2,5-dicarboxamide [2114];

1-isopropyl-N-(6-(1-(1-methylpiperidin-4-yl)-1H-pyrazol-4-yl)cinnolin-3-yl)-1H-pyrazole-4-carboxamide [2115];

2-methyl-N-(6-(1-(1-methylpiperidin-4-yl)-1H-pyrazol-4-yl)cinnolin-3-yl)thiazole-5-carboxamide [2116];

N-(6-(5-amino-1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [2117];

4-(difluoromethoxy)-N-(6-(5-(hydroxymethyl)-1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl) benzamide [2118];

N-(6-(5-(hydroxymethyl)-1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [2119];

N-(6-(5-(hydroxymethyl)-1-methyl-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(7-methyl-2,7-diazaspiro [3.5]nonan-2-yl)isonicotinamide [2120];

4-fluoro-N-(6-(1-methyl-5-(pyrrolidin-1-ylmethyl)-1H-pyrazol-4-yl)cinnolin-3-yl)benzamide [2121];

4-fluoro-N-(6-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)cinnolin-3-yl)benzamide [2122];

4-(difluoromethoxy)-N-(6-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)cinnolin-3-yl)benzamide [2123];

N-(6-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)cinnolin-3-yl)-3-(pyrrolidin-1-ylmethyl)benzamide [2124];

N-(6-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)cinnolin-3-yl)-2-(7-methyl-2,7-diazaspiro[3.5]nonan-2-yl)isonicotinamide [2125];

N-(6-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)cinnolin-3-yl)-2-morpholinoisonicotinamide [2126];

N-(6-(1-methyl-5-(morpholinomethyl)-1H-pyrazol-4-yl)cinnolin-3-yl)-2-morpholinoisonicotinamide [2127];

N-(6-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)cinnolin-3-yl)-1-((1-(trifluoromethyl) cyclopropyl)methyl)piperidine-4-carboxamide [2128];

3,3-difluoro-N-(6-(5-methyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)cinnolin-3-yl)cyclobutane-1-carboxamide [2129];

N-((4,4-difluorocyclohexyl)methyl)-6-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)cinnolin-3-amine [2130];

N-(6-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)cinnolin-3-yl)-1-((1-(trifluoromethyl)cyclopropyl)methyl)piperidine-4-carboxamide [2131];

N-(6-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)cinnolin-3-yl)-2-(pyrrolidin-1-yl)acetamide [2132];

2-(7-azabicyclo[2.2.1]heptan-7-yl)-N-(6-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)cinnolin-3-yl)acetamide [2133];

(R)—N-(6-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)cinnolin-3-yl)-1-isobutylpiperidine-3-carboxamide [2134];

N-(6-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)cinnolin-3-yl)piperidine-4-carboxamide [2135];

4-fluoro-N-(6-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)cinnolin-3-yl)-1-isobutylpiperidine-4-carboxamide [2136];

N-(6-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)acetamide [2137];

4-fluoro-N-(6-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)cinnolin-3-yl)benzamide [2138];

N-(6-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)cinnolin-3-yl)-3-(4-methylpiperazin-1-yl)benzamide [2139];

N 5 -(6-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)cinnolin-3-yl)-N 2 -methylpyridine-2,5-dicarboxamide [2140];

N-(6-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)cinnolin-3-yl)-6-(4-methylpiperazin-1-yl)nicotinamide [2141];

2-(azetidin-3-yloxy)-N-(6-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)cinnolin-3-yl)isonicotinamide [2142];

N-(6-(1-methyl-1H-pyrazol-5-yl)cinnolin-3-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [2143];

1-methyl-N-(6-(1-methyl-1H-pyrazol-3-yl)cinnolin-3-yl)piperidine-4-carboxamide [2144];

N-(6-(1-methyl-1H-pyrazol-3-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [2145];

2-fluoro-2-methyl-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)propanamide [2146];

2,2,3,3-tetramethyl-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)cyclopropane-1-carboxamide [2147];

trans-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)-4-(pyrrolidin-1-yl)cyclohexane-1-carboxamide [2148];

trans-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)-4-morpholinocyclohexane-1-carboxamide [2149];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)-2-(piperidin-1-yl)acetamide [2150];

1-ethyl-4-fluoro-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)piperidine-4-carboxamide [2151];

4-fluoro-1-isobutyl-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)piperidine-4-carboxamide [2152];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [2153];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)cyclopropanecarboxamide [2154];

4,4-difluoro-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)cyclohexane-1-carboxamide [2155];

trans-4-(dimethylamino)-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)cyclohexane-1-carboxamide [2156];

trans-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)-4-((4-methylpiperazin-1-yl)methyl) cyclohexane-1-carboxamide [2157];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)piperidine-4-carboxamide [2158];

1-isobutyl-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)piperidine-4-carboxamide [2159];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)-1-((1-(trifluoromethyl)cyclopropyl)methyl) piperidine-4-carboxamide [2160];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)-1-((3-methyloxetan-3-yl)methyl)piperidine-4-carboxamide [2161];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)-1-(2-(pyrrolidin-1-yl)acetyl)piperidine-4-carboxamide [2162];

1′-methyl-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)-[1,4′-bipiperidine]-4-carboxamide [2163];

(R)—N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)piperidine-3-carboxamide [2164];

(R)-1-isobutyl-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)piperidine-3-carboxamide [2165];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)-2-(pyrrolidin-1-yl)acetamide [2166];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)acetamide [2167];

2-(7-azabicyclo[2.2.1]heptan-7-yl)-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)acetamide [2168];

1-(2-hydroxy-2-methylpropyl)-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)piperidine-4-carboxamide [2169];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)-2-morpholinoacetamide [2170];

2-(4-methoxypiperidin-1-yl)-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)acetamide [2171];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)morpholine-4-carboxamide [2172];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)-1-(piperidin-4-yl)-1H-pyrazole-4-carboxamide [2173];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)-1-(1-methylpiperidin-4-yl)-1H-pyrazole-4-carboxamide [2174];

1-(1-ethylpiperidin-4-yl)-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)-1H-pyrazole-4-carboxamide [2175];

1-(1-isopropylpiperidin-4-yl)-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)-1H-pyrazole-4-carboxamide [2176];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)-1-(piperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide [2177];

1-(1-(2-fluoroethyl)piperidin-4-yl)-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)-1H-1,2,3-triazole-4-carboxamide [2178];

1-(1-isopropylpiperidin-4-yl)-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)-1H-1,2,3-triazole-4-carboxamide [2179];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)-2-(piperidin-4-yl)oxazole-4-carboxamide [2180];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)-2-(1-methylpiperidin-4-yl)oxazole-4-carboxamide [2181];

2-(1-isopropylpiperidin-4-yl)-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)oxazole-4-carboxamide [2182];

2-fluoro-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)benzamide [2183];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)-3-((1-methylpiperidin-4-yl)oxy)benzamide [2184];

N 2 -methyl-N 5 -(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)pyridine-2,5-dicarboxamide [2185];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)-6-(4-methylpiperazin-1-yl)nicotinamide [2186];

2-(3-(dimethylamino)azetidin-1-yl)-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl) isonicotinamide [2187];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)-2-(1-methylpiperidin-4-yl)isonicotinamide [2188];

2-(4-(dimethylamino)piperidin-1-yl)-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl) isonicotinamide [2189];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)-2-morpholinoisonicotinamide [2190];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [2191];

2-(4-methyl-1,4-diazepan-1-yl)-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl) isonicotinamide [2192];

2-(4-isopropylpiperazin-1-yl)-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)isonicotinamide [2193];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)-2-(piperidin-4-ylamino)isonicotinamide [2194];

2-(methyl(1-methylpiperidin-4-yl)amino)-N-(6-(1-methyl-1H-1,2,33-triazol-4-yl)cinnolin-3-yl)isonicotinamide [2195];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)-2-((1-methylpiperidin-4-yl)thio) isonicotinamide [2196];

2-methyl-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)-1,2,3,4-tetrahydroisoquinoline-6-carboxamide [2197];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)-2-(piperazin-1-yl)isonicotinamide [2198];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)-2-(2-(4-methylpiperazin-1-yl)pyridin-4-yl)acetamide [2199];

1,1-bis(methyl-d 3 )-4-(4-((6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)carbamoyl)pyridin-2-yl)piperazin-1-ium [2200];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)cinnolin-3-yl)-2-(4-(methyl-d 3 )piperazin-1-yl) isonicotinamide [2201];

N-(6-(1-methyl-1H-1,2,3-triazol-5-yl)cinnolin-3-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [2202];

N-(6-(4-methyl-4H-1,2,4-triazol-3-yl)cinnolin-3-yl)-2-morpholinoacetamide [2203];

N-(6-(4-methyl-4H-1,2,4-triazol-3-yl)cinnolin-3-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [2204];

4-fluoro-1-isobutyl-N-(6-(4-methyl-4H-1,2,4-triazol-3-yl)cinnolin-3-yl)piperidine-4-carboxamide [2205];

N-(6-(4,5-dimethyl-4H-1,2,4-triazol-3-yl)cinnolin-3-yl)-2-morpholinoacetamide [2206];

N-(6-(4,5-dimethyl-4H-1,2,4-triazol-3-yl)cinnolin-3-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [2207];

N-(6-(1H-1,2,3-triazol-1-yl)cinnolin-3-yl)-4-fluoro-1-isobutylpiperidine-4-carboxamide [2208];

N-(6-(2H-1,2,3-triazol-2-yl)cinnolin-3-yl)-4-fluoro-1-isobutylpiperidine-4-carboxamide [2209];

N-(6-(1H-1,2,4-triazol-1-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [2210];

1-isobutyl-N-(6-(1-methyl-1H-tetrazol-5-yl)cinnolin-3-yl)piperidine-4-carboxamide [2211];

2,2,3,3-tetramethyl-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)cyclopropane-1-carboxamide [2212];

4,4-difluoro-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)cyclohexane-1-carboxamide [2213];

N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)-2-(piperidin-1-yl)acetamide [2214];

2-fluoro-2-methyl-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)propanamide [2215];

1-fluoro-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)cyclopropane-1-carboxamide [2216];

2-methyl-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)-2-azaspiro[3.3]heptane-6-carboxamide [2217];

1-fluoro-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)cyclohexane-1-carboxamide [2218];

trans-4-methoxy-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)cyclohexane-1-carboxamide [2219];

trans-4-(hydroxymethyl)-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)cyclohexane-1-carboxamide [2220];

N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)azetidine-3-carboxamide [2221];

(R)—N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)tetrahydrofuran-2-carboxamide [2222];

1-(2-methoxyethyl)-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)piperidine-4-carboxamide [2223];

N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [2224];

1-isobutyl-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)piperidine-4-carboxamide [2225];

N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)-1-(methylsulfonyl)piperidine-4-carboxamide [2226];

N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)-2-(pyrrolidin-1-yl)propanamide [2227];

2-isopropoxy-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)acetamide [2228];

3-isopropoxy-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)propanamide [2229];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)cinnolin-3-yl)cyclopropanecarboxamide [2230];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)cinnolin-3-yl)cyclohexanecarboxamide [2231];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)cinnolin-3-yl)-4,4-difluorocyclohexane-1-carboxamide [2232];

(S)—N-(6-(1,2-dimethyl-1H-imidazol-5-yl)cinnolin-3-yl)tetrahydrofuran-2-carboxamide [2233];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)cinnolin-3-yl)-3,3-difluorocyclobutane-1-carboxamide [2234];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)cinnolin-3-yl)-1-fluorocyclopropane-1-carboxamide [2235];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)cinnolin-3-yl)morpholine-4-carboxamide [2236];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)cinnolin-3-yl)morpholine-d 8 -4-carboxamide [2237];

1-methyl-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)-1H-pyrazole-4-carboxamide [2238];

1-ethyl-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)-1H-pyrazole-4-carboxamide [2239];

1-isopropyl-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)-1H-pyrazole-4-carboxamide [2240];

1-cyclopropyl-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)-1H-pyrazole-4-carboxamide [2241];

1-isobutyl-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)-1H-pyrazole-4-carboxamide [2242];

1-methyl-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)-1H-pyrazole-3-carboxamide [2243];

N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)-2-(1-methyl-1H-pyrazol-4-yl)acetamide [2244];

1-methyl-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)-1H-imidazole-4-carboxamide [2245];

1-isopropyl-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)-1H-imidazole-4-carboxamide [2246];

N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)-1-(tetrahydro-2H-pyran-4-yl)-1H-imidazole-4-carboxamide [2247];

1,2-dimethyl-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)-1H-imidazole-5-carboxamide [2248];

1-methyl-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)-1H-1,2,4-triazole-3-carboxamide [2249];

2-methyl-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)oxazole-4-carboxamide [2250];

2-isopropyl-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)oxazole-4-carboxamide [2251];

4-methyl-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)oxazole-2-carboxamide [2252];

4-methyl-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)thiazole-2-carboxamide [2253];

2-methyl-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)thiazole-4-carboxamide [2254];

5-methyl-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)-1,3,4-oxadiazole-2-carboxamide [2255];

5-methyl-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)-1,3,4-thiadiazole-2-carboxamide [2256];

1-isopropyl-N-(6-(1-isopropyl-1H-imidazol-5-yl)cinnolin-3-yl)-1H-pyrazole-4-carboxamide [2257];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)cinnolin-3-yl)-1-methyl-1H-pyrazole-4-carboxamide [2258];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)cinnolin-3-yl)-1-isopropyl-1H-pyrazole-4-carboxamide [2259];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)cinnolin-3-yl)-2-methylthiazole-5-carboxamide [2260];

4-fluoro-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)benzamide [2261];

4-(difluoromethoxy)-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)benzamide [2262];

N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)-3-(pyrrolidin-1-ylmethyl)benzamide [2263];

2-fluoro-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)benzamide-3,4,5,6-d 4 [2264];

4-fluoro-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)benzamide-2,3,5,6-d 4 [2265];

2-chloro-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)benzamide-3,4,5,6-d 4 [2266];

4-chloro-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)benzamide-2,3,5,6-d 4 [2267];

4-(methyl-d 3 )—N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)benzamide [2268];

4-methyl-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)benzamide-2,3,5,6-d 4 [2269];

4-(methyl-d 3 )—N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)benzamide-2,3,5,6-d 4 [2270];

4-(methoxy-d 3 )—N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)benzamide [2271];

4-(methoxy-d 3 )—N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)benzamide-2,3,5,6-d 4 [2272];

4-methoxy-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)benzamide-2,3,5,6-d 4 [2273];

(E)-N-(6-(1,2-dimethyl-1H-imidazol-5-yl)cinnolin-3-yl)-3-(phenyl-2,3,4,5,6-d 5 )acrylamide [2274];

(E)-N-(6-(1,2-dimethyl-1H-imidazol-5-yl)cinnolin-3-yl)-3-(phenyl-2,3,4,5,6-d 5 )acrylamide-2,3-d 2 [2275];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)cinnolin-3-yl)-2-(4-fluorophenyl)acetamide-2,2-d 2 [2276];

(E)-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)-3-(phenyl-2,3,4,5,6-d 5 )acrylamide [2277];

(E)-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)-3-(phenyl-2,3,4,5,6-d 5 )acrylamide-2,3-d 2 [2278];

2-(4-fluorophenyl)-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)acetamide-2,2-d 2 [2279];

N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [2280];

2-(dimethylamino)-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)isonicotinamide [2281];

2-(3-aminoazetidin-1-yl)-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)isonicotinamide [2282];

N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)-2-(pyrrolidin-1-yl)isonicotinamide [2283];

N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)-2-(piperidin-1-yl)isonicotinamide [2284];

N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)-2-morpholinoisonicotinamide [2285];

2-(4-isopropylpiperazin-1-yl)-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)isonicotinamide [2286];

2-(4-cyclopropylpiperazin-1-yl)-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)isonicotinamide [2287];

N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)-2-(2,7-diazaspiro[3.5]nonan-2-yl) isonicotinamide [2288];

N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)-2-(7-methyl-2,7-diazaspiro[3.5]nonan-2-yl) isonicotinamide [2289];

N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)isoindoline-5-carboxamide [2290];

2-methyl-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)isoindoline-5-carboxamide [2291];

2-(azetidin-1-yl)-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)isonicotinamide [2292];

2-methoxy-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)isonicotinamide [2293];

2-methyl-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)isonicotinamide [2294];

2-cyano-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)isonicotinamide [2295];

2-(3,3-difluoroazetidin-1-yl)-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)isonicotinamide [2296];

2-(4,4-difluoropiperidin-1-yl)-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)isonicotinamide [2297];

2-isopropoxy-N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)isonicotinamide [2298];

N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)-2-(pyrrolidin-1-yl-2,2,5,5-d 4 )isonicotinamide [2299];

N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)-2-(pyrrolidin-1-yl-d 8 )isonicotinamide [2300];

N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)-2-(piperidin-1-yl-d 10 )isonicotinamide [2301];

N-(6-(1-methyl-1H-imidazol-5-yl)cinnolin-3-yl)-2-(morpholino-d 8 )isonicotinamide [2302];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)cinnolin-3-yl)-4-isopropoxybenzamide [2303];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)cinnolin-3-yl)-4-(piperidin-4-yloxy)benzamide [2304];

4-(benzyloxy)-N-(6-(1,2-dimethyl-1H-imidazol-5-yl)cinnolin-3-yl)benzamide [2305];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)cinnolin-3-yl)-2-fluorobenzamide-3,4,5,6-d 4 [2206];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)cinnolin-3-yl)-4-fluorobenzamide-2,3,5,6-d 4 [2307];

2-chloro-N-(6-(1,2-dimethyl-1H-imidazol-5-yl)cinnolin-3-yl)benzamide-3,4,5,6-d 4 [2308];

4-chloro-N-(6-(1,2-dimethyl-1H-imidazol-5-yl)cinnolin-3-yl)benzamide-2,3,5,6-d 4 [2309];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)cinnolin-3-yl)-4-(methyl-d 3 )benzamide [2310];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)cinnolin-3-yl)-4-methylbenzamide-2,3,5,6-d 4 [2311];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)cinnolin-3-yl)-4-(methyl-d 3 )benzamide-2,3,5,6-d 4 [2312];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)cinnolin-3-yl)-4-(methoxy-d 3 )benzamide [2313];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)cinnolin-3-yl)-4-(methoxy-d 3 )benzamide-2,3,5,6-d 4 [2314];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)cinnolin-3-yl)-4-methoxybenzamide-2,3,5,6-d 4 [2315];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [2316];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)cinnolin-3-yl)-2-morpholinoisonicotinamide [2317];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)cinnolin-3-yl)-2-(pyrrolidin-1-yl)isonicotinamide [2318];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)cinnolin-3-yl)-2-(dimethylamino)isonicotinamide [2319];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)cinnolin-3-yl)-2-(pyrrolidin-1-yl-2,2,5,5-d 4 ) isonicotinamide [2320];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)cinnolin-3-yl)-2-(pyrrolidin-1-yl-d 8 )isonicotinamide [2321];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)cinnolin-3-yl)-2-(piperidin-1-yl-d 10 )isonicotinamide [2322];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)cinnolin-3-yl)-2-(morpholino-d 8 )isonicotinamide [2323];

N-(6-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)cinnolin-3-yl)cyclopropanecarboxamide [2324];

N-(6-(7-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)cinnolin-3-yl) cyclopropanecarboxamide [2325];

3,3-difluoro-N-(6-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)cinnolin-3-yl)cyclobutane-1-carboxamide [2326];

(R)—N-(6-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)cinnolin-3-yl)pyrrolidine-2-carboxamide [2327];

(R)—N-(6-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)cinnolin-3-yl)piperidine-3-carboxamide [2328];

1-methyl-N-(6-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)cinnolin-3-yl)piperidine-4-carboxamide [2329];

N-(6-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)cinnolin-3-yl)-1-((1-(trifluoromethyl) cyclopropyl)methyl)piperidine-4-carboxamide [2330];

1-benzoyl-N-(6-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)cinnolin-3-yl)piperidine-4-carboxamide [2331];

4-fluoro-1-isobutyl-N-(6-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)cinnolin-3-yl)piperidine-4-carboxamide [2332];

(R)-2-(2-methylpyrrolidin-1-yl)-N-(6-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)cinnolin-3-yl)acetamide [2333];

2-(cyclobutyl(methyl)amino)-N-(6-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)cinnolin-3-yl)acetamide [2334];

4-fluoro-N-(6-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)cinnolin-3-yl)benzamide [2335];

4-isopropoxy-N-(6-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)cinnolin-3-yl)benzamide [2336];

4-(difluoromethoxy)-N-(6-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)cinnolin-3-yl) benzamide [2337];

2-((2-(dimethylamino)ethyl)amino)-N-(6-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)cinnolin-3-yl)isonicotinamide [2338];

2-((1-isopropylpiperidin-4-yl)oxy)-N-(6-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)cinnolin-3-yl)isonicotinamide [2339];

N-(6-(oxazol-5-yl)cinnolin-3-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [2340];

N-(6-(oxazol-5-yl)cinnolin-3-yl)cyclopropanecarboxamide [2341];

(R)—N-(6-(oxazol-5-yl)cinnolin-3-yl)tetrahydrofuran-2-carboxamide [2342];

(R)—N-(6-(oxazol-5-yl)cinnolin-3-yl)piperidine-3-carboxamide [2343];

N-(6-(oxazol-5-yl)cinnolin-3-yl)tetrahydro-2H-pyran-4-carboxamide [2344];

N-(6-(oxazol-5-yl)cinnolin-3-yl)-1-(2-(pyrrolidin-1-yl)acetyl)piperidine-4-carboxamide [2345];

1′-methyl-N-(6-(oxazol-5-yl)cinnolin-3-yl)-[1,4′-bipiperidine]-4-carboxamide [2346];

cis-4-morpholino-N-(6-(oxazol-5-yl)cinnolin-3-yl)cyclohexane-1-carboxamide [2347];

2-(cyclobutyl(methyl)amino)-N-(6-(oxazol-5-yl)cinnolin-3-yl)acetamide [2348];

N-(6-(oxazol-5-yl)cinnolin-3-yl)-2-(pyrrolidin-1-yl)acetamide [2349];

(R)-2-(2-methylpyrrolidin-1-yl)-N-(6-(oxazol-5-yl)cinnolin-3-yl)acetamide [2350];

2-(4-methylpiperazin-1-yl)-N-(6-(oxazol-5-yl)cinnolin-3-yl)acetamide [2351];

trans-4-((4-methylpiperazin-1-yl)methyl)-N-(6-(oxazol-5-yl)cinnolin-3-yl)cyclohexane-1-carboxamide [2352];

1-(2,2-difluoropropyl)-N-(6-(oxazol-5-yl)cinnolin-3-yl)piperidine-4-carboxamide [2353];

trans-4-(hydroxymethyl)-N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl)cyclohexane-1-carboxamide [2354];

trans-4-(methylamino)-N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl)cyclohexane-1-carboxamide [2355];

trans-4-((1,3-difluoropropan-2-yl)amino)-N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl)cyclohexane-1-carboxamide [2356];

trans-N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl)-4-((propan-2-yl-1,1,1,3,3,3-d 6 )amino) cyclohexane-1-carboxamide [2357];

trans-4-((2,2-difluoroethyl)amino)-N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl)cyclohexane-1-carboxamide [2358];

trans-N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl)-4-((3,3,3-trifluoropropyl)amino)cyclohexane-1-carboxamide [2359];

trans-4-((2-methoxyethyl)amino)-N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl)cyclohexane-1-carboxamide [2360];

trans-4-(dimethylamino)-N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl)cyclohexane-1-carboxamide [2361];

trans-4-(bis(methyl-d 3 )amino)-N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl)cyclohexane-1-carboxamide [2362];

cis-4-(dimethylamino)-N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl)cyclohexane-1-carboxamide [2363];

trans-4-((2,2-difluoroethyl)(methyl)amino)-N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl) cyclohexane-1-carboxamide [2364];

trans-4-(methyl(oxetan-3-yl)amino)-N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl)cyclohexane-1-carboxamide [2365];

trans-4-((2-fluoroethyl)amino)-N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl)cyclohexane-1-carboxamide [2366];

trans-4-(2-(fluoromethyl)aziridin-1-yl)-N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl)cyclohexane-1-carboxamide [2367];

trans-4-((3-fluoroazetidin-1-yl)methyl)-N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl)cyclohexane-1-carboxamide [2368];

trans-N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl)-3-morpholinocyclobutane-1-carboxamide [2369];

trans-N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl)-4-morpholinocyclohexane-1-carboxamide [2370];

N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl)-2-(piperidin-1-yl)acetamide [2371];

2-(4-methoxypiperidin-1-yl)-N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl)acetamide [2372];

N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)acetamide [2373];

N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl)morpholine-4-carboxamide [2374];

N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl)-2-morpholinoacetamide [2375];

N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl)-3-morpholinopropanamide [2376];

1-methyl-N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl)piperidine-4-carboxamide [2377];

1-(2,2-difluoropropyl)-N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl)piperidine-4-carboxamide [2378];

N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl)-4-morpholinopiperidine-1-carboxamide [2379];

4-((1,3-difluoropropan-2-yl)amino)-N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl)piperidine-1-carboxamide [2380];

(1R,3s,5S)-3-((1,3-difluoropropan-2-yl)amino)-N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl)-8-azabicyclo[3.2.1]octane-8-carboxamide [2381];

(1R,3s,5S)-3-((1,3-difluoropropan-2-yl)amino)-N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl)-8-azabicyclo[3.2.1]octane-8-carboxamide [2382];

4-(dimethylamino)-N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl)piperidine-1-carboxamide [2383];

4-((2,2-difluoroethyl)(methyl)amino)-N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl)piperidine-1-carboxamide [2384];

(3S,4S)-4-amino-3-fluoro-N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl)piperidine-1-carboxamide [2385];

(3S,4S)-3-fluoro-4-(methylamino)-N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl)piperidine-1-carboxamide [2386];

(3R,4R)-4-amino-3-fluoro-N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl)piperidine-1-carboxamide [2387];

(3R,4R)-3-fluoro-4-(methylamino)-N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl)piperidine-1-carboxamide [2388];

4-((2-fluoroethyl)amino)-N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl)piperidine-1-carboxamide [2389];

4-((2,2-difluoroethyl)amino)-N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl)piperidine-1-carboxamide [2390];

(1R,3 s,5 S)-3-amino-N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl)-8-azabicyclo [3.2.1]octane-8-carboxamide [2391];

(1R,3r,5 S)-3-amino-N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl)-8-azabicyclo[3.2.1]octane-8-carboxamide [2392];

(1R,3r,5 S)-3-((2-fluoroethyl)amino)-N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl)-8-azabicyclo [3.2.1]octane-8-carboxamide [2393];

(1R,3r,5S)-3-((2,2-difluoroethyl)amino)-N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl)-8-azabicyclo [3.2.1]octane-8-carboxamide [2394];

(1R,3s,5S)—N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl)-3-((3,3,3-trifluoropropyl)amino)-8-azabicyclo [3.2.1]octane-8-carboxamide [2395];

(3S,4S)-3-fluoro-4-(isopropylamino)-N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl)piperidine-1-carboxamide [2396];

N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl)-5,6-dihydroimidazo[1,2-a]pyrazine-7(8H)-carboxamide [2397];

2-methyl-N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl)-5,6-dihydroimidazo[1,2-a]pyrazine-7(8H)-carboxamide [2398];

N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl)-2-(morpholino-d 8 )acetamide [2399];

trans-N-(6-(2-methyloxazol-4-yl)cinnolin-3-yl)-4-(4-methylpiperazin-1-yl)cyclohexane-1-carboxamide [2400];

N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl)-1-(1-methylpiperidin-4-yl)-1H-pyrazole-4-carboxamide [2401];

2-(1H-imidazol-1-yl)-N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl)acetamide [2402];

4-(difluoromethoxy)-N-(6-(oxazol-5-yl)cinnolin-3-yl)benzamide [2403];

3-((1-methylpiperidin-4-yl)oxy)-N-(6-(oxazol-5-yl)cinnolin-3-yl)benzamide [2404];

N-(6-(oxazol-5-yl)cinnolin-3-yl)isonicotinamide [2405];

2-(3-aminoazetidin-1-yl)-N-(6-(oxazol-5-yl)cinnolin-3-yl)isonicotinamide [2406];

2-(1-methylpiperidin-4-yl)-N-(6-(oxazol-5-yl)cinnolin-3-yl)isonicotinamide [2407];

1′-methyl-N-(6-(oxazol-5-yl)cinnolin-3-yl)-1′,2′,3′,6′-tetrahydro-[2,4′-bipyridine]-4-carboxamide [2408];

2-(4-methylpiperazin-1-yl)-N-(6-(oxazol-5-yl)cinnolin-3-yl)isonicotinamide [2409];

2-(7-methyl-2,7-diazaspiro[3.5]nonan-2-yl)-N-(6-(oxazol-5-yl)cinnolin-3-yl)isonicotinamide [2410];

N-(6-(oxazol-5-yl)cinnolin-3-yl)-2-(2,7-diazaspiro[3.5]nonan-7-yl)isonicotinamide [2411];

N-(6-(oxazol-5-yl)cinnolin-3-yl)-2-(piperidin-4-ylamino)isonicotinamide [2412];

2-methyl-N-(6-(oxazol-5-yl)cinnolin-3-yl)isoindoline-5-carboxamide [2413];

N-(6-(oxazol-5-yl)cinnolin-3-yl)-1,2,3,4-tetrahydroisoquinoline-7-carboxamide [2414];

N-(6-(2-methyloxazol-5-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [2415];

N-(6-(3-methylisoxazol-5-yl)cinnolin-3-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [2416];

4-fluoro-1-isobutyl-N-(6-(5-methyl-1,3,4-oxadiazol-2-yl)cinnolin-3-yl)piperidine-4-carboxamide [2417];

1-isobutyl-N-(6-(5-methyl-1,3,4-oxadiazol-2-yl)cinnolin-3-yl)piperidine-4-carboxamide [2418];

N-(6-(5-(dimethylamino)-1,3,4-oxadiazol-2-yl)cinnolin-3-yl)piperidine-4-carboxamide [2419];

N-(6-(5-(dimethylamino)-1,3,4-oxadiazol-2-yl)cinnolin-3-yl)-1-methylpiperidine-4-carboxamide [2420];

N-(6-(5-methyl-1,3,4-oxadiazol-2-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [2421];

3,3-difluoro-N-(6-(thiazol-5-yl)cinnolin-3-yl)cyclobutane-1-carboxamide [2422];

2-methyl-N-(6-(thiazol-5-yl)cinnolin-3-yl)-2-azaspiro[3.3]heptane-6-carboxamide [2423];

1-fluoro-N-(6-(thiazol-5-yl)cinnolin-3-yl)cyclohexane-1-carboxamide [2424];

trans-4-(dimethylamino)-N-(6-(thiazol-5-yl)cinnolin-3-yl)cyclohexane-1-carboxamide [2425];

trans-4-((3-fluoroazetidin-1-yl)methyl)-N-(6-(thiazol-5-yl)cinnolin-3-yl)cyclohexane-1-carboxamide [2426];

N-(6-(thiazol-5-yl)cinnolin-3-yl)azetidine-3-carboxamide [2427];

1-methyl-N-(6-(thiazol-5-yl)cinnolin-3-yl)piperidine-4-carboxamide [2428];

1-(2,2-difluoropropyl)-N-(6-(thiazol-5-yl)cinnolin-3-yl)piperidine-4-carboxamide [2429];

1-(oxetan-3-yl)-N-(6-(thiazol-5-yl)cinnolin-3-yl)piperidine-4-carboxamide [2430];

1-(2-(pyrrolidin-1-yl)acetyl)-N-(6-(thiazol-5-yl)cinnolin-3-yl)piperidine-4-carboxamide [2431];

1′-methyl-N-(6-(thiazol-5-yl)cinnolin-3-yl)-[l 1,4′-bipiperidine]-4-carboxamide [2432];

2-(pyrrolidin-1-yl)-N-(6-(thiazol-5-yl)cinnolin-3-yl)propanamide [2433];

2-(piperidin-1-yl)-N-(6-(thiazol-5-yl)cinnolin-3-yl)acetamide [2434];

2-(4-methylpiperazin-1-yl)-N-(6-(thiazol-5-yl)cinnolin-3-yl)acetamide [2435];

2-morpholino-N-(6-(thiazol-5-yl)cinnolin-3-yl)acetamide [2436];

4-(piperidin-4-yloxy)-N-(6-(thiazol-5-yl)cinnolin-3-yl)benzamide [2437];

N-(6-(thiazol-5-yl)cinnolin-3-yl)isonicotinamide [2438];

6-(4-methylpiperazin-1-yl)-N-(6-(thiazol-5-yl)cinnolin-3-yl)nicotinamide [2439];

1′-methyl-N-(6-(thiazol-5-yl)cinnolin-3-yl)-1′,2′,3′,6′-tetrahydro-[2,4′-bipyridine]-4-carboxamide [2440];

2-(3-(dimethylamino)azetidin-1-yl)-N-(6-(thiazol-5-yl)cinnolin-3-yl)isonicotinamide [2441];

2-(4-(dimethylamino)piperidin-1-yl)-N-(6-(thiazol-5-yl)cinnolin-3-yl)isonicotinamide [2442];

2-(4-methylpiperazin-1-yl)-N-(6-(thiazol-5-yl)cinnolin-3-yl)isonicotinamide [2443];

2-((1-methylpiperidin-4-yl)thio)-N-(6-(thiazol-5-yl)cinnolin-3-yl)isonicotinamide [2444];

N-(6-(thiazol-5-yl)cinnolin-3-yl)-1,2,3,4-tetrahydroisoquinoline-7-carboxamide [2445];

trans-4-((1,3-difluoropropan-2-yl)amino)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl) cyclohexane-1-carboxamide [2446];

N-(6-(2-methylthiazol-5-yl)cinnolin-3-yl)morpholine-4-carboxamide [2447];

N-(6-(2-methylthiazol-5-yl)cinnolin-3-yl)-2-(pyrrolidin-1-yl)acetamide [2448];

2-((1R,4R)-2-oxa-5-azabicyclo[2.2.1]heptan-5-yl)-N-(6-(2-methylthiazol-5-yl)cinnolin-3-yl)acetamide [2449];

N-(6-(2-methylthiazol-5-yl)cinnolin-3-yl)-2-morpholinoacetamide [2450];

N-(6-(2-methylthiazol-5-yl)cinnolin-3-yl)-2-(morpholino-d 8 )acetamide [2451];

2-(4-methylpiperazin-1-yl)-N-(6-(2-methylthiazol-5-yl)cinnolin-3-yl)acetamide [2452];

1-methyl-N-(6-(2-methylthiazol-5-yl)cinnolin-3-yl)piperidine-4-carboxamide [2453];

N-(6-(2-methylthiazol-5-yl)cinnolin-3-yl)isonicotinamide [2454];

N-(6-(2-methylthiazol-5-yl)cinnolin-3-yl)nicotinamide [2455];

2-(4-methylpiperazin-1-yl)-N-(6-(2-methylthiazol-5-yl)cinnolin-3-yl)isonicotinamide [2456];

trans-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-4-morpholinocyclohexane-1-carboxamide [2457];

trans-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-4-(4-methylpiperazin-1-yl) cyclohexane-1-carboxamide [2458];

4-isopropyl-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)piperazine-1-carboxamide [2459];

4-((2-methoxyethyl)(methyl)amino)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl) piperidine-1-carboxamide [2460];

4-((1,3-difluoropropan-2-yl)amino)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl) piperidine-1-carboxamide [2461];

N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-4-((3,3,3-trifluoropropyl)amino)piperidine-1-carboxamide [2462];

4-((2-fluoroethyl)amino)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)piperidine-1-carboxamide [2463];

(3R,4S)-4-amino-3-fluoro-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)piperidine-1-carboxamide [2464];

(3R,4R)-4-amino-3-fluoro-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)piperidine-1-carboxamide [2465];

(3S,4S)-3-fluoro-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-4-(methylamino)piperidine-1-carboxamide [2466];

(3R,4R)-3-fluoro-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-4-(methylamino) piperidine-1-carboxamide [2467];

4-amino-3,3-difluoro-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)piperidine-1-carboxamide [2468];

(3R,4R)-3-fluoro-4-(isopropylamino)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl) piperidine-1-carboxamide [2469];

(3R,4S)-3-fluoro-4-(isopropylamino)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl) piperidine-1-carboxamide [2470];

3,3-difluoro-4-(isopropylamino)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)piperidine-1-carboxamide [2471];

(3S,4S)-3-fluoro-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-4-((propan-2-yl-1,1,1,3,3,3-d 6 )amino)piperidine-1-carboxamide [2472];

(1R,3s,5S)-3-((1,3-difluoropropan-2-yl)amino)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-8-azabicyclo[3.2.1]octane-8-carboxamide [2473];

(1R,3s,5S)-3-((1,3-difluoropropan-2-yl)amino)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-8-azabicyclo[3.2.1]octane-8-carboxamide [2474];

4-(dimethylamino)-N-(6-(2-methylthiazol-5-yl)cinnolin-3-yl)piperidine-1-carboxamide [2475];

4-((2,2-difluoroethyl)amino)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)piperidine-1-carboxamide [2476];

4-((2,2-difluoroethyl)(methyl-d 3 )amino)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)piperidine-1-carboxamide [2477];

N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-4-morpholinopiperidine-1-carboxamide [2478];

N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-4-(4-methylpiperazin-1-yl)piperidine-1-carboxamide [2479];

(R)-3,4-dimethyl-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)piperazine-1-carboxamide [2480];

(S)-3,4-dimethyl-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)piperazine-1-carboxamide [2481];

(1R,3r,5 S)-3-((2-fluoroethyl)amino)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-8-azabicyclo[3.2.1]octane-8-carboxamide [2482];

(1R,3r,5S)-3-((2,2-difluoroethyl)amino)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-8-azabicyclo[3.2.1]octane-8-carboxamide [2483];

(1R,3r,5 S)-3-amino-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-8-azabicyclo[3.2.1] octane-8-carboxamide [2484];

(1S,4S)-5-methyl-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-2,5-diazabicyclo[2.2.1] heptane-2-carboxamide [2485];

(1R,4R)-5-methyl-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-2,5-diazabicyclo[2.2.1] heptane-2-carboxamide [2486];

8-methyl-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-3,8-diazabicyclo[3.2.1]octane-3-carboxamide [2487];

3-methyl-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-3,8-diazabicyclo[3.2.1]octane-8-carboxamide [2488];

N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-5,6-dihydroimidazo[1,2-a]pyrazine-7(8H)-carboxamide [2489];

2-(4-methylpiperazin-1-yl)-N-(6-(5-methylthiazol-2-yl)cinnolin-3-yl)isonicotinamide [2490];

2-(4-methylpiperazin-1-yl)-N-(6-(4-methylthiazol-2-yl)cinnolin-3-yl)isonicotinamide [2491];

N-(6-(2-(methylamino)thiazol-5-yl)cinnolin-3-yl)piperidine-4-carboxamide [2492];

1-methyl-N-(6-(2-(methylamino)thiazol-5-yl)cinnolin-3-yl)piperidine-4-carboxamide [2493];

N-(6-(2-(diethylamino)thiazol-5-yl)cinnolin-3-yl)-2-(4-fluoropiperidin-1-yl)acetamide [2494];

N-(6-(2-(diethylamino)thiazol-5-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)acetamide [2495];

N-(6-(2-aminothiazol-5-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [2496];

N-(6-(2-(methylamino)thiazol-5-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [2497];

N-(6-(2-(dimethylamino)thiazol-5-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [2498];

2-(4-isopropylpiperazin-1-yl)-N-(6-(2-(methylamino)thiazol-5-yl)cinnolin-3-yl)isonicotinamide [2499];

2-(3-(dimethylamino)azetidin-1-yl)-N-(6-(2-(methylamino)thiazol-5-yl)cinnolin-3-yl) isonicotinamide [2500];

2-(3-(dimethylamino)azetidin-1-yl)-N-(6-(2-(dimethylamino)thiazol-5-yl)cinnolin-3-yl) isonicotinamide [2501];

2-(3-aminoazetidin-1-yl)-N-(6-(2-(dimethylamino)thiazol-5-yl)cinnolin-3-yl)isonicotinamide [2502];

N-(6-(5-chlorothiazol-2-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [2503];

2-(3-(2-(4-methylpiperazin-1-yl)isonicotinamido)cinnolin-6-yl)thiazole-5-carboxamide [2504];

N-(6-(isothiazol-4-yl)cinnolin-3-yl)-1-methylpiperidine-4-carboxamide [2505];

N-(6-(1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-4-(difluoromethoxy)benzamide [2506];

N-(6-(1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-4-(piperidin-4-yloxy)benzamide [2507];

N-(6-(1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-4-((l-methylpiperidin-4-yl)oxy)benzamide [2508];

N-(6-(1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-3-((1-methylpiperidin-4-yl)oxy)benzamide [2509];

N 5 -(6-(1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-N 2 -methylpyridine-2,5-dicarboxamide [2510];

N-(6-(1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-6-(4-methylpiperazin-1-yl)nicotinamide [2511];

N-(6-(1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-1′-methyl-1′,2′,3′,6′-tetrahydro-[2,4′-bipyridine]-4-carboxamide [2512];

N-(6-(1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-2-(3-(dimethylamino)azetidin-1-yl)isonicotinamide [2513];

N-(6-(1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [2514];

N-(6-(1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-2-(4-isopropylpiperazin-1-yl)isonicotinamide [2515];

N-(6-(1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-2-morpholinoisonicotinamide [2516];

1-fluoro-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)cyclohexane-1-carboxamide [2517];

trans-4-methoxy-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)cyclohexane-1-carboxamide [2518];

cis-4-methoxy-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)cyclohexane-1-carboxamide [2519];

trans-4-amino-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)cyclohexane-1-carboxamide [2520];

trans-4-(dimethylamino)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)cyclohexane-1-carboxamide [2521];

trans-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-4-morpholinocyclohexane-1-carboxamide [2522];

trans-4-(hydroxymethyl)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)cyclohexane-1-carboxamide [2523];

N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)piperidine-4-carboxamide [2524];

4-fluoro-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)piperidine-4-carboxamide [2525];

1-methyl-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)piperidine-4-carboxamide [2526];

4-fluoro-1-methyl-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)piperidine-4-carboxamide [2527];

1-(2-fluoroethyl)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)piperidine-4-carboxamide [2528];

1-(2,2-difluoroethyl)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)piperidine-4-carboxamide [2529];

N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [2530];

1-(2,2-difluoropropyl)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)piperidine-4-carboxamide [2531];

1-benzoyl-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)piperidine-4-carboxamide [2532];

N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-2-(pyrrolidin-1-yl)acetamide [2533];

N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-2-(piperidin-1-yl)acetamide [2534];

2-(4-methoxypiperidin-1-yl)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)acetamide [2535];

N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)acetamide [2536];

N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-2-morpholinoacetamide [2537];

(R)—N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-2-(3-methylmorpholino)acetamide [2538];

2-(7-azabicyclo[2.2.1]heptan-7-yl)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)acetamide [2539];

2-((1R,4R)-2-oxa-5-azabicyclo[2.2.1]heptan-5-yl)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)acetamide [2540];

2-(3-oxa-8-azabicyclo[3.2.1]octan-8-yl)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)acetamide [2541];

2-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)acetamide [2542];

N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-2-(1,4-oxazepan-4-yl)acetamide [2543];

N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-2-morpholinoacetamide-2,2-d 2 [2544];

N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-2-(morpholino-d 8 )acetamide [2545];

1-methyl-3-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-1-(1-methylpiperidin-4-yl)urea [2546];

(3S,4S)-4-amino-3-fluoro-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)piperidine-1-carboxamide [2547];

(3S,4S)-4-(dimethylamino)-3-fluor N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl) piperidine-1-carboxamide [2548];

N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)morpholine-4-carboxamide [2549];

N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-4-(methylamino)piperidine-1-carboxamide [2550];

4-(dimethylamino)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)piperidine-1-carboxamide [2551];

4-((2,2-difluoroethyl)(methyl)amino)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl) piperidine-1-carboxamide [2552];

(3S,4S)-3-fluoro-4-(isopropylamino)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl) piperidine-1-carboxamide [2553];

2-methyl-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-5,6-dihydroimidazo[1,2-a]pyrazine-7(8H)-carboxamide [2554];

4-methyl-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)piperazine-1-carboxamide [2555];

N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-1-(1-methylpiperidin-4-yl)-1H-pyrazole-4-carboxamide [2556];

1-(1-isopropylpiperidin-4-yl)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-1H-pyrazole-4-carboxamide [2557];

N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-1-(1-methylpiperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide [2558];

N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-2-(piperidin-4-yl)oxazole-4-carboxamide [2559];

N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-2-(1-methylpiperidin-4-yl)oxazole-4-carboxamide [2560];

2-(3-(dimethylamino)azetidin-1-yl)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)isonicotinamide [2561];

1′-methyl-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-1′,2′,3′,6′-tetrahydro-[2,4′-bipyridine]-4-carboxamide [2562];

N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [2563];

2-(methyl(1-methylpiperidin-4-yl)amino)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl) isonicotinamide [2564];

2-(azetidin-3-yloxy)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)isonicotinamide [2565];

N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-3-((1-methylpiperidin-4-yl)oxy)benzamide [2566];

N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-2-((1-methylpiperidin-4-yl)thio) isonicotinamide [2567];

6-(4-methylpiperazin-1-yl)-N-(6-(5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl)cinnolin-3-yl) nicotinamide [2568];

2-(4-methylpiperazin-1-yl)-N-(6-(5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl)cinnolin-3-yl) isonicotinamide [2569];

N-(6-(5-amino-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [2570];

N-(6-(5-(dimethylamino)-1,3,4-thiadiazol-2-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [2571];

N-(6-(3-amino-5-fluorophenyl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [2572];

N-(6-(3-fluoro-5-(isopropylamino)phenyl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [2573];

1-methyl-N-(6-(pyridin-2-yl)cinnolin-3-yl)piperidine-4-carboxamide [2574];

2-(4-methylpiperazin-1-yl)-N-(6-(pyridin-2-yl)cinnolin-3-yl)isonicotinamide [2575];

2-(4-methylpiperazin-1-yl)-N-(6-(pyridin-4-yl)cinnolin-3-yl)isonicotinamide [2576];

N-(6-(pyridin-3-yl)cinnolin-3-yl)cyclopropanecarboxamide [2577];

N-(6-(pyridin-3-yl)cinnolin-3-yl)-2-(pyrrolidin-1-yl)acetamide [2578];

1-methyl-N-(6-(pyridin-3-yl)cinnolin-3-yl)piperidine-4-carboxamide [2579];

N-(6-(pyridin-3-yl)cinnolin-3-yl)quinuclidine-4-carboxamide [2580];

2-morpholino-N-(6-(pyridin-3-yl)cinnolin-3-yl)acetamide [2581];

2-(morpholino-d 8 )—N-(6-(pyridin-3-yl)cinnolin-3-yl)acetamide [2582];

2-(4-methylpiperazin-1-yl)-N-(6-(pyridin-3-yl)cinnolin-3-yl)acetamide [2583];

2-(4-methyl-1,4-diazepan-1-yl)-N-(6-(pyridin-3-yl)cinnolin-3-yl)acetamide [2584];

2-(4-methylpiperazin-1-yl)-N-(6-(pyridin-3-yl)cinnolin-3-yl)isonicotinamide [2585];

2-(2-methyl-1H-imidazol-1-yl)-N-(6-(pyridin-3-yl)cinnolin-3-yl)acetamide [2586];

2-(1H-imidazol-1-yl)-N-(6-(pyridin-3-yl)cinnolin-3-yl)acetamide [2587];

2-(piperidin-4-yl)-N-(6-(pyridin-3-yl)cinnolin-3-yl)oxazole-4-carboxamide [2588];

2-(1-methylpiperidin-4-yl)-N-(6-(pyridin-3-yl)cinnolin-3-yl)oxazole-4-carboxamide [2589];

2-(1-isopropylpiperidin-4-yl)-N-(6-(pyridin-3-yl)cinnolin-3-yl)oxazole-4-carboxamide [2590];

trans-N-(6-(5-fluoropyridin-3-yl)cinnolin-3-yl)-3-morpholinocyclobutane-1-carboxamide [2591];

trans-N-(6-(5-fluoropyridin-3-yl)cinnolin-3-yl)-4-((4-methylpiperazin-1-yl)methyl)cyclohexane-1-carboxamide [2592];

N-(6-(5-fluoropyridin-3-yl)cinnolin-3-yl)-2-(pyrrolidin-1-yl)acetamide [2593];

N-(6-(5-fluoropyridin-3-yl)cinnolin-3-yl)-1-methylpiperidine-4-carboxamide [2594];

N-(6-(5-fluoropyridin-3-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)acetamide [2595];

N-(6-(6-fluoropyridin-3-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)acetamide [2596];

N-(6-(5-fluoropyridin-3-yl)cinnolin-3-yl)-2-morpholinoacetamide [2597];

N-(6-(5-fluoropyridin-3-yl)cinnolin-3-yl)-3-morpholinopropanamide [2598];

N-(6-(5-fluoropyridin-3-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [2599];

N-(6-(5-fluoropyridin-3-yl)cinnolin-3-yl)-2-(piperidin-4-yl)oxazole-4-carboxamide [2600];

N-(6-(5-fluoropyridin-3-yl)cinnolin-3-yl)-2-(1-methylpiperidin-4-yl)oxazole-4-carboxamide [2601];

N-(6-(5-fluoropyridin-3-yl)cinnolin-3-yl)-2-(1-isopropylpiperidin-4-yl)oxazole-4-carboxamide [2602];

N-(6-(5-chloropyridin-3-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [2603];

N-(6-(5-methylpyridin-3-yl)cinnolin-3-yl)-2-morpholinoacetamide [2604];

N-(6-(5-(difluoromethyl)pyridin-3-yl)cinnolin-3-yl)-3-(piperidin-4-yl)benzamide [2605];

N-(6-(5-(difluoromethyl)pyridin-3-yl)cinnolin-3-yl)-3-(1-methylpiperidin-4-yl)benzamide [2606];

N-(6-(5-(difluoromethyl)pyridin-3-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [2607];

2-(4-methylpiperazin-1-yl)-N-(6-(5-(trifluoromethyl)pyridin-3-yl)cinnolin-3-yl)acetamide [2608];

2-(4-methylpiperazin-1-yl)-N-(6-(6-(trifluoromethyl)pyridin-3-yl)cinnolin-3-yl)acetamide [2609];

N-(6-(5-(hydroxymethyl)pyridin-3-yl)cinnolin-3-yl)-1-methylpiperidine-4-carboxamide [2610];

N-(6-(5-cyanopyridin-3-yl)cinnolin-3-yl)-1-methylpiperidine-4-carboxamide [2611];

N-(6-(5-methoxypyridin-3-yl)cinnolin-3-yl)-1-methylpiperidine-4-carboxamide [2612];

N-(6-(5-methoxypyridin-3-yl)cinnolin-3-yl)-2-morpholinoacetamide [2613];

N-(6-(5-methoxypyridin-3-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [2614];

4-fluoro-N-(6-(5-(piperidin-4-yloxy)pyridin-3-yl)cinnolin-3-yl)benzamide [2615];

N-(6-(5-aminopyridin-3-yl)cinnolin-3-yl)-4-fluorobenzamide [2616];

N-(6-(5-aminopyridin-3-yl)cinnolin-3-yl)-4-(piperidin-4-yloxy)benzamide [2617];

N-(6-(5-aminopyridin-3-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [2618];

N-(6-(5-aminopyridin-3-yl)cinnolin-3-yl)-2-(piperidin-4-yl)oxazole-4-carboxamide [2619];

N-(6-(6-aminopyridin-3-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [2620];

N-(6-(6-(methylamino)pyridin-3-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [2621];

N-(6-(5-(isopropylamino)pyridin-3-yl)cinnolin-3-yl)-3-(piperidin-4-yl)benzamide [2622];

N-(6-(5-(isopropylamino)pyridin-3-yl)cinnolin-3-yl)-3-(1-methylpiperidin-4-yl)benzamide [2623];

N-(6-(5-(isopropylamino)pyridin-3-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [2624];

N-(6-(5-(piperidin-4-ylamino)pyridin-3-yl)cinnolin-3-yl)cyclohexanecarboxamide [2625];

4-fluoro-N-(6-(5-(piperidin-4-ylamino)pyridin-3-yl)cinnolin-3-yl)benzamide [2626];

4-fluoro-N-(6-(5-((1-methylpiperidin-4-yl)amino)pyridin-3-yl)cinnolin-3-yl)benzamide [2627];

N-(6-(5-acetamidopyridin-3-yl)cinnolin-3-yl)-1-methylpiperidine-4-carboxamide [2628];

N-(6-(5-(dimethylamino)pyridin-3-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [2629];

N-(6-(6-(dimethylamino)pyridin-3-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [2630];

1-methyl-N-(6-(5-(pyrrolidin-1-yl)pyridin-3-yl)cinnolin-3-yl)piperidine-4-carboxamide [2631];

N-(6-(5-(pyrrolidin-1-ylmethyl)pyridin-3-yl)cinnolin-3-yl)cyclopropanecarboxamide [2632];

4-fluoro-N-(6-(5-(pyrrolidin-1-ylmethyl)pyridin-3-yl)cinnolin-3-yl)benzamide [2633];

N-(6-(5-((4-hydroxypiperidin-1-yl)methyl)pyridin-3-yl)cinnolin-3-yl)cyclopropanecarboxamide [2634];

4-fluoro-N-(6-(5-((4-hydroxypiperidin-1-yl)methyl)pyridin-3-yl)cinnolin-3-yl)benzamide [2635];

N-(6-(5-(piperazin-1-ylmethyl)pyridin-3-yl)cinnolin-3-yl)cyclopropanecarboxamide [2636];

N-(6-(5-((4-methylpiperazin-1-yl)methyl)pyridin-3-yl)cinnolin-3-yl)cyclopropanecarboxamide [2637];

N-(6-(5-(morpholinomethyl)pyridin-3-yl)cinnolin-3-yl)cyclopropanecarboxamide [2638];

N-methyl-5-(3-(1-methylpiperidine-4-carboxamido)cinnolin-6-yl)nicotinamide [2639];

N-methyl-5-(3-(2-(4-methylpiperazin-1-yl)isonicotinamido)cinnolin-6-yl)nicotinamide [2640];

N-(6-(pyridin-3-yl-d 4 )cinnolin-3-yl)-2-(pyrrolidin-1-yl)acetamide [2641];

2-(4-methylpiperazin-1-yl)-N-(6-(pyridin-3-yl-d 4 )cinnolin-3-yl)acetamide [2642];

2-morpholino-N-(6-(pyridin-3-yl-d 4 )cinnolin-3-yl)acetamide [2643];

1-methyl-N-(6-(2-methylpyrimidin-5-yl)cinnolin-3-yl)piperidine-4-carboxamide [2644];

2-(4-methylpiperazin-1-yl)-N-(6-(2-methylpyrimidin-5-yl)cinnolin-3-yl)isonicotinamide [2645];

N-(6-(2-aminopyrimidin-5-yl)cinnolin-3-yl)-1-methylpiperidine-4-carboxamide [2646];

2-morpholino-N-(6-(pyridazin-3-yl)cinnolin-3-yl)acetamide [2647];

2-morpholino-N-(6-(pyridazin-4-yl)cinnolin-3-yl)acetamide [2648];

N-(6-(pyridazin-4-yl)cinnolin-3-yl)-2-(pyrrolidin-1-yl)acetamide [2649];

trans-3-morpholino-N-(6-(pyrazin-2-yl)cinnolin-3-yl)cyclobutane-1-carboxamide [2650];

trans-4-(dimethylamino)-N-(6-(pyrazin-2-yl)cinnolin-3-yl)cyclohexane-1-carboxamide [2651];

trans-4-morpholino-N-(6-(pyrazin-2-yl)cinnolin-3-yl)cyclohexane-1-carboxamide [2652];

trans-4-((3-fluoroazetidin-1-yl)methyl)-N-(6-(pyrazin-2-yl)cinnolin-3-yl)cyclohexane-1-carboxamide [2653];

trans-4-((4-methylpiperazin-1-yl)methyl)-N-(6-(pyrazin-2-yl)cinnolin-3-yl)cyclohexane-1-carboxamide [2654];

N-(6-(pyrazin-2-yl)cinnolin-3-yl)-2-(pyrrolidin-1-yl)acetamide [2655];

1-methyl-N-(6-(pyrazin-2-yl)cinnolin-3-yl)piperidine-4-carboxamide [2656];

4-fluoro-1-methyl-N-(6-(pyrazin-2-yl)cinnolin-3-yl)piperidine-4-carboxamide [2657];

1-(2-fluoroethyl)-N-(6-(pyrazin-2-yl)cinnolin-3-yl)piperidine-4-carboxamide [2658];

1-(oxetan-3-yl)-N-(6-(pyrazin-2-yl)cinnolin-3-yl)piperidine-4-carboxamide [2659];

2-morpholino-N-(6-(pyrazin-2-yl)cinnolin-3-yl)acetamide [2660];

1-methyl-N-(6-(pyrazin-2-yl)cinnolin-3-yl)azepane-4-carboxamide [2661];

1-isobutyl-N-(6-(pyrazin-2-yl)cinnolin-3-yl)azepane-4-carboxamide [2662];

1-(2-hydroxy-2-methylpropyl)-N-(6-(pyrazin-2-yl)cinnolin-3-yl)azepane-4-carboxamide [2663];

4-(morpholinomethyl)-N-(6-(pyrazin-2-yl)cinnolin-3-yl)benzamide [2664];

2-(4-methylpiperazin-1-yl)-N-(6-(pyrazin-2-yl)cinnolin-3-yl)isonicotinamide [2665];

N-(6-(6-(methylamino)pyrazin-2-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [2666];

N-(6-(6-(isopropylamino)pyrazin-2-yl)cinnolin-3-yl)azetidine-3-carboxamide [2667];

N-(6-(6-(isopropylamino)pyrazin-2-yl)cinnolin-3-yl)piperidine-4-carboxamide [2668];

N-(6-(6-(isopropylamino)pyrazin-2-yl)cinnolin-3-yl)-1-methylpiperidine-4-carboxamide [2669];

1-(2-fluoroethyl)-N-(6-(6-(isopropylamino)pyrazin-2-yl)cinnolin-3-yl)piperidine-4-carboxamide [2670];

1-isopropyl-N-(6-(6-(isopropylamino)pyrazin-2-yl)cinnolin-3-yl)piperidine-4-carboxamide [2671];

1-isopentyl-N-(6-(6-(isopropylamino)pyrazin-2-yl)cinnolin-3-yl)piperidine-4-carboxamide [2672];

N-(6-(6-(isopropylamino)pyrazin-2-yl)cinnolin-3-yl)-3-(piperidin-4-yl)benzamide [2673];

N-(6-(6-(isopropylamino)pyrazin-2-yl)cinnolin-3-yl)-3-(1-methylpiperidin-4-yl)benzamide [2674];

N-(6-(6-(isopropylamino)pyrazin-2-yl)cinnolin-3-yl)-1-(piperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide [2675];

1-(1-(2-fluoroethyl)piperidin-4-yl)-N-(6-(6-(isopropylamino)pyrazin-2-yl)cinnolin-3-yl)-1H-1,2,3-triazole-4-carboxamide [2676];

N-(6-(6-(isopropylamino)pyrazin-2-yl)cinnolin-3-yl)-1-(1-isopropylpiperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide [2677];

N-(6-(6-(isopropylamino)pyrazin-2-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [2678];

N-(6-(6-(tert-butylamino)pyrazin-2-yl)cinnolin-3-yl)-2-(3-(dimethylamino)azetidin-1-yl) isonicotinamide [2679];

N-(6-(6-(tert-butylamino)pyrazin-2-yl)cinnolin-3-yl)-1′-methyl-1′,2′,3′,6′-tetrahydro-[2,4′-bipyridine]-4-carboxamide [2680];

N-(6-(6-(tert-butylamino)pyrazin-2-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [2681];

N-(6-(6-(tert-butylamino)pyrazin-2-yl)cinnolin-3-yl)-2-(4-isopropylpiperazin-1-yl) isonicotinamide [2682];

N-(6-(6-(tert-butylamino)pyrazin-2-yl)cinnolin-3-yl)-2-morpholinoisonicotinamide [2683];

N-(6-(6-(((3-fluoroazetidin-3-yl)methyl)amino)pyrazin-2-yl)cinnolin-3-yl) cyclopropanecarboxamide [2684];

4-fluoro-N-(6-(6-(((3-fluoroazetidin-3-yl)methyl)amino)pyrazin-2-yl)cinnolin-3-yl)benzamide [2685];

N-(6-(6-(piperidin-4-ylamino)pyrazin-2-yl)cinnolin-3-yl)cyclobutanecarboxamide [2686];

3,3-difluoro-N-(6-(6-(piperidin-4-ylamino)pyrazin-2-yl)cinnolin-3-yl)cyclobutane-1-carboxamide [2687];

N-(6-(6-(piperidin-4-ylamino)pyrazin-2-yl)cinnolin-3-yl)cyclopentanecarboxamide [2688];

4,4-difluoro-N-(6-(6-(piperidin-4-ylamino)pyrazin-2-yl)cinnolin-3-yl)cyclohexane-1-carboxamide [2689];

N-(6-(6-(piperidin-4-ylamino)pyrazin-2-yl)cinnolin-3-yl)tetrahydro-2H-pyran-4-carboxamide [2690];

4-fluoro-N-(6-(6-(piperidin-4-ylamino)pyrazin-2-yl)cinnolin-3-yl)benzamide [2691];

N-(6-(6-(((3 S,4S)-3-fluoropiperidin-4-yl)amino)pyrazin-2-yl)cinnolin-3-yl) cyclopropanecarboxamide [2692];

4-fluoro-N-(6-(6-(((3S,4S)-3-fluoropiperidin-4-yl)amino)pyrazin-2-yl)cinnolin-3-yl)benzamide [2693];

N-(6-(6-((1-methylpiperidin-4-yl)amino)pyrazin-2-yl)cinnolin-3-yl)cyclobutanecarboxamide [2694];

N-(6-(6-((1-methylpiperidin-4-yl)amino)pyrazin-2-yl)cinnolin-3-yl)cyclopentanecarboxamide [2695];

4-fluoro-N-(6-(6-((1-methylpiperidin-4-yl)amino)pyrazin-2-yl)cinnolin-3-yl)benzamide [2696];

N-(6-(6-((1-isopropylpiperidin-4-yl)amino)pyrazin-2-yl)cinnolin-3-yl)cyclopropanecarboxamide [2697];

3,3-difluoro-N-(6-(6-((1-isopropylpiperidin-4-yl)amino)pyrazin-2-yl)cinnolin-3-yl)cyclobutane-1-carboxamide [2698];

N-(6-(6-((1-isopropylpiperidin-4-yl)amino)pyrazin-2-yl)cinnolin-3-yl)cyclopentanecarboxamide [2699];

4-fluoro-N-(6-(6-((1-isopropylpiperidin-4-yl)amino)pyrazin-2-yl)cinnolin-3-yl)benzamide [2700];

N-(6-(6-(dimethylamino)pyrazin-2-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [2701];

N-(6-(6-(diethylamino)pyrazin-2-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [2702];

N-(6-(6-(3-aminoazetidin-1-yl)pyrazin-2-yl)cinnolin-3-yl)-4-fluorobenzamide [2703];

2-(4-methylpiperazin-1-yl)-N-(6-(6-(pyrrolidin-1-yl)pyrazin-2-yl)cinnolin-3-yl)isonicotinamide [2704];

N-(6-(6-(azetidin-3-ylmethoxy)pyrazin-2-yl)cinnolin-3-yl)-4-fluorobenzamide [2705];

N-(6-(6-(azetidin-3-yloxy)pyrazin-2-yl)cinnolin-3-yl)-4-fluorobenzamide [2706];

N-(6-(1H-pyrrolo[2,3-b]pyridin-5-yl)cinnolin-3-yl)-1-(1-methylpiperidin-4-yl)-1H-pyrazole-4-carboxamide [2707];

N-(6-(1H-pyrrolo[3,2-b]pyridin-6-yl)cinnolin-3-yl)-1-(1-methylpiperidin-4-yl)-1H-pyrazole-4-carboxamide [2708];

N-(6-(1H-pyrrolo[2,3-c]pyridin-4-yl)cinnolin-3-yl)-1-(1-methylpiperidin-4-yl)-1H-pyrazole-4-carboxamide [2709];

N-(6-(1H-pyrrolo[2,3-b]pyridin-5-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [2710];

N-(6-(1H-pyrrolo[3,2-b]pyridin-6-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [2711];

N-(6-(1H-pyrrolo[2,3-c]pyridin-4-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [2712];

2-(4-methylpiperazin-1-yl)-N-(6-(oxazolo[5,4-b]pyridin-6-yl)cinnolin-3-yl)isonicotinamide [2713];

N-(6-(2-methyl-1H-pyrrolo[2,3-b]pyridin-5-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [2714];

N-(6-(3-methyl-1H-pyrrolo[2,3-b]pyridin-5-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [2715];

N-(6-(2-methyl-1H-pyrrolo[3,2-b]pyridin-6-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [2716];

N-(6-(5H-pyrrolo[2,3-b]pyrazin-2-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [2717];

N-(6-(5H-pyrrolo[2,3-b]pyrazin-3-yl)cinnolin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [2718];

1-isopropyl-N-(6-(6-(piperidin-4-ylamino)pyrazin-2-yl)cinnolin-3-yl)-1H-pyrazole-4-carboxamide [2719];

1-isopropyl-N-(6-(6-((1-methylpiperidin-4-yl)amino)pyrazin-2-yl)cinnolin-3-yl)-1H-pyrazole-4-carboxamide [2720]; or a pharmaceutically acceptable salt thereof.

15. The compound of claim 1 , wherein the compound of Formula I is selected from the group consisting of:

N-(3-(1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-1-isobutylpiperidine-4-carboxamide [2721];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)cyclopropanecarboxamide [2722];

4,4-difluoro-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)cyclohexane-1-carboxamide [2723];

trans-4-methoxy-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)cyclohexane-1-carboxamide [2724];

trans-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-4-morpholinocyclohexane-1-carboxamide [2725];

trans-4-((3-fluoroazetidin-1-yl)methyl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl) cyclohexane-1-carboxamide [2726];

trans-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-4-((4-methylpiperazin-1-yl) methyl)cyclohexane-1-carboxamide [2727];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(pyrrolidin-1-yl)acetamide [2728];

(S)-2-(3-fluoropyrrolidin-1-yl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl) acetamide [2729];

(S)—N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)tetrahydrofuran-2-carboxamide [2730];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [2731];

1-methyl-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [2732];

1-isopropyl-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [2733];

1-(tert-butyl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [2734];

1-cyclopropyl-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [2735];

1-isobutyl-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [2736];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-1-neopentylpiperidine-4-carboxamide [2737];

1-(2-fluoroethyl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [2738];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [2739];

1-butyl-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [2740];

1-benzoyl-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [2741];

1-(2,2-difluoropropyl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [2742];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)azetidine-3-carboxamide [2743];

1-(2,2-difluoroethyl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [2744];

1-(2-fluoro-2-methylpropyl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [2745];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-1-(oxetan-3-yl)piperidine-4-carboxamide [2746];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-1-((3-methyloxetan-3-yl)methyl) piperidine-4-carboxamide [2747];

1-(2-methoxyethyl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [2748];

1-(2-isopropoxyethyl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [2749];

1,1-diisobutyl-4-((3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)carbamoyl)piperidin-1-ium [2750];

4-fluoro-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [2751];

4-fluoro-1-methyl-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [2752];

4-fluoro-1-isobutyl-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [2753];

(S)—N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)piperidine-3-carboxamide [2754];

(R)—N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)piperidine-3-carboxamide [2755];

(S)-1-isobutyl-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)piperidine-3-carboxamide [2756];

(R)-1-isobutyl-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)piperidine-3-carboxamide [2757];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)tetrahydro-2H-pyran-4-carboxamide [2758];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(piperidin-1-yl)acetamide [2759];

2-(4-fluoropiperidin-1-yl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)acetamide [2760];

trans-4-amino-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)cyclohexane-1-carboxamide [2761];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl)acetamide [2762];

(S)—N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)piperidine-2-carboxamide [2763];

2-(4-isobutylpiperazin-1-yl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)acetamide [2764];

2-(3,3-dimethylazetidin-1-yl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)acetamide [2765];

(R)-2-(3-fluoropyrrolidin-1-yl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl) acetamide [2766];

(S)—N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(2-methylpyrrolidin-1-yl) acetamide [2767];

2-(3-azabicyclo[3.1.0]hexan-3-yl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl) acetamide [2768];

2-(7-azabicyclo[2.2.1]heptan-7-yl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl) acetamide [2769];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperidin-1-yl)acetamide [2770];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(4-(trifluoromethyl)piperidin-1-yl) acetamide [2771];

2-(4-(difluoromethyl)piperidin-1-yl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl) acetamide [2772];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(6-azaspiro[2.5]octan-6-yl)acetamide [2773];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(pyrrolidin-1-yl)propanamide [2774];

(R)—N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(2-methylpyrrolidin-1-yl) acetamide [2775];

2-(cyclobutyl(methyl)amino)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)acetamide [2776];

2-(diethylamino)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)acetamide [2777];

7-(2-fluoroethyl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-7-azaspiro[3.5]nonane-2-carboxamide [2778];

4-methyl-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)piperazine-1-carboxamide [2779];

(S)—N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(pyrrolidin-1-yl)propanamide [2780];

(R)—N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(pyrrolidin-1-yl)propanamide [2781];

(R)—N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)pyrrolidine-2-carboxamide [2782];

2-methyl-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-azaspiro [3.3]heptane-6-carboxamide [2783];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(2,2,2-trifluoroacetyl)-2-azaspiro [3.3]heptane-6-carboxamide [2784];

2-(2-fluoroethyl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-azaspiro[3.3]heptane-6-carboxamide [2785];

trans-4-(dimethylamino)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)cyclohexane-1-carboxamide [2786];

1-acetyl-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [2787];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-1-((1-(trifluoromethyl)cyclopropyl) methyl)piperidine-4-carboxamide [2788];

(S)-1-(2-fluoropropyl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [2789];

(R)-1-(2-fluoropropyl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [2790];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(piperidin-1-yl)propanamide [2791];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-1-(methylsulfonyl)piperidine-4-carboxamide [2792];

1′-methyl-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-[1,4′-bipiperidine]-4-carboxamide [2793];

trans-4-(hydroxymethyl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)cyclohexane-1-carboxamide [2794];

methyl 2-(4-((3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)carbamoyl)piperidin-1-yl) acetate [2795];

1-benzyl-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [2796];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-1-(2-(pyrrolidin-1-yl)acetyl)piperidine-4-carboxamide [2797];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-morpholinoacetamide [2798];

(S)—N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(3-methylmorpholino)acetamide [2799];

(R)—N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(3-methylmorpholino)acetamide [2800];

(S)—N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(2-methylmorpholino)acetamide [2801];

2-((2R,6S)-2,6-dimethylmorpholino)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl) acetamide [2802];

2-((1S,4S)-2-oxa-5-azabicyclo[2.2.1]heptan-5-yl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)acetamide [2803];

2-((1R,4R)-2-oxa-5-azabicyclo[2.2.1]heptan-5-yl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)acetamide [2804];

2-(3-oxa-8-azabicyclo[3.2.1]octan-8-yl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl) acetamide [2805];

(S)—N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-morpholinopropanamide [2806];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(morpholin-2-yl)acetamide [2807];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(4-methylmorpholin-2-yl)acetamide [2808];

2-(4-ethylpiperazin-1-yl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)acetamide [2809];

2-(4-isopropylpiperazin-1-yl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)acetamide [2810];

2-(4-cyclopropylpiperazin-1-yl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl) acetamide [2911];

2-(4-(2-fluoroethyl)piperazin-1-yl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl) acetamide [2812];

(S)-2-(2,4-dimethylpiperazin-1-yl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl) acetamide [2813];

1-(2-hydroxyethyl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [2814];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-1-(pyridin-2-ylmethyl)piperidine-4-carboxamide [2815];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-1-(oxazol-2-ylmethyl)piperidine-4-carboxamide [2816];

(R)—N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-1-oxotetrahydro-1H-pyrrolo[1,2-c]imidazole-2(3H)-carboxamide [2817];

(R)-1-methyl-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)pyrrolidine-2-carboxamide [2818];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-1-(tetrahydro-2H-pyran-4-yl)piperidine-4-carboxamide [2819];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-1-(pyrimidin-2-ylmethyl)piperidine-4-carboxamide [2820];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-1-(pyrazin-2-ylmethyl)piperidine-4-carboxamide [2821];

1-((5-methyl-1,2,4-oxadiazol-3-yl)methyl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [2822];

1-(2-hydroxy-2-methylpropyl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl) piperidine-4-carboxamide [2823];

tert-butyl 2-(4-((3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)carbamoyl)piperidin-1-yl) acetate [2824];

2-(4-((3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)carbamoyl)piperidin-1-yl)acetic acid [2825];

2-(4-methyl-1,4-diazepan-1-yl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl) acetamide [2826];

tert-butyl (3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)carbamate [2827];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)but-2-ynamide [2828];

trans-4-((3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)carbamoyl)cyclohexane-1-carboxylic acid [2829];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-3-morpholinopropanamide [2830];

trans-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-3-morpholinocyclobutane-1-carboxamide [2831];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)quinuclidine-4-carboxamide [2832];

1-isobutyl-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)azepane-4-carboxamide [2833];

2-(4-methoxypiperidin-1-yl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)acetamide [2834];

2-(4-hydroxypiperidin-1-yl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)acetamide [2835];

3-(hydroxymethyl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)bicyclo[1.1.1]pentane-1-carboxamide [2836];

1-methyl-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)azepane-4-carboxamide [2837];

trans-4-(dimethylamino)-N-(3 (1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)cyclohexane-1,7-naphthyridin-6-yl)c carboxamide [2838];

trans-4-(bis(methyl-d 3 )amino)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl) cyclohexane-1-carboxamide [2839];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-3-((4-methylpiperazin-1-yl)methyl) bicyclo[1.1.1]pentane-1-carboxamide [2840];

methyl trans-4-((3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)carbamoyl)cyclohexane-1-carboxylate [2841];

2-(1-isobutylpyrrolidin-3-yl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)acetamide [2842];

trans-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-4-(4-methylpiperazine-1-carbonyl)cyclohexane-1-carboxamide [2843];

1-isobutyl-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [2844];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-1-(phenylsulfonyl)piperidine-4-carboxamide [2845];

8-methyl-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-3,8-diazabicyclo[3.2.1]octane-3-carboxamide [2846];

3-methyl-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-3,8-diazabicyclo[3.2.1]octane-8-carboxamide [2847];

(1R,3s,5S)-3-amino-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-8-azabicyclo[3.2.1] octane-8-carboxamide [2848];

(1R,3s,5S)—N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-3-((3,3,3-trifluoropropyl) amino)-8-azabicyclo[3.2.1]octane-8-carboxamide [2849];

(1R,3s,5S)-3-((1,3-difluoropropan-2-yl)amino)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-8-azabicyclo[3.2.1]octane-8-carboxamide [2850];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)morpholine-4-carboxamide [2851];

4-(dimethylamino)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)piperidine-1-carboxamide [2852];

(S)-2,4-dimethyl-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)piperazine-1-carboxamide [2853];

1-methyl-3-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-1-(1-methylpiperidin-4-yl)urea [2854];

1-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-3-(1-methylpiperidin-4-yl)urea [2855];

4-isopropyl-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)piperazine-1-carboxamide [2856];

(R)-3,4-dimethyl-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)piperazine-1-carboxamide [2857];

N-(3-(1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [2858];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-3-(piperazin-1-yl)benzamide [2859];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-3-(4-methylpiperazin-1-yl)benzamide [2860];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-3-(pyrrolidin-1-ylmethyl)benzamide [2861];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-3-(piperidin-4-yloxy)benzamide [2862];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-3-((1-methylpiperidin-4-yl)oxy) benzamide [2863];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-4-(piperidin-4-yloxy)benzamide [2864];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-4-((1-methylpiperidin-4-yl)oxy) benzamide [2865];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(piperazin-1-yl)isonicotinamide [2866];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [2867];

2-(4-isopropylpiperazin-1-yl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl) isonicotinamide [2868];

2-(4-cyclopropylpiperazin-1-yl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl) isonicotinamide [2869];

2-(4-(2-fluoroethyl)piperazin-1-yl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl) isonicotinamide [2870];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-6-(4-methylpiperazin-1-yl)nicotinamide [2871];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-5-(piperidin-4-yloxy)nicotinamide [2872];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(piperidin-4-yloxy)isonicotinamide [2873];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-((1-methylpiperidin-4-yl)oxy) isonicotinamide [2874];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-5-(piperidin-4-ylamino)nicotinamide [2875];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-5-((1-methylpiperidin-4-yl)amino) nicotinamide [2876];

2-(4-aminopiperidin-1-yl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl) isonicotinamide [2877];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(4-(methylamino)piperidin-1-yl) isonicotinamide [2878];

2-(4-(dimethylamino)piperidin-1-yl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl) isonicotinamide [2879];

2-((1-isopropylpiperidin-4-yl)oxy)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl) isonicotinamide [2880];

2-(3-aminoazetidin-1-yl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl) isonicotinamide [2881];

2-(3-(dimethylamino)azetidin-1-yl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl) isonicotinamide [2882];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-morpholinoisonicotinamide [2883];

2-((2-(dimethylamino)ethyl)amino)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl) isonicotinamide [2884];

2-(2-(dimethylamino)ethoxy)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl) isonicotinamide [2885];

2-(4-isobutylpiperazin-1-yl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl) isonicotinamide [2886];

2-(azetidin-3-yloxy)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)isonicotinamide [2887];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-((1-methylazetidin-3-yl)oxy) isonicotinamide [2888];

2-(4-ethylpiperazin-1-yl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl) isonicotinamide [2889];

4-((dimethylamino)methyl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)benzamide [2890];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-3-(1-methylpiperidin-4-yl)benzamide [2891];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-3-((4-methylpiperazin-1-yl)methyl) benzamide [2892];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)isonicotinamide [2893];

2-hydroxy-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)isonicotinamide [2894];

2-isopropoxy-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)isonicotinamide [2895];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(1-methylpiperidin-4-yl) isonicotinamide [2896];

1′-methyl-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-1′,2′,3′,6′-tetrahydro-[2,4′-bipyridine]-4-carboxamide [2897];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(4-(6-(4-methylpiperazin-1-yl) nicotinoyl)piperazin-1-yl)isonicotinamide [2898];

2-(4-hydroxy-4-methyl-4λ4-piperazin-1-yl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)isonicotinamide [2899];

2-methyl-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-6-(4-methylpiperazin-1-yl) isonicotinamide [2900];

3-methyl-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [2901];

2-(4-methyl-1,4-diazepan-1-yl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl) isonicotinamide [2902];

2-((2S,6R)-2,6-dimethylmorpholino)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)isonicotinamide [2903];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(2,7-diazaspiro[3.5]nonan-2-yl) isonicotinamide [2904];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(7-methyl-2,7-diazaspiro[3.5]nonan-2-yl)isonicotinamide [2905];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(2,7-diazaspiro[3.5]nonan-7-yl) isonicotinamide [2906];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(2-methyl-2,7-diazaspiro[3.5]nonan-7-yl)isonicotinamide [2907];

2-(methyl(1-methylpiperidin-4-yl)amino)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)isonicotinamide [2908];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-((1-methylpiperidin-4-yl)thio) isonicotinamide [2909];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl)pyrimidine-4-carboxamide [2910];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-6-(4-methylpiperazin-1-yl)pyridazine-4-carboxamide [2911];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-6-(4-methylpiperazin-1-yl)pyrimidine-4-carboxamide [2912];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-phenylacetamide [2913];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-3-phenylpropanamide [2914];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(pyridin-3-yl)acetamide [2915];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-3-(pyridin-3-yl)propanamide [2916];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(pyridin-4-yl)acetamide [2917];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-3-(pyridin-4-yl)propanamide [2918];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)isoindoline-5-carboxamide [2919];

2-methyl-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)isoindoline-5-carboxamide [2920];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-1,2,3,4-tetrahydroisoquinoline-7-carboxamide [2921];

2-methyl-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-1,2,3,4-tetrahydroisoquinoline-7-carboxamide [2922];

2-methyl-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-1,2,3,4-tetrahydroisoquinoline-6-carboxamide [2923];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-1,2,3,4-tetrahydroisoquinoline-6-carboxamide [2924];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-1H-indole-5-carboxamide [2925];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)benzofuran-5-carboxamide [2926];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)furo[2,3-c]pyridine-5-carboxamide [2927];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)benzo[b]thiophene-5-carboxamide [2928];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)benzofuran-6-carboxamide [2929];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)benzo[d]oxazole-6-carboxamide [2930];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)benzo[d]thiazole-6-carboxamide [2931];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)benzo[d]oxazole-5-carboxamide [2932];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)benzo[d]thiazole-5-carboxamide [2933];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)quinoline-3-carboxamide [2934];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)quinoline-6-carboxamide [2935];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)quinoxaline-6-carboxamide [2936];

5-chloro-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [2937];

3-chloro-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [2938];

2-(2,5-diazabicyclo[2.2.1]heptan-2-yl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl) isonicotinamide [2939];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(5-methyl-2,5-diazabicyclo[2.2.1] heptan-2-yl)isonicotinamide [2940];

3-fluoro-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [2941];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-((4-methylpiperazin-1-yl)methyl) isonicotinamide [2942];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(morpholinomethyl)isonicotinamide [2943];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(pyrrolidin-1-ylmethyl) isonicotinamide [2944];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(2-(4-methylpiperazin-1-yl)pyridin-4-yl)acetamide [2945];

1-methyl-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-1H-indazole-5-carboxamide [2946];

1-methyl-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-1H-benzo[d]imidazole-5-carboxamide [2947];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-1-(piperidin-4-yl)-1H-pyrazole-4-carboxamide [2948];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-1-(1-methylpiperidin-4-yl)-1H-pyrazole-4-carboxamide [2949];

1-(1-ethylpiperidin-4-yl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-1H-pyrazole-4-carboxamide [2950];

1-(1-(2-fluoroethyl)piperidin-4-yl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-1H-pyrazole-4-carboxamide [2951];

1-(1-isopropylpiperidin-4-yl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-1H-pyrazole-4-carboxamide [2952];

1-(1-cyclopropylpiperidin-4-yl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-1H-pyrazole-4-carboxamide [2953];

isopropyl 4-(4-((3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)carbamoyl)-1H-pyrazol-1-yl)piperidine-1-carboxylate [2954];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-1-(piperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide [2955];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-1-(1-methylpiperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide [2956];

1-(1-(2-fluoroethyl)piperidin-4-yl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-1H-1,2,3-triazole-4-carboxamide [2957];

1-(1-isopropylpiperidin-4-yl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-1H-1,2,3-triazole-4-carboxamide [2958];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl)oxazole-5-carboxamide [2959];

2-(3-(dimethylamino)azetidin-1-yl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl) oxazole-4-carboxamide [2960];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(piperidin-4-yl)oxazole-4-carboxamide [2961];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(1-methylpiperidin-4-yl)oxazole-4-carboxamide [2962];

2-(1-(2-fluoroethyl)piperidin-4-yl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl) oxazole-4-carboxamide [2963];

2-(1-isopropylpiperidin-4-yl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)oxazole-4-carboxamide [2964];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl)oxazole-4-carboxamide [2965];

2-(3-(dimethylamino)azetidin-1-yl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl) thiazole-5-carboxamide [2966];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(piperidin-4-yl)thiazole-4-carboxamide [2967];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl)thiazole-4-carboxamide [2968];

2-(1-(2-fluoroethyl)piperidin-4-yl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl) thiazole-4-carboxamide [2969];

2-(1-isopropylpiperidin-4-yl)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)thiazole-4-carboxamide [2970];

1-methyl-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl-5-d)piperidine-4-carboxamide [2971];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-1-(2-(methyl-d 3 )propyl-1,1,2,3,3,3-d 6 ) piperidine-4-carboxamide [2972];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(pyrrolidin-1-yl-2,2,5,5-d 4 )acetamide [2973];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(4-(methyl-d 3 )piperazin-1-yl) acetamide [2974];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(morpholino-d 8 )acetamide [2975];

(S)—N-(3-(1-(methyl-d 3 )-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(pyrrolidin-1-yl)propanamide [2976];

1-isobutyl-N-(3-(1-(methyl-d 3 )-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [2977];

N-(3-(1-(methyl-d 3 )-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl) acetamide [2978];

N-(3-(1-(methyl-d 3 )-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(pyrrolidin-1-yl)acetamide [2979];

N-(3-(1-(methyl-d 3 )-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(piperidin-1-yl)acetamide [2980];

N-(3-(1-(methyl-d 3 )-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [2981];

N-(3-(1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(4-(methyl-d 3 )piperazin-1-yl)isonicotinamide [2982];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(4-(methyl-d 3 )piperazin-1-yl) isonicotinamide [2983];

N-(3-(1-(methyl-d 3 )-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [2984];

N-(3-(1-(methyl-d 3 )-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(4-(methyl-d 3 )piperazin-1-yl) isonicotinamide [2985];

N-(3-(1-(methyl-d 3 )-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-1-(piperidin-4-yl)-1H-pyrazole-4-carboxamide [2986];

N-(3-(1-(methyl-d 3 )-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-1-(1-methylpiperidin-4-yl)-1H-pyrazole-4-carboxamide [2987];

N-(3-(1-(methyl-d 3 )-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(piperidin-4-yl)oxazole-4-carboxamide [2988];

N-(3-(1-(methyl-d 3 )-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(1-methylpiperidin-4-yl)oxazole-4-carboxamide [2989];

N-(3-(1-ethyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(pyrrolidin-1-yl)acetamide [2990];

N-(3-(1-cyclopropyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(pyrrolidin-1-yl)acetamide [2991];

N-(3-(1-cyclopropyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [2992];

N-(3-(1-(1-methylpiperidin-4-yl)-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl) cyclohexanecarboxamide [2993];

2-(pyrrolidin-1-yl)-N-(3-(5-(trifluoromethyl)-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)acetamide [2994];

N-(3-(5-(hydroxymethyl)-1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-1-methylpiperidine-4-carboxamide [2995];

N-(3-(5-(hydroxymethyl)-1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)tetrahydro-2H-pyran-4-carboxamide [2996];

N-(3-(5-(azetidin-1-ylmethyl)-1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-4,4-difluorocyclohexane-1-carboxamide [2997];

4,4-difluoro-N-(3-(1-methyl-5-(pyrrolidin-1-ylmethyl)-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl) cyclohexane-1-carboxamide [2998];

4,4-difluoro-N-(3-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl) cyclohexane-1-carboxamide [2999];

2-(2-fluoroethyl)-N-(3-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-azaspiro[3.3]heptane-6-carboxamide [3000];

tert-butyl 6-((3-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl) carbamoyl)-2-azaspiro[3.3]heptane-2-carboxylate [3001];

2-fluoro-2-methyl-N-(3-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)propanamide [3002];

2-(diethylamino)-N-(3-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)acetamide [3003];

trans-4-methoxy-N-(3-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)cyclohexane-1-carboxamide [3004];

trans-4-(hydroxymethyl)-N-(3-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)cyclohexane-1-carboxamide [3005];

(R)—N-(3-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)pyrrolidine-2-carboxamide [3006];

1-isobutyl-N-(3-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl) piperidine-4-carboxamide [3007];

N-(3-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-1-(oxetan-3-yl) piperidine-4-carboxamide [3008];

1-benzoyl-N-(3-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl) piperidine-4-carboxamide [3009];

N-(3-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)tetrahydro-2H-pyran-4-carboxamide [3010];

N-(3-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperidin-1-yl)acetamide [3011];

N-(3-(1-(difluoromethyl)-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [3012];

N-(3-(1-ethyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [3013];

N-(3-(1-isopropyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-3-(piperidin-4-yloxy)benzamide [3014];

N-(3-(1-isopropyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-3-((1-methylpiperidin-4-yl)oxy) benzamide [3015];

N-(3-(1-isopropyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-4-(piperidin-4-yloxy)benzamide [3016];

N-(3-(1-cyclopropyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [3017];

4-fluoro-N-(3-(1-(1-methylpiperidin-4-yl)-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)benzamide [3018];

4-(difluoromethoxy)-N-(3-(1-(1-methylpiperidin-4-yl)-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl) benzamide [3019];

5-fluoro-N-(3-(1-(1-methylpiperidin-4-yl)-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)nicotinamide [3020];

N 2 -methyl-N 5 -(3-(1-(1-methylpiperidin-4-yl)-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)pyridine-2,5-dicarboxamide [3021];

1-isopropyl-N-(3-(1-(1-methylpiperidin-4-yl)-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-1H-pyrazole-4-carboxamide [3022];

2-methyl-N-(3-(1-(1-methylpiperidin-4-yl)-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)thiazole-5-carboxamide [3023];

N-(3-(5-amino-1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [3024];

4-(difluoromethoxy)-N-(3-(5-(hydroxymethyl)-1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl) benzamide [3025];

N-(3-(5-(hydroxymethyl)-1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [3026];

N-(3-(5-(hydroxymethyl)-1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(7-methyl-2,7-diazaspiro[3.5]nonan-2-yl)isonicotinamide [3027];

4-fluoro-N-(3-(1-methyl-5-(pyrrolidin-1-ylmethyl)-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl) benzamide [3028];

4-fluoro-N-(3-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl) benzamide [3029];

4-(difluoromethoxy)-N-(3-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)benzamide [3030];

N-(3-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-3-(pyrrolidin-1-ylmethyl)benzamide [3031];

N-(3-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(7-methyl-2,7-diazaspiro[3.5]nonan-2-yl)isonicotinamide [3032];

N-(3-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-morpholinoisonicotinamide [3033];

N-(3-(1-methyl-5-(morpholinomethyl)-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-morpholinoisonicotinamide [3034];

N-(3-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)-1,7-naphthyridin-6-yl)-1-((1-(trifluoromethyl)cyclopropyl)methyl)piperidine-4-carboxamide [3035];

3,3-difluoro-N-(3-(5-methyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)-1,7-naphthyridin-6-yl)cyclobutane-1-carboxamide [3036];

N-((4,4-difluorocyclohexyl)methyl)-3-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a] pyrazin-3-yl)-1,7-naphthyridin-6-amine [3037];

N-(3-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)-1,7-naphthyridin-6-yl)-1-((1-(trifluoromethyl)cyclopropyl)methyl)piperidine-4-carboxamide [3038];

N-(3-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)-1,7-naphthyridin-6-yl)-2-(pyrrolidin-1-yl)acetamide [3039];

2-(7-azabicyclo[2.2.1]heptan-7-yl)-N-(3-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)-1,7-naphthyridin-6-yl)acetamide [3040];

(R)—N-(3-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)-1,7-naphthyridin-6-yl)-1-isobutylpiperidine-3-carboxamide [3041];

N-(3-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)-1,7-naphthyridin-6-yl) piperidine-4-carboxamide [3042];

4-fluoro-N-(3-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)-1,7-naphthyridin-6-yl)-1-isobutylpiperidine-4-carboxamide [3043];

N-(3-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl)acetamide [3044];

4-fluoro-N-(3-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)-1,7-naphthyridin-6-yl)benzamide [3045];

N-(3-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)-1,7-naphthyridin-6-yl)-3-(4-methylpiperazin-1-yl)benzamide [3046];

N 5 -(3-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)-1,7-naphthyridin-6-yl)-N 2 -methylpyridine-2,5-dicarboxamide [3047];

N-(3-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)-1,7-naphthyridin-6-yl)-6-(4-methylpiperazin-1-yl)nicotinamide [3048];

2-(azetidin-3-yloxy)-N-(3-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)-1,7-naphthyridin-6-yl)isonicotinamide [3049];

N-(3-(1-methyl-1H-pyrazol-5-yl)-1,7-naphthyridin-6-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [3050];

1-methyl-N-(3-(1-methyl-1H-pyrazol-3-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [3051];

N-(3-(1-methyl-1H-pyrazol-3-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [3052];

2-fluoro-2-methyl-N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)propanamide [3053];

2,2,3,3-tetramethyl-N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)cyclopropane-1-carboxamide [3054];

trans-N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)-4-(pyrrolidin-1-yl) cyclohexane-1-carboxamide [3055];

trans-N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)-4-morpholinocyclohexane-1-carboxamide [3056];

N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)-2-(piperidin-1-yl)acetamide [3057];

1-ethyl-4-fluoro-N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [3058];

4-fluoro-1-isobutyl-N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [3059];

N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [3060];

N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)cyclopropanecarboxamide [3061];

4,4-difluoro-N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)cyclohexane-1-carboxamide [3062];

trans-4-(dimethylamino)-N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl) cyclohexane-1-carboxamide [3063];

trans-N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)-4-((4-methylpiperazin-1-yl) methyl)cyclohexane-1-carboxamide [3064];

N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [3065];

1-isobutyl-N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [3066];

N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)-1-((1-(trifluoromethyl)cyclopropyl) methyl)piperidine-4-carboxamide [3067];

N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)-1-((3-methyloxetan-3-yl) methyl)piperidine-4-carboxamide [3068];

N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)-1-(2-(pyrrolidin-1-yl) acetyl)piperidine-4-carboxamide [3069];

1′-methyl-N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)-[1,4′-bipiperidine]-4-carboxamide [3070];

(R)—N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)piperidine-3-carboxamide [3071];

(R)-1-isobutyl-N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)piperidine-3-carboxamide [3072];

N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)-2-(pyrrolidin-1-yl)acetamide [3073];

N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl) acetamide [3074];

2-(7-azabicyclo[2.2.1]heptan-7-yl)-N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl) acetamide [3075];

1-(2-hydroxy-2-methylpropyl)-N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl) piperidine-4-carboxamide [3076];

N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)-2-morpholinoacetamide [3077];

2-(4-methoxypiperidin-1-yl)-N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl) acetamide [3078];

N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)morpholine-4-carboxamide [3079];

N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)-1-(piperidin-4-yl)-1H-pyrazole-4-carboxamide [3080];

N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)-1-(1-methylpiperidin-4-yl)-1H-pyrazole-4-carboxamide [3081];

1-(1-ethylpiperidin-4-yl)-N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)-1H-pyrazole-4-carboxamide [3082];

1-(1-isopropylpiperidin-4-yl)-N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)-1H-pyrazole-4-carboxamide [3083];

N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)-1-(piperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide [3084];

1-(1-(2-fluoroethyl)piperidin-4-yl)-N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)-1H-1,2,3-triazole-4-carboxamide [3085];

1-(1-isopropylpiperidin-4-yl)-N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)-1H-1,2,3-triazole-4-carboxamide [3086];

N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)-2-(piperidin-4-yl)oxazole-4-carboxamide [3087];

N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)-2-(1-methylpiperidin-4-yl)oxazole-4-carboxamide [3088];

2-(1-isopropylpiperidin-4-yl)-N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl) oxazole-4-carboxamide [3089];

2-fluoro-N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)benzamide [3090];

N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)-3-((1-methylpiperidin-4-yl)oxy) benzamide [3091];

N 2 -methyl-N 5 -(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)pyridine-2,5-dicarboxamide [3092];

N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)-6-(4-methylpiperazin-1-yl) nicotinamide [3093];

2-(3-(dimethylamino)azetidin-1-yl)-N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl) isonicotinamide [3094];

N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)-2-(1-methylpiperidin-4-yl) isonicotinamide [3095];

2-(4-(dimethylamino)piperidin-1-yl)-N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)isonicotinamide [3096];

N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)-2-morpholinoisonicotinamide [3097];

N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [3098];

2-(4-methyl-1,4-diazepan-1-yl)-N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl) isonicotinamide [3099];

2-(4-isopropylpiperazin-1-yl)-N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl) isonicotinamide [3100];

N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)-2-(piperidin-4-ylamino) isonicotinamide [3101];

2-(methyl(1-methylpiperidin-4-yl)amino)-N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)isonicotinamide [3102];

N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)-2-((1-methylpiperidin-4-yl)thio) isonicotinamide [3103];

2-methyl-N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)-1,2,3,4-tetrahydroisoquinoline-6-carboxamide [3104];

N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)-2-(piperazin-1-yl)isonicotinamide [3105];

N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)-2-(2-(4-methylpiperazin-1-yl) pyridin-4-yl)acetamide [3106];

1,1-bis(methyl-d 3 )-4-(4-((3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)carbamoyl) pyridin-2-yl)piperazin-1-ium iodide [3107];

N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)-2-(4-(methyl-d 3 )piperazin-1-yl) isonicotinamide [3108];

N-(3-(1-methyl-1H-1,2,3-triazol-5-yl)-1,7-naphthyridin-6-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [3109];

N-(3-(4-methyl-4H-1,2,4-triazol-3-yl)-1,7-naphthyridin-6-yl)-2-morpholinoacetamide [3110];

N-(3-(4-methyl-4H-1,2,4-triazol-3-yl)-1,7-naphthyridin-6-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [3111];

4-fluoro-1-isobutyl-N-(3-(4-methyl-4H-1,2,4-triazol-3-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [3112];

N-(3-(4,5-dimethyl-4H-1,2,4-triazol-3-yl)-1,7-naphthyridin-6-yl)-2-morpholinoacetamide [3113];

N-(3-(4,5-dimethyl-4H-1,2,4-triazol-3-yl)-1,7-naphthyridin-6-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [3114];

N-(3-(1H-1,2,3-triazol-1-yl)-1,7-naphthyridin-6-yl)-4-fluoro-1-isobutylpiperidine-4-carboxamide [3115];

N-(3-(2H-1,2,3-triazol-2-yl)-1,7-naphthyridin-6-yl)-4-fluoro-1-isobutylpiperidine-4-carboxamide [3116];

N-(3-(1H-1,2,4-triazol-1-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [3117];

1-isobutyl-N-(3-(1-methyl-1H-tetrazol-5-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [3118];

2,2,3,3-tetramethyl-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)cyclopropane-1-carboxamide [3119];

4,4-difluoro-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)cyclohexane-1-carboxamide [3120];

N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-2-(piperidin-1-yl)acetamide [3121];

2-fluoro-2-methyl-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)propanamide [3122];

1-fluoro-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)cyclopropane-1-carboxamide [3123];

2-methyl-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-2-azaspiro[3.3]heptane-6-carboxamide [3124];

1-fluoro-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)cyclohexane-1-carboxamide [3125];

trans-4-methoxy-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)cyclohexane-1-carboxamide [3126];

trans-4-(hydroxymethyl)-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)cyclohexane-1-carboxamide [3127];

N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)azetidine-3-carboxamide [3128];

(R)—N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)tetrahydrofuran-2-carboxamide [3129];

1-(2-methoxyethyl)-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [3130];

N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [3131];

1-isobutyl-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [3132];

N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-1-(methylsulfonyl)piperidine-4-carboxamide [3133];

N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-2-(pyrrolidin-1-yl)propanamide [3134];

2-isopropoxy-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)acetamide [3135];

3-isopropoxy-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)propanamide [3136];

N-(3-(1,2-dimethyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)cyclopropanecarboxamide [3137];

N-(3-(1,2-dimethyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)cyclohexanecarboxamide [3138];

N-(3-(1,2-dimethyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-4,4-difluorocyclohexane-1-carboxamide [3139];

(S)—N-(3-(1,2-dimethyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)tetrahydrofuran-2-carboxamide [3140];

N-(3-(1,2-dimethyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-3,3-difluorocyclobutane-1-carboxamide [3141];

N-(3-(1,2-dimethyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-1-fluorocyclopropane-1-carboxamide [3142];

N-(3-(1,2-dimethyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)morpholine-4-carboxamide [3143];

N-(3-(1,2-dimethyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)morpholine-d 8 -4-carboxamide [3144];

1-methyl-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-1H-pyrazole-4-carboxamide [3145];

1-ethyl-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-1H-pyrazole-4-carboxamide [3146];

1-isopropyl-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-1H-pyrazole-4-carboxamide [3147];

1-cyclopropyl-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-1H-pyrazole-4-carboxamide [3148];

1-isobutyl-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-1H-pyrazole-4-carboxamide [3149];

1-methyl-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-1H-pyrazole-3-carboxamide [3150];

N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-2-(1-methyl-1H-pyrazol-4-yl) acetamide [3151];

1-methyl-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-1H-imidazole-4-carboxamide [3152];

1-isopropyl-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-1H-imidazole-4-carboxamide [3153];

N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-1-(tetrahydro-2H-pyran-4-yl)-1H-imidazole-4-carboxamide [3154];

1,2-dimethyl-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-1H-imidazole-5-carboxamide [3155];

1-methyl-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-1H-1,2,4-triazole-3-carboxamide [3156];

2-methyl-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)oxazole-4-carboxamide [3157];

2-isopropyl-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)oxazole-4-carboxamide [3158];

4-methyl-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)oxazole-2-carboxamide [3159];

4-methyl-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)thiazole-2-carboxamide [3160];

2-methyl-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)thiazole-4-carboxamide [3161];

5-methyl-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-1,3,4-oxadiazole-2-carboxamide [3162];

5-methyl-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-1,3,4-thiadiazole-2-carboxamide [3163];

1-isopropyl-N-(3-(1-isopropyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-1H-pyrazole-4-carboxamide [3164];

N-(3-(1,2-dimethyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-1-methyl-1H-pyrazole-4-carboxamide [3165];

N-(3-(1,2-dimethyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-1-isopropyl-1H-pyrazole-4-carboxamide [3166];

N-(3-(1,2-dimethyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-2-methylthiazole-5-carboxamide [3167];

4-fluoro-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)benzamide [3168];

4-fluoro-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)benzamide-2,3,5,6-d 4 [3169];

2-chloro-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)benzamide-3,4,5,6-d 4 [3170];

4-chloro-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)benzamide-2,3,5,6-d 4 [3171];

4-(methyl-d 3 )—N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)benzamide [3172];

4-methyl-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)benzamide-2,3,5,6-d 4 [3173];

4-(methyl-d 3 )—N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)benzamide-2,3,5,6-d 4 [3174];

4-(methoxy-d 3 )—N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)benzamide [3175];

4-(methoxy-d 3 )—N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)benzamide-2,3,56-d 4 [3176];

4-methoxy-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)benzamide-2,3,5,6-d 4 [3177];

(E)-N-(3-(1,2-dimethyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-3-(phenyl-2,3,4,5,6-d 5 ) acrylamide [3178];

(E)-N-(3-(1,2-dimethyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-3-(phenyl-2,3,4,5,6-d 5 ) acrylamide-2,3-d 2 [3179];

N-(3-(1,2-dimethyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-2-(4-fluorophenyl)acetamide-2,2-d 2 [3180];

(E)-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-3-(phenyl-2,3,4,5,6-d 5 )acrylamide [3181];

(E)-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-3-(phenyl-2,3,4,5,6-d 5 )acrylamide-2,3-d 2 [3182];

2-(4-fluorophenyl)-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)acetamide-2,2-d 2 [3183];

N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [3184];

2-(dimethylamino)-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)isonicotinamide [3185];

2-(3-aminoazetidin-1-yl)-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl) isonicotinamide [3186];

N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-2-(pyrrolidin-1-yl)isonicotinamide [3187];

N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-2-(piperidin-1-yl)isonicotinamide [3188];

N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-2-morpholinoisonicotinamide [3189];

2-(4-isopropylpiperazin-1-yl)-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl) isonicotinamide [3190];

2-(4-cyclopropylpiperazin-1-yl)-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl) isonicotinamide [3191];

N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-2-(2,7-diazaspiro[3.5]nonan-2-yl) isonicotinamide [3192];

N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-2-(7-methyl-2,7-diazaspiro[3.5]nonan-2-yl)isonicotinamide [3193];

N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)isoindoline-5-carboxamide [3194];

2-methyl-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)isoindoline-5-carboxamide [3195];

2-(azetidin-1-yl)-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)isonicotinamide [3196];

2-methoxy-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)isonicotinamide [3197];

2-methyl-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)isonicotinamide [3198];

2-cyano-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)isonicotinamide [3199];

2-(3,3-difluoroazetidin-1-yl)-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl) isonicotinamide [3200];

2-(4,4-difluoropiperidin-1-yl)-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl) isonicotinamide [3201];

2-isopropoxy-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)isonicotinamide [3202];

N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-2-(pyrrolidin-1-yl-2,2,5,5-d 4 ) isonicotinamide [3203];

N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-2-(pyrrolidin-1-yl-d 8 )isonicotinamide [3204];

N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-2-(piperidin-1-yl-d 10 )isonicotinamide [3205];

N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-2-(morpholino-d 8 )isonicotinamide [3206];

N-(3-(1,2-dimethyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-4-isopropoxybenzamide [3207];

N-(3-(1,2-dimethyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-4-(piperidin-4-yloxy)benzamide [3208];

4-(benzyloxy)-N-(3-(1,2-dimethyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)benzamide [3209];

N-(3-(1,2-dimethyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-2-fluorobenzamide-3,4,5,6-d 4 [3210];

N-(3-(1,2-dimethyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-4-fluorobenzamide-2,3,5,6-d 4 [3211];

2-chloro-N-(3-(1,2-dimethyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)benzamide-3,4,5,6-d 4 [3212];

4-chloro-N-(3-(1,2-dimethyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)benzamide-2,3,5,6-d 4 [3213];

N-(3-(1,2-dimethyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-4-(methyl-d 3 )benzamide [3214];

N-(3-(1,2-dimethyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-4-methylbenzamide-2,3,5,6-d 4 [3215];

N-(3-(1,2-dimethyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-4-(methyl-d3)benzamide-2,3,5,6-d 4 [3216];

N-(3-(1,2-dimethyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-4-(methoxy-d 3 )benzamide [3217];

N-(3-(1,2-dimethyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-4-(methoxy-d 3 )benzamide-2,3,5,6-d 4 [3218];

N-(3-(1,2-dimethyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-4-methoxybenzamide-2,3,5,6-d 4 [3219];

N-(3-(1,2-dimethyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [3220];

N-(3-(1,2-dimethyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-2-morpholinoisonicotinamide [3221];

N-(3-(1,2-dimethyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-2-(pyrrolidin-1-yl)isonicotinamide [3222];

N-(3-(1,2-dimethyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-2-(dimethylamino)isonicotinamide [3223];

N-(3-(1,2-dimethyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-2-(pyrrolidin-1-yl-2,2,5,5-d 4 ) isonicotinamide [3324];

N-(3-(1,2-dimethyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-2-(pyrrolidin-1-yl-d 8 ) isonicotinamide [3225];

N-(3-(1,2-dimethyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-2-(piperidin-1-yl-d 10 ) isonicotinamide [3226];

N-(3-(1,2-dimethyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-2-(morpholino-d 8 )isonicotinamide [3227];

N-(3-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-1,7-naphthyridin-6-yl) cyclopropanecarboxamide [3228];

N-(3-(7-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-1,7-naphthyridin-6-yl) cyclopropanecarboxamide [3229];

3,3-difluoro-N-(3-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-1,7-naphthyridin-6-yl) cyclobutane-1-carboxamide [3230];

(R)—N-(3-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-1,7-naphthyridin-6-yl)pyrrolidine-2-carboxamide [3231];

(R)—N-(3-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-1,7-naphthyridin-6-yl)piperidine-3-carboxamide [3232];

1-methyl-N-(3-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [3233];

N-(3-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-1,7-naphthyridin-6-yl)-1-((1-(trifluoromethyl)cyclopropyl)methyl)piperidine-4-carboxamide [3234];

1-benzoyl-N-(3-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [3235];

4-fluoro-1-isobutyl-N-(3-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-1,7-naphthyridin-6-yl) piperidine-4-carboxamide [3236];

(R)-2-(2-methylpyrrolidin-1-yl)-N-(3-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-1,7-naphthyridin-6-yl)acetamide [3237];

2-(cyclobutyl(methyl)amino)-N-(3-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-1,7-naphthyridin-6-yl)acetamide [3238];

4-fluoro-N-(3-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-1,7-naphthyridin-6-yl)benzamide [3239];

4-isopropoxy-N-(3-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-1,7-naphthyridin-6-yl) benzamide [3240];

4-(difluoromethoxy)-N-(3-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-1,7-naphthyridin-6-yl)benzamide [3241];

2-((2-(dimethylamino)ethyl)amino)-N-(3-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-1,7-naphthyridin-6-yl)isonicotinamide [3242];

2-((1-isopropylpiperidin-4-yl)oxy)-N-(3-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-1,7-naphthyridin-6-yl)isonicotinamide [3243];

N-(3-(oxazol-5-yl)-1,7-naphthyridin-6-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [3244];

N-(3-(oxazol-5-yl)-1,7-naphthyridin-6-yl)cyclopropanecarboxamide [3245];

(R)—N-(3-(oxazol-5-yl)-1,7-naphthyridin-6-yl)tetrahydrofuran-2-carboxamide [3246];

(R)—N-(3-(oxazol-5-yl)-1,7-naphthyridin-6-yl)piperidine-3-carboxamide [3247];

N-(3-(oxazol-5-yl)-1,7-naphthyridin-6-yl)tetrahydro-2H-pyran-4-carboxamide [3248];

N-(3-(oxazol-5-yl)-1,7-naphthyridin-6-yl)-1-(2-(pyrrolidin-1-yl)acetyl)piperidine-4-carboxamide [3249];

1′-methyl-N-(3-(oxazol-5-yl)-1,7-naphthyridin-6-yl)-[1,4′-bipiperidine]-4-carboxamide [3250];

cis-4-morpholino-N-(3-(oxazol-5-yl)-1,7-naphthyridin-6-yl)cyclohexane-1-carboxamide [3251];

2-(cyclobutyl(methyl)amino)-N-(3-(oxazol-5-yl)-1,7-naphthyridin-6-yl)acetamide [3252];

N-(3-(oxazol-5-yl)-1,7-naphthyridin-6-yl)-2-(pyrrolidin-1-yl)acetamide [3253];

(R)-2-(2-methylpyrrolidin-1-yl)-N-(3-(oxazol-5-yl)-1,7-naphthyridin-6-yl)acetamide [3254];

2-(4-methylpiperazin-1-yl)-N-(3-(oxazol-5-yl)-1,7-naphthyridin-6-yl)acetamide [3255];

trans-4-((4-methylpiperazin-1-yl)methyl)-N-(3-(oxazol-5-yl)-1,7-naphthyridin-6-yl)cyclohexane-1-carboxamide [3256];

1-(2,2-difluoropropyl)-N-(3-(oxazol-5-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [3257];

4-(difluoromethoxy)-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)benzamide [3258];

N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-3-(pyrrolidin-1-ylmethyl)benzamide [3259];

2-fluoro-N-(3-(1-methyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)benzamide-3,4,5,6-d 4 [3260];

trans-4-(hydroxymethyl)-N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl)cyclohexane-1-carboxamide [3261];

trans-4-(methylamino)-N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl)cyclohexane-1-carboxamide [3262];

trans-4-((1,3-difluoropropan-2-yl)amino)-N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl) cyclohexane-1-carboxamide [3263];

trans-N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl)-4-((propan-2-yl-1,1,1,3,3,3-d 6 ) amino)cyclohexane-1-carboxamide [3264];

trans-4-((2,2-difluoroethyl)amino)-N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl) cyclohexane-1-carboxamide [3265];

trans-N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl)-4-((3,3,3-trifluoropropyl)amino)cyclohexane-1-carboxamide [3266];

trans-4-((2-methoxyethyl)amino)-N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl) cyclohexane-1-carboxamide [3267];

trans-4-(dimethylamino)-N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl)cyclohexane-1-carboxamide [3268];

trans-4-(bis(methyl-d 3 )amino)-N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl)cyclohexane-1-carboxamide [3269];

cis-4-(dimethylamino)-N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl)cyclohexane-1-carboxamide [3270];

trans-4-((2,2-difluoroethyl)(methyl)amino)-N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl) cyclohexane-1-carboxamide [3271];

trans-4-(methyl(oxetan-3-yl)amino)-N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl) cyclohexane-1-carboxamide [3272];

trans-4-((2-fluoroethyl)amino)-N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl)cyclohexane-1-carboxamide [3273];

trans-4-(2-(fluoromethyl)aziridin-1-yl)-N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl) cyclohexane-1-carboxamide [3274];

trans-4-((3-fluoroazetidin-1-yl)methyl)-N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl) cyclohexane-1-carboxamide [3275];

trans-N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl)-3-morpholinocyclobutane-1-carboxamide [3276];

trans-N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl)-4-morpholinocyclohexane-1-carboxamide [3277];

N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl)-2-(piperidin-1-yl)acetamide [3278];

2-(4-methoxypiperidin-1-yl)-N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl)acetamide [3279];

N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl)acetamide [3280];

N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl)morpholine-4-carboxamide [3281];

N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl)-2-morpholinoacetamide [3282];

N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl)-3-morpholinopropanamide [3283];

1-methyl-N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [3284];

1-(2,2-difluoropropyl)-N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [3285];

N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl)-4-morpholinopiperidine-1-carboxamide [3286];

4-((1,3-difluoropropan-2-yl)amino)-N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl) piperidine-1-carboxamide [3287];

(1R,3s,5S)-3-((1,3-difluoropropan-2-yl)amino)-N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl)-8-azabicyclo[3.2.1]octane-8-carboxamide [3288];

(1R,3s,5S)-3-((1,3-difluoropropan-2-yl)amino)-N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl)-8-azabicyclo[3.2.1]octane-8-carboxamide [3289];

4-(dimethylamino)-N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl)piperidine-1-carboxamide [3290];

4-((2,2-difluoroethyl)(methyl)amino)-N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl) piperidine-1-carboxamide [3291];

(3S,4S)-4-amino-3-fluoro-N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl)piperidine-1-carboxamide [3292];

(3S,4S)-3-fluoro-4-(methylamino)-N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl)piperidine-1-carboxamide [3293];

(3R,4R)-4-amino-3-fluoro-N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl)piperidine-1-carboxamide [3294];

(3R,4R)-3-fluoro-4-(methylamino)-N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl)piperidine-1-carboxamide [3295];

4-((2-fluoroethyl)amino)-N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl)piperidine-1-carboxamide [3296];

4-((2,2-difluoroethyl)amino)-N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl)piperidine-1-carboxamide [3297];

(1R,3s,5S)-3-amino-N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl)-8-azabicyclo[3.2.1] octane-8-carboxamide [3298];

(1R,3r,5S)-3-amino-N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl)-8-azabicyclo[3.2.1] octane-8-carboxamide [3299];

(1R,3r,5S)-3-((2-fluoroethyl)amino)-N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl)-8-azabicyclo[3.2.1]octane-8-carboxamide [3300];

(1R,3r,5S)-3-((2,2-difluoroethyl)amino)-N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl)-8-azabicyclo[3.2.1]octane-8-carboxamide [3301];

(1R,3s,5S)—N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl)-3-((3,3,3-trifluoropropyl)amino)-8-azabicyclo[3.2.1]octane-8-carboxamide [3302];

(3S,4S)-3-fluoro-4-(isopropylamino)-N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl)piperidine-1-carboxamide [3303];

N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl)-5,6-dihydroimidazo[1,2-a]pyrazine-7(8H)-carboxamide [3304];

2-methyl-N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl)-5,6-dihydroimidazo[1,2-a]pyrazine-7(8H)-carboxamide [3305];

N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl)-2-(morpholino-d 8 )acetamide [3306];

trans-N-(3-(2-methyloxazol-4-yl)-1,7-naphthyridin-6-yl)-4-(4-methylpiperazin-1-yl)cyclohexane-1-carboxamide [3307];

N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl)-1-(1-methylpiperidin-4-yl)-1H-pyrazole-4-carboxamide [3308];

2-(1H-imidazol-1-yl)-N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl)acetamide [3309];

4-(difluoromethoxy)-N-(3-(oxazol-5-yl)-1,7-naphthyridin-6-yl)benzamide [3310];

3-((1-methylpiperidin-4-yl)oxy)-N-(3-(oxazol-5-yl)-1,7-naphthyridin-6-yl)benzamide [3311];

N-(3-(oxazol-5-yl)-1,7-naphthyridin-6-yl)isonicotinamide [3312];

2-(3-aminoazetidin-1-yl)-N-(3-(oxazol-5-yl)-1,7-naphthyridin-6-yl)isonicotinamide [3313];

2-(1-methylpiperidin-4-yl)-N-(3-(oxazol-5-yl)-1,7-naphthyridin-6-yl)isonicotinamide [3314];

1′-methyl-N-(3-(oxazol-5-yl)-1,7-naphthyridin-6-yl)-1′,2′,3′,6′-tetrahydro-[2,4′-bipyridine]-4-carboxamide [3315];

2-(4-methylpiperazin-1-yl)-N-(3-(oxazol-5-yl)-1,7-naphthyridin-6-yl)isonicotinamide [3316];

2-(7-methyl-2,7-diazaspiro[3.5]nonan-2-yl)-N-(3-(oxazol-5-yl)-1,7-naphthyridin-6-yl) isonicotinamide [3317];

N-(3-(oxazol-5-yl)-1,7-naphthyridin-6-yl)-2-(2,7-diazaspiro[3.5]nonan-7-yl)isonicotinamide [3318];

N-(3-(oxazol-5-yl)-1,7-naphthyridin-6-yl)-2-(piperidin-4-ylamino)isonicotinamide [3319];

2-methyl-N-(3-(oxazol-5-yl)-1,7-naphthyridin-6-yl)isoindoline-5-carboxamide [3320];

N-(3-(oxazol-5-yl)-1,7-naphthyridin-6-yl)-1,2,3,4-tetrahydroisoquinoline-7-carboxamide [3321];

N-(3-(2-methyloxazol-5-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [3322];

N-(3-(3-methylisoxazol-5-yl)-1,7-naphthyridin-6-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [3323];

4-fluoro-1-isobutyl-N-(3-(5-methyl-1,3,4-oxadiazol-2-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [3324];

1-isobutyl-N-(3-(5-methyl-1,3,4-oxadiazol-2-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [3325];

N-(3-(5-(dimethylamino)-1,3,4-oxadiazol-2-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [3326];

N-(3-(5-(dimethylamino)-1,3,4-oxadiazol-2-yl)-1,7-naphthyridin-6-yl)-1-methylpiperidine-4-carboxamide [3327];

N-(3-(5-methyl-1,3,4-oxadiazol-2-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [3328];

3,3-difluoro-N-(3-(thiazol-5-yl)-1,7-naphthyridin-6-yl)cyclobutane-1-carboxamide [3329];

2-methyl-N-(3-(thiazol-5-yl)-1,7-naphthyridin-6-yl)-2-azaspiro [3.3]heptane-6-carboxamide [3330];

1-fluoro-N-(3-(thiazol-5-yl)-1,7-naphthyridin-6-yl)cyclohexane-1-carboxamide [3331];

trans-4-(dimethylamino)-N-(3-(thiazol-5-yl)-1,7-naphthyridin-6-yl)cyclohexane-1-carboxamide [3332];

trans-4-((3-fluoroazetidin-1-yl)methyl)-N-(3-(thiazol-5-yl)-1,7-naphthyridin-6-yl)cyclohexane-1-carboxamide [3333];

N-(3-(thiazol-5-yl)-1,7-naphthyridin-6-yl)azetidine-3-carboxamide [3334];

1-methyl-N-(3-(thiazol-5-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [3335];

1-(2,2-difluoropropyl)-N-(3-(thiazol-5-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [3336];

1-(oxetan-3-yl)-N-(3-(thiazol-5-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [3337];

1-(2-(pyrrolidin-1-yl)acetyl)-N-(3-(thiazol-5-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [3338];

1′-methyl-N-(3-(thiazol-5-yl)-1,7-naphthyridin-6-yl)-[1,4′-bipiperidine]-4-carboxamide [3339];

2-(pyrrolidin-1-yl)-N-(3-(thiazol-5-yl)-1,7-naphthyridin-6-yl)propanamide [3340];

2-(piperidin-1-yl)-N-(3-(thiazol-5-yl)-1,7-naphthyridin-6-yl)acetamide [3341];

2-(4-methylpiperazin-1-yl)-N-(3-(thiazol-5-yl)-1,7-naphthyridin-6-yl)acetamide [3342];

2-morpholino-N-(3-(thiazol-5-yl)-1,7-naphthyridin-6-yl)acetamide [3343];

4-(piperidin-4-yloxy)-N-(3-(thiazol-5-yl)-1,7-naphthyridin-6-yl)benzamide [3344];

N-(3-(thiazol-5-yl)-1,7-naphthyridin-6-yl)isonicotinamide [3345];

6-(4-methylpiperazin-1-yl)-N-(3-(thiazol-5-yl)-1,7-naphthyridin-6-yl)nicotinamide [3346];

1′-methyl-N-(3-(thiazol-5-yl)-1,7-naphthyridin-6-yl)-1′,2′,3′,6′-tetrahydro-[2,4′-bipyridine]-4-carboxamide [3347];

2-(3-(dimethylamino)azetidin-1-yl)-N-(3-(thiazol-5-yl)-1,7-naphthyridin-6-yl)isonicotinamide [3348];

2-(4-(dimethylamino)piperidin-1-yl)-N-(3-(thiazol-5-yl)-1,7-naphthyridin-6-yl)isonicotinamide [3349];

2-(4-methylpiperazin-1-yl)-N-(3-(thiazol-5-yl)-1,7-naphthyridin-6-yl)isonicotinamide [3350];

2-((1-methylpiperidin-4-yl)thio)-N-(3-(thiazol-5-yl)-1,7-naphthyridin-6-yl)isonicotinamide [3351];

N-(3-(thiazol-5-yl)-1,7-naphthyridin-6-yl)-1,2,3,4-tetrahydroisoquinoline-7-carboxamide [3352];

trans-4-((1,3-difluoropropan-2-yl)amino)-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)cyclohexane-1-carboxamide [3353];

N-(3-(2-methylthiazol-5-yl)-1,7-naphthyridin-6-yl)morpholine-4-carboxamide [3354];

N-(3-(2-methylthiazol-5-yl)-1,7-naphthyridin-6-yl)-2-(pyrrolidin-1-yl)acetamide [3355];

2-((1R,4R)-2-oxa-5-azabicyclo [2.2.1]heptan-5-yl)-N-(3-(2-methylthiazol-5-yl)-1,7-naphthyridin-6-yl)acetamide [3356];

N-(3-(2-methylthiazol-5-yl)-1,7-naphthyridin-6-yl)-2-morpholinoacetamide [3357];

N-(3-(2-methylthiazol-5-yl)-1,7-naphthyridin-6-yl)-2-(morpholino-d 8 )acetamide [3358];

2-(4-methylpiperazin-1-yl)-N-(3-(2-methylthiazol-5-yl)-1,7-naphthyridin-6-yl)acetamide [3359];

1-methyl-N-(3-(2-methylthiazol-5-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [3360];

N-(3-(2-methylthiazol-5-yl)-1,7-naphthyridin-6-yl)isonicotinamide [3361];

N-(3-(2-methylthiazol-5-yl)-1,7-naphthyridin-6-yl)nicotinamide [3362];

2-(4-methylpiperazin-1-yl)-N-(3-(2-methylthiazol-5-yl)-1,7-naphthyridin-6-yl)isonicotinamide [3363];

trans-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-4-morpholinocyclohexane-1-carboxamide [3364];

trans-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-4-(4-methylpiperazin-1-yl) cyclohexane-1-carboxamide [3365];

4-isopropyl-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)piperazine-1-carboxamide [3366];

4-((2-methoxyethyl)(methyl)amino)-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl) piperidine-1-carboxamide [3367];

4-((1,3-difluoropropan-2-yl)amino)-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl) piperidine-1-carboxamide [3368];

N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-4-((3,3,3-trifluoropropyl)amino) piperidin 1-carboxamide [3369];

4-((2-fluoroethyl)amino)-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)piperidine-1-carboxamide [3370];

(3R,4S)-4-amino-3-fluoro-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl) piperidine-1-carboxamide [3371];

(3R,4R)-4-amino-3-fluoro-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl) piperidine-1-carboxamide [3372];

(3 S,4S)-3-fluoro-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-4-(methylamino) piperidine-1-carboxamide [3373];

(3R,4R)-3-fluoro-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-4-(methylamino) piperidine-1-carboxamide [3374];

4-amino-3,3-difluoro-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)piperidine-1-carboxamide [3375];

(3R,4R)-3-fluoro-4-(isopropylamino)-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)piperidine-1-carboxamide [3376];

(3R,4S)-3-fluoro-4-(isopropylamino)-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)piperidine-1-carboxamide [3377];

3,3-difluoro-4-(isopropylamino)-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl) piperidine-1-carboxamide [3378];

(3 S,4S)-3-fluoro-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-4-((propan-2-yl-1,1,1,3,3,3-d 6 )amino)piperidine-1-carboxamide [3379];

(1R,3s,5S)-3-((1,3-difluoropropan-2-yl)amino)-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-8-azabicyclo[3.2.1]octane-8-carboxamide [3380];

(1R,3 s,5 S)-3-((1,3-difluoropropan-2-yl)amino)-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-8-azabicyclo[3.2.1]octane-8-carboxamide [3381];

4-(dimethylamino)-N-(3-(2-methylthiazol-5-yl)-1,7-naphthyridin-6-yl)piperidine-1-carboxamide [3382];

4-((2,2-difluoroethyl)amino)-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl) piperidine-1-carboxamide [3383];

4-((2,2-difluoroethyl)(methyl-d3)amino)-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)piperidine-1-carboxamide [3384];

N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-4-morpholinopiperidine-1-carboxamide [3385];

N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-4-(4-methylpiperazin-1-yl) piperidine-1-carboxamide [3386];

(R)-3,4-dimethyl-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)piperazine-1-carboxamide [3387];

(S)-3,4-dimethyl-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)piperazine-1-carboxamide [3388];

(1R,3r,5 S)-3-((2-fluoroethyl)amino)-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-8-azabicyclo[3.2.1]octane-8-carboxamide [3389];

(1R,3r,5 S)-3-((2,2-difluoroethyl)amino)-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-8-azabicyclo[3.2.1]octane-8-carboxamide [3390];

(1R,3r,5 S)-3-amino-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-8-azabicyclo [3.2.1]octane-8-carboxamide [3391];

(1 S,4S)-5-methyl-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-2,5-diazabicyclo [2.2.1]heptane-2-carboxamide [3392];

(1R,4R)-5-methyl-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-2,5-diazabicyclo [2.2.1]heptane-2-carboxamide [3393];

8-methyl-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-3,8-diazabicyclo [3.2.1]octane-3-carboxamide [3394];

3-methyl-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-3,8-diazabicyclo [3.2.1]octane-8-carboxamide [3395];

N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-5,6-dihydroimidazo[1,2-a]pyrazine-7(8H)-carboxamide [3396];

2-(4-methylpiperazin-1-yl)-N-(3-(5-methylthiazol-2-yl)-1,7-naphthyridin-6-yl)isonicotinamide [3397];

2-(4-methylpiperazin-1-yl)-N-(3-(4-methylthiazol-2-yl)-1,7-naphthyridin-6-yl)isonicotinamide [3398];

N-(3-(2-(methylamino)thiazol-5-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [3399];

1-methyl-N-(3-(2-(methylamino)thiazol-5-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [3400];

N-(3-(2-(diethylamino)thiazol-5-yl)-1,7-naphthyridin-6-yl)-2-(4-fluoropiperidin-1-yl)acetamide [3401];

N-(3-(2-(diethylamino)thiazol-5-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl)acetamide [3402];

N-(3-(2-aminothiazol-5-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [3403];

N-(3-(2-(methylamino)thiazol-5-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [3404];

N-(3-(2-(dimethylamino)thiazol-5-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [3405];

2-(4-isopropylpiperazin-1-yl)-N-(3-(2-(methylamino)thiazol-5-yl)-1,7-naphthyridin-6-yl) isonicotinamide [3406];

2-(3-(dimethylamino)azetidin-1-yl)-N-(3-(2-(methylamino)thiazol-5-yl)-1,7-naphthyridin-6-yl) isonicotinamide [3407];

2-(3-(dimethylamino)azetidin-1-yl)-N-(3-(2-(dimethylamino)thiazol-5-yl)-1,7-naphthyridin-6-yl) isonicotinamide [3408];

2-(3-aminoazetidin-1-yl)-N-(3-(2-(dimethylamino)thiazol-5-yl)-1,7-naphthyridin-6-yl) isonicotinamide [3409];

N-(3-(5-chlorothiazol-2-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [3410];

2-(6-(2-(4-methylpiperazin-1-yl)isonicotinamido)-1,7-naphthyridin-3-yl)thiazole-5-carboxamide [3411];

N-(3-(isothiazol-4-yl)-1,7-naphthyridin-6-yl)-1-methylpiperidine-4-carboxamide [3412];

N-(3-(1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-4-(difluoromethoxy)benzamide [3413];

N-(3-(1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-4-(piperidin-4-yloxy)benzamide [3414];

N-(3-(1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-4-((1-methylpiperidin-4-yl)oxy)benzamide [3415];

N-(3-(1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-3-((1-methylpiperidin-4-yl)oxy)benzamide [3416];

N 5 -(3-(1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-N 2 -methylpyridine-2,5-dicarboxamide [3417];

N-(3-(1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-6-(4-methylpiperazin-1-yl)nicotinamide [3418];

N-(3-(1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-1′-methyl-1′,2′,3′,6′-tetrahydro-[2,4′-bipyridine]-4-carboxamide [3419];

N-(3-(1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-2-(3-(dimethylamino)azetidin-1-yl) isonicotinamide [3420];

N-(3-(1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [3421];

N-(3-(1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-2-(4-isopropylpiperazin-1-yl)isonicotinamide [3422];

N-(3-(1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-2-morpholinoisonicotinamide [3423];

1-fluoro-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)cyclohexane-1-carboxamide [3424];

trans-4-methoxy-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)cyclohexane-1-carboxamide [3425];

cis-4-methoxy-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)cyclohexane-1-carboxamide [3426];

trans-4-amino-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)cyclohexane-1-carboxamide [3427];

trans-4-(dimethylamino)-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl) cyclohexane-1-carboxamide [3428];

trans-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-4-morpholinocyclohexane-1-carboxamide [3429];

trans-4-(hydroxymethyl)-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl) cyclohexane-1-carboxamide [3430];

N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [3431];

4-fluoro-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [3432];

1-methyl-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [3433];

4-fluoro-1-methyl-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [3434];

1-(2-fluoroethyl)-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [3435];

1-(2,2-difluoroethyl)-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [3436];

N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [3437];

1-(2,2-difluoropropyl)-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [3438];

1-benzoyl-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [3439];

N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-2-(pyrrolidin-1-yl)acetamide [3440];

N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-2-(piperidin-1-yl)acetamide [3441];

2-(4-methoxypiperidin-1-yl)-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl) acetamide [3442];

N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl) acetamide [3443];

N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-2-morpholinoacetamide [3444];

(R)—N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-2-(3-methylmorpholino) acetamide [3445];

2-(7-azabicyclo[2.2.1]heptan-7-yl)-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl) acetamide [3446];

2-((1R,4R)-2-oxa-5-azabicyclo [2.2.1]heptan-5-yl)-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)acetamide [3447];

2-(3-oxa-8-azabicyclo[3.2.1]octan-8-yl)-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)acetamide [3448];

2-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)acetamide [3449];

N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-2-(1,4-oxazepan-4-yl)acetamide [3450];

N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-2-morpholinoacetamide-2,2-d 2 [3451];

N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-2-(morpholino-d)acetamide [3452];

1-methyl-3-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-1-(1-methylpiperidin-4-yl) urea [3453];

(3S,4S)-4-amino-3-fluoro-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl) piperidine-1-carboxamide [3454];

(3S,4S)-4-(dimethylamino)-3-fluoro-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl) piperidine-1-carboxamide [3455];

N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)morpholine-4-carboxamide [3456];

N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-4-(methylamino)piperidine-1-carboxamide [3457];

4-(dimethylamino)-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)piperidine-1-carboxamide [3458];

4-((2,2-difluoroethyl)(methyl)amino)-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)piperidine-1-carboxamide [3459];

(3 S,4S)-3-fluoro-4-(isopropylamino)-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)piperidine-1-carboxamide [3460];

2-methyl-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-5,6-dihydroimidazo[1,2-a]pyrazine-7(8H)-carboxamide [3461];

4-methyl-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)piperazine-1-carboxamide [3462];

N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-1-(1-methylpiperidin-4-yl)-1H-pyrazole-4-carboxamide [3463];

1-(1-isopropylpiperidin-4-yl)-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-1H-pyrazole-4-carboxamide [3464];

N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-1-(1-methylpiperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide [3465];

N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-2-(piperidin-4-yl)oxazole-4-carboxamide [3466];

N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-2-(1-methylpiperidin-4-yl)oxazole-4-carboxamide [3467];

2-(3-(dimethylamino)azetidin-1-yl)-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl) isonicotinamide [3468];

1′-methyl-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-1′,2′,3′,6′-tetrahydro-[2,4′-bipyridine]-4-carboxamide [3469];

N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [3470];

2-(methyl(1-methylpiperidin-4-yl)amino)-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)isonicotinamide [3471];

2-(azetidin-3-yloxy)-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)isonicotinamide [3472];

N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-3-((1-methylpiperidin-4-yl)oxy) benzamide [3473];

N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-2-((1-methylpiperidin-4-yl)thio) isonicotinamide [3474];

6-(4-methylpiperazin-1-yl)-N-(3-(5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)nicotinamide [3475];

2-(4-methylpiperazin-1-yl)-N-(3-(5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)isonicotinamide [3476];

N-(3-(5-amino-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [3477];

N-(3-(5-(dimethylamino)-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [3478];

N-(3-(3-amino-5-fluorophenyl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [3479];

N-(3-(3-fluoro-5-(isopropylamino)phenyl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [3480];

1-methyl-N-(3-(pyridin-2-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [3481];

2-(4-methylpiperazin-1-yl)-N-(3-(pyridin-2-yl)-1,7-naphthyridin-6-yl)isonicotinamide [3482];

2-(4-methylpiperazin-1-yl)-N-(3-(pyridin-4-yl)-1,7-naphthyridin-6-yl)isonicotinamide [3483];

N-(3-(pyridin-3-yl)-1,7-naphthyridin-6-yl)cyclopropanecarboxamide [3484];

N-(3-(pyridin-3-yl)-1,7-naphthyridin-6-yl)-2-(pyrrolidin-1-yl)acetamide [3485];

1-methyl-N-(3-(pyridin-3-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [3486];

N-(3-(pyridin-3-yl)-1,7-naphthyridin-6-yl)quinuclidine-4-carboxamide [3487];

2-morpholino-N-(3-(pyridin-3-yl)-1,7-naphthyridin-6-yl)acetamide [3488];

2-(morpholino-d 8 )—N-(3-(pyridin-3-yl)-1,7-naphthyridin-6-yl)acetamide [3489];

2-(4-methylpiperazin-1-yl)-N-(3-(pyridin-3-yl)-1,7-naphthyridin-6-yl)acetamide [3490];

2-(4-methyl-1,4-diazepan-1-yl)-N-(3-(pyridin-3-yl)-1,7-naphthyridin-6-yl)acetamide [3491];

2-(4-methylpiperazin-1-yl)-N-(3-(pyridin-3-yl)-1,7-naphthyridin-6-yl)isonicotinamide [3492];

2-(2-methyl-1H-imidazol-1-yl)-N-(3-(pyridin-3-yl)-1,7-naphthyridin-6-yl)acetamide [3493];

2-(1H-imidazol-1-yl)-N-(3-(pyridin-3-yl)-1,7-naphthyridin-6-yl)acetamide [3494];

2-(piperidin-4-yl)-N-(3-(pyridin-3-yl)-1,7-naphthyridin-6-yl)oxazole-4-carboxamide [3495];

2-(1-methylpiperidin-4-yl)-N-(3-(pyridin-3-yl)-1,7-naphthyridin-6-yl)oxazole-4-carboxamide [3496];

2-(1-isopropylpiperidin-4-yl)-N-(3-(pyridin-3-yl)-1,7-naphthyridin-6-yl)oxazole-4-carboxamide [3497];

trans-N-(3-(5-fluoropyridin-3-yl)-1,7-naphthyridin-6-yl)-3-morpholinocyclobutane-1-carboxamide [3498];

trans-N-(3-(5-fluoropyridin-3-yl)-1,7-naphthyridin-6-yl)-4-((4-methylpiperazin-1-yl)methyl) cyclohexane-1-carboxamide [3499];

N-(3-(5-fluoropyridin-3-yl)-1,7-naphthyridin-6-yl)-2-(pyrrolidin-1-yl)acetamide [3500];

N-(3-(5-fluoropyridin-3-yl)-1,7-naphthyridin-6-yl)-1-methylpiperidine-4-carboxamide [3501];

N-(3-(5-fluoropyridin-3-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl)acetamide [3502];

N-(3-(6-fluoropyridin-3-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl)acetamide [3503];

N-(3-(5-fluoropyridin-3-yl)-1,7-naphthyridin-6-yl)-2-morpholinoacetamide [3504];

N-(3-(5-fluoropyridin-3-yl)-1,7-naphthyridin-6-yl)-3-morpholinopropanamide [3505];

N-(3-(5-fluoropyridin-3-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [3506];

N-(3-(5-fluoropyridin-3-yl)-1,7-naphthyridin-6-yl)-2-(piperidin-4-yl)oxazole-4-carboxamide [3507];

N-(3-(5-fluoropyridin-3-yl)-1,7-naphthyridin-6-yl)-2-(1-methylpiperidin-4-yl)oxazole-4-carboxamide [3508];

N-(3-(5-fluoropyridin-3-yl)-1,7-naphthyridin-6-yl)-2-(1-isopropylpiperidin-4-yl)oxazole-4-carboxamide [3509];

N-(3-(5-chloropyridin-3-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [3510];

N-(3-(5-methylpyridin-3-yl)-1,7-naphthyridin-6-yl)-2-morpholinoacetamide [3511];

N-(3-(5-(difluoromethyl)pyridin-3-yl)-1,7-naphthyridin-6-yl)-3-(piperidin-4-yl)benzamide [3512];

N-(3-(5-(difluoromethyl)pyridin-3-yl)-1,7-naphthyridin-6-yl)-3-(1-methylpiperidin-4-yl) benzamide [3513];

N-(3-(5-(difluoromethyl)pyridin-3-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [3514];

2-(4-methylpiperazin-1-yl)-N-(3-(5-(trifluoromethyl)pyridin-3-yl)-1,7-naphthyridin-6-yl) acetamide [3515];

2-(4-methylpiperazin-1-yl)-N-(3-(6-(trifluoromethyl)pyridin-3-yl)-1,7-naphthyridin-6-yl) acetamide [3516];

N-(3-(5-(hydroxymethyl)pyridin-3-yl)-1,7-naphthyridin-6-yl)-1-methylpiperidine-4-carboxamide [3517];

N-(3-(5-cyanopyridin-3-yl)-1,7-naphthyridin-6-yl)-1-methylpiperidine-4-carboxamide [3518];

N-(3-(5-methoxypyridin-3-yl)-1,7-naphthyridin-6-yl)-1-methylpiperidine-4-carboxamide [3519];

N-(3-(5-methoxypyridin-3-yl)-1,7-naphthyridin-6-yl)-2-morpholinoacetamide [3520];

N-(3-(5-methoxypyridin-3-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [3521];

4-fluoro-N-(3-(5-(piperidin-4-yloxy)pyridin-3-yl)-1,7-naphthyridin-6-yl)benzamide [3522];

N-(3-(5-aminopyridin-3-yl)-1,7-naphthyridin-6-yl)-4-fluorobenzamide [3523];

N-(3-(5-aminopyridin-3-yl)-1,7-naphthyridin-6-yl)-4-(piperidin-4-yloxy)benzamide [3524];

N-(3-(5-aminopyridin-3-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [3525];

N-(3-(5-aminopyridin-3-yl)-1,7-naphthyridin-6-yl)-2-(piperidin-4-yl)oxazole-4-carboxamide [3526];

N-(3-(6-aminopyridin-3-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [3527];

N-(3-(6-(methylamino)pyridin-3-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [3528];

N-(3-(5-(isopropylamino)pyridin-3-yl)-1,7-naphthyridin-6-yl)-3-(piperidin-4-yl)benzamide [3529];

N-(3-(5-(isopropylamino)pyridin-3-yl)-1,7-naphthyridin-6-yl)-3-(1-methylpiperidin-4-yl) benzamide [3530];

N-(3-(5-(isopropylamino)pyridin-3-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [3531];

N-(3-(5-(piperidin-4-ylamino)pyridin-3-yl)-1,7-naphthyridin-6-yl)cyclohexanecarboxamide [3532];

4-fluoro-N-(3-(5-(piperidin-4-ylamino)pyridin-3-yl)-1,7-naphthyridin-6-yl)benzamide [3533];

4-fluoro-N-(3-(5-((1-methylpiperidin-4-yl)amino)pyridin-3-yl)-1,7-naphthyridin-6-yl)benzamide [3534];

N-(3-(5-acetamidopyridin-3-yl)-1,7-naphthyridin-6-yl)-1-methylpiperidine-4-carboxamide [3535];

N-(3-(5-(dimethylamino)pyridin-3-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [3536];

N-(3-(6-(dimethylamino)pyridin-3-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [3537];

1-methyl-N-(3-(5-(pyrrolidin-1-yl)pyridin-3-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [3538];

N-(3-(5-(pyrrolidin-1-ylmethyl)pyridin-3-yl)-1,7-naphthyridin-6-yl)cyclopropanecarboxamide [3539];

4-fluoro-N-(3-(5-(pyrrolidin-1-ylmethyl)pyridin-3-yl)-1,7-naphthyridin-6-yl)benzamide [3540];

N-(3-(5-((4-hydroxypiperidin-1-yl)methyl)pyridin-3-yl)-1,7-naphthyridin-6-yl) cyclopropanecarboxamide [3541];

4-fluoro-N-(3-(5-((4-hydroxypiperidin-1-yl)methyl)pyridin-3-yl)-1,7-naphthyridin-6-yl) benzamide [3542];

N-(3-(5-(piperazin-1-ylmethyl)pyridin-3-yl)-1,7-naphthyridin-6-yl)cyclopropanecarboxamide [3543];

N-(3-(5-((4-methylpiperazin-1-yl)methyl)pyridin-3-yl)-1,7-naphthyridin-6-yl) cyclopropanecarboxamide [3544];

N-(3-(5-(morpholinomethyl)pyridin-3-yl)-1,7-naphthyridin-6-yl)cyclopropanecarboxamide [3545];

N-methyl-5-(6-(1-methylpiperidine-4-carboxamido)-1,7-naphthyridin-3-yl)nicotinamide [3546];

N-methyl-5-(6-(2-(4-methylpiperazin-1-yl)isonicotinamido)-1,7-naphthyridin-3-yl)nicotinamide [3547];

N-(3-(pyridin-3-yl-d 4 )-1,7-naphthyridin-6-yl)-2-(pyrrolidin-1-yl)acetamide [3548];

2-(4-methylpiperazin-1-yl)-N-(3-(pyridin-3-yl-d 4 )-1,7-naphthyridin-6-yl)acetamide [3549];

2-morpholino-N-(3-(pyridin-3-yl-d 4 )-1,7-naphthyridin-6-yl)acetamide [3550];

1-methyl-N-(3-(2-methylpyrimidin-5-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [3551];

2-(4-methylpiperazin-1-yl)-N-(3-(2-methylpyrimidin-5-yl)-1,7-naphthyridin-6-yl)isonicotinamide [3552];

N-(3-(2-aminopyrimidin-5-yl)-1,7-naphthyridin-6-yl)-1-methylpiperidine-4-carboxamide [3553];

2-morpholino-N-(3-(pyridazin-3-yl)-1,7-naphthyridin-6-yl)acetamide [3554];

2-morpholino-N-(3-(pyridazin-4-yl)-1,7-naphthyridin-6-yl)acetamide [3555];

N-(3-(pyridazin-4-yl)-1,7-naphthyridin-6-yl)-2-(pyrrolidin-1-yl)acetamide [3556];

trans-3-morpholino-N-(3-(pyrazin-2-yl)-1,7-naphthyridin-6-yl)cyclobutane-1-carboxamide [3557];

trans-4-(dimethylamino)-N-(3-(pyrazin-2-yl)-1,7-naphthyridin-6-yl)cyclohexane-1-carboxamide [3558];

trans-4-morpholino-N-(3-(pyrazin-2-yl)-1,7-naphthyridin-6-yl)cyclohexane-1-carboxamide [3559];

trans-4-((3-fluoroazetidin-1-yl)methyl)-N-(3-(pyrazin-2-yl)-1,7-naphthyridin-6-yl)cyclohexane-1-carboxamide [3560];

trans-4-((4-methylpiperazin-1-yl)methyl)-N-(3-(pyrazin-2-yl)-1,7-naphthyridin-6-yl) cyclohexane-1-carboxamide [3561];

N-(3-(pyrazin-2-yl)-1,7-naphthyridin-6-yl)-2-(pyrrolidin-1-yl)acetamide [3562];

1-methyl-N-(3-(pyrazin-2-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [3563];

4-fluoro-1-methyl-N-(3-(pyrazin-2-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [3564];

1-(2-fluoroethyl)-N-(3-(pyrazin-2-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [3565];

1-(oxetan-3-yl)-N-(3-(pyrazin-2-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [3566];

2-morpholino-N-(3-(pyrazin-2-yl)-1,7-naphthyridin-6-yl)acetamide [3567];

1-methyl-N-(3-(pyrazin-2-yl)-1,7-naphthyridin-6-yl)azepane-4-carboxamide [3568];

1-isobutyl-N-(3-(pyrazin-2-yl)-1,7-naphthyridin-6-yl)azepane-4-carboxamide [3569];

1-(2-hydroxy-2-methylpropyl)-N-(3-(pyrazin-2-yl)-1,7-naphthyridin-6-yl)azepane-4-carboxamide [3570];

4-(morpholinomethyl)-N-(3-(pyrazin-2-yl)-1,7-naphthyridin-6-yl)benzamide [3571];

2-(4-methylpiperazin-1-yl)-N-(3-(pyrazin-2-yl)-1,7-naphthyridin-6-yl)isonicotinamide[3572];

N-(3-(6-(methylamino)pyrazin-2-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [3573];

N-(3-(6-(isopropylamino)pyrazin-2-yl)-1,7-naphthyridin-6-yl)azetidine-3-carboxamide [3574];

N-(3-(6-(isopropylamino)pyrazin-2-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [3575];

N-(3-(6-(isopropylamino)pyrazin-2-yl)-1,7-naphthyridin-6-yl)-1-methylpiperidine-4-carboxamide [3576];

1-(2-fluoroethyl)-N-(3-(6-(isopropylamino)pyrazin-2-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [3577];

1-isopropyl-N-(3-(6-(isopropylamino)pyrazin-2-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [3578];

1-isopentyl-N-(3-(6-(isopropylamino)pyrazin-2-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [3579];

N-(3-(6-(isopropylamino)pyrazin-2-yl)-1,7-naphthyridin-6-yl)-3-(piperidin-4-yl)benzamide [3580];

N-(3-(6-(isopropylamino)pyrazin-2-yl)-1,7-naphthyridin-6-yl)-3-(1-methylpiperidin-4-yl) benzamide [3581];

N-(3-(6-(isopropylamino)pyrazin-2-yl)-1,7-naphthyridin-6-yl)-1-(piperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide [3582];

1-(1-(2-fluoroethyl)piperidin-4-yl)-N-(3-(6-(isopropylamino)pyrazin-2-yl)-1,7-naphthyridin-6-yl)-1H-1,2,3-triazole-4-carboxamide [3583];

N-(3-(6-(isopropylamino)pyrazin-2-yl)-1,7-naphthyridin-6-yl)-1-(1-isopropylpiperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide [3584];

N-(3-(6-(isopropylamino)pyrazin-2-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [3585];

N-(3-(6-(tert-butylamino)pyrazin-2-yl)-1,7-naphthyridin-6-yl)-2-(3-(dimethylamino)azetidin-1-yl)isonicotinamide [3586];

N-(3-(6-(tert-butylamino)pyrazin-2-yl)-1,7-naphthyridin-6-yl)-1′-methyl-1′,2′,3′,6′-tetrahydro-[2,4′-bipyridine]-4-carboxamide [3587];

N-(3-(6-(tert-butylamino)pyrazin-2-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1l-yl) isonicotinamide [3588];

N-(3-(6-(tert-butylamino)pyrazin-2-yl)-1,7-naphthyridin-6-yl)-2-(4-isopropylpiperazin-1l-yl) isonicotinamide [3589];

N-(3-(6-(tert-butylamino)pyrazin-2-yl)-1,7-naphthyridin-6-yl)-2-morpholinoisonicotinamide [3590];

N-(3-(6-(((3-fluoroazetidin-3-yl)methyl)amino)pyrazin-2-yl)-1,7-naphthyridin-6-yl) cyclopropanecarboxamide [3591];

4-fluoro-N-(3-(6-(((3-fluoroazetidin-3-yl)methyl)amino)pyrazin-2-yl)-1,7-naphthyridin-6-yl) benzamide [3592];

N-(3-(6-(piperidin-4-ylamino)pyrazin-2-yl)-1,7-naphthyridin-6-yl)cyclobutanecarboxamide [3593];

3,3-difluoro-N-(3-(6-(piperidin-4-ylamino)pyrazin-2-yl)-1,7-naphthyridin-6-yl)cyclobutane-1-carboxamide [3594];

N-(3-(6-(piperidin-4-ylamino)pyrazin-2-yl)-1,7-naphthyridin-6-yl)cyclopentanecarboxamide [3595];

4,4-difluoro-N-(3-(6-(piperidin-4-ylamino)pyrazin-2-yl)-1,7-naphthyridin-6-yl)cyclohexane-1-carboxamide [3596];

N-(3-(6-(piperidin-4-ylamino)pyrazin-2-yl)-1,7-naphthyridin-6-yl)tetrahydro-2H-pyran-4-carboxamide [3597];

4-fluoro-N-(3-(6-(piperidin-4-ylamino)pyrazin-2-yl)-1,7-naphthyridin-6-yl)benzamide [3598];

N-(3-(6-(((3S,4S)-3-fluoropiperidin-4-yl)amino)pyrazin-2-yl)-1,7-naphthyridin-6-yl) cyclopropanecarboxamide [3599];

4-fluoro-N-(3-(6-(((3S,4S)-3-fluoropiperidin-4-yl)amino)pyrazin-2-yl)-1,7-naphthyridin-6-yl) benzamide [3600];

N-(3-(6-((1-methylpiperidin-4-yl)amino)pyrazin-2-yl)-1,7-naphthyridin-6-yl) cyclobutanecarboxamide [3601];

N-(3-(6-((1-methylpiperidin-4-yl)amino)pyrazin-2-yl)-1,7-naphthyridin-6-yl) cyclopentanecarboxamide [3602];

4-fluoro-N-(3-(6-((1-methylpiperidin-4-yl)amino)pyrazin-2-yl)-1,7-naphthyridin-6-yl)benzamide [3603];

N-(3-(6-((1-isopropylpiperidin-4-yl)amino)pyrazin-2-yl)-1,7-naphthyridin-6-yl) cyclopropanecarboxamide [3604];

3,3-difluoro-N-(3-(6-((1-isopropylpiperidin-4-yl)amino)pyrazin-2-yl)-1,7-naphthyridin-6-yl) cyclobutane-1-carboxamide [3605];

N-(3-(6-((1-isopropylpiperidin-4-yl)amino)pyrazin-2-yl)-1,7-naphthyridin-6-yl) cyclopentanecarboxamide [3606];

4-fluoro-N-(3-(6-((1-isopropylpiperidin-4-yl)amino)pyrazin-2-yl)-1,7-naphthyridin-6-yl) benzamide [3607];

N-(3-(6-(dimethylamino)pyrazin-2-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [3608];

N-(3-(6-(diethylamino)pyrazin-2-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [3609];

N-(3-(6-(3-aminoazetidin-1-yl)pyrazin-2-yl)-1,7-naphthyridin-6-yl)-4-fluorobenzamide [3610];

2-(4-methylpiperazin-1-yl)-N-(3-(6-(pyrrolidin-1-yl)pyrazin-2-yl)-1,7-naphthyridin-6-yl) isonicotinamide [3611];

N-(3-(6-(azetidin-3-ylmethoxy)pyrazin-2-yl)-1,7-naphthyridin-6-yl)-4-fluorobenzamide [3612];

N-(3-(6-(azetidin-3-yloxy)pyrazin-2-yl)-1,7-naphthyridin-6-yl)-4-fluorobenzamide [3613];

N-(3-(1H-pyrrolo[2,3-b]pyridin-5-yl)-1,7-naphthyridin-6-yl)-1-(1-methylpiperidin-4-yl)-1H-pyrazole-4-carboxamide [3614];

N-(3-(1H-pyrrolo[3,2-b]pyridin-6-yl)-1,7-naphthyridin-6-yl)-1-(1-methylpiperidin-4-yl)-1H-pyrazole-4-carboxamide [3615];

N-(3-(1H-pyrrolo[2,3-c]pyridin-4-yl)-1,7-naphthyridin-6-yl)-1-(1-methylpiperidin-4-yl)-1H-pyrazole-4-carboxamide [3616];

N-(3-(1H-pyrrolo[2,3-b]pyridin-5-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [3617];

N-(3-(1H-pyrrolo[3,2-b]pyridin-6-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [3618];

N-(3-(1H-pyrrolo[2,3-c]pyridin-4-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [3619];

2-(4-methylpiperazin-1-yl)-N-(3-(oxazolo[5,4-b]pyridin-6-yl)-1,7-naphthyridin-6-yl) isonicotinamide [3620];

N-(3-(2-methyl-1H-pyrrolo[2,3-b]pyridin-5-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [3621];

N-(3-(3-methyl-1H-pyrrolo[2,3-b]pyridin-5-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [3622];

N-(3-(2-methyl-1H-pyrrolo[3,2-b]pyridin-6-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [3623];

N-(3-(5H-pyrrolo[2,3-b]pyrazin-2-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [3624];

N-(3-(5H-pyrrolo[2,3-b]pyrazin-3-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [3625];

1-isopropyl-N-(3-(6-(piperidin-4-ylamino)pyrazin-2-yl)-1,7-naphthyridin-6-yl)-1H-pyrazole-4-carboxamide [3626];

1-isopropyl-N-(3-(6-((1-methylpiperidin-4-yl)amino)pyrazin-2-yl)-1,7-naphthyridin-6-yl)-1H-pyrazole-4-carboxamide [3627];

trans-4-((2-fluoroethyl)amino)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl) cyclohexane-1-carboxamide [4597];

trans-4-((2-methoxyethyl)amino)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl) cyclohexane-1-carboxamide [4598];

tert-butyl (trans-4-((6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)carbamoyl)cyclohexyl) carbamate [4599];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-((1-methylpiperidin-4-yl)amino) isonicotinamide [4600];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl)thiazole-5-carboxamide [4601];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl)thiazole-5-carboxamide [4602];

N-(6-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(2,7-diazaspiro[3.5]nonan-2-yl)isonicotinamide [4603];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)-4-(piperidin-4-yloxy)benzamide [4604];

N-(6-(1-methyl-1H-tetrazol-5-yl)-2,7-naphthyridin-3-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [4605];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-2-(pyrrolidin-1-yl)propanamide [4606];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-2-(piperidin-1-yl)propanamide [4607];

4-isopropoxy-N-(6-(7-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-2,7-naphthyridin-3-yl)benzamide [4608];

trans-3-morpholino-N-(6-(oxazol-5-yl)-2,7-naphthyridin-3-yl)cyclobutane-1-carboxamide [4609];

trans-4-(hydroxymethyl)-N-(6-(oxazol-5-yl)-2,7-naphthyridin-3-yl)cyclohexane-1-carboxamide [4610];

N-(6-(oxazol-5-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [4611];

4-morpholino-N-(6-(oxazol-5-yl)-2,7-naphthyridin-3-yl)piperidine-1-carboxamide [4612];

N-(6-(oxazol-5-yl)-2,7-naphthyridin-3-yl)-4-(piperidin-4-yloxy)benzamide [4613];

N-(6-(oxazol-5-yl)-2,7-naphthyridin-3-yl)-3-(piperidin-4-yloxy)benzamide [4614];

2-methyl-N-(6-(oxazol-5-yl)-2,7-naphthyridin-3-yl)-5,6-dihydroimidazo[1,2-a]pyrazine-7(8H)-carboxamide [4615];

2-(1H-imidazol-1-yl)-N-(6-(oxazol-5-yl)-2,7-naphthyridin-3-yl)acetamide [4616];

trans-4-(hydroxymethyl)-N-(6-(thiazol-5-yl)-2,7-naphthyridin-3-yl)cyclohexane-1-carboxamide [4617];

trans-4-(dimethylamino)-N-(6-(thiazol-5-yl)-2,7-naphthyridin-3-yl)cyclohexane-1-carboxamide [4618];

N-(6-(thiazol-5-yl)-2,7-naphthyridin-3-yl)-1-((1-(trifluoromethyl)cyclopropyl)methyl)piperidine-4-carboxamide [4619];

trans-4-(hydroxymethyl)-N-(6-(2-methylthiazol-5-yl)-2,7-naphthyridin-3-yl)cyclohexane-1-carboxamide [4620];

trans-4-(dimethylamino)-N-(6-(2-methylthiazol-5-yl)-2,7-naphthyridin-3-yl)cyclohexane-1-carboxamide [4621];

N-(6-(2-methylthiazol-5-yl)-2,7-naphthyridin-3-yl)-1-(oxetan-3-yl)piperidine-4-carboxamide [4622];

N-(6-(2-methylthiazol-5-yl)-2,7-naphthyridin-3-yl)-1-(2-(pyrrolidin-1-yl)acetyl)piperidine-4-carboxamide [4623];

2-((1S,4S)-2-oxa-5-azabicyclo [2.2.1]heptan-5-yl)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)acetamide [4624];

N-(6-(5-(cyano(4-hydroxypiperidin-1-yl)methyl)pyridin-3-yl)-2,7-naphthyridin-3-yl) cyclopropanecarboxamide [4625];

4-fluoro-N-(6-(6-((1-methylazetidin-3-yl)methoxy)pyrazin-2-yl)-2,7-naphthyridin-3-yl) benzamide [4626];

1-isopropyl-N-(6-(6-((1-methylpiperidin-4-yl)amino)pyrazin-2-yl)-2,7-naphthyridin-3-yl)-1H-pyrazole-4-carboxamide [4627]; or a pharmaceutically acceptable salt thereof.

16. The compound of claim 1 , wherein the compound of Formula I is selected from the group consisting of:

N-(6-(1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-1-isobutylpiperidine-4-carboxamide [3628];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)cyclopropanecarboxamide [3629];

4,4-difluoro-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)cyclohexane-1-carboxamide [3630];

trans-4-methoxy-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)cyclohexane-1-carboxamide [3631];

trans-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-4-morpholinocyclohexane-1-carboxamide [3632];

trans-4-((3-fluoroazetidin-1-yl)methyl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl) cyclohexane-1-carboxamide [3633];

trans-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-4-((4-methylpiperazin-1-yl) methyl)cyclohexane-1-carboxamide [3634];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide [3635];

(S)-2-(3-fluoropyrrolidin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl) acetamide [3636];

(S)—N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)tetrahydrofuran-2-carboxamide [3637];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [3638];

1-methyl-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [3639];

1-isopropyl-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [3640];

1-(tert-butyl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [3641];

1-cyclopropyl-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [3642];

1-isobutyl-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [3643];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-1-neopentylpiperidine-4-carboxamide [3644];

1-(2-fluoroethyl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [3645];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [3646];

1-butyl-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [3647];

1-benzoyl-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [3648];

1-(2,2-difluoropropyl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [3649];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)azetidine-3-carboxamide [3650];

1-(2,2-difluoroethyl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [3651];

1-(2-fluoro-2-methylpropyl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [3652];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-1-(oxetan-3-yl)piperidine-4-carboxamide [3653];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-1-((3-methyloxetan-3-yl)methyl) piperidine-4-carboxamide [3654];

1-(2-methoxyethyl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [3655];

1-(2-isopropoxyethyl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [3656];

1,1-diisobutyl-4-((6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)carbamoyl)piperidin-1-ium [3657];

4-fluoro-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [3658];

4-fluoro-1-methyl-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [3659];

4-fluoro-1-isobutyl-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [3660];

(S)—N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)piperidine-3-carboxamide [3661];

(R)—N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)piperidine-3-carboxamide [3662];

(S)-1-isobutyl-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)piperidine-3-carboxamide [3663];

(R)-1-isobutyl-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)piperidine-3-carboxamide [3664];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)tetrahydro-2H-pyran-4-carboxamide [3665];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(piperidin-1-yl)acetamide [3666];

2-(4-fluoropiperidin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)acetamide [3667];

trans-4-amino-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)cyclohexane-1-carboxamide [3668];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl)acetamide [3669];

(S)—N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)piperidine-2-carboxamide [3670];

2-(4-isobutylpiperazin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)acetamide [3671];

2-(3,3-dimethylazetidin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)acetamide [3672];

(R)-2-(3-fluoropyrrolidin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl) acetamide [3673];

(S)—N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(2-methylpyrrolidin-1-yl) acetamide [3674];

2-(3-azabicyclo[3.1.0]hexan-3-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl) acetamide [3675];

2-(7-azabicyclo[2.2.1]heptan-7-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl) acetamide [3676];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperidin-1-yl)acetamide [3677];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(4-(trifluoromethyl)piperidin-1-yl) acetamide [3678];

2-(4-(difluoromethyl)piperidin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl) acetamide [3679];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(6-azaspiro[2.5]octan-6-yl)acetamide [3680];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(pyrrolidin-1-yl)propanamide [3681];

(R)—N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(2-methylpyrrolidin-1-yl) acetamide [3682];

2-(cyclobutyl(methyl)amino)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)acetamide [3683];

2-(diethylamino)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)acetamide [3684];

7-(2-fluoroethyl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-7-azaspiro[3.5]nonane-2-carboxamide [3685];

4-methyl-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)piperazine-1-carboxamide [3686];

(S)—N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(pyrrolidin-1-yl)propanamide [3687];

(R)—N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(pyrrolidin-1-yl)propanamide [3688];

(R)—N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)pyrrolidine-2-carboxamide [3689];

2-methyl-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-azaspiro [3.3]heptane-6-carboxamide [3690];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(2,2,2-trifluoroacetyl)-2-azaspiro[3.3]heptane-6-carboxamide [3691];

2-(2-fluoroethyl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-azaspiro[3.3]heptane-6-carboxamide [3692];

trans-4-(dimethylamino)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)cyclohexane-1-carboxamide [3693];

1-acetyl-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [3694];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-1-((1-(trifluoromethyl)cyclopropyl) methyl)piperidine-4-carboxamide [3695];

(S)-1-(2-fluoropropyl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [3696];

(R)-1-(2-fluoropropyl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [3697];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(piperidin-1-yl)propanamide [3698];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-1-(methylsulfonyl)piperidine-4-carboxamide [3699];

1′-methyl-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-[1,4′-bipiperidine]-4-carboxamide [3700];

trans-4-(hydroxymethyl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)cyclohexane-1-carboxamide [3701];

methyl 2-(4-((6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)carbamoyl)piperidin-1-yl) acetate [3702];

1-benzyl-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [3703];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-1-(2-(pyrrolidin-1-yl)acetyl)piperidine-4-carboxamide [3704];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-morpholinoacetamide [3705];

(S)—N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(3-methylmorpholino)acetamide [3706];

(R)—N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(3-methylmorpholino)acetamide [3707];

(S)—N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(2-methylmorpholino)acetamide [3708];

2-((2R,6S)-2,6-dimethylmorpholino)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl) acetamide [3709];

2-((1S,4S)-2-oxa-5-azabicyclo [2.2.1]heptan-5-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)acetamide [3710];

2-((1R,4R)-2-oxa-5-azabicyclo[2.2.1]heptan-5-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)acetamide [3711];

2-(3-oxa-8-azabicyclo[3.2.1]octan-8-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl) acetamide [3712];

(S)—N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-morpholinopropanamide [3713];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(morpholin-2-yl)acetamide [3714];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(4-methylmorpholin-2-yl)acetamide [3715];

2-(4-ethylpiperazin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)acetamide [3716];

2-(4-isopropylpiperazin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)acetamide [3717];

2-(4-cyclopropylpiperazin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl) acetamide [3718];

2-(4-(2-fluoroethyl)piperazin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl) acetamide [3719];

(S)-2-(2,4-dimethylpiperazin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl) acetamide [3720];

1-(2-hydroxyethyl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [3721];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-1-(pyridin-2-ylmethyl)piperidine-4-carboxamide [3722];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-1-(oxazol-2-ylmethyl)piperidine-4-carboxamide [3723];

(R)—N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-1-oxotetrahydro-1H-pyrrolo[1,2-c]imidazole-2(3H)-carboxamide [3724];

(R)-1-methyl-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)pyrrolidine-2-carboxamide [3725];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-1-(tetrahydro-2H-pyran-4-yl)piperidine-4-carboxamide [3726];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-1-(pyrimidin-2-ylmethyl)piperidine-4-carboxamide [3727];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-1-(pyrazin-2-ylmethyl)piperidine-4-carboxamide [3728];

1-((5-methyl-1,2,4-oxadiazol-3-yl)methyl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [3729];

1-(2-hydroxy-2-methylpropyl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl) piperidine-4-carboxamide [3730];

tert-butyl 2-(4-((6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)carbamoyl)piperidin-1-yl) acetate [3731];

2-(4-((6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)carbamoyl)piperidin-1-yl)acetic acid [3732];

2-(4-methyl-1,4-diazepan-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl) acetamide [3733];

tert-butyl (6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)carbamate [3734];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)but-2-ynamide [3735];

trans-4-((6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)carbamoyl)cyclohexane-1-carboxylic acid [3736];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-3-morpholinopropanamide [3737];

trans-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-3-morpholinocyclobutane-1-carboxamide [3738];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)quinuclidine-4-carboxamide [3739];

1-isobutyl-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)azepane-4-carboxamide [3740];

2-(4-methoxypiperidin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)acetamide [3741];

2-(4-hydroxypiperidin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)acetamide [3742];

3-(hydroxymethyl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)bicyclo[1.1.1]pentane-1-carboxamide [3743];

1-methyl-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)azepane-4-carboxamide [3744];

trans-4-(dimethylamino)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)cyclohexane-1-carboxamide [3745];

trans-4-(bis(methyl-d 3 )amino)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl) cyclohexane-1-carboxamide [3746];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-3-((4-methylpiperazin-1-yl)methyl) bicyclo[1.1.1]pentane-1-carboxamide [3747];

methyl trans-4-((6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)carbamoyl)cyclohexane-1-carboxylate [3748];

2-(1-isobutylpyrrolidin-3-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)acetamide [3749];

trans-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-4-(4-methylpiperazine-1-carbonyl)cyclohexane-1-carboxamide [3750];

1-isobutyl-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [3751];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-1-(phenylsulfonyl)piperidine-4-carboxamide [3752];

8-methyl-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-3,8-diazabicyclo[3.2.1]octane-3-carboxamide [3753];

3-methyl-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-3,8-diazabicyclo[3.2.1]octane-8-carboxamide [3754];

(1R,3s,5S)-3-amino-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-8-azabicyclo[3.2.1] octane-8-carboxamide [3755];

(1R,3s,5S)—N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-3-((3,3,3-trifluoropropyl) amino)-8-azabicyclo[3.2.1]octane-8-carboxamide [3756];

(1R,3s,5S)-3-((1,3-difluoropropan-2-yl)amino)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-8-azabicyclo[3.2.1]octane-8-carboxamide [3757];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)morpholine-4-carboxamide [3758];

4-(dimethylamino)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)piperidine-1-carboxamide [3759];

(S)-2,4-dimethyl-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)piperazine-1-carboxamide [3760];

1-methyl-3-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-1-(1-methylpiperidin-4-yl)urea [3761];

1-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-3-(1-methylpiperidin-4-yl)urea [3762];

4-isopropyl-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)piperazine-1-carboxamide [3763];

(R)-3,4-dimethyl-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)piperazine-1-carboxamide [3764];

N-(6-(1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [3765];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-3-(piperazin-1-yl)benzamide [3766];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-3-(4-methylpiperazin-1-yl)benzamide [3767];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-3-(pyrrolidin-1-ylmethyl)benzamide [3768];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-3-(piperidin-4-yloxy)benzamide [3769];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-3-((1-methylpiperidin-4-yl)oxy) benzamide [3770];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-4-(piperidin-4-yloxy)benzamide [3771];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-4-((1-methylpiperidin-4-yl)oxy) benzamide [3772];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(piperazin-1-yl)isonicotinamide [3773];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [3774];

2-(4-isopropylpiperazin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl) isonicotinamide [3775];

2-(4-cyclopropylpiperazin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl) isonicotinamide [3776];

2-(4-(2-fluoroethyl)piperazin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl) isonicotinamide [3777];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-6-(4-methylpiperazin-1-yl)nicotinamide [3778];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-5-(piperidin-4-yloxy)nicotinamide [3779];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(piperidin-4-yloxy)isonicotinamide [3780];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-((1-methylpiperidin-4-yl)oxy) isonicotinamide [3781];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-5-(piperidin-4-ylamino)nicotinamide [3782];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-5-((1-methylpiperidin-4-yl)amino) nicotinamide [3783];

2-(4-aminopiperidin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl) isonicotinamide [3784];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(4-(methylamino)piperidin-1-yl) isonicotinamide [3785];

2-(4-(dimethylamino)piperidin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl) isonicotinamide [3786];

2-((1-isopropylpiperidin-4-yl)oxy)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl) isonicotinamide [3787];

2-(3-aminoazetidin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl) isonicotinamide [3788];

2-(3-(dimethylamino)azetidin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl) isonicotinamide [3789];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-morpholinoisonicotinamide [3790];

2-((2-(dimethylamino)ethyl)amino)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl) isonicotinamide [3791];

2-(2-(dimethylamino)ethoxy)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl) isonicotinamide [3792];

2-(4-isobutylpiperazin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl) isonicotinamide [3793];

2-(azetidin-3-yloxy)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)isonicotinamide [3794];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-((1-methylazetidin-3-yl)oxy) isonicotinamide [3795];

2-(4-ethylpiperazin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl) isonicotinamide [3796];

4-((dimethylamino)methyl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)benzamide [3797];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-3-(1-methylpiperidin-4-yl)benzamide [3798];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-3-((4-methylpiperazin-1-yl)methyl) benzamide [3799];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)isonicotinamide [3800];

2-hydroxy-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)isonicotinamide [3801];

2-isopropoxy-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)isonicotinamide [3802];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(1-methylpiperidin-4-yl) isonicotinamide [3803];

1′-methyl-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-1′,2′,3′,6′-tetrahydro-[2,4′-bipyridine]-4-carboxamide [3804];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(4-(6-(4-methylpiperazin-1-yl) nicotinoyl)piperazin-1-yl)isonicotinamide [3805];

2-(4-hydroxy-4-methyl-4λ4-piperazin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)isonicotinamide [3806];

2-methyl-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-6-(4-methylpiperazin-1-yl) isonicotinamide [3807];

3-methyl-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [3808];

2-(4-methyl-1,4-diazepan-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl) isonicotinamide [3809];

2-((2S,6R)-2,6-dimethylmorpholino)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl) isonicotinamide [3810];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(2,7-diazaspiro[3.5]nonan-2-yl) isonicotinamide [3811];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(7-methyl-2,7-diazaspiro[3.5]nonan-2-yl)isonicotinamide [3812];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(2,7-diazaspiro[3.5]nonan-7-yl) isonicotinamide [3813];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(2-methyl-2,7-diazaspiro[3.5]nonan-7-yl)isonicotinamide [3814];

2-(methyl(1-methylpiperidin-4-yl)amino)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)isonicotinamide [3815];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-((1-methylpiperidin-4-yl)thio) isonicotinamide [3816];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl)pyrimidine-4-carboxamide [3817];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-6-(4-methylpiperazin-1-yl)pyridazine-4-carboxamide [3818];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-6-(4-methylpiperazin-1-yl)pyrimidine-4-carboxamide [3819];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-phenylacetamide [3820];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-3-phenylpropanamide [3821];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(pyridin-3-yl)acetamide [3822];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-3-(pyridin-3-yl)propanamide [3823];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(pyridin-4-yl)acetamide [3824];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-3-(pyridin-4-yl)propanamide [3825];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)isoindoline-5-carboxamide [3826];

2-methyl-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)isoindoline-5-carboxamide [3827];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-1,2,3,4-tetrahydroisoquinoline-7-carboxamide [3828];

2-methyl-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-1,2,3,4-tetrahydroisoquinoline-7-carboxamide [3829];

2-methyl-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-1,2,3,4-tetrahydroisoquinoline-6-carboxamide [3830];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-1,2,3,4-tetrahydroisoquinoline-6-carboxamide [3831];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-1H-indole-5-carboxamide [3832];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)benzofuran-5-carboxamide [3833];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)furo[2,3-c]pyridine-5-carboxamide [3834];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)benzo[b]thiophene-5-carboxamide [3835];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)benzofuran-6-carboxamide [3836];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)benzo[d]oxazole-6-carboxamide [3837];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)benzo[d]thiazole-6-carboxamide [3838];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)benzo[d]oxazole-5-carboxamide [3839];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)benzo[d]thiazole-5-carboxamide [3840];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)quinoline-3-carboxamide [3841];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)quinoline-6-carboxamide [3842];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)quinoxaline-6-carboxamide [3843];

5-chloro-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [3844];

3-chloro-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [3845];

2-(2,5-diazabicyclo[2.2.1]heptan-2-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl) isonicotinamide [3846];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(5-methyl-2,5-diazabicyclo[2.2.1] heptan-2-yl)isonicotinamide [3847];

3-fluoro-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [3848];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-((4-methylpiperazin-1-yl)methyl) isonicotinamide [3849];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(morpholinomethyl)isonicotinamide [3850];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(pyrrolidin-1-ylmethyl) isonicotinamide [3851];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(2-(4-methylpiperazin-1-yl)pyridin-4-yl)acetamide [3852];

1-methyl-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-1H-indazole-5-carboxamide [3853];

1-methyl-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-1H-benzo[d]imidazole-5-carboxamide [3854];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-1-(piperidin-4-yl)-1H-pyrazole-4-carboxamide [3855];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-1-(1-methylpiperidin-4-yl)-1H-pyrazole-4-carboxamide [3856];

1-(1-ethylpiperidin-4-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-1H-pyrazole-4-carboxamide [3857];

1-(1-(2-fluoroethyl)piperidin-4-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-1H-pyrazole-4-carboxamide [3858];

1-(1-isopropylpiperidin-4-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-1H-pyrazole-4-carboxamide [3859];

1-(1-cyclopropylpiperidin-4-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-1H-pyrazole-4-carboxamide [3860];

isopropyl 4-(4-((6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)carbamoyl)-1H-pyrazol-1-yl)piperidine-1-carboxylate [3861];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-1-(piperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide [3862];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-1-(1-methylpiperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide [3863];

1-(1-(2-fluoroethyl)piperidin-4-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-1H-1,2,3-triazole-4-carboxamide [3864];

1-(1-isopropylpiperidin-4-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-1H-1,2,3-triazole-4-carboxamide [3865];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl)oxazole-5-carboxamide [3866];

2-(3-(dimethylamino)azetidin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl) oxazole-4-carboxamide [3867];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(piperidin-4-yl)oxazole-4-carboxamide [3868];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(1-methylpiperidin-4-yl)oxazole-4-carboxamide [3869];

2-(1-(2-fluoroethyl)piperidin-4-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl) oxazole-4-carboxamide [3870];

2-(1-isopropylpiperidin-4-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)oxazole-4-carboxamide [3871];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl)oxazole-4-carboxamide [3872];

2-(3-(dimethylamino)azetidin-1-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl) thiazole-5-carboxamide [3873];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(piperidin-4-yl)thiazole-4-carboxamide [3874];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl)thiazole-4-carboxamide [3875];

2-(1-(2-fluoroethyl)piperidin-4-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl) thiazole-4-carboxamide [3876];

2-(1-isopropylpiperidin-4-yl)-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)thiazole-4-carboxamide [3877];

1-methyl-N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl-4-d)piperidine-4-carboxamide [3878];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-1-(2-(methyl-d3)propyl-1,1,2,3,3,3-d6) piperidine-4-carboxamide [3879];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(pyrrolidin-1-yl-2,2,5,5-d 4 )acetamide [3880];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(4-(methyl-d 3 )piperazin-1-yl) acetamide [3881];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(morpholino-d 8 )acetamide [3882];

(S)—N-(6-(1-(methyl-d 3 )-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(pyrrolidin-1-yl)propanamide [3883];

1-isobutyl-N-(6-(1-(methyl-d 3 )-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [3884];

N-(6-(1-(methyl-d 3 )-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl) acetamide [3885];

N-(6-(1-(methyl-d 3 )-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide [3886];

N-(6-(1-(methyl-d 3 )-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(piperidin-1-yl)acetamide [3887];

N-(6-(1-(methyl-d 3 )-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [3888];

N-(6-(1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(4-(methyl-d 3 )piperazin-1-yl)isonicotinamide [3889];

N-(6-(1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(4-(methyl-d 3 )piperazin-1-yl) isonicotinamide [3890];

N-(6-(1-(methyl-d 3 )-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [3891];

N-(6-(1-(methyl-d 3 )-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(4-(methyl-d 3 )piperazin-1-yl) isonicotinamide [3892];

N-(6-(1-(methyl-d 3 )-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-1-(piperidin-4-yl)-1H-pyrazole-4-carboxamide [3893];

N-(6-(1-(methyl-d 3 )-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-1-(1-methylpiperidin-4-yl)-1H-pyrazole-4-carboxamide [3894];

N-(6-(1-(methyl-d 3 )-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(piperidin-4-yl)oxazole-4-carboxamide [3895];

N-(6-(1-(methyl-d 3 )-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(1-methylpiperidin-4-yl)oxazole-4-carboxamide [3896];

N-(6-(1-ethyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide [3897];

N-(6-(1-cyclopropyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide [3898];

N-(6-(1-cyclopropyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [3899];

N-(6-(1-(1-methylpiperidin-4-yl)-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl) cyclohexanecarboxamide [3900];

2-(pyrrolidin-1-yl)-N-(6-(5-(trifluoromethyl)-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)acetamide [3901];

N-(6-(5-(hydroxymethyl)-1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-1-methylpiperidine-4-carboxamide [3902];

N-(6-(5-(hydroxymethyl)-1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)tetrahydro-2H-pyran-4-carboxamide [3903];

N-(6-(5-(azetidin-1-ylmethyl)-1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-4,4-difluorocyclohexane-1-carboxamide [3904];

4,4-difluoro-N-(6-(1-methyl-5-(pyrrolidin-1-ylmethyl)-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl) cyclohexane-1-carboxamide [3905];

4,4-difluoro-N-(6-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl) cyclohexane-1-carboxamide [3906];

2-(2-fluoroethyl)-N-(6-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-azaspiro[3.3]heptane-6-carboxamide [3907];

tert-butyl 6-((6-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl) carbamoyl)-2-azaspiro[3.3]heptane-2-carboxylate [3908];

2-fluoro-2-methyl-N-(6-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)propanamide [3909];

2-(diethylamino)-N-(6-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)acetamide [3910];

trans-4-methoxy-N-(6-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)cyclohexane-1-carboxamide [3911];

trans-4-(hydroxymethyl)-N-(6-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)cyclohexane-1-carboxamide [3912];

(R)—N-(6-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)pyrrolidine-2-carboxamide [3913];

1-isobutyl-N-(6-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl) piperidine-4-carboxamide [3914];

N-(6-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-1-(oxetan-3-yl) piperidine-4-carboxamide [3915];

1-benzoyl-N-(6-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl) piperidine-4-carboxamide [3916];

N-(6-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)tetrahydro-2H-pyran-4-carboxamide [3917];

N-(6-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperidin-1-yl)acetamide [3918];

N-(6-(1-(difluoromethyl)-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [3919];

N-(6-(1-ethyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [3920];

N-(6-(1-isopropyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-3-(piperidin-4-yloxy)benzamide [3921];

N-(6-(1-isopropyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-3-((1-methylpiperidin-4-yl)oxy) benzamide [3922];

N-(6-(1-isopropyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-4-(piperidin-4-yloxy)benzamide [3923];

N-(6-(1-cyclopropyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [3924];

4-fluoro-N-(6-(1-(1-methylpiperidin-4-yl)-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)benzamide [3925];

4-(difluoromethoxy)-N-(6-(1-(1-methylpiperidin-4-yl)-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl) benzamide [3926];

5-fluoro-N-(6-(1-(1-methylpiperidin-4-yl)-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)nicotinamide [3927];

N 2 -methyl-N 5 -(6-(1-(1-methylpiperidin-4-yl)-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)pyridine-2,5-dicarboxamide [3928];

1-isopropyl-N-(6-(1-(1-methylpiperidin-4-yl)-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-1H-pyrazole-4-carboxamide [3929];

2-methyl-N-(6-(1-(1-methylpiperidin-4-yl)-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)thiazole-5-carboxamide [3930];

N-(6-(5-amino-1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [3931];

4-(difluoromethoxy)-N-(6-(5-(hydroxymethyl)-1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl) benzamide [3932];

N-(6-(5-(hydroxymethyl)-1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [3933];

N-(6-(5-(hydroxymethyl)-1-methyl-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(7-methyl-2,7-diazaspiro[3.5]nonan-2-yl)isonicotinamide [3934];

4-fluoro-N-(6-(1-methyl-5-(pyrrolidin-1-ylmethyl)-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl) benzamide [3935];

4-fluoro-N-(6-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl) benzamide [3936];

4-(difluoromethoxy)-N-(6-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)benzamide [3937];

N-(6-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-3-(pyrrolidin-1-ylmethyl)benzamide [3938];

N-(6-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-(7-methyl-2,7-diazaspiro[3.5]nonan-2-yl)isonicotinamide [3939];

N-(6-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-morpholinoisonicotinamide [3940];

N-(6-(1-methyl-5-(morpholinomethyl)-1H-pyrazol-4-yl)-2,7-naphthyridin-3-yl)-2-morpholinoisonicotinamide [3941];

N-(6-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)-2,7-naphthyridin-3-yl)-1-((1-(trifluoromethyl)cyclopropyl)methyl)piperidine-4-carboxamide [3942];

3,3-difluoro-N-(6-(5-methyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)-2,7-naphthyridin-3-yl)cyclobutane-1-carboxamide [3943];

4,4-difluoro-N-(6-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)-2,7-naphthyridin-3-yl)cyclohexane-1-carboxamide [3944];

N-(6-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)-2,7-naphthyridin-3-yl)-1-((1-(trifluoromethyl)cyclopropyl)methyl)piperidine-4-carboxamide [3945];

N-(6-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)-2,7-naphthyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide [3946];

2-(7-azabicyclo[2.2.1]heptan-7-yl)-N-(6-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)-2,7-naphthyridin-3-yl)acetamide [3947];

(R)—N-(6-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)-2,7-naphthyridin-3-yl)-1-isobutylpiperidine-3-carboxamide [3948];

N-(6-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)-2,7-naphthyridin-3-yl) piperidine-4-carboxamide [3949];

4-fluoro-N-(6-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)-2,7-naphthyridin-3-yl)-1-isobutylpiperidine-4-carboxamide [3950];

N-(6-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl)acetamide [3951];

4-fluoro-N-(6-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)-2,7-naphthyridin-3-yl)benzamide [3952];

N-(6-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)-2,7-naphthyridin-3-yl)-3-(4-methylpiperazin-1-yl)benzamide [3953];

N 5 -(6-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)-2,7-naphthyridin-3-yl)-N 2 -methylpyridine-2,5-dicarboxamide [3954];

N-(6-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)-2,7-naphthyridin-3-yl)-6-(4-methylpiperazin-1-yl)nicotinamide [3955];

2-(azetidin-3-yloxy)-N-(6-(5-(2-fluoroethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl)-2,7-naphthyridin-3-yl)isonicotinamide [3956];

N-(6-(1-methyl-1H-pyrazol-5-yl)-2,7-naphthyridin-3-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [3957];

1-methyl-N-(6-(1-methyl-1H-pyrazol-3-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [3958];

N-(6-(1-methyl-1H-pyrazol-3-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [3959];

2-fluoro-2-methyl-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)propanamide [3960];

2,2,3,3-tetramethyl-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)cyclopropane-1-carboxamide [3961];

trans-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)-4-(pyrrolidin-1-yl) cyclohexane-1-carboxamide [3962];

trans-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)-4-morpholinocyclohexane-1-carboxamide [3963];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)-2-(piperidin-1-yl)acetamide [3964];

1-ethyl-4-fluoro-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [3965];

4-fluoro-1-isobutyl-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [3966];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [3967];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)cyclopropanecarboxamide [3968];

4,4-difluoro-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)cyclohexane-1-carboxamide [3969];

trans-4-(dimethylamino)-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl) cyclohexane-1-carboxamide [3970];

trans-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)-4-((4-methylpiperazin-1-yl) methyl)cyclohexane-1-carboxamide [3971];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [3972];

1-isobutyl-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [3973];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)-1-((1-(trifluoromethyl)cyclopropyl) methyl)piperidine-4-carboxamide [3974];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)-1-((3-methyloxetan-3-yl)methyl) piperidine-4-carboxamide [3975];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)-1-(2-(pyrrolidin-1-yl)acetyl) piperidine-4-carboxamide [3976];

1′-methyl-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)-[1,4′-bipiperidine]-4-carboxamide [3977];

(R)—N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)piperidine-3-carboxamide [3978];

(R)-1-isobutyl-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)piperidine-3-carboxamide [3979];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide [3980];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl) acetamide [3981];

2-(7-azabicyclo[2.2.1]heptan-7-yl)-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl) acetamide [3982];

1-(2-hydroxy-2-methylpropyl)-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl) piperidine-4-carboxamide [3983];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)-2-morpholinoacetamide [3984];

2-(4-methoxypiperidin-1-yl)-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl) acetamide [3985];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)morpholine-4-carboxamide [3986];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)-1-(piperidin-4-yl)-1H-pyrazole-4-carboxamide [3987];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)-1-(1-methylpiperidin-4-yl)-1H-pyrazole-4-carboxamide [3988];

1-(1-ethylpiperidin-4-yl)-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)-1H-pyrazole-4-carboxamide [3989];

1-(1-isopropylpiperidin-4-yl)-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)-1H-pyrazole-4-carboxamide [3990];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)-1-(piperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide [3991];

1-(1-(2-fluoroethyl)piperidin-4-yl)-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)-1H-1,2,3-triazole-4-carboxamide [3992];

1-(1-isopropylpiperidin-4-yl)-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)-1H-1,2,3-triazole-4-carboxamide [3993];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)-2-(piperidin-4-yl)oxazole-4-carboxamide [3994];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)-2-(1-methylpiperidin-4-yl)oxazole-4-carboxamide [3995];

2-(1-isopropylpiperidin-4-yl)-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl) oxazole-4-carboxamide [3996];

2-fluoro-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)benzamide [3997];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)-3-((1-methylpiperidin-4-yl)oxy) benzamide [3998];

N 2 -methyl-N 5 -(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)pyridine-2,5-dicarboxamide [3999];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)-6-(4-methylpiperazin-1-yl) nicotinamide [4000];

2-(3-(dimethylamino)azetidin-1-yl)-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl) isonicotinamide [4001];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)-2-(1-methylpiperidin-4-yl) isonicotinamide [4002];

2-(4-(dimethylamino)piperidin-1-yl)-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)isonicotinamide [4003];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)-2-morpholinoisonicotinamide [4004];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [4005];

2-(4-methyl-1,4-diazepan-1-yl)-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl) isonicotinamide [4006];

2-(4-isopropylpiperazin-1-yl)-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl) isonicotinamide [4007];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)-2-(piperidin-4-ylamino) isonicotinamide [4008];

2-(methyl(1-methylpiperidin-4-yl)amino)-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)isonicotinamide [4009];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)-2-((1-methylpiperidin-4-yl)thio) isonicotinamide [4010];

2-methyl-N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)-1,2,3,4-tetrahydroisoquinoline-6-carboxamide [4011];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)-2-(piperazin-1-yl)isonicotinamide [4012];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)-2-(2-(4-methylpiperazin-1-yl) pyridin-4-yl)acetamide [4013];

1,1-bis(methyl-d 3 )-4-(4-((6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)carbamoyl) pyridin-2-yl)piperazin-1-ium iodide [4014];

N-(6-(1-methyl-1H-1,2,3-triazol-4-yl)-2,7-naphthyridin-3-yl)-2-(4-(methyl-d 3 )piperazin-1-yl) isonicotinamide [4015];

N-(6-(1-methyl-1H-1,2,3-triazol-5-yl)-2,7-naphthyridin-3-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [4016];

N-(6-(4-methyl-4H-1,2,4-triazol-3-yl)-2,7-naphthyridin-3-yl)-2-morpholinoacetamide [4017];

N-(6-(4-methyl-4H-1,2,4-triazol-3-yl)-2,7-naphthyridin-3-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [4018];

4-fluoro-1-isobutyl-N-(6-(4-methyl-4H-1,2,4-triazol-3-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [4019];

N-(6-(4,5-dimethyl-4H-1,2,4-triazol-3-yl)-2,7-naphthyridin-3-yl)-2-morpholinoacetamide [4020];

N-(6-(4,5-dimethyl-4H-1,2,4-triazol-3-yl)-2,7-naphthyridin-3-yl)-1-(3,3,3-trifluoropropyl) piperidine-4-carboxamide [4021];

N-(6-(1H-1,2,3-triazol-1-yl)-2,7-naphthyridin-3-yl)-4-fluoro-1-isobutylpiperidine-4-carboxamide [4022];

N-(6-(2H-1,2,3-triazol-2-yl)-2,7-naphthyridin-3-yl)-4-fluoro-1-isobutylpiperidine-4-carboxamide [4023];

N-(6-(1H-1,2,4-triazol-1-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [4024];

1-isobutyl-N-(6-(1-methyl-1H-tetrazol-5-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [4025];

2,2,3,3-tetramethyl-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)cyclopropane-1-carboxamide [4026];

4,4-difluoro-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)cyclohexane-1-carboxamide [4027];

N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-2-(piperidin-1-yl)acetamide [4028];

2-fluoro-2-methyl-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)propanamide [4029];

1-fluoro-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)cyclopropane-1-carboxamide [4030];

2-methyl-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-2-azaspiro[3.3]heptane-6-carboxamide [4031];

1-fluoro-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)cyclohexane-1-carboxamide [4032];

trans-4-methoxy-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)cyclohexane-1-carboxamide [4033];

trans-4-(hydroxymethyl)-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)cyclohexane-1-carboxamide [4034];

N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)azetidine-3-carboxamide [4035];

(R)—N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)tetrahydrofuran-2-carboxamide [4036];

1-(2-methoxyethyl)-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [4037];

N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [4038];

1-isobutyl-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [4039];

N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-1-(methylsulfonyl)piperidine-4-carboxamide [4040];

N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-2-(pyrrolidin-1-yl)propanamide [4041];

2-isopropoxy-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)acetamide [4042];

3-isopropoxy-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)propanamide [4043];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)cyclopropanecarboxamide [4044];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)cyclohexanecarboxamide [4045];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-4,4-difluorocyclohexane-1-carboxamide [4046];

(S)—N-(6-(1,2-dimethyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)tetrahydrofuran-2-carboxamide [4047];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-3,3-difluorocyclobutane-1-carboxamide [4048];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-1-fluorocyclopropane-1-carboxamide [4049];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)morpholine-4-carboxamide [4050];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)morpholine-d 8 -4-carboxamide [4051];

1-methyl-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-1H-pyrazole-4-carboxamide [4052];

1-ethyl-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-1H-pyrazole-4-carboxamide [4053];

1-isopropyl-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-1H-pyrazole-4-carboxamide [4054];

1-cyclopropyl-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-1H-pyrazole-4-carboxamide [4055];

1-isobutyl-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-1H-pyrazole-4-carboxamide [4056];

1-methyl-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-1H-pyrazole-3-carboxamide [4057];

N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-2-(1-methyl-1H-pyrazol-4-yl) acetamide [4058];

1-methyl-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-1H-imidazole-4-carboxamide [4059];

1-isopropyl-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-1H-imidazole-4-carboxamide [4060];

N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-1-(tetrahydro-2H-pyran-4-yl)-1H-imidazole-4-carboxamide [4061];

1,2-dimethyl-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-1H-imidazole-5-carboxamide [4062];

1-methyl-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-1H-1,2,4-triazole-3-carboxamide [4063];

2-methyl-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)oxazole-4-carboxamide [4064];

2-isopropyl-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)oxazole-4-carboxamide [4065];

4-methyl-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)oxazole-2-carboxamide [4066];

4-methyl-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)thiazole-2-carboxamide [4067];

2-methyl-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)thiazole-4-carboxamide [4068];

5-methyl-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-1,3,4-oxadiazole-2-carboxamide [4069];

5-methyl-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-1,3,4-thiadiazole-2-carboxamide [4070];

1-isopropyl-N-(6-(1-isopropyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-1H-pyrazole-4-carboxamide [4071];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-1-methyl-1H-pyrazole-4-carboxamide [4072];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-1-isopropyl-1H-pyrazole-4-carboxamide [4073];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-2-methylthiazole-5-carboxamide [4074];

4-fluoro-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)benzamide [4075];

4-(difluoromethoxy)-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)benzamide [4076];

N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-3-(pyrrolidin-1-ylmethyl)benzamide [4077];

2-fluoro-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)benzamide-3,4,5,6-d 4 [4078];

4-fluoro-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)benzamide-2,3,5,6-d 4 [4079];

2-chloro-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)benzamide-3,4,5,6-d 4 [4080];

4-chloro-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)benzamide-2,3,5,6-d 4 [4081];

4-(methyl-d 3 )—N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)benzamide [4082];

4-methyl-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)benzamide-2,3,5,6-d 4 [4083];

4-(methyl-d 3 )—N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)benzamide-2,3,5,6-d 4 [4084];

4-(methoxy-d 3 )—N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)benzamide [4085];

4-(methoxy-d 3 )—N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)benzamide-2,3,5,6-d 4 [4086];

4-methoxy-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)benzamide-2,3,5,6-d 4 [4087];

(E)-N-(6-(1,2-dimethyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-3-(phenyl-2,3,4,5,6-d 5 ) acrylamide [4088];

(E)-N-(6-(1,2-dimethyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-3-(phenyl-2,3,4,5,6-d 5 ) acrylamide-2,3-d 2 [4089];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-2-(4-fluorophenyl)acetamide-2,2-d 2 [4090];

(E)-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-3-(phenyl-2,3,4,5,6-d 5 )acrylamide [4091];

(E)-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-3-(phenyl-2,3,4,5,6-d 5 )acrylamide-2,3-d 2 [4092];

2-(4-fluorophenyl)-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)acetamide-2,2-d 2 [4093];

N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [4094];

2-(dimethylamino)-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)isonicotinamide [4095];

2-(3-aminoazetidin-1-yl)-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl) isonicotinamide [4096];

N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-2-(pyrrolidin-1-yl)isonicotinamide [4097];

N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-2-(piperidin-1-yl)isonicotinamide [4098];

N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-2-morpholinoisonicotinamide [4099];

2-(4-isopropylpiperazin-1-yl)-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl) isonicotinamide [4100];

2-(4-cyclopropylpiperazin-1-yl)-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl) isonicotinamide [4101];

N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-2-(2,7-diazaspiro[3.5]nonan-2-yl) isonicotinamide [4102];

N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-2-(7-methyl-2,7-diazaspiro[3.5]nonan-2-yl)isonicotinamide [4103];

N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)isoindoline-5-carboxamide [4104];

2-methyl-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)isoindoline-5-carboxamide [4105];

2-(azetidin-1-yl)-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)isonicotinamide [4106];

2-methoxy-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)isonicotinamide [4107];

2-methyl-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)isonicotinamide [4108];

2-cyano-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)isonicotinamide [4109];

2-(3,3-difluoroazetidin-1-yl)-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl) isonicotinamide [4110];

2-(4,4-difluoropiperidin-1-yl)-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl) isonicotinamide [4111];

2-isopropoxy-N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)isonicotinamide [4112];

N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-2-(pyrrolidin-1-yl-2,2,5,5-d 4 ) isonicotinamide [4113];

N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-2-(pyrrolidin-1-yl-d 8 )isonicotinamide [4114];

N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-2-(piperidin-1-yl-d 10 )isonicotinamide [4115];

N-(6-(1-methyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-2-(morpholino-d 8 )isonicotinamide [4116];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-4-isopropoxybenzamide [4117];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-4-(piperidin-4-yloxy)benzamide [4118];

4-(benzyloxy)-N-(6-(1,2-dimethyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)benzamide [4119];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-2-fluorobenzamide-3,4,5,6-d 4 [4120];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-4-fluorobenzamide-2,3,5,6-d 4 [4121];

2-chloro-N-(6-(1,2-dimethyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)benzamide-3,4,5,6-d 4 [4122];

4-chloro-N-(6-(1,2-dimethyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)benzamide-2,3,5,6-d 4 [4123];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-4-(methyl-d 3 )benzamide [4124];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-4-methylbenzamide-2,3,5,6-d 4 [4125];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-4-(methyl-d 3 )benzamide-2,3,5,6-d 4 [4126];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-4-(methoxy-d 3 )benzamide [4127];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-4-(methoxy-d 3 )benzamide-2,3,5,6-d 4 [4128];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-4-methoxybenzamide-2,3,5,6-d 4 [4129];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [4130];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-2-morpholinoisonicotinamide [4131];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-2-(pyrrolidin-1-yl)isonicotinamide [4132];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-2-(dimethylamino)isonicotinamide [4133];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-2-(pyrrolidin-1-yl-2,2,5,5-d 4 ) isonicotinamide [4134];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-2-(pyrrolidin-1-yl-d 8 ) isonicotinamide [4135];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-2-(piperidin-1-yl-d 10 ) isonicotinamide [4136];

N-(6-(1,2-dimethyl-1H-imidazol-5-yl)-2,7-naphthyridin-3-yl)-2-(morpholino-d 8 )isonicotinamide [4137];

N-(6-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-2,7-naphthyridin-3-yl) cyclopropanecarboxamide [4138];

N-(6-(7-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-2,7-naphthyridin-3-yl) cyclopropanecarboxamide [4139];

3,3-difluoro-N-(6-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-2,7-naphthyridin-3-yl) cyclobutane-1-carboxamide [4140];

(R)—N-(6-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-2,7-naphthyridin-3-yl)pyrrolidine-2-carboxamide [4141];

(R)—N-(6-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-2,7-naphthyridin-3-yl)piperidine-3-carboxamide [4142];

1-methyl-N-(6-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [4143];

N-(6-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-2,7-naphthyridin-3-yl)-1-((1-(trifluoromethyl)cyclopropyl)methyl)piperidine-4-carboxamide [4144];

1-benzoyl-N-(6-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [4145];

4-fluoro-1-isobutyl-N-(6-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-2,7-naphthyridin-3-yl) piperidine-4-carboxamide [4146];

(R)-2-(2-methylpyrrolidin-1-yl)-N-(6-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-2,7-naphthyridin-3-yl)acetamide [4147];

2-(cyclobutyl(methyl)amino)-N-(6-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-2,7-naphthyridin-3-yl)acetamide [4148];

4-fluoro-N-(6-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-2,7-naphthyridin-3-yl)benzamide [4149];

4-isopropoxy-N-(6-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-2,7-naphthyridin-3-yl) benzamide [4150];

4-(difluoromethoxy)-N-(6-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-2,7-naphthyridin-3-yl) benzamide [4151];

2-((2-(dimethylamino)ethyl)amino)-N-(6-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-2,7-naphthyridin-3-yl)isonicotinamide [4152];

2-((1-isopropylpiperidin-4-yl)oxy)-N-(6-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-2,7-naphthyridin-3-yl)isonicotinamide [4153];

N-(6-(oxazol-5-yl)-2,7-naphthyridin-3-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [4154];

N-(6-(oxazol-5-yl)-2,7-naphthyridin-3-yl)cyclopropanecarboxamide [4155];

(R)—N-(6-(oxazol-5-yl)-2,7-naphthyridin-3-yl)tetrahydrofuran-2-carboxamide [4156];

(R)—N-(6-(oxazol-5-yl)-2,7-naphthyridin-3-yl)piperidine-3-carboxamide [4157];

N-(6-(oxazol-5-yl)-2,7-naphthyridin-3-yl)tetrahydro-2H-pyran-4-carboxamide [4158];

N-(6-(oxazol-5-yl)-2,7-naphthyridin-3-yl)-1-(2-(pyrrolidin-1-yl)acetyl)piperidine-4-carboxamide [4159];

1′-methyl-N-(6-(oxazol-5-yl)-2,7-naphthyridin-3-yl)-[1,4′-bipiperidine]-4-carboxamide [4160];

cis-4-morpholino-N-(6-(oxazol-5-yl)-2,7-naphthyridin-3-yl)cyclohexane-1-carboxamide [4161];

2-(cyclobutyl(methyl)amino)-N-(6-(oxazol-5-yl)-2,7-naphthyridin-3-yl)acetamide [4162];

N-(6-(oxazol-5-yl)-2,7-naphthyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide [4163];

(R)-2-(2-methylpyrrolidin-1-yl)-N-(6-(oxazol-5-yl)-2,7-naphthyridin-3-yl)acetamide [4164];

2-(4-methylpiperazin-1-yl)-N-(6-(oxazol-5-yl)-2,7-naphthyridin-3-yl)acetamide [4165];

trans-4-((4-methylpiperazin-1-yl)methyl)-N-(6-(oxazol-5-yl)-2,7-naphthyridin-3-yl)cyclohexane-1-carboxamide [4166];

1-(2,2-difluoropropyl)-N-(6-(oxazol-5-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [4167];

trans-4-(hydroxymethyl)-N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl)cyclohexane-1-carboxamide [4168];

trans-4-(methylamino)-N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl)cyclohexane-1-carboxamide [4169];

trans-4-((1,3-difluoropropan-2-yl)amino)-N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl) cyclohexane-1-carboxamide [4170];

trans-N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl)-4-((propan-2-yl-1,1,1,3,3,3-d 6 )amino) cyclohexane-1-carboxamide [4171];

trans-4-((2,2-difluoroethyl)amino)-N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl) cyclohexane-1-carboxamide [4172];

trans-N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl)-4-((3,3,3-trifluoropropyl)amino) cyclohexane-1-carboxamide [4173];

trans-4-((2-methoxyethyl)amino)-N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl) cyclohexane-1-carboxamide [4174];

trans-4-(dimethylamino)-N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl)cyclohexane-1-carboxamide [4175];

trans-4-(bis(methyl-d 3 )amino)-N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl)cyclohexane-1-carboxamide [4176];

cis-4-(dimethylamino)-N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl)cyclohexane-1-carboxamide [4177];

trans-4-((2,2-difluoroethyl)(methyl)amino)-N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl) cyclohexane-1-carboxamide [4178];

trans-4-(methyl(oxetan-3-yl)amino)-N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl) cyclohexane-1-carboxamide [4179];

trans-4-((2-fluoroethyl)amino)-N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl)cyclohexane-1-carboxamide [4180];

trans-4-(2-(fluoromethyl)aziridin-1-yl)-N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl) cyclohexane-1-carboxamide [4181];

trans-4-((3-fluoroazetidin-1-yl)methyl)-N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl) cyclohexane-1-carboxamide [4182];

trans-N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl)-3-morpholinocyclobutane-1-carboxamide [4183];

trans-N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl)-4-morpholinocyclohexane-1-carboxamide [4184];

N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl)-2-(piperidin-1-yl)acetamide [4185];

2-(4-methoxypiperidin-1-yl)-N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl)acetamide [4186];

N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl)acetamide [4187];

N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl)morpholine-4-carboxamide [4188];

N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl)-2-morpholinoacetamide [4189];

N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl)-3-morpholinopropanamide [4190];

1-methyl-N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [4191];

1-(2,2-difluoropropyl)-N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [4192];

N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl)-4-morpholinopiperidine-1-carboxamide [4193];

4-((1,3-difluoropropan-2-yl)amino)-N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl) piperidine-1-carboxamide [4194];

(1R,3s,5S)-3-((1,3-difluoropropan-2-yl)amino)-N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl)-8-azabicyclo[3.2.1]octane-8-carboxamide [4195];

(1R,3s,5S)-3-((1,3-difluoropropan-2-yl)amino)-N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl)-8-azabicyclo[3.2.1]octane-8-carboxamide [4196];

4-(dimethylamino)-N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl)piperidine-1-carboxamide [4197];

4-((2,2-difluoroethyl)(methyl)amino)-N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl) piperidine-1-carboxamide [4198];

(3S,4S)-4-amino-3-fluoro-N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl)piperidine-1-carboxamide [4199];

(3S,4S)-3-fluoro-4-(methylamino)-N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl)piperidine-1-carboxamide [4200];

(3 R,4R)-4-amino-3-fluoro-N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl)piperidine-1-carboxamide [4201];

(3R,4R)-3-fluoro-4-(methylamino)-N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl)piperidine-1-carboxamide [4202];

4-((2-fluoroethyl)amino)-N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl)piperidine-1-carboxamide [4203];

4-((2,2-difluoroethyl)amino)-N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl)piperidine-1-carboxamide [4204];

(1R,3s,5S)-3-amino-N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl)-8-azabicyclo[3.2.1] octane-8-carboxamide [4205];

(1R,3r,5S)-3-amino-N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl)-8-azabicyclo[3.2.1] octane-8-carboxamide [4206];

(1R,3r,5S)-3-((2-fluoroethyl)amino)-N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl)-8-azabicyclo[3.2.1]octane-8-carboxamide [4207];

(1R,3r,5S)-3-((2,2-difluoroethyl)amino)-N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl)-8-azabicyclo[3.2.1]octane-8-carboxamide [4208];

(1R,3s,5 S)—N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl)-3-((3,3,3-trifluoropropyl)amino)-8-azabicyclo[3.2.1]octane-8-carboxamide [4209];

(3 S,4S)-3-fluoro-4-(isopropylamino)-N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl) piperidine-1-carboxamide [4210];

N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl)-5,6-dihydroimidazo[1,2-a]pyrazine-7(8H)-carboxamide [4211];

2-methyl-N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl)-5,6-dihydroimidazo[1,2-a]pyrazine-7(8H)-carboxamide [4212];

N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl)-2-(morpholino-d 8 )acetamide [4213];

trans-N-(6-(2-methyloxazol-4-yl)-2,7-naphthyridin-3-yl)-4-(4-methylpiperazin-1-yl)cyclohexane-1-carboxamide [4214];

N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl)-1-(1-methylpiperidin-4-yl)-1H-pyrazole-4-carboxamide [4215];

2-(1H-imidazol-1-yl)-N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl)acetamide [4216];

4-(difluoromethoxy)-N-(6-(oxazol-5-yl)-2,7-naphthyridin-3-yl)benzamide [4217];

3-((1-methylpiperidin-4-yl)oxy)-N-(6-(oxazol-5-yl)-2,7-naphthyridin-3-yl)benzamide [4218];

N-(6-(oxazol-5-yl)-2,7-naphthyridin-3-yl)isonicotinamide [4219];

2-(3-aminoazetidin-1-yl)-N-(6-(oxazol-5-yl)-2,7-naphthyridin-3-yl)isonicotinamide [4220];

2-(1-methylpiperidin-4-yl)-N-(6-(oxazol-5-yl)-2,7-naphthyridin-3-yl)isonicotinamide [4221];

1′-methyl-N-(6-(oxazol-5-yl)-2,7-naphthyridin-3-yl)-1′,2′,3′,6′-tetrahydro-[2,4′-bipyridine]-4-carboxamide [4222];

2-(4-methylpiperazin-1-yl)-N-(6-(oxazol-5-yl)-2,7-naphthyridin-3-yl)isonicotinamide [4223];

2-(7-methyl-2,7-diazaspiro[3.5]nonan-2-yl)-N-(6-(oxazol-5-yl)-2,7-naphthyridin-3-yl) isonicotinamide [4224];

N-(6-(oxazol-5-yl)-2,7-naphthyridin-3-yl)-2-(2,7-diazaspiro[3.5]nonan-7-yl)isonicotinamide [4225];

N-(6-(oxazol-5-yl)-2,7-naphthyridin-3-yl)-2-(piperidin-4-ylamino)isonicotinamide [4226];

2-methyl-N-(6-(oxazol-5-yl)-2,7-naphthyridin-3-yl)isoindoline-5-carboxamide [4227];

N-(6-(oxazol-5-yl)-2,7-naphthyridin-3-yl)-1,2,3,4-tetrahydroisoquinoline-7-carboxamide [4228];

N-(6-(2-methyloxazol-5-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [4229];

N-(6-(3-methylisoxazol-5-yl)-2,7-naphthyridin-3-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [4230];

4-fluoro-1-isobutyl-N-(6-(5-methyl-1,3,4-oxadiazol-2-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [4231];

1-isobutyl-N-(6-(5-methyl-1,3,4-oxadiazol-2-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [4232];

N-(6-(5-(dimethylamino)-1,3,4-oxadiazol-2-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [4233];

N-(6-(5-(dimethylamino)-1,3,4-oxadiazol-2-yl)-2,7-naphthyridin-3-yl)-1-methylpiperidine-4-carboxamide [4234];

N-(6-(5-methyl-1,3,4-oxadiazol-2-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [4235];

3,3-difluoro-N-(6-(thiazol-5-yl)-2,7-naphthyridin-3-yl)cyclobutane-1-carboxamide [4236];

2-methyl-N-(6-(thiazol-5-yl)-2,7-naphthyridin-3-yl)-2-azaspiro[3.3]heptane-6-carboxamide [4237];

1-fluoro-N-(6-(thiazol-5-yl)-2,7-naphthyridin-3-yl)cyclohexane-1-carboxamide [4238];

trans-4-(dimethylamino)-N-(6-(thiazol-5-yl)-2,7-naphthyridin-3-yl)cyclohexane-1-carboxamide [4239];

trans-4-((3-fluoroazetidin-1-yl)methyl)-N-(6-(thiazol-5-yl)-2,7-naphthyridin-3-yl)cyclohexane-1-carboxamide [4240];

N-(6-(thiazol-5-yl)-2,7-naphthyridin-3-yl)azetidine-3-carboxamide [4241];

1-methyl-N-(6-(thiazol-5-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [4242];

1-(2,2-difluoropropyl)-N-(6-(thiazol-5-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [4243];

1-(oxetan-3-yl)-N-(6-(thiazol-5-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [4244];

1-(2-(pyrrolidin-1-yl)acetyl)-N-(6-(thiazol-5-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [4245];

1′-methyl-N-(6-(thiazol-5-yl)-2,7-naphthyridin-3-yl)-[1,4′-bipiperidine]-4-carboxamide [4246];

2-(pyrrolidin-1-yl)-N-(6-(thiazol-5-yl)-2,7-naphthyridin-3-yl)propanamide [4247];

2-(piperidin-1-yl)-N-(6-(thiazol-5-yl)-2,7-naphthyridin-3-yl)acetamide [4248];

2-(4-methylpiperazin-1-yl)-N-(6-(thiazol-5-yl)-2,7-naphthyridin-3-yl)acetamide [4249];

2-morpholino-N-(6-(thiazol-5-yl)-2,7-naphthyridin-3-yl)acetamide [4250];

4-(piperidin-4-yloxy)-N-(6-(thiazol-5-yl)-2,7-naphthyridin-3-yl)benzamide [4251];

N-(6-(thiazol-5-yl)-2,7-naphthyridin-3-yl)isonicotinamide [4252];

6-(4-methylpiperazin-1-yl)-N-(6-(thiazol-5-yl)-2,7-naphthyridin-3-yl)nicotinamide [5253];

1′-methyl-N-(6-(thiazol-5-yl)-2,7-naphthyridin-3-yl)-1′,2′,3′,6′-tetrahydro-[2,4′-bipyridine]-4-carboxamide [4254];

2-(3-(dimethylamino)azetidin-1-yl)-N-(6-(thiazol-5-yl)-2,7-naphthyridin-3-yl)isonicotinamide [4255];

2-(4-(dimethylamino)piperidin-1-yl)-N-(6-(thiazol-5-yl)-2,7-naphthyridin-3-yl)isonicotinamide [4256];

2-(4-methylpiperazin-1-yl)-N-(6-(thiazol-5-yl)-2,7-naphthyridin-3-yl)isonicotinamide [4257];

2-((1-methylpiperidin-4-yl)thio)-N-(6-(thiazol-5-yl)-2,7-naphthyridin-3-yl)isonicotinamide [4258];

N-(6-(thiazol-5-yl)-2,7-naphthyridin-3-yl)-1,2,3,4-tetrahydroisoquinoline-7-carboxamide [4259];

trans-4-((1,3-difluoropropan-2-yl)amino)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)cyclohexane-1-carboxamide [4260];

N-(6-(2-methylthiazol-5-yl)-2,7-naphthyridin-3-yl)morpholine-4-carboxamide [4261];

N-(6-(2-methylthiazol-5-yl)-2,7-naphthyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide [4262];

2-((1R,4R)-2-oxa-5-azabicyclo[2.2.1]heptan-5-yl)-N-(6-(2-methylthiazol-5-yl)-2,7-naphthyridin-3-yl)acetamide [4263];

N-(6-(2-methylthiazol-5-yl)-2,7-naphthyridin-3-yl)-2-morpholinoacetamide [4264];

N-(6-(2-methylthiazol-5-yl)-2,7-naphthyridin-3-yl)-2-(morpholino-d 8 )acetamide [4265];

2-(4-methylpiperazin-1-yl)-N-(6-(2-methylthiazol-5-yl)-2,7-naphthyridin-3-yl)acetamide [4266];

1-methyl-N-(6-(2-methylthiazol-5-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [4267];

N-(6-(2-methylthiazol-5-yl)-2,7-naphthyridin-3-yl)isonicotinamide [4268];

N-(6-(2-methylthiazol-5-yl)-2,7-naphthyridin-3-yl)nicotinamide [4269];

2-(4-methylpiperazin-1-yl)-N-(6-(2-methylthiazol-5-yl)-2,7-naphthyridin-3-yl)isonicotinamide [4270];

trans-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-4-morpholinocyclohexane-1-carboxamide [4271];

trans-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-4-(4-methylpiperazin-1-yl) cyclohexane-1-carboxamide [4272];

4-isopropyl-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)piperazine-1-carboxamide [4273];

4-((2-methoxyethyl)(methyl)amino)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl) piperidine-1-carboxamide [4274];

4-((1,3-difluoropropan-2-yl)amino)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl) piperidine-1-carboxamide [4275];

N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-4-((3,3,3-trifluoropropyl)amino) piperidine-1-carboxamide [4276];

4-((2-fluoroethyl)amino)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)piperidine-1-carboxamide [4277];

(3R,4S)-4-amino-3-fluoro-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl) piperidine-1-carboxamide [4278];

(3R,4R)-4-amino-3-fluoro-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl) piperidine-1-carboxamide [4279];

(3S,4S)-3-fluoro-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-4-(methylamino) piperidine-1-carboxamide [4280];

(3R,4R)-3-fluoro-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-4-(methylamino) piperidine-1-carboxamide [4281];

4-amino-3,3-difluoro-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)piperidine-1-carboxamide [4282];

(3R,4R)-3-fluoro-4-(isopropylamino)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)piperidine-1-carboxamide [4283];

(3R,4S)-3-fluoro-4-(isopropylamino)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)piperidine-1-carboxamide [4284];

3,3-difluoro-4-(isopropylamino)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl) piperidine-1-carboxamide [4285];

(3S,4S)-3-fluoro-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-4-((propan-2-yl-1,1,1,3,3,3-d 6 )amino)piperidine-1-carboxamide [4286];

(1R,3s,5S)-3-((1,3-difluoropropan-2-yl)amino)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-8-azabicyclo[3.2.1]octane-8-carboxamide [4287];

(1R,3s,5S)-3-((1,3-difluoropropan-2-yl)amino)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-8-azabicyclo[3.2.1]octane-8-carboxamide [4288];

4-(dimethylamino)-N-(6-(2-methylthiazol-5-yl)-2,7-naphthyridin-3-yl)piperidine-1-carboxamide [4289];

4-((2,2-difluoroethyl)amino)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl) piperidine-1-carboxamide [4290];

4-((2,2-difluoroethyl)(methyl-d3)amino)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)piperidine-1-carboxamide [4291];

N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-4-morpholinopiperidine-1-carboxamide [4292];

N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-4-(4-methylpiperazin-1-yl) piperidine-1-carboxamide [4293];

(R)-3,4-dimethyl-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)piperazine-1-carboxamide [4294];

(S)-3,4-dimethyl-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)piperazine-1-carboxamide [4295];

(1R,3r,5S)-3-((2-fluoroethyl)amino)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-8-azabicyclo[3.2.1]octane-8-carboxamide [4296];

(1R,3r,5S)-3-((2,2-difluoroethyl)amino)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-8-azabicyclo[3.2.1]octane-8-carboxamide [4297];

(1R,3r,5S)-3-amino-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-8-azabicyclo [3.2.1]octane-8-carboxamide [4298];

(1 S,4S)-5-methyl-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-2,5-diazabicyclo [2.2.1]heptane-2-carboxamide [4299];

(1R,4R)-5-methyl-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-2,5-diazabicyclo [2.2.1]heptane-2-carboxamide [4300];

8-methyl-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-3,8-diazabicyclo[3.2.1]octane-3-carboxamide [4301];

3-methyl-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-3,8-diazabicyclo[3.2.1]octane-8-carboxamide [4302];

N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-5,6-dihydroimidazo[1,2-a]pyrazine-7(8H)-carboxamide [4303];

2-(4-methylpiperazin-1-yl)-N-(6-(5-methylthiazol-2-yl)-2,7-naphthyridin-3-yl)isonicotinamide [4304];

2-(4-methylpiperazin-1-yl)-N-(6-(4-methylthiazol-2-yl)-2,7-naphthyridin-3-yl)isonicotinamide [4305];

N-(6-(2-(methylamino)thiazol-5-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [4306];

1-methyl-N-(6-(2-(methylamino)thiazol-5-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [4307];

N-(6-(2-(diethylamino)thiazol-5-yl)-2,7-naphthyridin-3-yl)-2-(4-fluoropiperidin-1-yl)acetamide [4308];

N-(6-(2-(diethylamino)thiazol-5-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl)acetamide [4309];

N-(6-(2-aminothiazol-5-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [4310];

N-(6-(2-(methylamino)thiazol-5-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [4311];

N-(6-(2-(dimethylamino)thiazol-5-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [4312];

2-(4-isopropylpiperazin-1-yl)-N-(6-(2-(methylamino)thiazol-5-yl)-2,7-naphthyridin-3-yl) isonicotinamide [4313];

2-(3-(dimethylamino)azetidin-1-yl)-N-(6-(2-(methylamino)thiazol-5-yl)-2,7-naphthyridin-3-yl) isonicotinamide [4314];

2-(3-(dimethylamino)azetidin-1-yl)-N-(6-(2-(dimethylamino)thiazol-5-yl)-2,7-naphthyridin-3-yl) isonicotinamide [4315];

2-(3-aminoazetidin-1-yl)-N-(6-(2-(dimethylamino)thiazol-5-yl)-2,7-naphthyridin-3-yl) isonicotinamide [4316];

N-(6-(5-chlorothiazol-2-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [4317];

2-(6-(2-(4-methylpiperazin-1-yl)isonicotinamido)-2,7-naphthyridin-3-yl)thiazole-5-carboxamide [4318];

N-(6-(isothiazol-4-yl)-2,7-naphthyridin-3-yl)-1-methylpiperidine-4-carboxamide [4319];

N-(6-(1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-4-(difluoromethoxy)benzamide [4320];

N-(6-(1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-4-(piperidin-4-yloxy)benzamide [4321];

N-(6-(1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-4-((1-methylpiperidin-4-yl)oxy)benzamide [4322];

N-(6-(1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-3-((1-methylpiperidin-4-yl)oxy)benzamide [4323];

N 5 -(6-(1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-N 2 -methylpyridine-2,5-dicarboxamide [4324];

N-(6-(1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-6-(4-methylpiperazin-1-yl)nicotinamide [4325];

N-(6-(1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-′-methyl-1′,2′,3′,6′-tetrahydro-[2,4′-bipyridine]-4-carboxamide [4326];

N-(6-(1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-2-(3-(dimethylamino)azetidin-1-yl) isonicotinamide [4327];

N-(6-(1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [4328];

N-(6-(1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-2-(4-isopropylpiperazin-1-yl)isonicotinamide [4329];

N-(6-(1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-2-morpholinoisonicotinamide [4330];

1-fluoro-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)cyclohexane-1-carboxamide [4331];

trans-4-methoxy-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)cyclohexane-1-carboxamide [4332];

cis-4-methoxy-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)cyclohexane-1-carboxamide [4333];

trans-4-amino-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)cyclohexane-1-carboxamide [4334];

trans-4-(dimethylamino)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl) cyclohexane-1-carboxamide [4335];

trans-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-4-morpholinocyclohexane-1-carboxamide [4336];

trans-4-(hydroxymethyl)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl) cyclohexane-1-carboxamide [4337];

N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [4338];

4-fluoro-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [4339];

1-methyl-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [4340];

4-fluoro-1-methyl-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [4341];

1-(2-fluoroethyl)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [4342];

1-(2,2-difluoroethyl)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [4343];

N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [4344];

1-(2,2-difluoropropyl)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [4345];

1-benzoyl-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [4346];

N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide [4347];

N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-2-(piperidin-1-yl)acetamide [4348];

2-(4-methoxypiperidin-1-yl)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl) acetamide [4349];

N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl) acetamide [4350];

N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-2-morpholinoacetamide [4351];

(R)—N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-2-(3-methylmorpholino) acetamide [4352];

2-(7-azabicyclo[2.2.1]heptan-7-yl)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl) acetamide [4353];

2-((1R,4R)-2-oxa-5-azabicyclo[2.2.1]heptan-5-yl)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)acetamide [4354];

2-(3-oxa-8-azabicyclo[3.2.1]octan-8-yl)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)acetamide [4355];

2-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)acetamide [4356];

N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-2-(1,4-oxazepan-4-yl)acetamide [4357];

N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-2-morpholinoacetamide-2,2-d 2 [4358];

N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-2-(morpholino-d 8 )acetamide [4359];

1-methyl-3-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-1-(1-methylpiperidin-4-yl) urea [4360];

(3S,4S)-4-amino-3-fluoro-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl) piperidine-1-carboxamide [4361];

(3 S,4S)-4-(dimethylamino)-3-fluoro-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl) piperidine-1-carboxamide [4362];

N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)morpholine-4-carboxamide [4363];

N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-4-(methylamino)piperidine-1-carboxamide [4364];

4-(dimethylamino)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)piperidine-1-carboxamide [4365];

4-((2,2-difluoroethyl)(methyl)amino)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)piperidine-1-carboxamide [4366];

(3S,4S)-3-fluoro-4-(isopropylamino)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)piperidine-1-carboxamide [4367];

2-methyl-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-5,6-dihydroimidazo[1,2-a]pyrazine-7(8H)-carboxamide [4368];

4-methyl-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)piperazine-1-carboxamide [4369];

N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-1-(1-methylpiperidin-4-yl)-1H-pyrazole-4-carboxamide [4370];

1-(1-isopropylpiperidin-4-yl)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-1H-pyrazole-4-carboxamide [4371];

N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-1-(1-methylpiperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide [4372];

N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-2-(piperidin-4-yl)oxazole-4-carboxamide [4373];

N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-2-(1-methylpiperidin-4-yl)oxazole-4-carboxamide [4374];

2-(3-(dimethylamino)azetidin-1-yl)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl) isonicotinamide [4375];

1′-methyl-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-1′,2′,3′,6′-tetrahydro-[2,4′-bipyridine]-4-carboxamide [4376];

N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [4377];

2-(methyl(1-methylpiperidin-4-yl)amino)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)isonicotinamide [4378];

2-(azetidin-3-yloxy)-N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)isonicotinamide [4379];

N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-3-((1-methylpiperidin-4-yl)oxy) benzamide [4380];

N-(6-(5-methyl-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-2-((1-methylpiperidin-4-yl)thio) isonicotinamide [4381];

6-(4-methylpiperazin-1-yl)-N-(6-(5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)nicotinamide [4382];

2-(4-methylpiperazin-1-yl)-N-(6-(5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)isonicotinamide [4383];

N-(6-(5-amino-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [4384];

N-(6-(5-(dimethylamino)-1,3,4-thiadiazol-2-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [4385];

N-(6-(3-amino-5-fluorophenyl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [4386];

N-(6-(3-fluoro-5-(isopropylamino)phenyl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [4387];

1-methyl-N-(6-(pyridin-2-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [4388];

2-(4-methylpiperazin-1-yl)-N-(6-(pyridin-2-yl)-2,7-naphthyridin-3-yl)isonicotinamide [4389];

2-(4-methylpiperazin-1-yl)-N-(6-(pyridin-4-yl)-2,7-naphthyridin-3-yl)isonicotinamide [4390];

N-(6-(pyridin-3-yl)-2,7-naphthyridin-3-yl)cyclopropanecarboxamide [4391];

N-(6-(pyridin-3-yl)-2,7-naphthyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide [4392];

1-methyl-N-(6-(pyridin-3-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [4393];

N-(6-(pyridin-3-yl)-2,7-naphthyridin-3-yl)quinuclidine-4-carboxamide [4394];

2-morpholino-N-(6-(pyridin-3-yl)-2,7-naphthyridin-3-yl)acetamide [4395];

2-(morpholino-d 8 )—N-(6-(pyridin-3-yl)-2,7-naphthyridin-3-yl)acetamide [4396];

2-(4-methylpiperazin-1-yl)-N-(6-(pyridin-3-yl)-2,7-naphthyridin-3-yl)acetamide [4397];

2-(4-methyl-1,4-diazepan-1-yl)-N-(6-(pyridin-3-yl)-2,7-naphthyridin-3-yl)acetamide [4398];

2-(4-methylpiperazin-1-yl)-N-(6-(pyridin-3-yl)-2,7-naphthyridin-3-yl)isonicotinamide [4399];

2-(2-methyl-1H-imidazol-1-yl)-N-(6-(pyridin-3-yl)-2,7-naphthyridin-3-yl)acetamide [4400];

2-(1H-imidazol-1-yl)-N-(6-(pyridin-3-yl)-2,7-naphthyridin-3-yl)acetamide [4401];

2-(piperidin-4-yl)-N-(6-(pyridin-3-yl)-2,7-naphthyridin-3-yl)oxazole-4-carboxamide [4402];

2-(1-methylpiperidin-4-yl)-N-(6-(pyridin-3-yl)-2,7-naphthyridin-3-yl)oxazole-4-carboxamide [4403];

2-(1-isopropylpiperidin-4-yl)-N-(6-(pyridin-3-yl)-2,7-naphthyridin-3-yl)oxazole-4-carboxamide [4404];

trans-N-(6-(5-fluoropyridin-3-yl)-2,7-naphthyridin-3-yl)-3-morpholinocyclobutane-1-carboxamide [4405];

trans-N-(6-(5-fluoropyridin-3-yl)-2,7-naphthyridin-3-yl)-4-((4-methylpiperazin-1-yl)methyl) cyclohexane-1-carboxamide [4406];

N-(6-(5-fluoropyridin-3-yl)-2,7-naphthyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide [4407];

N-(6-(5-fluoropyridin-3-yl)-2,7-naphthyridin-3-yl)-1-methylpiperidine-4-carboxamide [4408];

N-(6-(5-fluoropyridin-3-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl)acetamide [4409];

N-(6-(6-fluoropyridin-3-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl)acetamide [4410];

N-(6-(5-fluoropyridin-3-yl)-2,7-naphthyridin-3-yl)-2-morpholinoacetamide [4411];

N-(6-(5-fluoropyridin-3-yl)-2,7-naphthyridin-3-yl)-3-morpholinopropanamide [4412];

N-(6-(5-fluoropyridin-3-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [4413];

N-(6-(5-fluoropyridin-3-yl)-2,7-naphthyridin-3-yl)-2-(piperidin-4-yl)oxazole-4-carboxamide [4414];

N-(6-(5-fluoropyridin-3-yl)-2,7-naphthyridin-3-yl)-2-(1-methylpiperidin-4-yl)oxazole-4-carboxamide [4415];

N-(6-(5-fluoropyridin-3-yl)-2,7-naphthyridin-3-yl)-2-(1-isopropylpiperidin-4-yl)oxazole-4-carboxamide [4416];

N-(6-(5-chloropyridin-3-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [4417];

N-(6-(5-methylpyridin-3-yl)-2,7-naphthyridin-3-yl)-2-morpholinoacetamide [4418];

N-(6-(5-(difluoromethyl)pyridin-3-yl)-2,7-naphthyridin-3-yl)-3-(piperidin-4-yl)benzamide [4419];

N-(6-(5-(difluoromethyl)pyridin-3-yl)-2,7-naphthyridin-3-yl)-3-(1-methylpiperidin-4-yl) benzamide [4420];

N-(6-(5-(difluoromethyl)pyridin-3-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [4421];

2-(4-methylpiperazin-1-yl)-N-(6-(5-(trifluoromethyl)pyridin-3-yl)-2,7-naphthyridin-3-yl) acetamide [4422];

2-(4-methylpiperazin-1-yl)-N-(6-(6-(trifluoromethyl)pyridin-3-yl)-2,7-naphthyridin-3-yl) acetamide [4423];

N-(6-(5-(hydroxymethyl)pyridin-3-yl)-2,7-naphthyridin-3-yl)-1-methylpiperidine-4-carboxamide [4424];

N-(6-(5-cyanopyridin-3-yl)-2,7-naphthyridin-3-yl)-1-methylpiperidine-4-carboxamide [4425];

N-(6-(5-methoxypyridin-3-yl)-2,7-naphthyridin-3-yl)-1-methylpiperidine-4-carboxamide [4426];

N-(6-(5-methoxypyridin-3-yl)-2,7-naphthyridin-3-yl)-2-morpholinoacetamide [4427];

N-(6-(5-methoxypyridin-3-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [4428];

4-fluoro-N-(6-(5-(piperidin-4-yloxy)pyridin-3-yl)-2,7-naphthyridin-3-yl)benzamide [4429];

N-(6-(5-aminopyridin-3-yl)-2,7-naphthyridin-3-yl)-4-fluorobenzamide [4430];

N-(6-(5-aminopyridin-3-yl)-2,7-naphthyridin-3-yl)-4-(piperidin-4-yloxy)benzamide [4431];

N-(6-(5-aminopyridin-3-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [4432];

N-(6-(5-aminopyridin-3-yl)-2,7-naphthyridin-3-yl)-2-(piperidin-4-yl)oxazole-4-carboxamide [4433];

N-(6-(6-aminopyridin-3-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [4434];

N-(6-(6-(methylamino)pyridin-3-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [4435];

N-(6-(5-(isopropylamino)pyridin-3-yl)-2,7-naphthyridin-3-yl)-3-(piperidin-4-yl)benzamide [4436];

N-(6-(5-(isopropylamino)pyridin-3-yl)-2,7-naphthyridin-3-yl)-3-(1-methylpiperidin-4-yl) benzamide [4437];

N-(6-(5-(isopropylamino)pyridin-3-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [4438];

N-(6-(5-(piperidin-4-ylamino)pyridin-3-yl)-2,7-naphthyridin-3-yl)cyclohexanecarboxamide [4439];

4-fluoro-N-(6-(5-(piperidin-4-ylamino)pyridin-3-yl)-2,7-naphthyridin-3-yl)benzamide [4440];

4-fluoro-N-(6-(5-((1-methylpiperidin-4-yl)amino)pyridin-3-yl)-2,7-naphthyridin-3-yl)benzamide [4441];

N-(6-(5-acetamidopyridin-3-yl)-2,7-naphthyridin-3-yl)-1-methylpiperidine-4-carboxamide [4442];

N-(6-(5-(dimethylamino)pyridin-3-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [4443];

N-(6-(6-(dimethylamino)pyridin-3-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [4444];

1-methyl-N-(6-(5-(pyrrolidin-1-yl)pyridin-3-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [4445];

N-(6-(5-(pyrrolidin-1-ylmethyl)pyridin-3-yl)-2,7-naphthyridin-3-yl)cyclopropanecarboxamide [4446];

4-fluoro-N-(6-(5-(pyrrolidin-1-ylmethyl)pyridin-3-yl)-2,7-naphthyridin-3-yl)benzamide [4447];

N-(6-(5-((4-hydroxypiperidin-1-yl)methyl)pyridin-3-yl)-2,7-naphthyridin-3-yl) cyclopropanecarboxamide [4448];

4-fluoro-N-(6-(5-((4-hydroxypiperidin-1-yl)methyl)pyridin-3-yl)-2,7-naphthyridin-3-yl) benzamide [4449];

N-(6-(5-(piperazin-1-ylmethyl)pyridin-3-yl)-2,7-naphthyridin-3-yl)cyclopropanecarboxamide [4450];

N-(6-(5-((4-methylpiperazin-1-yl)methyl)pyridin-3-yl)-2,7-naphthyridin-3-yl) cyclopropanecarboxamide [4451];

N-(6-(5-(morpholinomethyl)pyridin-3-yl)-2,7-naphthyridin-3-yl)cyclopropanecarboxamide [4452];

N-methyl-5-(6-(1-methylpiperidine-4-carboxamido)-2,7-naphthyridin-3-yl)nicotinamide [4453];

N-methyl-5-(6-(2-(4-methylpiperazin-1-yl)isonicotinamido)-2,7-naphthyridin-3-yl)nicotinamide [4454];

N-(6-(pyridin-3-yl-d 4 )-2,7-naphthyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide [4455];

2-(4-methylpiperazin-1-yl)-N-(6-(pyridin-3-yl-d 4 )-2,7-naphthyridin-3-yl)acetamide [4456];

2-morpholino-N-(6-(pyridin-3-yl-d 4 )-2,7-naphthyridin-3-yl)acetamide [4457];

1-methyl-N-(6-(2-methylpyrimidin-5-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [4458];

2-(4-methylpiperazin-1-yl)-N-(6-(2-methylpyrimidin-5-yl)-2,7-naphthyridin-3-yl)isonicotinamide [4459];

N-(6-(2-aminopyrimidin-5-yl)-2,7-naphthyridin-3-yl)-1-methylpiperidine-4-carboxamide [4460];

2-morpholino-N-(6-(pyridazin-3-yl)-2,7-naphthyridin-3-yl)acetamide [4461];

2-morpholino-N-(6-(pyridazin-4-yl)-2,7-naphthyridin-3-yl)acetamide [4462];

N-(6-(pyridazin-4-yl)-2,7-naphthyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide [4463];

trans-3-morpholino-N-(6-(pyrazin-2-yl)-2,7-naphthyridin-3-yl)cyclobutane-1-carboxamide [4464];

trans-4-(dimethylamino)-N-(6-(pyrazin-2-yl)-2,7-naphthyridin-3-yl)cyclohexane-1-carboxamide [4465];

trans-4-morpholino-N-(6-(pyrazin-2-yl)-2,7-naphthyridin-3-yl)cyclohexane-1-carboxamide [4466];

trans-4-((3-fluoroazetidin-1-yl)methyl)-N-(6-(pyrazin-2-yl)-2,7-naphthyridin-3-yl) cyclohexane-1-carboxamide [4467];

trans-4-((4-methylpiperazin-1-yl)methyl)-N-(6-(pyrazin-2-yl)-2,7-naphthyridin-3-yl) cyclohexane-1-carboxamide [4468];

N-(6-(pyrazin-2-yl)-2,7-naphthyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide [4469];

1-methyl-N-(6-(pyrazin-2-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [4470];

4-fluoro-1-methyl-N-(6-(pyrazin-2-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [4471];

1-(2-fluoroethyl)-N-(6-(pyrazin-2-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [4472];

1-(oxetan-3-yl)-N-(6-(pyrazin-2-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [4473];

2-morpholino-N-(6-(pyrazin-2-yl)-2,7-naphthyridin-3-yl)acetamide [4474];

1-methyl-N-(6-(pyrazin-2-yl)-2,7-naphthyridin-3-yl)azepane-4-carboxamide [4475];

1-isobutyl-N-(6-(pyrazin-2-yl)-2,7-naphthyridin-3-yl)azepane-4-carboxamide [4476];

1-(2-hydroxy-2-methylpropyl)-N-(6-(pyrazin-2-yl)-2,7-naphthyridin-3-yl)azepane-4-carboxamide [4477];

4-(morpholinomethyl)-N-(6-(pyrazin-2-yl)-2,7-naphthyridin-3-yl)benzamide [4478];

2-(4-methylpiperazin-1-yl)-N-(6-(pyrazin-2-yl)-2,7-naphthyridin-3-yl)isonicotinamide [4479], N-(6-(6-(methylamino)pyrazin-2-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [4480];

N-(6-(6-(isopropylamino)pyrazin-2-yl)-2,7-naphthyridin-3-yl)azetidine-3-carboxamide [4481];

N-(6-(6-(isopropylamino)pyrazin-2-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [4482];

N-(6-(6-(isopropylamino)pyrazin-2-yl)-2,7-naphthyridin-3-yl)-1-methylpiperidine-4-carboxamide [4483];

1-(2-fluoroethyl)-N-(6-(6-(isopropylamino)pyrazin-2-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [4484];

1-isopropyl-N-(6-(6-(isopropylamino)pyrazin-2-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [4485];

1-isopentyl-N-(6-(6-(isopropylamino)pyrazin-2-yl)-2,7-naphthyridin-3-yl)piperidine-4-carboxamide [4486];

N-(6-(6-(isopropylamino)pyrazin-2-yl)-2,7-naphthyridin-3-yl)-3-(piperidin-4-yl)benzamide [4487];

N-(6-(6-(isopropylamino)pyrazin-2-yl)-2,7-naphthyridin-3-yl)-3-(1-methylpiperidin-4-yl) benzamide [4488];

N-(6-(6-(isopropylamino)pyrazin-2-yl)-2,7-naphthyridin-3-yl)-1-(piperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide [4489];

1-(1-(2-fluoroethyl)piperidin-4-yl)-N-(6-(6-(isopropylamino)pyrazin-2-yl)-2,7-naphthyridin-3-yl)-1H-1,2,3-triazole-4-carboxamide [4490];

N-(6-(6-(isopropylamino)pyrazin-2-yl)-2,7-naphthyridin-3-yl)-1-(1-isopropylpiperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide [4491];

N-(6-(6-(isopropylamino)pyrazin-2-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [4492], N-(6-(6-(tert-butylamino)pyrazin-2-yl)-2,7-naphthyridin-3-yl)-2-(3-(dimethylamino)azetidin-1-yl)isonicotinamide [4493];

N-(6-(6-(tert-butylamino)pyrazin-2-yl)-2,7-naphthyridin-3-yl)-1′-methyl-1′,2′,3′,6′-tetrahydro-[2,4′-bipyridine]-4-carboxamide [4494];

N-(6-(6-(tert-butylamino)pyrazin-2-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1l-yl) isonicotinamide [4495];

N-(6-(6-(tert-butylamino)pyrazin-2-yl)-2,7-naphthyridin-3-yl)-2-(4-isopropylpiperazin-1l-yl) isonicotinamide [4496];

N-(6-(6-(tert-butylamino)pyrazin-2-yl)-2,7-naphthyridin-3-yl)-2-morpholinoisonicotinamide [4497];

N-(6-(6-(((3-fluoroazetidin-3-yl)methyl)amino)pyrazin-2-yl)-2,7-naphthyridin-3-yl) cyclopropanecarboxamide [4498];

4-fluoro-N-(6-(6-(((3-fluoroazetidin-3-yl)methyl)amino)pyrazin-2-yl)-2,7-naphthyridin-3-yl) benzamide [4499];

N-(6-(6-(piperidin-4-ylamino)pyrazin-2-yl)-2,7-naphthyridin-3-yl)cyclobutanecarboxamide [4500];

3,3-difluoro-N-(6-(6-(piperidin-4-ylamino)pyrazin-2-yl)-2,7-naphthyridin-3-yl)cyclobutane-1-carboxamide [4501];

N-(6-(6-(piperidin-4-ylamino)pyrazin-2-yl)-2,7-naphthyridin-3-yl)cyclopentanecarboxamide [4502];

4,4-difluoro-N-(6-(6-(piperidin-4-ylamino)pyrazin-2-yl)-2,7-naphthyridin-3-yl)cyclohexane-1-carboxamide [4503];

N-(6-(6-(piperidin-4-ylamino)pyrazin-2-yl)-2,7-naphthyridin-3-yl)tetrahydro-2H-pyran-4-carboxamide [4504];

4-fluoro-N-(6-(6-(piperidin-4-ylamino)pyrazin-2-yl)-2,7-naphthyridin-3-yl)benzamide [4505];

N-(6-(6-(((3 S,4S)-3-fluoropiperidin-4-yl)amino)pyrazin-2-yl)-2,7-naphthyridin-3-yl) cyclopropanecarboxamide [4506];

4-fluoro-N-(6-(6-(((3 S,4S)-3-fluoropiperidin-4-yl)amino)pyrazin-2-yl)-2,7-naphthyridin-3-yl) benzamide [4507];

N-(6-(6-((1-methylpiperidin-4-yl)amino)pyrazin-2-yl)-2,7-naphthyridin-3-yl) cyclobutanecarboxamide [4508];

N-(6-(6-((1-methylpiperidin-4-yl)amino)pyrazin-2-yl)-2,7-naphthyridin-3-yl) cyclopentanecarboxamide [4509];

4-fluoro-N-(6-(6-((1-methylpiperidin-4-yl)amino)pyrazin-2-yl)-2,7-naphthyridin-3-yl)benzamide [4510];

N-(6-(6-((1-isopropylpiperidin-4-yl)amino)pyrazin-2-yl)-2,7-naphthyridin-3-yl) cyclopropanecarboxamide [4511];

3,3-difluoro-N-(6-(6-((1-isopropylpiperidin-4-yl)amino)pyrazin-2-yl)-2,7-naphthyridin-3-yl) cyclobutane-1-carboxamide [4512];

N-(6-(6-((1-isopropylpiperidin-4-yl)amino)pyrazin-2-yl)-2,7-naphthyridin-3-yl) cyclopentanecarboxamide [4513];

4-fluoro-N-(6-(6-((1-isopropylpiperidin-4-yl)amino)pyrazin-2-yl)-2,7-naphthyridin-3-yl) benzamide [4514];

N-(6-(6-(dimethylamino)pyrazin-2-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [4515];

N-(6-(6-(diethylamino)pyrazin-2-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [4516];

N-(6-(6-(3-aminoazetidin-1-yl)pyrazin-2-yl)-2,7-naphthyridin-3-yl)-4-fluorobenzamide [4517];

2-(4-methylpiperazin-1-yl)-N-(6-(6-(pyrrolidin-1-yl)pyrazin-2-yl)-2,7-naphthyridin-3-yl) isonicotinamide [4518];

N-(6-(6-(azetidin-3-ylmethoxy)pyrazin-2-yl)-2,7-naphthyridin-3-yl)-4-fluorobenzamide [4519];

N-(6-(6-(azetidin-3-yloxy)pyrazin-2-yl)-2,7-naphthyridin-3-yl)-4-fluorobenzamide [4520];

N-(6-(1H-pyrrolo[2,3-b]pyridin-5-yl)-2,7-naphthyridin-3-yl)-1-(1-methylpiperidin-4-yl)-1H-pyrazole-4-carboxamide [4521];

N-(6-(1H-pyrrolo[3,2-b]pyridin-6-yl)-2,7-naphthyridin-3-yl)-1-(1-methylpiperidin-4-yl)-1H-pyrazole-4-carboxamide [4522];

N-(6-(1H-pyrrolo[2,3-c]pyridin-4-yl)-2,7-naphthyridin-3-yl)-1-(1-methylpiperidin-4-yl)-1H-pyrazole-4-carboxamide [4523];

N-(6-(1H-pyrrolo[2,3-b]pyridin-5-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [4524];

N-(6-(1H-pyrrolo[3,2-b]pyridin-6-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [4525];

N-(6-(1H-pyrrolo[2,3-c]pyridin-4-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [4526];

2-(4-methylpiperazin-1-yl)-N-(6-(oxazolo[5,4-b]pyridin-6-yl)-2,7-naphthyridin-3-yl) isonicotinamide [4527];

N-(6-(2-methyl-1H-pyrrolo[2,3-b]pyridin-5-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [4528];

N-(6-(3-methyl-1H-pyrrolo[2,3-b]pyridin-5-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [4529];

N-(6-(2-methyl-1H-pyrrolo[3,2-b]pyridin-6-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl)isonicotinamide [4530];

N-(6-(5H-pyrrolo[2,3-b]pyrazin-2-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [4531];

N-(6-(5H-pyrrolo[2,3-b]pyrazin-3-yl)-2,7-naphthyridin-3-yl)-2-(4-methylpiperazin-1-yl) isonicotinamide [4532];

1-isopropyl-N-(6-(6-(piperidin-4-ylamino)pyrazin-2-yl)-2,7-naphthyridin-3-yl)-1H-pyrazole-4-carboxamide [4533];

1-isopropyl-N-(6-(6-((1-methylpiperidin-4-yl)amino)pyrazin-2-yl)-2,7-naphthyridin-3-yl)-1H-pyrazole-4-carboxamide [4534];

trans-4-((2-fluoroethyl)amino)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl) cyclohexane-1-carboxamide [4628];

trans-4-((2-methoxyethyl)amino)-N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl) cyclohexane-1-carboxamide [4629];

tert-butyl (trans-4-((3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)carbamoyl)cyclohexyl) carbamate [4630];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-((1-methylpiperidin-4-yl)amino) isonicotinamide [4631];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl)thiazole-5-carboxamide [4632];

N-(3-(1-methyl-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(4-methylpiperazin-1-yl)thiazole-5-carboxamide [4633];

N-(3-(1-methyl-5-(piperidin-1-ylmethyl)-1H-pyrazol-4-yl)-1,7-naphthyridin-6-yl)-2-(2,7-diazaspiro[3.5]nonan-2-yl)isonicotinamide [4634];

N-(3-(1-methyl-1H-1,2,3-triazol-4-yl)-1,7-naphthyridin-6-yl)-4-(piperidin-4-yloxy)benzamide [4635];

N-(3-(1-methyl-1H-tetrazol-5-yl)-1,7-naphthyridin-6-yl)-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide [4636];

N-(3-(1,2-dimethyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-2-(pyrrolidin-1-yl)propanamide [4637];

N-(3-(1,2-dimethyl-1H-imidazol-5-yl)-1,7-naphthyridin-6-yl)-2-(piperidin-1-yl)propanamide [4638];

4-isopropoxy-N-(3-(7-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-yl)-1,7-naphthyridin-6-yl)benzamide [4639];

trans-3-morpholino-N-(3-(oxazol-5-yl)-1,7-naphthyridin-6-yl)cyclobutane-1-carboxamide [4640];

trans-4-(hydroxymethyl)-N-(3-(oxazol-5-yl)-1,7-naphthyridin-6-yl)cyclohexane-1-carboxamide [4641];

N-(3-(oxazol-5-yl)-1,7-naphthyridin-6-yl)piperidine-4-carboxamide [4642];

4-morpholino-N-(3-(oxazol-5-yl)-1,7-naphthyridin-6-yl)piperidine-1-carboxamide [4643];

N-(3-(oxazol-5-yl)-1,7-naphthyridin-6-yl)-4-(piperidin-4-yloxy)benzamide [4644];

N-(3-(oxazol-5-yl)-1,7-naphthyridin-6-yl)-3-(piperidin-4-yloxy)benzamide [4645];

2-methyl-N-(3-(oxazol-5-yl)-1,7-naphthyridin-6-yl)-5,6-dihydroimidazo[1,2-a]pyrazine-7(8H)-carboxamide [4646];

2-(1H-imidazol-1-yl)-N-(3-(oxazol-5-yl)-1,7-naphthyridin-6-yl)acetamide [4647];

trans-4-(hydroxymethyl)-N-(3-(thiazol-5-yl)-1,7-naphthyridin-6-yl)cyclohexane-1-carboxamide [4648];

trans-4-(dimethylamino)-N-(3-(thiazol-5-yl)-1,7-naphthyridin-6-yl)cyclohexane-1-carboxamide [4649];

N-(3-(thiazol-5-yl)-1,7-naphthyridin-6-yl)-1-((1-(trifluoromethyl)cyclopropyl)methyl)piperidine-4-carboxamide [4650];

trans-4-(hydroxymethyl)-N-(3-(2-methylthiazol-5-yl)-1,7-naphthyridin-6-yl)cyclohexane-1-carboxamide [4651];

trans-4-(dimethylamino)-N-(3-(2-methylthiazol-5-yl)-1,7-naphthyridin-6-yl)cyclohexane-1-carboxamide [4652];

N-(3-(2-methylthiazol-5-yl)-1,7-naphthyridin-6-yl)-1-(oxetan-3-yl)piperidine-4-carboxamide [4653];

N-(3-(2-methylthiazol-5-yl)-1,7-naphthyridin-6-yl)-1-(2-(pyrrolidin-1-yl)acetyl)piperidine-4-carboxamide [4654];

2-((1S,4S)-2-oxa-5-azabicyclo [2.2.1]heptan-5-yl)-N-(3-(5-methyl-1,3,4-thiadiazol-2-yl)-1,7-naphthyridin-6-yl)acetamide [4655];

N-(3-(5-(cyano(4-hydroxypiperidin-1-yl)methyl)pyridin-3-yl)-1,7-naphthyridin-6-yl) cyclopropanecarboxamide [4656];

4-fluoro-N-(3-(6-((1-methylazetidin-3-yl)methoxy)pyrazin-2-yl)-1,7-naphthyridin-6-yl) benzamide [4657];

1-isopropyl-N-(3-(6-((1-methylpiperidin-4-yl)amino)pyrazin-2-yl)-1,7-naphthyridin-6-yl)-1H-pyrazole-4-carboxamide [4658]; or a pharmaceutically acceptable salt thereof.

17. A pharmaceutical composition comprising a therapeutically effective amount of a compound of claim 1 , or a pharmaceutically acceptable salt thereof, and a pharmaceutically acceptable excipient.

Assignments (4)
RELEASE OF SECURITY INTEREST Recorded Mar 12, 2026
From: TMF GROUP NEW YORK, LLC, NOT INDIVIDUALLY BUT SOLELY AS COLLATERAL AGENT
To: BIOSPLICE THERAPEUTICS, INC.
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SECURITY INTEREST Recorded Sep 14, 2022
From: BIOSPLICE THERAPEUTICS, INC.
To: VICKERS VENTURE FUND VI PTE. LTD.; VICKERS VENTURE FUND VI (PLAN) PTE. LTD.; VICKERS-SPLICE CO-INVESTMENT LLC; MED-PATHWAYS II LIMITED
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ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 23, 2021
From: SAMUMED, LLC
To: BIOSPLICE THERAPEUTICS, INC.
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ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 4, 2019
From: KC, SUNIL KUMAR; MAK, CHI CHING; CAO, JIANGUO; BOLLU, VENKATAIAH; CHIRUTA, CHANDRAMOULI; MITTAPALLI, GOPI KUMAR; EASTMAN, BRIAN WALTER; HOFILENA, BRIAN JOSEPH
To: SAMUMED, LLC
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Continuity (2)
Provisional Application 62579883 · Oct 31, 2017
Related Publication 20190127370A1 · May 2, 2019